8WQ9
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8JE0
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![BU of 8je0 by Molmil](/molmil-images/mine/8je0) | A novel amidohydrolase | 分子名称: | 1,2-ETHANEDIOL, Amidase, ZINC ION | 著者 | Ma, D, Feng, R. | 登録日 | 2023-05-15 | 公開日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | A novel amidohydrolase catalyze the degradation of PAM by Klebsiella sp. PCX To Be Published
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8PBG
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![BU of 8pbg by Molmil](/molmil-images/mine/8pbg) | Mutant K1556T of the dihydroorotase domain of human CAD protein bound to the inhibitor fluoroorotate | 分子名称: | 5-FLUORO-2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID, CAD protein, FORMIC ACID, ... | 著者 | del Cano-Ochoa, F, Ramon-Maiques, S. | 登録日 | 2023-06-09 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.46 Å) | 主引用文献 | Beyond genetics: Deciphering the impact of missense variants in CAD deficiency. J Inherit Metab Dis, 46, 2023
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8PBP
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8PBI
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![BU of 8pbi by Molmil](/molmil-images/mine/8pbi) | Mutant R1617Q of the dihydroorotase domain of human CAD protein bound to the inhibitor fluoroorotate | 分子名称: | 5-FLUORO-2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID, CAD protein, FORMIC ACID, ... | 著者 | del Cano-Ochoa, F, Ramon-Maiques, S. | 登録日 | 2023-06-09 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Beyond genetics: Deciphering the impact of missense variants in CAD deficiency. J Inherit Metab Dis, 46, 2023
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8PBE
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8PBM
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8PBQ
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8PBR
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8PBJ
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8PBN
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![BU of 8pbn by Molmil](/molmil-images/mine/8pbn) | Mutant R1789Q of the dihydroorotase domain of human CAD protein bound to the inhibitor fluoorotate | 分子名称: | 5-FLUORO-2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID, CAD protein, FORMIC ACID, ... | 著者 | del Cano-Ochoa, F, Ramon-Maiques, S. | 登録日 | 2023-06-09 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Beyond genetics: Deciphering the impact of missense variants in CAD deficiency. J Inherit Metab Dis, 46, 2023
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8PBT
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8PBU
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![BU of 8pbu by Molmil](/molmil-images/mine/8pbu) | Mutant K1482M of the dihydroorotase domain of human CAD protein bound to the inhibitor fluoorotate | 分子名称: | 5-FLUORO-2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID, CAD protein, FORMIC ACID, ... | 著者 | del Cano-Ochoa, F, Ramon-Maiques, S. | 登録日 | 2023-06-09 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Beyond genetics: Deciphering the impact of missense variants in CAD deficiency. J Inherit Metab Dis, 46, 2023
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8PBH
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8PBK
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![BU of 8pbk by Molmil](/molmil-images/mine/8pbk) | Mutant R1722W of the dihydroorotase domain of human CAD protein bound to the inhibitor fluoorotate | 分子名称: | 5-FLUORO-2,6-DIOXO-1,2,3,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID, CAD protein, FORMIC ACID, ... | 著者 | del Cano-Ochoa, F, Ramon-Maiques, S. | 登録日 | 2023-06-09 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Beyond genetics: Deciphering the impact of missense variants in CAD deficiency. J Inherit Metab Dis, 46, 2023
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8PBS
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8Q2E
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![BU of 8q2e by Molmil](/molmil-images/mine/8q2e) | The 1.68-A X-ray crystal structure of Sporosarcina pasteurii urease inhibited by thiram and bound to dimethylditiocarbamate | 分子名称: | 1,2-ETHANEDIOL, HYDROXIDE ION, NICKEL (II) ION, ... | 著者 | Mazzei, L, Cianci, M, Ciurli, S. | 登録日 | 2023-08-02 | 公開日 | 2023-11-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Kinetic and structural details of urease inactivation by thiuram disulphides. J.Inorg.Biochem., 250, 2023
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8HFD
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![BU of 8hfd by Molmil](/molmil-images/mine/8hfd) | Crystal structure of allantoinase from E. coli BL21 | 分子名称: | Allantoinase, DI(HYDROXYETHYL)ETHER, ZINC ION | 著者 | Lin, E.S, Huang, H.Y, Yang, P.C, Liu, H.W, Huang, C.Y. | 登録日 | 2022-11-10 | 公開日 | 2023-10-18 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.07 Å) | 主引用文献 | Crystal Structure of Allantoinase from Escherichia coli BL21: A Molecular Insight into a Role of the Active Site Loops in Catalysis. Molecules, 28, 2023
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8GW0
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![BU of 8gw0 by Molmil](/molmil-images/mine/8gw0) | Crystal structure of the human dihydroorotase domain in complex with malic acid | 分子名称: | (2S)-2-hydroxybutanedioic acid, CAD protein, ZINC ION | 著者 | Yang, P.C, Liu, H.W, Huang, H.Y, Huang, C.Y. | 登録日 | 2022-09-16 | 公開日 | 2023-09-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.64 Å) | 主引用文献 | Complexed Crystal Structure of the Dihydroorotase Domain of Human CAD Protein with the Anticancer Drug 5-Fluorouracil. Biomolecules, 13, 2023
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8GVZ
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![BU of 8gvz by Molmil](/molmil-images/mine/8gvz) | Crystal structure of the human dihydroorotase domain in complex with the anticancer drug 5-fluorouracil | 分子名称: | 5-FLUOROURACIL, CAD protein, ZINC ION | 著者 | Liu, H.W, Yang, P.C, Huang, H.Y, Huang, C.Y. | 登録日 | 2022-09-16 | 公開日 | 2023-09-20 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Complexed Crystal Structure of the Dihydroorotase Domain of Human CAD Protein with the Anticancer Drug 5-Fluorouracil. Biomolecules, 13, 2023
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8IHQ
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![BU of 8ihq by Molmil](/molmil-images/mine/8ihq) | Cryo-EM structure of ochratoxin A-detoxifying amidohydrolase ADH3 | 分子名称: | Amidohydrolase family protein, ZINC ION | 著者 | Dai, L.H, Niu, D, Huang, J.-W, Li, X, Shen, P.P, Li, H, Hu, Y.M, Yang, Y, Chen, C.-C, Guo, R.-T. | 登録日 | 2023-02-23 | 公開日 | 2023-08-30 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.71 Å) | 主引用文献 | Cryo-EM structure and rational engineering of a superefficient ochratoxin A-detoxifying amidohydrolase. J Hazard Mater, 458, 2023
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8J85
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![BU of 8j85 by Molmil](/molmil-images/mine/8j85) | Cryo-EM structure of ochratoxin A-detoxifying amidohydrolase ADH3 mutant S88E in complex with ochratoxin A | 分子名称: | (2~{S})-2-[[(3~{R})-5-chloranyl-3-methyl-8-oxidanyl-1-oxidanylidene-3,4-dihydroisochromen-7-yl]carbonylamino]-3-phenyl-propanoic acid, Amidohydrolase family protein, ZINC ION | 著者 | Dai, L.H, Niu, D, Huang, J.-W, Li, X, Shen, P.P, Li, H, Hu, Y.M, Yang, Y, Chen, C.-C, Guo, R.-T. | 登録日 | 2023-04-30 | 公開日 | 2023-08-30 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Cryo-EM structure and rational engineering of a superefficient ochratoxin A-detoxifying amidohydrolase. J Hazard Mater, 458, 2023
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8IHS
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![BU of 8ihs by Molmil](/molmil-images/mine/8ihs) | Cryo-EM structure of ochratoxin A-detoxifying amidohydrolase ADH3 in complex with ochratoxin A | 分子名称: | (2~{S})-2-[[(3~{R})-5-chloranyl-3-methyl-8-oxidanyl-1-oxidanylidene-3,4-dihydroisochromen-7-yl]carbonylamino]-3-phenyl-propanoic acid, Amidohydrolase family protein, ZINC ION | 著者 | Dai, L.H, Niu, D, Huang, J.-W, Li, X, Shen, P.P, Li, H, Hu, Y.M, Yang, Y, Chen, C.-C, Guo, R.-T. | 登録日 | 2023-02-23 | 公開日 | 2023-08-30 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Cryo-EM structure and rational engineering of a superefficient ochratoxin A-detoxifying amidohydrolase. J Hazard Mater, 458, 2023
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8IHR
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![BU of 8ihr by Molmil](/molmil-images/mine/8ihr) | Cryo-EM structure of ochratoxin A-detoxifying amidohydrolase ADH3 in complex with Phe | 分子名称: | Amidohydrolase family protein, PHENYLALANINE, ZINC ION | 著者 | Dai, L.H, Niu, D, Huang, J.-W, Li, X, Shen, P.P, Li, H, Hu, Y.M, Yang, Y, Chen, C.-C, Guo, R.-T. | 登録日 | 2023-02-23 | 公開日 | 2023-08-30 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Cryo-EM structure and rational engineering of a superefficient ochratoxin A-detoxifying amidohydrolase. J Hazard Mater, 458, 2023
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8A18
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![BU of 8a18 by Molmil](/molmil-images/mine/8a18) | 1.63 A resolution hydroquinone inhibited Sporosarcina pasteurii urease | 分子名称: | 1,2-ETHANEDIOL, HYDROXIDE ION, NICKEL (II) ION, ... | 著者 | Mazzei, L, Ciurli, S, Cianci, M. | 登録日 | 2022-06-01 | 公開日 | 2023-06-14 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Inhibition of Urease by Hydroquinones: A Structural and Kinetic Study. Chemistry, 28, 2022
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