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8TLV
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Crystal structure of MBP and AF9 AHD fusion protein 4AQK in complex with peptidomimetic inhibitor 28
分子名称: GLUTATHIONE, MBP and AF9 AHD fusion protein 4AQK, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ...
著者Yang, Y, Nikolovska-Coleska, Z.
登録日2023-07-27
公開日2024-05-29
実験手法X-RAY DIFFRACTION (2.659 Å)
主引用文献Structural studies of intrinsically disordered MLL-fusion protein AF9 in complex with peptidomimetic inhibitors.
Protein Sci., 33, 2024
8TLW
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Crystal structure of MBP and AF9 AHD fusion protein 3AQA in complex with peptidomimetic inhibitor 28
分子名称: MBP and AF9 AHD fusion protein 3AQA, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, peptidomimetic inhibitor 28
著者Yang, Y, Nikolovska-Coleska, Z.
登録日2023-07-27
公開日2024-05-29
実験手法X-RAY DIFFRACTION (2.106 Å)
主引用文献Structural studies of intrinsically disordered MLL-fusion protein AF9 in complex with peptidomimetic inhibitors.
Protein Sci., 33, 2024
1AQJ
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STRUCTURE OF ADENINE-N6-DNA-METHYLTRANSFERASE TAQI
分子名称: ADENINE-N6-DNA-METHYLTRANSFERASE TAQI, SINEFUNGIN
著者Schluckebier, G, Saenger, W.
登録日1996-07-25
公開日1997-02-12
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Differential binding of S-adenosylmethionine S-adenosylhomocysteine and Sinefungin to the adenine-specific DNA methyltransferase M.TaqI.
J.Mol.Biol., 265, 1997
8TC5
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Cryo-EM Structure of Spike Glycoprotein from Civet Coronavirus SZ3 in Closed Conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bostina, M, Hills, F.R, Eruera, A.
登録日2023-06-29
公開日2024-05-15
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (2.11 Å)
主引用文献Variation in structural motifs within SARS-related coronavirus spike proteins.
Plos Pathog., 20, 2024
1AQL
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CRYSTAL STRUCTURE OF BOVINE BILE-SALT ACTIVATED LIPASE COMPLEXED WITH TAUROCHOLATE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, BILE-SALT ACTIVATED LIPASE, TAUROCHOLIC ACID
著者Wang, X, Zhang, X.
登録日1997-07-30
公開日1998-08-05
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The crystal structure of bovine bile salt activated lipase: insights into the bile salt activation mechanism.
Structure, 5, 1997
4XKW
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Tailspike protein mutant D339N of E. coli bacteriophage HK620 in complex with pentasaccharide
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, FORMIC ACID, SODIUM ION, ...
著者Gohlke, U, Broeker, N.K, Heinemann, U, Seckler, R, Barbirz, S.
登録日2015-01-12
公開日2016-01-20
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Enthalpic cost of water removal from a hydrophobic glucose binding cavity on HK620 tailspike protein.
to be published
6Y6A
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BU of 6y6a by Molmil
Structure of Finch Polyomavirus VP1 in complex with 2-O-Methyl-5-N-acetyl-alpha-D-neuraminic acid
分子名称: CHLORIDE ION, Capsid protein VP1, MAGNESIUM ION, ...
著者Stroh, L.J, Rustmeier, N.H, Stehle, T.
登録日2020-02-26
公開日2020-07-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Structural Basis and Evolution of Glycan Receptor Specificities within the Polyomavirus Family.
Mbio, 11, 2020
8TR3
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BU of 8tr3 by Molmil
Cryo-EM structure of HmAb64 scFv in complex with CNE40 SOSIP trimer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CNE40 SOSIP Envelope glycoprotein gp120, ...
著者Chan, K.-W, Kong, X.P.
登録日2023-08-09
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.74 Å)
主引用文献Human CD4-binding site antibody elicited by polyvalent DNA prime-protein boost vaccine neutralizes cross-clade tier-2-HIV strains.
Nat Commun, 15, 2024
1B9S
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NOVEL AROMATIC INHIBITORS OF INFLUENZA VIRUS NEURAMINIDASE MAKE SELECTIVE INTERACTIONS WITH CONSERVED RESIDUES AND WATER MOLECULES IN THE ACTIVE SITE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(N-ACETYLAMINO)-3-[N-(2-ETHYLBUTANOYLAMINO)]BENZOIC ACID, CALCIUM ION, ...
著者Finley, J.B, Atigadda, V.R, Duarte, F, Zhao, J.J, Brouillette, W.J, Air, G.M, Luo, M.
登録日1999-02-15
公開日1999-02-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Novel aromatic inhibitors of influenza virus neuraminidase make selective interactions with conserved residues and water molecules in the active site.
J.Mol.Biol., 293, 1999
8T2E
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BU of 8t2e by Molmil
BG505 Boost2 SOSIP.664 in complex with NHP polyclonal antibody FP3
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, FP3 Heavy Chain, ...
著者Pratap, P.P, Antansijevic, A, Ozorowski, G, Ward, A.B.
登録日2023-06-05
公開日2024-06-12
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Priming antibody responses to the fusion peptide in rhesus macaques.
Npj Vaccines, 9, 2024
1B0M
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BU of 1b0m by Molmil
ACONITASE R644Q:FLUOROCITRATE COMPLEX
分子名称: CITRATE ANION, IRON/SULFUR CLUSTER, PROTEIN (ACONITASE)
著者Lloyd, S.J, Lauble, H, Prasad, G.S, Stout, C.D.
登録日1998-11-11
公開日1998-11-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The mechanism of aconitase: 1.8 A resolution crystal structure of the S642a:citrate complex.
Protein Sci., 8, 1999
1APY
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BU of 1apy by Molmil
HUMAN ASPARTYLGLUCOSAMINIDASE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ASPARTYLGLUCOSAMINIDASE, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
著者Rouvinen, J, Oinonen, C.
登録日1995-06-14
公開日1996-12-23
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Three-dimensional structure of human lysosomal aspartylglucosaminidase.
Nat.Struct.Biol., 2, 1995
8T2F
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BU of 8t2f by Molmil
BG505 Boost2 SOSIP.664 in complex with NHP polyclonal antibody N289
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N289 Heavy Chain, ...
著者Pratap, P.P, Antansijevic, A, Ozorowski, G, Ward, A.B.
登録日2023-06-05
公開日2024-06-12
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Priming antibody responses to the fusion peptide in rhesus macaques.
Npj Vaccines, 9, 2024
6ZGY
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BU of 6zgy by Molmil
Structure of human galactokinase 1 bound with 2-(4-chlorophenyl)-N-(pyrimidin-2-yl)acetamide
分子名称: (2,5-dimethylphenyl) pyridine-4-carboxylate, 2-(1,3-benzoxazol-2-ylamino)spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclohexane]-5-one, Galactokinase, ...
著者Mackinnon, S.R, Bezerra, G.A, Zhang, M, Foster, W, Krojer, T, Brandao-Neto, J, Douangamath, A, Arrowsmith, C, Edwards, A, Bountra, C, Brennan, P, Lai, K, Yue, W.W.
登録日2020-06-20
公開日2020-07-29
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Fragment Screening Reveals Starting Points for Rational Design of Galactokinase 1 Inhibitors to Treat Classic Galactosemia.
Acs Chem.Biol., 16, 2021
1BZE
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BU of 1bze by Molmil
TERTIARY STRUCTURES OF THREE AMYLOIDOGENIC TRANSTHYRETIN VARIANTS AND IMPLICATIONS FOR AMYLOID FIBRIL FORMATION
分子名称: PROTEIN (TRANSTHYRETIN)
著者Schormann, N, Murrell, J.R, Benson, M.D.
登録日1998-10-28
公開日1998-11-04
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Tertiary structures of amyloidogenic and non-amyloidogenic transthyretin variants: new model for amyloid fibril formation.
Amyloid, 5, 1998
1BZR
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BU of 1bzr by Molmil
ATOMIC RESOLUTION CRYSTAL STRUCTURE ANALYSIS OF NATIVE DEOXY AND CO MYOGLOBIN FROM SPERM WHALE AT ROOM TEMPERATURE
分子名称: CARBON MONOXIDE, PROTEIN (MYOGLOBIN), PROTOPORPHYRIN IX CONTAINING FE, ...
著者Kachalova, G.S, Popov, A.N, Bartunik, H.D.
登録日1998-11-03
公開日1999-05-10
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献A steric mechanism for inhibition of CO binding to heme proteins.
Science, 284, 1999
8TG9
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Complex of NPR1 ectodomain with ANP plus an allosteric activating antibody, REGN5381
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Atrial natriuretic peptide, ...
著者Franklin, M.C, Romero Hernandez, A.
登録日2023-07-12
公開日2024-07-17
実験手法ELECTRON MICROSCOPY (3.08 Å)
主引用文献Complex of NPR1 ectodomain with ANP plus an allosteric activating antibody, REGN5381
To Be Published
7A9D
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BU of 7a9d by Molmil
Crystal structure of H12 Haemagglutinin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Hemagglutinin
著者Xiong, X, Walker, P, Zhang, J, Gamblin, S, Skehel, J.J.
登録日2020-09-01
公開日2020-12-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Hemagglutinin Structure and Activities.
Cold Spring Harb Perspect Med, 11, 2021
6ZGW
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BU of 6zgw by Molmil
Structure of human galactokinase 1 bound with (4-chlorophenyl)methyl pyridine-3-carboxylate
分子名称: (4-chlorophenyl)methyl pyridine-3-carboxylate, 2-(1,3-benzoxazol-2-ylamino)spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclohexane]-5-one, Galactokinase, ...
著者Mackinnon, S.R, Bezerra, G.A, Zhang, M, Foster, W, Krojer, T, Brandao-Neto, J, Douangamath, A, Arrowsmith, C, Edwards, A, Bountra, C, Brennan, P, Lai, K, Yue, W.W.
登録日2020-06-20
公開日2020-07-29
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Fragment Screening Reveals Starting Points for Rational Design of Galactokinase 1 Inhibitors to Treat Classic Galactosemia.
Acs Chem.Biol., 16, 2021
5INE
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BU of 5ine by Molmil
Crystal structure of the prefusion glycoprotein of LCMV
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Pre-glycoprotein polyprotein GP complex, ...
著者Hastie, K.M, Saphire, E.O.
登録日2016-03-07
公開日2016-04-20
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Crystal structure of the prefusion surface glycoprotein of the prototypic arenavirus LCMV.
Nat.Struct.Mol.Biol., 23, 2016
8TGV
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CryoEM structure of Fab HC84.26-HCV E2 complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HC84.26 Heavy chain, ...
著者Shahid, S, Liqun, J, LIu, Y, Hasan, S.S, Mariuzza, R.A.
登録日2023-07-13
公開日2024-07-24
実験手法ELECTRON MICROSCOPY (3.75 Å)
主引用文献CryoEM structure of Fab HC84.26-HCV E2 complex
To Be Published
8THZ
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BU of 8thz by Molmil
CryoEM structure of neutralizing antibodies CBH-7 and HC84.26 in complex with Hepatitis C virus envelope glycoprotein E2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CBH-7 Heavy chain, ...
著者Shahid, S, Jiang, L, Liu, Y, Hasan, S.S, Mariuzza, R.A.
登録日2023-07-18
公開日2024-07-24
実験手法ELECTRON MICROSCOPY (3.25 Å)
主引用文献CryoEM structure of neutralizing antibodies CBH-7 and HC84.26 in complex with Hepatitis C virus envelope glycoprotein E2
To Be Published
8TJR
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BU of 8tjr by Molmil
CRYO-EM STRUCTURE OF HIV-1 BG505DS-SOSIP.664 ENV TRIMER BOUND TO HERH-c.01 FAB
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody HERH-a.01 Heavy Chain, ...
著者Morano, N.C, Hoyt, F, Hansen, B, Fischer, E, Shapiro, L.
登録日2023-07-24
公開日2024-07-31
実験手法ELECTRON MICROSCOPY (3.29 Å)
主引用文献CRYO-EM STRUCTURE OF HIV-1 BG505DS-SOSIP.664 ENV TRIMER BOUND TO HERH-c.01 FAB
To Be Published
8TGZ
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BU of 8tgz by Molmil
CryoEM structure of neutralizing antibody HC84.26 in complex with Hepatitis C virus envelope glycoprotein E2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HC84.26 Heavy chain, ...
著者Shahid, S, Liqun, J, Liu, Y, Hasan, S.S, Mariuzza, R.A.
登録日2023-07-13
公開日2024-07-24
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献CryoEM structure of neutralizing antibody HC84.26 in complex with Hepatitis C virus envelope glycoprotein E2
To Be Published
6XS3
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BU of 6xs3 by Molmil
X-ray structure of the monoclinic crystal form at 2.48 A resolution of lipase from Thermomyces (Humicola) lanuginosa at 298 K
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-hydroxy-3-(octadecanoyloxy)propyl pentacosanoate, CALCIUM ION, ...
著者McPherson, A.
登録日2020-07-14
公開日2020-10-14
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.48 Å)
主引用文献The crystal Structures of Thermomyces (Humicola) lanuginosa lipase in complex with enzymatic reactants
Current Enzyme Inhibition, 16, 2020

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件を2024-08-21に公開中

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