5C1V
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![BU of 5c1v by Molmil](/molmil-images/mine/5c1v) | CRYSTAL STRUCTURE ANALYSIS OF CATALYTIC SUBUNIT OF HUMAN CALCINEURIN | 分子名称: | FE (III) ION, PHOSPHATE ION, Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform, ... | 著者 | Guasch, A, Fita, I, Perez-Luque, R, Aparicio, D, Aranguren-Ibanez, A, Perez-Riba, M. | 登録日 | 2015-06-15 | 公開日 | 2016-02-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.35 Å) | 主引用文献 | Calcineurin Undergoes a Conformational Switch Evoked via Peptidyl-Prolyl Isomerization. Plos One, 10, 2015
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6PIB
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![BU of 6pib by Molmil](/molmil-images/mine/6pib) | Structure of the Klebsiella pneumoniae LpxH-AZ1 complex | 分子名称: | 1-[5-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}sulfonyl)-2,3-dihydro-1H-indol-1-yl]ethan-1-one, MANGANESE (II) ION, TETRAETHYLENE GLYCOL, ... | 著者 | Cho, J, Zhou, P. | 登録日 | 2019-06-26 | 公開日 | 2020-02-12 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Structural basis of the UDP-diacylglucosamine pyrophosphohydrolase LpxH inhibition by sulfonyl piperazine antibiotics. Proc.Natl.Acad.Sci.USA, 117, 2020
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4TUG
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![BU of 4tug by Molmil](/molmil-images/mine/4tug) | Crystal structure of MjMre11-DNA2 complex | 分子名称: | DNA (5'-D(P*CP*TP*GP*TP*CP*CP*TP*AP*CP*GP*TP*GP*CP*CP*A)-3'), DNA (5'-D(P*GP*CP*AP*CP*GP*TP*AP*GP*GP*AP*CP*AP*GP*C)-3'), DNA double-strand break repair protein Mre11, ... | 著者 | Sung, S, Cho, Y. | 登録日 | 2014-06-24 | 公開日 | 2014-10-15 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.55 Å) | 主引用文献 | DNA end recognition by the Mre11 nuclease dimer: insights into resection and repair of damaged DNA. Embo J., 33, 2014
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4O24
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![BU of 4o24 by Molmil](/molmil-images/mine/4o24) | DNA Double-Strand Break Repair Pathway Choice Is Directed by Distinct MRE11 Nuclease Activities | 分子名称: | (5~{Z})-5-[(4-hydroxyphenyl)methylidene]-3-(2-methylpropyl)-2-sulfanylidene-1,3-thiazolidin-4-one, Exonuclease, putative, ... | 著者 | Shibata, A, Moiani, D, Arvai, A.S, Perry, J, Harding, S.M, Genois, M, Maity, R, Rossum-Fikkert, S, Kertokalio, A, Romoli, F, Ismail, A, Ismalaj, E, Petricci, E, Neale, M.J, Bristow, R.G, Masson, J, Wyman, C, Jeggo, P.A, Tainer, J.A. | 登録日 | 2013-12-16 | 公開日 | 2014-01-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | DNA Double-Strand Break Repair Pathway Choice Is Directed by Distinct MRE11 Nuclease Activities. Mol.Cell, 53, 2014
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4NZV
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![BU of 4nzv by Molmil](/molmil-images/mine/4nzv) | DNA Double-Strand Break Repair Pathway Choice Is Directed by Distinct MRE11 Nuclease Activities | 分子名称: | Exonuclease, putative, MANGANESE (II) ION | 著者 | Shibata, A, Moiani, D, Arvai, A.S, Perry, J, Harding, S.M, Genois, M, Maity, R, Rossum-Fikkert, S, Kertokalio, A, Romoli, F, Ismail, A, Ismalaj, E, Petricci, E, Neale, M.J, Bristow, R.G, Masson, J, Wyman, C, Jeggo, P.A, Tainer, J.A. | 登録日 | 2013-12-12 | 公開日 | 2014-01-08 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.901 Å) | 主引用文献 | DNA Double-Strand Break Repair Pathway Choice Is Directed by Distinct MRE11 Nuclease Activities. Mol.Cell, 53, 2014
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4TUI
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![BU of 4tui by Molmil](/molmil-images/mine/4tui) | Crystal structure of MjMre11-DNA1 complex | 分子名称: | DNA (5'-D(P*TP*CP*CP*TP*AP*CP*GP*TP*GP*CP*CP*AP*G)-3'), DNA (5'-D(P*TP*GP*GP*CP*AP*CP*GP*TP*AP*GP*GP*AP*C)-3'), DNA double-strand break repair protein Mre11 | 著者 | Sung, S, Cho, Y. | 登録日 | 2014-06-24 | 公開日 | 2014-10-15 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.59 Å) | 主引用文献 | DNA end recognition by the Mre11 nuclease dimer: insights into resection and repair of damaged DNA. Embo J., 33, 2014
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1G5B
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![BU of 1g5b by Molmil](/molmil-images/mine/1g5b) | BACTERIOPHAGE LAMBDA SER/THR PROTEIN PHOSPHATASE | 分子名称: | MANGANESE (II) ION, MERCURY (II) ION, SERINE/THREONINE PROTEIN PHOSPHATASE, ... | 著者 | Voegtli, W.C, White, D.J, Reiter, N.J, Rusnak, F, Rosenzweig, A.C. | 登録日 | 2000-10-31 | 公開日 | 2001-03-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structure of the bacteriophage lambda Ser/Thr protein phosphatase with sulfate ion bound in two coordination modes. Biochemistry, 39, 2000
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3JYF
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![BU of 3jyf by Molmil](/molmil-images/mine/3jyf) | The crystal structure of a 2,3-cyclic nucleotide 2-phosphodiesterase/3-nucleotidase bifunctional periplasmic precursor protein from Klebsiella pneumoniae subsp. pneumoniae MGH 78578 | 分子名称: | 2',3'-cyclic nucleotide 2'-phosphodiesterase/3'-nucleotidase bifunctional periplasmic protein, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, ... | 著者 | Fan, Y, Volkart, L, Cobb, G, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2009-09-21 | 公開日 | 2009-09-29 | 最終更新日 | 2017-11-01 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | The crystal structure of a 2,3-cyclic nucleotide 2-phosphodiesterase/3-nucleotidase bifunctional periplasmic precursor protein from Klebsiella pneumoniae subsp. pneumoniae MGH 78578 To be Published
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6HMF
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![BU of 6hmf by Molmil](/molmil-images/mine/6hmf) | D-family DNA polymerase - DP1 subunit (3'-5' proof-reading exonuclease) H451 proof-reading deficient variant | 分子名称: | ACETATE ION, CACODYLATE ION, CALCIUM ION, ... | 著者 | Raia, P, Delarue, M, Sauguet, L. | 登録日 | 2018-09-12 | 公開日 | 2019-01-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure of the DP1-DP2 PolD complex bound with DNA and its implications for the evolutionary history of DNA and RNA polymerases. PLoS Biol., 17, 2019
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3THN
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![BU of 3thn by Molmil](/molmil-images/mine/3thn) | |
3TGH
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![BU of 3tgh by Molmil](/molmil-images/mine/3tgh) | GAP50 the anchor in the inner membrane complex of Plasmodium | 分子名称: | COBALT (II) ION, DIMETHYL SULFOXIDE, Glideosome-associated protein 50, ... | 著者 | Bosch, J, Paige, M.H, Vaidya, A, Bergman, L, Hol, W.G.J. | 登録日 | 2011-08-17 | 公開日 | 2012-03-07 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of GAP50, the anchor of the invasion machinery in the inner membrane complex of Plasmodium falciparum. J.Struct.Biol., 178, 2012
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4B2O
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![BU of 4b2o by Molmil](/molmil-images/mine/4b2o) | Crystal structure of Bacillus subtilis YmdB, a global regulator of late adaptive responses. | 分子名称: | FE (II) ION, PHOSPHATE ION, YMDB PHOSPHODIESTERASE | 著者 | Newman, J.A, Diethmaier, C, Kovacs, A.T, Rodrigues, C, Kuipers, O.P, Stulke, J, Lewis, R.J. | 登録日 | 2012-07-17 | 公開日 | 2013-07-24 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.64 Å) | 主引用文献 | The Ymdb Phosphodiesterase is a Global Regulator of Late Adaptive Responses in Bacillus Subtilis. J.Bacteriol., 196, 2014
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6ASC
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![BU of 6asc by Molmil](/molmil-images/mine/6asc) | Mre11 dimer in complex with Endonuclease inhibitor PFM04 | 分子名称: | (5E)-3-butyl-5-[(4-hydroxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one, 1,2-ETHANEDIOL, MANGANESE (II) ION, ... | 著者 | Moiani, D, Arvai, A.S, Tainer, J.A. | 登録日 | 2017-08-24 | 公開日 | 2018-03-07 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Targeting Allostery with Avatars to Design Inhibitors Assessed by Cell Activity: Dissecting MRE11 Endo- and Exonuclease Activities. Meth. Enzymol., 601, 2018
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2QJC
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![BU of 2qjc by Molmil](/molmil-images/mine/2qjc) | Crystal structure of a putative diadenosine tetraphosphatase | 分子名称: | Diadenosine tetraphosphatase, putative, MANGANESE (II) ION, ... | 著者 | Sugadev, R, Burley, S.K, Swaminathan, S, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2007-07-06 | 公開日 | 2007-07-24 | 最終更新日 | 2021-02-03 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural genomics of protein phosphatases. J.Struct.Funct.Genom., 8, 2007
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2Q8U
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![BU of 2q8u by Molmil](/molmil-images/mine/2q8u) | |
1UTE
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![BU of 1ute by Molmil](/molmil-images/mine/1ute) | PIG PURPLE ACID PHOSPHATASE COMPLEXED WITH PHOSPHATE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ISOPROPYL ALCOHOL, MU-OXO-DIIRON, ... | 著者 | Guddat, L.W, Mcalpine, A, Hume, D, Hamilton, S, De Jersey, J, Martin, J.L. | 登録日 | 1999-01-18 | 公開日 | 1999-10-01 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Crystal structure of mammalian purple acid phosphatase. Structure Fold.Des., 7, 1999
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6PH9
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![BU of 6ph9 by Molmil](/molmil-images/mine/6ph9) | Crystal Structure of the Klebsiella pneumoniae LpxH-lipid X complex | 分子名称: | (R)-((2R,3S,4R,5R,6R)-3-HYDROXY-2-(HYDROXYMETHYL)-5-((R)-3-HYDROXYTETRADECANAMIDO)-6-(PHOSPHONOOXY)TETRAHYDRO-2H-PYRAN-4-YL) 3-HYDROXYTETRADECANOATE, 1,2-ETHANEDIOL, CALCIUM ION, ... | 著者 | Cho, J, Zhou, P. | 登録日 | 2019-06-25 | 公開日 | 2020-02-12 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Structural basis of the UDP-diacylglucosamine pyrophosphohydrolase LpxH inhibition by sulfonyl piperazine antibiotics. Proc.Natl.Acad.Sci.USA, 117, 2020
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6PJ3
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![BU of 6pj3 by Molmil](/molmil-images/mine/6pj3) | Crystal structure of the Klebsiella pneumoniae LpxH/JH-LPH-33 complex | 分子名称: | 1,2-ETHANEDIOL, 1-[5-({4-[3-chloro-5-(trifluoromethyl)phenyl]piperazin-1-yl}sulfonyl)-2,3-dihydro-1H-indol-1-yl]ethan-1-one, MANGANESE (II) ION, ... | 著者 | Cho, J, Zhou, P. | 登録日 | 2019-06-27 | 公開日 | 2020-02-12 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural basis of the UDP-diacylglucosamine pyrophosphohydrolase LpxH inhibition by sulfonyl piperazine antibiotics. Proc.Natl.Acad.Sci.USA, 117, 2020
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1WAR
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![BU of 1war by Molmil](/molmil-images/mine/1war) | Recombinant Human Purple Acid Phosphatase expressed in Pichia Pastoris | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, FE (III) ION, HUMAN PURPLE ACID PHOSPHATASE, ... | 著者 | Duff, A.P, Langley, D.B, Han, R, Averill, B.A, Freeman, H.C, Guss, J.M. | 登録日 | 2004-10-28 | 公開日 | 2005-07-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Crystal Structures of Recombinant Human Purple Acid Phosphatase with and without an Inhibitory Conformation of the Repression Loop. J.Mol.Biol., 351, 2005
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1XM7
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![BU of 1xm7 by Molmil](/molmil-images/mine/1xm7) | |
1V73
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![BU of 1v73 by Molmil](/molmil-images/mine/1v73) | Crystal Structure of Cold-Active Protein-Tyrosine Phosphatase of a Psychrophile Shewanella SP. | 分子名称: | ACETIC ACID, CALCIUM ION, psychrophilic phosphatase I | 著者 | Tsuruta, H, Mikami, B, Aizono, Y. | 登録日 | 2003-12-09 | 公開日 | 2005-03-01 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Crystal Structure of Cold-Active Protein-Tyrosine Phosphatase from a Psychrophile, Shewanella sp J.Biochem.(Tokyo), 137, 2005
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2AHD
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![BU of 2ahd by Molmil](/molmil-images/mine/2ahd) | |
1II7
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![BU of 1ii7 by Molmil](/molmil-images/mine/1ii7) | Crystal structure of P. furiosus Mre11 with manganese and dAMP | 分子名称: | 2'-DEOXYADENOSINE-5'-MONOPHOSPHATE, MANGANESE (II) ION, Mre11 nuclease, ... | 著者 | Hopfner, K.-P, Karcher, A, Craig, L, Woo, T.T, Carney, J.P, Tainer, J.A. | 登録日 | 2001-04-20 | 公開日 | 2001-05-30 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural biochemistry and interaction architecture of the DNA double-strand break repair Mre11 nuclease and Rad50-ATPase. Cell(Cambridge,Mass.), 105, 2001
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6WII
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![BU of 6wii by Molmil](/molmil-images/mine/6wii) | Crystal structure of the K. pneumoniae LpxH/JH-LPH-41 complex | 分子名称: | 5-({[4-({4-[3-chloro-5-(trifluoromethyl)phenyl]piperazin-1-yl}sulfonyl)phenyl]carbamoyl}amino)-N-hydroxypentanamide, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Cochrane, C.S, Cho, J, Fenton, B.A, Zhou, P. | 登録日 | 2020-04-09 | 公開日 | 2020-07-29 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Synthesis and evaluation of sulfonyl piperazine LpxH inhibitors. Bioorg.Chem., 102, 2020
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6X1Z
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![BU of 6x1z by Molmil](/molmil-images/mine/6x1z) | Mre11 dimer in complex with small molecule modulator PFMJ | 分子名称: | (5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, MAGNESIUM ION, ... | 著者 | Arvai, A.S, Moiani, D, Tainer, J.A. | 登録日 | 2020-05-19 | 公開日 | 2020-06-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Fragment- and structure-based drug discovery for developing therapeutic agents targeting the DNA Damage Response. Prog.Biophys.Mol.Biol., 163, 2021
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