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2PKG
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Structure of a complex between the A subunit of protein phosphatase 2A and the small t antigen of SV40
分子名称: Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform, Small T antigen, ZINC ION
著者Jeffrey, P.D, Shi, Y.
登録日2007-04-17
公開日2007-05-15
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural and biochemical insights into the regulation of protein phosphatase 2A by small t antigen of SV40.
Nat.Struct.Mol.Biol., 14, 2007
2PSP
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Porcine pancreatic spasmolytic polypeptide
分子名称: PORCINE PANCREATIC SPASMOLYTIC POLYPEPTIDE
著者Petersen, T.N, Henriksen, A, Gajhede, M.
登録日1996-02-01
公開日1996-07-11
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of porcine pancreatic spasmolytic polypeptide at 1.95 A resolution.
Acta Crystallogr.,Sect.D, 52, 1996
2PZX
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Structure of the methuselah ectodomain with peptide inhibitor
分子名称: G-protein coupled receptor Mth
著者West Jr, A.P, Ja, W.W, Delker, S.L, Bjorkman, P.J, Benzer, S, Roberts, R.W.
登録日2007-05-18
公開日2007-08-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Extension of Drosophila melanogaster life span with a GPCR peptide inhibitor.
Nat.Chem.Biol., 3, 2007
2Q9C
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Structure of FTSY:GMPPNP with MGCL Complex
分子名称: Cell division protein ftsY, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, SULFATE ION
著者Reyes, C.L, Stroud, R.M.
登録日2007-06-12
公開日2007-07-03
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献X-ray Structures of the Signal Recognition Particle Receptor Reveal Targeting Cycle Intermediates.
Plos One, 2, 2007
2PGD
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THE STRUCTURE OF 6-PHOSPHOGLUCONATE DEHYDROGENASE REFINED AT 2 ANGSTROMS RESOLUTION
分子名称: 6-PHOSPHOGLUCONATE DEHYDROGENASE, SULFATE ION
著者Adams, M.J, Phillips, C, Gover, S.
登録日1994-07-18
公開日1995-02-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The structure of 6-phosphogluconate dehydrogenase refined at 2.5 A resolution.
Acta Crystallogr.,Sect.B, 47, 1991
2PGG
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BU of 2pgg by Molmil
Crystal Structure of a Birnavirus (IBDV) RNA-dependent RNA Polymerase VP1
分子名称: RNA-directed RNA polymerase
著者Pan, J, Vakharia, V.N, Tao, Y.J.
登録日2007-04-09
公開日2007-05-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The structure of a birnavirus polymerase reveals a distinct active site topology.
Proc.Natl.Acad.Sci.Usa, 104, 2007
2PA2
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Crystal structure of human Ribosomal protein L10 core domain
分子名称: 60S ribosomal protein L10, POTASSIUM ION
著者Nishimura, M, Kaminishi, T, Takemoto, C, Kawazoe, M, Yoshida, T, Tanaka, A, Sugano, S, Shirouzu, M, Ohkubo, T, Yokoyama, S, Kobayashi, Y, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-03-27
公開日2008-03-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal Structure of Human Ribosomal Protein L10 Core Domain Reveals Eukaryote-Specific Motifs in Addition to the Conserved Fold
J.Mol.Biol., 377, 2008
2P3T
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Crystal structure of human factor XA complexed with 3-Chloro-4-(2-methylamino-imidazol-1-ylmethyl)-thiophene-2-carboxylic acid [4-chloro-2-(5-chloro-pyridin-2-ylcarbamoyl)-6-methoxy-phenyl]-amide
分子名称: 3-CHLORO-4-(2-METHYLAMINO-IMIDAZOL-1-YLMETHYL)-THIOPHENE-2-CARBOXYLIC ACID [4-CHLORO-2-(5-CHLORO-PYRIDIN-2-YLCARBAMOYL)-6-METHOXY-PHENYL]-AMIDE, CALCIUM ION, CHLORIDE ION, ...
著者Adler, M, Whitlow, M.
登録日2007-03-09
公開日2008-01-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Thiophene-anthranilamides as highly potent and orally available factor xa inhibitors.
J.Med.Chem., 50, 2007
2P4X
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Crystal Structure of Atp12 from Paracoccus Denitrificans
分子名称: ATP12 ATPase
著者Ludlam, A.V, Brunzelle, J.S, Gatti, D.L, Ackerman, S.H.
登録日2007-03-13
公開日2008-03-11
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal Structure of Atp12 from Paracoccus Denitrificans
To be Published
2P8H
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Crystal structure of human beta secretase complexed with inhibitor
分子名称: Beta-secretase 1, N-{(1S,2S)-1-BENZYL-2-HYDROXY-2-[(4S)-1,2,2-TRIMETHYL-5-OXOIMIDAZOLIDIN-4-YL]ETHYL}-N'-[(1R)-1-(4-FLUOROPHENYL)ETHYL]-5-[METHYL(METHYLSULFONYL)AMINO]ISOPHTHALAMIDE
著者Munshi, S.
登録日2007-03-22
公開日2007-08-14
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Design and Synthesis of 2,3,5-Substituted Imidazolidin-4-one Inhibitors of BACE-1.
Chemmedchem, 2, 2007
2PE6
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Non-covalent complex between human SUMO-1 and human Ubc9
分子名称: SUMO-conjugating enzyme UBC9, Small ubiquitin-related modifier 1
著者Capili, A.D, Lima, C.D.
登録日2007-04-02
公開日2007-04-17
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure and Analysis of a Complex between SUMO and Ubc9 Illustrates Features of a Conserved E2-Ubl Interaction.
J.Mol.Biol., 369, 2007
2PCQ
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Crystal structure of putative dihydrodipicolinate synthase (TTHA0737) from Thermus Thermophilus HB8
分子名称: GLYCEROL, POTASSIUM ION, Putative dihydrodipicolinate synthase
著者Jeyakanthan, J, Kanaujia, S.P, Vasuki Ranjani, C, Sekar, K, Kitamura, Y, Ebihara, A, Kuramitsu, S, Shinkai, A, Shiro, Y, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-03-30
公開日2007-10-02
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of putative dihydrodipicolinate synthase (TTHA0737) from Thermus Thermophilus HB8
To be Published
2PE1
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CRYSTAL STRUCTURE OF HUMAN PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1 (PDK1) {2-Oxo-3-[1-(1H-pyrrol-2-yl)-eth-(Z)-ylidene]-2,3-dihydro-1H-indol-5-yl}-urea {BX-517} COMPLEX
分子名称: 1-{2-OXO-3-[(1R)-1-(1H-PYRROL-2-YL)ETHYL]-2H-INDOL-5-YL}UREA, 3-phosphoinositide-dependent protein kinase 1, GLYCEROL, ...
著者Whitlow, M, Adler, M.
登録日2007-04-01
公開日2007-06-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Indolinone based phosphoinositide-dependent kinase-1 (PDK1) inhibitors. Part 1: Design, synthesis and biological activity.
Bioorg.Med.Chem.Lett., 17, 2007
2P4B
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BU of 2p4b by Molmil
Crystal structure of E.coli RseB
分子名称: Sigma-E factor regulatory protein rseB, octyl beta-D-glucopyranoside
著者Kim, D.Y, Kim, K.K.
登録日2007-03-12
公開日2007-05-22
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of RseB and a model of its binding mode to RseA
Proc.Natl.Acad.Sci.Usa, 104, 2007
2PBG
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6-PHOSPHO-BETA-D-GALACTOSIDASE FORM-B
分子名称: 6-PHOSPHO-BETA-D-GALACTOSIDASE, SULFATE ION
著者Wiesmann, C, Schulz, G.E.
登録日1997-02-21
公開日1997-07-23
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structures and mechanism of 6-phospho-beta-galactosidase from Lactococcus lactis.
J.Mol.Biol., 269, 1997
2PJ1
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CRYSTAL STRUCTURE OF ACTIVATED PORCINE PANCREATIC CARBOXYPEPTIDASE B (3-Aminomethyl-phenyl)-[((R)-1-benzyloxycarbonylamino-2-methyl-propyl)-hydroxy-phosphinoyloxy]-acetic acid COMPLEX
分子名称: (5R,6S,8S)-8-[3-(AMINOMETHYL)PHENYL]-6-HYDROXY-5-ISOPROPYL-3-OXO-1-PHENYL-2,7-DIOXA-4-AZA-6-PHOSPHANONAN-9-OIC ACID 6-OXIDE, Carboxypeptidase B, ZINC ION
著者Adler, M, Whitlow, M.
登録日2007-04-15
公開日2008-01-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献Structures of potent selective peptide mimetics bound to carboxypeptidase B.
Acta Crystallogr.,Sect.D, 64, 2008
2Q21
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CRYSTAL STRUCTURES AT 2.2 ANGSTROMS RESOLUTION OF THE CATALYTIC DOMAINS OF NORMAL RAS PROTEIN AND AN ONCOGENIC MUTANT COMPLEXED WITH GSP
分子名称: C-H-RAS P21 PROTEIN CATALYTIC DOMAIN, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION
著者Kim, S.-H.
登録日1991-09-25
公開日1992-07-15
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structures at 2.2 A resolution of the catalytic domains of normal ras protein and an oncogenic mutant complexed with GDP.
J.Mol.Biol., 217, 1991
2Q8W
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Crystal structure of PAP-S1aci, a pokeweed antiviral protein from seeds of Phytolacca acinosa
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, POKEWEED ANTIVIRAL PROTEIN
著者Hogg, T, Hilgenfeld, R.
登録日2007-06-12
公開日2008-06-17
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The complete covalent structure and 1.7 A crystal structure of PAP-S1aci reveals a RIP glycoprotein with multiple Asn-GlcNAc modifications
To be Published
2Q9A
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Structure of Apo FTSY
分子名称: 1,2-ETHANEDIOL, Cell division protein ftsY, SULFATE ION
著者Reyes, C.L, Stroud, R.M.
登録日2007-06-12
公開日2007-07-03
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献X-ray Structures of the Signal Recognition Particle Receptor Reveal Targeting Cycle Intermediates.
Plos One, 2, 2007
2PJ5
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CRYSTAL STRUCTURE OF ACTIVATED PORCINE PANCREATIC CARBOXYPEPTIDASE B [((R)-1-Benzyloxycarbonylamino-hexyl)-hydroxy-phosphinoyloxy]-(3-guanidino-phenyl)-acetic acid COMPLEX
分子名称: (5R,6S,8S)-8-(3-{[AMINO(IMINO)METHYL]AMINO}PHENYL)-6-HYDROXY-3-OXO-5-PENTYL-1-PHENYL-2,7-DIOXA-4-AZA-6-PHOSPHANONAN-9-OIC ACID 6-OXIDE, Carboxypeptidase B, ZINC ION
著者Adler, M, Whitlow, M.
登録日2007-04-15
公開日2008-01-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structures of potent selective peptide mimetics bound to carboxypeptidase B.
Acta Crystallogr.,Sect.D, 64, 2008
2PJR
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HELICASE PRODUCT COMPLEX
分子名称: DNA (5'-D(*AP*CP*TP*GP*C)-3'), DNA (5'-D(*GP*C)-3'), DNA (5'-D(*TP*TP*TP*TP*T)-3'), ...
著者Velankar, S.S, Soultanas, P, Dillingham, M.S, Subramanya, H.S, Wigley, D.B.
登録日1999-03-12
公開日1999-04-08
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structures of complexes of PcrA DNA helicase with a DNA substrate indicate an inchworm mechanism.
Cell(Cambridge,Mass.), 97, 1999
2PMI
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Structure of the Pho85-Pho80 CDK-cyclin Complex of the Phosphate-responsive Signal Transduction Pathway with Bound ATP-gamma-S
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Cyclin-dependent protein kinase PHO85, PHO85 cyclin PHO80, ...
著者Huang, K, Ferrin-O'Connell, I, Zhang, W, Leonard, G.A, O'Shea, E.K, Quiocho, F.A.
登録日2007-04-23
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structure of the Pho85-Pho80 CDK-Cyclin Complex of the Phosphate-Responsive Signal Transduction Pathway
Mol.Cell, 28, 2007
2POZ
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Crystal structure of a putative dehydratase from Mesorhizobium loti
分子名称: Putative dehydratase
著者Sugadev, R, Eswaramoorthy, S, Burley, S.K, Swaminathan, S, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2007-04-27
公開日2007-05-15
最終更新日2021-02-03
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Crystal structure of a putative dehydratase from Mesorhizobium loti.
To be Published
2PRO
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PRO REGION OF ALPHA-LYTIC PROTEASE
分子名称: ALPHA-LYTIC PROTEASE
著者Sauter, N.K, Mau, T, Rader, S.D, Agard, D.A.
登録日1998-08-20
公開日1999-04-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of alpha-lytic protease complexed with its pro region.
Nat.Struct.Biol., 5, 1998
2PRI
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BINDING OF 2-DEOXY-GLUCOSE-6-PHOSPHATE TO GLYCOGEN PHOSPHORYLASE B
分子名称: 2-deoxy-6-O-phosphono-alpha-D-glucopyranose, GLYCOGEN PHOSPHORYLASE B, PYRIDOXAL-5'-PHOSPHATE
著者Oikonomakos, N.G, Zographos, S.E, Johnson, L.N, Papageorgiou, A.C, Acharya, K.R.
登録日1998-12-11
公開日1998-12-14
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The binding of 2-deoxy-D-glucose 6-phosphate to glycogen phosphorylase b: kinetic and crystallographic studies.
J.Mol.Biol., 254, 1995

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