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4UYO
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BU of 4uyo by Molmil
Structure of delta7-DgkA in 7.9 MAG by serial femtosecond crystatallography to 2.18 angstrom resolution
分子名称: (2R)-2,3-dihydroxypropyl (7Z)-hexadec-7-enoate, (2S)-2,3-dihydroxypropyl (7Z)-hexadec-7-enoate, CITRATE ANION, ...
著者Li, D, Howe, N, Other, O, Caffrey, M.
登録日2014-09-02
公開日2015-09-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Ternary Structure Reveals Mechanism of a Membrane Diacylglycerol Kinase.
Nat.Commun., 6, 2015
3SFC
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BU of 3sfc by Molmil
Structure-Based Optimization of Potent 4- and 6-Azaindole-3-Carboxamides as Renin Inhibitors
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, Renin, ...
著者Scheiper, B, Matter, H, Steinhagen, H, Bocskei, Z, Fleury, V, McCort, G.
登録日2011-06-13
公開日2011-08-31
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure-based optimization of potent 4- and 6-azaindole-3-carboxamides as renin inhibitors.
Bioorg.Med.Chem.Lett., 21, 2011
4UXX
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BU of 4uxx by Molmil
Structure of delta4-DgkA with AMPPCP in 9.9 MAG
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (4S)-2-METHYL-2,4-PENTANEDIOL, ACETATE ION, ...
著者Li, D, Vogeley, L, Caffrey, M.
登録日2014-08-27
公開日2015-09-30
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.701 Å)
主引用文献Ternary Structure Reveals Mechanism of a Membrane Diacylglycerol Kinase.
Nat.Commun., 6, 2015
3S9N
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BU of 3s9n by Molmil
Complex between transferrin receptor 1 and transferrin with iron in the N-Lobe, room temperature
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, CARBONATE ION, ...
著者Eckenroth, B.E, Steere, A.N, Mason, A.B, Everse, S.J.
登録日2011-06-01
公開日2011-08-10
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献How the binding of human transferrin primes the transferrin receptor potentiating iron release at endosomal pH.
Proc.Natl.Acad.Sci.USA, 108, 2011
4V2W
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BU of 4v2w by Molmil
JMJD2A COMPLEXED WITH NI(II), NOG AND HISTONE H3K27me3 PEPTIDE (16-35)
分子名称: CHLORIDE ION, GLYCEROL, HISTONE H3.1T, ...
著者Chowdhury, R, Zafred, D, Schofield, C.J.
登録日2014-10-15
公開日2014-11-26
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Studies on the Catalytic Domains of Multiple Jmjc Oxygenases Using Peptide Substrates.
Epigenetics, 9, 2014
4V1U
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BU of 4v1u by Molmil
Heterocyclase in complex with substrate and Cofactor
分子名称: ADENOSINE MONOPHOSPHATE, CALCIUM ION, LYND, ...
著者Koehnke, J, Naismith, J.H.
登録日2014-10-02
公開日2015-01-14
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.86 Å)
主引用文献Structural Analysis of Leader Peptide Binding Enables Leader-Free Cyanobactin Processing.
Nat.Chem.Biol., 11, 2015
4W5S
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BU of 4w5s by Molmil
Tankyrase in complex with compound
分子名称: 8-(hydroxymethyl)-2-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]quinazolin-4(3H)-one, GLYCEROL, Tankyrase-1, ...
著者Johannes, J, Kazmirski, S.L, Boriack-Sjodin, P.A, Howard, T.
登録日2014-08-18
公開日2015-05-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Pyrimidinone nicotinamide mimetics as selective tankyrase and wnt pathway inhibitors suitable for in vivo pharmacology.
Acs Med.Chem.Lett., 6, 2015
4W7M
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BU of 4w7m by Molmil
CRYSTAL STRUCTURE OF A DECOLORIZING PEROXIDASE (DYP) FROM AURICULARIA AURICULA-JUDAE. W377S MUTANT
分子名称: Dye-decolorizing peroxidase, PROTOPORPHYRIN IX CONTAINING FE
著者Medrano, F.J, Romero, A.
登録日2014-08-22
公開日2015-03-11
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Catalytic surface radical in dye-decolorizing peroxidase: a computational, spectroscopic and site-directed mutagenesis study.
Biochem.J., 466, 2015
4UVA
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BU of 4uva by Molmil
LSD1(KDM1A)-CoREST in complex with 1-Methyl-Tranylcypromine (1R,2S)
分子名称: LYSINE-SPECIFIC HISTONE DEMETHYLASE 1A, REST COREPRESSOR 1, [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl (2R,3S,4S)-2,3,4-trihydroxy-5-[(4aS)-4a-[(1S,3E)-3-imino-1-phenylbutyl]-7,8-dimethyl-2,4-dioxo-3,4,4a,5-tetrahydrobenzo[g]pteridin-10(2H)-yl]pentyl dihydrogen diphosphate
著者Vianello, P, Botrugno, O, Cappa, A, Ciossani, G, Dessanti, P, Mai, A, Mattevi, A, Meroni, G, Minucci, S, Thaler, F, Tortorici, M, Trifiro, P, Valente, S, Villa, M, Varasi, M, Mercurio, C.
登録日2014-08-05
公開日2014-09-10
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Synthesis, Biological Activity and Mechanistic Insights of 1-Substituted Cyclopropylamine Derivatives: A Novel Class of Irreversible Inhibitors of Histone Demethylase Kdm1A.
Eur.J.Med.Chem., 86C, 2014
7MZX
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BU of 7mzx by Molmil
AUGalpha - FAM150B - ALKL2 77-152
分子名称: ALK and LTK ligand 2
著者Rossi, P, Sowaileh, M, Reshetnyak, A.V, Kalodimos, C.G.
登録日2021-05-24
公開日2021-11-24
最終更新日2024-10-23
実験手法SOLUTION NMR
主引用文献Mechanism for the activation of the anaplastic lymphoma kinase receptor.
Nature, 600, 2021
4V0K
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BU of 4v0k by Molmil
Crystal structure of the CrARL6DN in the GDP bound form
分子名称: ARF-LIKE SMALL GTPASE, CADMIUM ION, GUANOSINE-5'-DIPHOSPHATE
著者Mourao, A, Lorentzen, E.
登録日2014-09-17
公開日2014-11-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.438 Å)
主引用文献Structural Basis for Membrane Targeting of the Bbsome by Arl6
Nat.Struct.Mol.Biol., 21, 2014
4V1T
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BU of 4v1t by Molmil
Heterocyclase in complex with substrate and Cofactor
分子名称: ADENOSINE-5'-DIPHOSPHATE, LYND, MAGNESIUM ION, ...
著者Koehnke, J, Naismith, J.H.
登録日2014-10-02
公開日2015-01-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Structural Analysis of Leader Peptide Binding Enables Leader-Free Cyanobactin Processing
Nat.Chem.Biol., 11, 2015
3S8R
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BU of 3s8r by Molmil
Crystal Structures of Glutaryl 7-Aminocephalosporanic Acid Acylase: Insight into Autoproteolytic Activation
分子名称: GLYCEROL, Glutaryl-7-aminocephalosporanic-acid acylase
著者Kim, J.K, Yang, I.S, Park, S.S, Kim, K.H.
登録日2011-05-30
公開日2011-07-06
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structures of glutaryl 7-aminocephalosporanic acid acylase: insight into autoproteolytic activation.
Biochemistry, 42, 2003
4V1V
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BU of 4v1v by Molmil
Heterocyclase in complex with substrate and Cofactor
分子名称: LYND, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
著者Koehnke, J, Naismith, J.H.
登録日2014-10-02
公開日2015-01-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.01 Å)
主引用文献Structural Analysis of Leader Peptide Binding Enables Leader-Free Cyanobactin Processing.
Nat.Chem.Biol., 11, 2015
3J2P
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BU of 3j2p by Molmil
CryoEM structure of Dengue virus envelope protein heterotetramer
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope protein E, ...
著者Zhang, X, Ge, P, Yu, X, Brannan, J.M, Bi, G, Zhang, Q, Schein, S, Zhou, Z.H.
登録日2012-11-30
公開日2012-12-19
最終更新日2024-10-16
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Cryo-EM structure of the mature dengue virus at 3.5-A resolution.
Nat.Struct.Mol.Biol., 20, 2012
4V0O
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BU of 4v0o by Molmil
Crystal structure of BBS1N in complex with ARL6DN, soaked with lead
分子名称: ARF-LIKE SMALL GTPASE, BARDET-BIEDL SYNDROME 1 PROTEIN, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Mourao, A, Lorentzen, E.
登録日2014-09-17
公開日2014-11-19
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (3.351 Å)
主引用文献Structural Basis for Membrane Targeting of the Bbsome by Arl6
Nat.Struct.Mol.Biol., 21, 2014
4UZ7
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BU of 4uz7 by Molmil
STRUCTURE OF THE WNT DEACYLASE NOTUM - CRYSTAL FORM VI - 2.2A
分子名称: CHLORIDE ION, PROTEIN NOTUM HOMOLOG
著者Zebisch, M, Jones, E.Y.
登録日2014-09-04
公開日2015-02-25
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Notum Deacylates Wnt Proteins to Suppress Signalling Activity.
Nature, 519, 2015
4V0L
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BU of 4v0l by Molmil
Crystal structure of the CrARL6DN in the GTP bound form
分子名称: ARF-LIKE SMALL GTPASE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION
著者Mourao, A, Lorentzen, E.
登録日2014-09-17
公開日2014-11-19
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.197 Å)
主引用文献Structural Basis for Membrane Targeting of the Bbsome by Arl6
Nat.Struct.Mol.Biol., 21, 2014
3S97
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BU of 3s97 by Molmil
PTPRZ CNTN1 complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Contactin-1, Receptor-type tyrosine-protein phosphatase zeta
著者Bouyain, S.
登録日2011-05-31
公開日2011-09-28
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.2971 Å)
主引用文献A complex between contactin-1 and the protein tyrosine phosphatase PTPRZ controls the development of oligodendrocyte precursor cells.
Proc.Natl.Acad.Sci.USA, 108, 2011
4WF0
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BU of 4wf0 by Molmil
Crystal Structure of iLID - an Improved Light-Inducible Dimer
分子名称: CHLORIDE ION, FLAVIN MONONUCLEOTIDE, NPH1-1
著者Hallett, R, Williams, T, Kuhlman, B.
登録日2014-09-11
公開日2014-12-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Engineering an improved light-induced dimer (iLID) for controlling the localization and activity of signaling proteins.
Proc.Natl.Acad.Sci.USA, 112, 2015
4WGZ
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BU of 4wgz by Molmil
Crystal Structure of Cytochrome c' from Alcaligenes xylosoxidans NCIMB 11015 at pH 6.0
分子名称: Cytochrome c', HEME C
著者Takashina, A, Unno, M, Kohzuma, T.
登録日2014-09-19
公開日2015-03-18
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.11 Å)
主引用文献X-ray Crystallographic Elucidation for the Alkaline High-spin State Transition of Iron(III) Cytochrome c' from Alcaligenes xylosoxidans NCIMB 11015
CHEM LETT., 44, 2015
3S29
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BU of 3s29 by Molmil
The crystal structure of sucrose synthase-1 from Arabidopsis thaliana and its functional implications.
分子名称: MALONIC ACID, POTASSIUM ION, SULFATE ION, ...
著者Zheng, Y.I, Garavito, R.M.
登録日2011-05-16
公開日2011-08-24
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献The Structure of Sucrose Synthase-1 from Arabidopsis thaliana and Its Functional Implications.
J.Biol.Chem., 286, 2011
3S4B
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BU of 3s4b by Molmil
Cellobiose phosphorylase from Cellulomonas uda in complex with glucose
分子名称: Cellobiose phosphorylase, alpha-D-glucopyranose
著者Van Hoorebeke, A, Stout, J, Soetaert, W, Van Beeumen, J, Desmet, T, Savvides, S.
登録日2011-05-19
公開日2012-06-27
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Cellobiose phosphorylase: reconstructing the structural itinerary along the catalytic pathway
To be Published
3SEK
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BU of 3sek by Molmil
Crystal Structure of the Myostatin:Follistatin-like 3 Complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Follistatin-related protein 3, Growth/differentiation factor 8
著者Cash, J.N, Thompson, T.B.
登録日2011-06-10
公開日2011-11-02
最終更新日2024-11-27
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献Structure of myostatinfollistatin-like 3: N-terminal domains of follistatin-type molecules exhibit alternate modes of binding.
J.Biol.Chem., 287, 2012
3S9L
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BU of 3s9l by Molmil
Complex between transferrin receptor 1 and transferrin with iron in the N-Lobe, cryocooled 2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, CARBONATE ION, ...
著者Eckenroth, B.E, Steere, A.N, Mason, A.B, Everse, S.J.
登録日2011-06-01
公開日2011-08-10
最終更新日2024-10-30
実験手法X-RAY DIFFRACTION (3.22 Å)
主引用文献How the binding of human transferrin primes the transferrin receptor potentiating iron release at endosomal pH.
Proc.Natl.Acad.Sci.USA, 108, 2011

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