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1M8O
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Platelet integrin alfaIIb-beta3 cytoplasmic domain
分子名称: platelet integrin alfaIIb subunit: cytoplasmic domain, platelet integrin beta3 subunit: cytoplasmic domain
著者Vinogradova, O, Velyvis, A, Velyviene, A, Hu, B, Haas, T, Plow, E.F, Qin, J.
登録日2002-07-25
公開日2002-09-18
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献A Structural mechanism of integrin alfaiib beta3 "Inside-out" Activation as regulated by its cytoplasmic face.
Cell(Cambridge,Mass.), 110, 2002
1M2J
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BU of 1m2j by Molmil
Sir2 homologue H80N mutant-ADP ribose complex
分子名称: ADENOSINE-5-DIPHOSPHORIBOSE, Silent Information Regulator 2, ZINC ION
著者Chang, J, Cho, Y.
登録日2002-06-24
公開日2003-04-08
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural basis for the NAD-dependent deacetylase mechanism of Sir2
J.BIOL.CHEM., 277, 2002
4YXQ
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PksG, a HMG-CoA Synthase from Bacillus subtilis
分子名称: DI(HYDROXYETHYL)ETHER, Polyketide biosynthesis 3-hydroxy-3-methylglutaryl-ACP synthase PksG
著者Nair, A.V, Race, P.R, Till, M.
登録日2015-03-23
公開日2016-06-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献PksG, a HMG-CoA Synthase from Bacillus subtilis
To Be Published
1M2X
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Crystal Structure of the metallo-beta-lactamase BlaB of Chryseobacterium meningosepticum in complex with the inhibitor D-captopril
分子名称: 1-(3-MERCAPTO-2-METHYL-PROPIONYL)-PYRROLIDINE-2-CARBOXYLIC ACID, GLYCEROL, SODIUM ION, ...
著者Garcia-Saez, I, Dideberg, O.
登録日2002-06-26
公開日2003-07-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The 1.5 A structure of Chryseobacterium meningosepticum Zn-beta-lactamase in complex with the inhibitor, D-captopril
J.Biol.Chem., 278, 2003
4YYF
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The crystal structure of a glycosyl hydrolase of GH3 family member from [Mycobacterium smegmatis str. MC2 155
分子名称: ACETATE ION, Beta-N-acetylhexosaminidase, FORMIC ACID, ...
著者Tan, K, Hatzos-Skintges, C, Clancy, S, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2015-03-23
公開日2015-04-08
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献The crystal structure of a glycosyl hydrolase of GH3 family member from [Mycobacterium smegmatis str. MC2 155
To Be Published
4YZ2
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Crystal Structure of Streptococcus pneumoniae NanC, in complex with 2-deoxy-2,3-didehydro-N-acetylneuraminic acid.
分子名称: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, SULFATE ION, Sialidase NanC
著者Lukacik, P, Owen, C.D, Potter, J.A, Taylor, G.L, Walsh, M.A.
登録日2015-03-24
公開日2015-09-23
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Streptococcus pneumoniae NanC: STRUCTURAL INSIGHTS INTO THE SPECIFICITY AND MECHANISM OF A SIALIDASE THAT PRODUCES A SIALIDASE INHIBITOR.
J.Biol.Chem., 290, 2015
1M9Y
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X-ray crystal structure of Cyclophilin A/HIV-1 CA N-terminal domain (1-146) M-type H87A,G89A Complex.
分子名称: Cyclophilin A, HIV-1 Capsid
著者Howard, B.R, Vajdos, F.F, Li, S, Sundquist, W.I, Hill, C.P.
登録日2002-07-30
公開日2003-05-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural insights into the catalytic mechanism of cyclophilin A
Nat.Struct.Biol., 10, 2003
1M3A
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Solution structure of a circular form of the truncated N-terminal SH3 domain from oncogene protein c-Crk.
分子名称: Proto-oncogene C-crk
著者Schumann, F.H, Varadan, R, Tayakuniyil, P.P, Hall, J.B, Camarero, J.A, Fushman, D.
登録日2002-06-27
公開日2003-08-05
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献Changing protein backbone topology: Structural and dynamic consequences of the backbone cyclization in SH3 domain
To be Published
4YZV
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Precleavage 70S structure of the P. vulgaris HigB deltaH92 toxin bound to the ACA codon
分子名称: 16S rRNA, 23S rRNA, 30S ribosomal protein S10, ...
著者Schureck, M.A, Dunkle, J.A, Maehigashi, T, Dunham, C.M.
登録日2015-03-25
公開日2015-10-21
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Defining the mRNA recognition signature of a bacterial toxin protein.
Proc.Natl.Acad.Sci.USA, 112, 2015
1MAJ
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SOLUTION STRUCTURE OF AN ISOLATED ANTIBODY VL DOMAIN
分子名称: IGG2A-KAPPA 26-10 FV (LIGHT CHAIN)
著者Constantine, K.L, Friedrichs, M.S, Metzler, W.J, Wittekind, M, Hensley, P, Mueller, L.
登録日1993-09-16
公開日1994-01-31
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Solution structure of an isolated antibody VL domain.
J.Mol.Biol., 236, 1994
4ZJI
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PAK1 in complex with 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine
分子名称: 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine, MAGNESIUM ION, Serine/threonine-protein kinase PAK 1
著者Gutmann, S, Rummel, G.
登録日2015-04-29
公開日2015-06-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor.
Acs Med.Chem.Lett., 6, 2015
1M3K
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biosynthetic thiolase, inactive C89A mutant
分子名称: Acetyl-CoA acetyltransferase, GLYCEROL, SULFATE ION
著者Kursula, P, Ojala, J, Lambeir, A.-M, Wierenga, R.K.
登録日2002-06-28
公開日2002-11-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The catalytic cycle of biosynthetic thiolase: A conformational journey of an acetyl group through four binding modes and two oxyanion holes
Biochemistry, 41, 2002
4ZJQ
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Crystal structure of AcrB deletion mutant in complex with antibiotic in P21 space group
分子名称: DODECYL-BETA-D-MALTOSIDE, ERYTHROMYCIN A, Multidrug efflux pump subunit AcrB, ...
著者Ababou, A, Koronakis, V.
登録日2015-04-29
公開日2016-07-27
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.592 Å)
主引用文献Structures of Gate Loop Variants of the AcrB Drug Efflux Pump Bound by Erythromycin Substrate.
Plos One, 11, 2016
1MBQ
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Anionic Trypsin from Pacific Chum Salmon
分子名称: BENZAMIDINE, CALCIUM ION, Trypsin
著者Toyota, E, Ng, K.K.S, Kuninaga, S, Sekizaki, H, Itoh, K, Tanizawa, K, James, M.N.G.
登録日2002-08-03
公開日2002-12-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure and Nucleotide Sequence of an Anionic Trypsin from Chum Salmon (Oncorhynchus keta) in Comparison with Atlantic Salmon (Salmo salar) and Bovine Trypsin
J.Mol.Biol., 324, 2002
1MBZ
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BETA-LACTAM SYNTHETASE WITH TRAPPED INTERMEDIATE
分子名称: ARGININE-N-METHYLCARBONYL PHOSPHORIC ACID 5'-ADENOSINE ESTER, BETA-LACTAM SYNTHETASE, GLYCEROL, ...
著者Miller, M.T, Bachmann, B.O, Townsend, C.A, Rosenzweig, A.C.
登録日2002-08-04
公開日2002-10-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献The catalytic cycle of beta -lactam synthetase observed by x-ray crystallographic snapshots
Proc.Natl.Acad.Sci.USA, 99, 2002
4YXK
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Crystal structure of Elk prion protein complexed with POM1 FAB
分子名称: Major prion protein, POM1 FAB HEAVY CHAIN, POM1 FAB LIGHT CHAIN, ...
著者Baral, P.K, Swayampakula, M, James, M.N.G.
登録日2015-03-23
公開日2015-09-23
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.805 Å)
主引用文献X-ray structural and molecular dynamical studies of the globular domains of cow, deer, elk and Syrian hamster prion proteins.
J.Struct.Biol., 192, 2015
4YXY
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Computationally designed left-handed alpha/alpha toroid with 9 repeats; two linked rings of 12 repeats each structure
分子名称: dTor_9x31L
著者Doyle, L, Stoddard, B.L, Bradley, P.
登録日2015-03-23
公開日2015-12-16
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.203 Å)
主引用文献Rational design of alpha-helical tandem repeat proteins with closed architectures.
Nature, 528, 2015
1M47
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Crystal Structure of Human Interleukin-2
分子名称: SULFATE ION, interleukin-2
著者Arkin, M.A, Randal, M, DeLano, W.L, Hyde, J, Luong, T.N, Oslob, J.D, Raphael, D.R, Taylor, L, Wang, J, Wells, J.A, McDowell, R.S, Wells, J.A, Braisted, A.C.
登録日2002-07-02
公開日2002-07-31
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Binding of small molecules to an adaptive protein-protein interface.
Proc.Natl.Acad.Sci.USA, 100, 2003
4YYA
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The structure of hemagglutinin from a H6N1 influenza virus (A/Taiwan/2/2013) in complex with avian receptor analog 3'SLNLN
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, HA1, HA2, ...
著者Wang, F, Qi, J, Bi, Y, Zhang, W, Wang, M, Wang, M, Liu, J, Yan, J, Shi, Y, Gao, G.F.
登録日2015-03-23
公開日2016-04-13
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.595 Å)
主引用文献Structure of hemagglutinin from a H6N1 influenza virus (A/chicken/Taiwan/A2837/2013)
To Be Published
1MCJ
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PRINCIPLES AND PITFALLS IN DESIGNING SITE DIRECTED PEPTIDE LIGANDS
分子名称: ACETYL GROUP, AMINO GROUP, D-PHENYLALANINE, ...
著者Edmundson, A.B, Harris, D.L, Fan, Z.-C, Guddat, L.W.
登録日1993-02-25
公開日1994-01-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Principles and pitfalls in designing site-directed peptide ligands.
Proteins, 16, 1993
4YYL
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Phenolic acid derivative bound to influenza strain H1N1 polymerase subunit PA endonuclease
分子名称: 2-(4-fluorophenoxy)-1-(2,3,4-trihydroxyphenyl)ethanone, MANGANESE (II) ION, Polymerase acidic protein, ...
著者Fudo, S, Yamamoto, N, Nukaga, M, Odagiri, T, Tashiro, M, Neya, S, Hoshino, T.
登録日2015-03-24
公開日2015-04-29
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.905 Å)
主引用文献Structural and computational study on inhibitory compounds for endonuclease activity of influenza virus polymerase
Bioorg.Med.Chem., 23, 2015
1MCW
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THREE-DIMENSIONAL STRUCTURE OF A HYBRID LIGHT CHAIN DIMER. PROTEIN ENGINEERING OF A BINDING CAVITY
分子名称: IMMUNOGLOBULIN MCG (LIGHT CHAIN), IMMUNOGLOBULIN WEIR (LIGHT CHAIN)
著者Ely, K.R, Herron, J.N, Edmundson, A.B.
登録日1989-05-09
公開日1990-10-15
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Three-dimensional structure of a hybrid light chain dimer: protein engineering of a binding cavity.
Mol.Immunol., 27, 1990
1M4C
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Crystal Structure of Human Interleukin-2
分子名称: interleukin-2
著者Arkin, M.A, Randal, M, DeLano, W.L, Hyde, J, Luong, T.N, Oslob, J.D, Raphael, D.R, Taylor, L, Wang, J, McDowell, R.S, Wells, J.A, Braisted, A.C.
登録日2002-07-02
公開日2002-07-31
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Binding of small molecules to an adaptive protein-protein interface
Proc.Natl.Acad.Sci.USA, 100, 2003
4YYP
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Crystal structure of human PLK4-PB3 in complex with STIL-CC
分子名称: CHLORIDE ION, SCL-interrupting locus protein, Serine/threonine-protein kinase PLK4
著者Imseng, S, Arquint, C, Gabryjonczyk, A, Boehm, R, Sauer, E, Hiller, S, Nigg, E.A, Maier, T.
登録日2015-03-24
公開日2015-07-29
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献STIL binding to Polo-box 3 of PLK4 regulates centriole duplication.
Elife, 4, 2015
4YZ1
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Crystal Structure of Streptococcus pneumoniae NanC, apo structure.
分子名称: Putative neuraminidase, SULFATE ION
著者Lukacik, P, Owen, D.O, Potter, J.A, Taylor, G.L, Walsh, M.A.
登録日2015-03-24
公開日2015-09-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Streptococcus pneumoniae NanC: STRUCTURAL INSIGHTS INTO THE SPECIFICITY AND MECHANISM OF A SIALIDASE THAT PRODUCES A SIALIDASE INHIBITOR.
J.Biol.Chem., 290, 2015

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