6QAO
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6TXC
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![BU of 6txc by Molmil](/molmil-images/mine/6txc) | Crystal structure of tetrameric human wt-SAMHD1 (residues 109-626) with GTP, dATP, dCMPNPP and Mg | 分子名称: | 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]cytidine, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, ... | 著者 | Morris, E.R, Kunzelmann, S, Caswell, S.J, Arnold, L.H, Purkiss, A, Kelly, G, Taylor, I.A. | 登録日 | 2020-01-14 | 公開日 | 2020-06-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.84 Å) | 主引用文献 | Crystal structures of SAMHD1 inhibitor complexes reveal the mechanism of water-mediated dNTP hydrolysis. Nat Commun, 11, 2020
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6FGK
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6TXF
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![BU of 6txf by Molmil](/molmil-images/mine/6txf) | Crystal structure of tetrameric human D137N-SAMHD1 (residues 109-626) with XTP, dAMPNPP and Mn | 分子名称: | 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]adenosine, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION, ... | 著者 | Morris, E.R, Kunzelmann, S, Caswell, S.J, Arnold, L.H, Purkiss, A.G, Kelly, G, Taylor, I.A. | 登録日 | 2020-01-14 | 公開日 | 2020-06-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Crystal structures of SAMHD1 inhibitor complexes reveal the mechanism of water-mediated dNTP hydrolysis. Nat Commun, 11, 2020
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6TX0
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![BU of 6tx0 by Molmil](/molmil-images/mine/6tx0) | Crystal structure of tetrameric human D137N-SAMHD1 (residues 109-626) with XTP, dAMPNPP and Mg | 分子名称: | 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]adenosine, Deoxynucleoside triphosphate triphosphohydrolase SAMHD1, FE (III) ION, ... | 著者 | Morris, E.R, Kunzelmann, S, Caswell, S.J, Arnold, L.H, Purkiss, A.G, Kelly, G, Taylor, I.A. | 登録日 | 2020-01-13 | 公開日 | 2020-06-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Crystal structures of SAMHD1 inhibitor complexes reveal the mechanism of water-mediated dNTP hydrolysis. Nat Commun, 11, 2020
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3BG3
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6GNO
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![BU of 6gno by Molmil](/molmil-images/mine/6gno) | Crystal Structure Of Sea Bream Transthyretin in complex with Tetrabromobisphenol A (TBBPA) | 分子名称: | 4,4'-propane-2,2-diylbis(2,6-dibromophenol), SULFATE ION, Transthyretin | 著者 | Grundstrom, C, Zhang, J, Olofsson, A, Andersson, P.L, Sauer-Eriksson, A.E. | 登録日 | 2018-05-31 | 公開日 | 2018-07-11 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Interspecies Variation between Fish and Human Transthyretins in Their Binding of Thyroid-Disrupting Chemicals. Environ. Sci. Technol., 52, 2018
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4U4F
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![BU of 4u4f by Molmil](/molmil-images/mine/4u4f) | Structure of GluA2* in complex with partial agonist (S)-5-Nitrowillardiine | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3-(5-nitro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-L-alanine, ... | 著者 | Yelshanskaya, M.V, Li, M, Sobolevsky, A.I. | 登録日 | 2014-07-23 | 公開日 | 2014-08-27 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (4.79 Å) | 主引用文献 | Structure of an agonist-bound ionotropic glutamate receptor. Science, 345, 2014
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3SSO
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3AK3
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3T2A
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![BU of 3t2a by Molmil](/molmil-images/mine/3t2a) | TMAO-grown cubic insulin (porcine) | 分子名称: | Insulin A chain, Insulin B chain, trimethylamine oxide | 著者 | Cahn, J, Venkat, M, Marshall, H, Juers, D. | 登録日 | 2011-07-22 | 公開日 | 2011-12-28 | 最終更新日 | 2012-01-11 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The use of trimethylamine N-oxide as a primary precipitating agent and related methylamine osmolytes as cryoprotective agents for macromolecular crystallography. Acta Crystallogr.,Sect.D, 68, 2012
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6R2U
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![BU of 6r2u by Molmil](/molmil-images/mine/6r2u) | Zinc-alpha2-Glycoprotein with a Fluorescent Dansyl C 11 Fatty Acid | 分子名称: | 11-({[5-(dimethylamino)naphthalen-1-yl]sulfonyl}amino)undecanoic acid, AZIDE ION, SULFATE ION, ... | 著者 | Lau, A.M, Gor, J, Perkins, S.J, Coker, A.R, McDermott, L.C. | 登録日 | 2019-03-18 | 公開日 | 2019-09-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Crystal structure of zinc-alpha 2-glycoprotein in complex with a fatty acid reveals multiple different modes of protein-lipid binding. Biochem.J., 476, 2019
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6H4J
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![BU of 6h4j by Molmil](/molmil-images/mine/6h4j) | Usp25 catalytic domain | 分子名称: | CHLORIDE ION, Ubiquitin carboxyl-terminal hydrolase 25 | 著者 | Klemm, T.A, Sauer, F, Kisker, C. | 登録日 | 2018-07-21 | 公開日 | 2019-03-27 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.07 Å) | 主引用文献 | Differential Oligomerization of the Deubiquitinases USP25 and USP28 Regulates Their Activities. Mol.Cell, 74, 2019
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4U4G
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![BU of 4u4g by Molmil](/molmil-images/mine/4u4g) | Structure of GluA2* in complex with competitive antagonist ZK 200775 | 分子名称: | Glutamate receptor 2, beta-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid | 著者 | Yelshanskaya, M.V, Li, M, Sobolevsky, A.I. | 登録日 | 2014-07-23 | 公開日 | 2014-10-22 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (4.49 Å) | 主引用文献 | Structure of an agonist-bound ionotropic glutamate receptor. Science, 345, 2014
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3SSM
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3SSN
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![BU of 3ssn by Molmil](/molmil-images/mine/3ssn) | MycE Methyltransferase from the Mycinamycin Biosynthetic Pathway in Complex with Mg, SAH, and Mycinamycin VI | 分子名称: | DIMETHYL SULFOXIDE, GLYCEROL, MAGNESIUM ION, ... | 著者 | Akey, D.L, Smith, J.L. | 登録日 | 2011-07-08 | 公開日 | 2011-08-24 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.392 Å) | 主引用文献 | A new structural form in the SAM/metal-dependent o‑methyltransferase family: MycE from the mycinamicin biosynthetic pathway. J.Mol.Biol., 413, 2011
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3C2U
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![BU of 3c2u by Molmil](/molmil-images/mine/3c2u) | Structure of the two subsite D-xylosidase from Selenomonas ruminantium in complex with 1,3-bis[tris(hydroxymethyl)methylamino]propane | 分子名称: | 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Xylosidase/arabinosidase | 著者 | Brunzelle, J.S, Jordan, D.B, McCaslin, D.R, Olczak, A, Wawrzak, A. | 登録日 | 2008-01-25 | 公開日 | 2008-04-22 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structure of the two-subsite beta-d-xylosidase from Selenomonas ruminantium in complex with 1,3-bis[tris(hydroxymethyl)methylamino]propane. Arch.Biochem.Biophys., 474, 2008
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1J1Y
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![BU of 1j1y by Molmil](/molmil-images/mine/1j1y) | Crystal Structure of PaaI from Thermus thermophilus HB8 | 分子名称: | CHLORIDE ION, MAGNESIUM ION, PaaI protein | 著者 | Kunishima, N, Sugahara, M, Kuramitsu, S, Yokoyama, S, Miyano, M, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2002-12-24 | 公開日 | 2004-02-17 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A Novel Induced-fit Reaction Mechanism of Asymmetric Hot Dog Thioesterase PaaI J.Mol.Biol., 352, 2005
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3AK2
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3TM2
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![BU of 3tm2 by Molmil](/molmil-images/mine/3tm2) | Crystal structure of mature ThnT with a covalently bound product mimic | 分子名称: | (2R)-N-(4-chloro-3-oxobutyl)-2,4-dihydroxy-3,3-dimethylbutanamide, cysteine transferase | 著者 | Schildbach, J.F, Wright, N.T, Buller, A.R. | 登録日 | 2011-08-30 | 公開日 | 2012-07-04 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Autoproteolytic Activation of ThnT Results in Structural Reorganization Necessary for Substrate Binding and Catalysis. J.Mol.Biol., 422, 2012
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3AK1
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1TF1
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![BU of 1tf1 by Molmil](/molmil-images/mine/1tf1) | Crystal Structure of the E. coli Glyoxylate Regulatory Protein Ligand Binding Domain | 分子名称: | Negative regulator of allantoin and glyoxylate utilization operons | 著者 | Walker, J.R, Skarina, T, Kudrytska, M, Joachimiak, A, Arrowsmith, C, Edwards, A, Savchenko, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2004-05-26 | 公開日 | 2004-08-03 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural and biochemical study of effector molecule recognition by the E.coli glyoxylate and allantoin utilization regulatory protein AllR. J.Mol.Biol., 358, 2006
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7ECH
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![BU of 7ech by Molmil](/molmil-images/mine/7ech) | Crystal Structure of d(G4C2)2-K in F222 space group | 分子名称: | DNA (5'-D(*GP*GP*GP*GP*CP*CP*GP*GP*GP*GP*CP*C)-3'), POTASSIUM ION | 著者 | Geng, Y, Liu, C, Cai, Q, Luo, Z, Zhu, G. | 登録日 | 2021-03-12 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Crystal structure of parallel G-quadruplex formed by the two-repeat ALS- and FTD-related GGGGCC sequence. Nucleic Acids Res., 49, 2021
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2K1E
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![BU of 2k1e by Molmil](/molmil-images/mine/2k1e) | NMR studies of a channel protein without membranes: structure and dynamics of water-solubilized KcsA | 分子名称: | water soluble analogue of potassium channel, KcsA | 著者 | Ma, D, Xu, Y, Tillman, T, Tang, P, Meirovitch, E, Eckenhoff, R, Carnini, A. | 登録日 | 2008-02-29 | 公開日 | 2008-11-11 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR studies of a channel protein without membranes: structure and dynamics of water-solubilized KcsA. Proc.Natl.Acad.Sci.Usa, 105, 2008
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7ECG
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![BU of 7ecg by Molmil](/molmil-images/mine/7ecg) | Crystal Structure of d(G4C2)2-Ba in F222 space group | 分子名称: | BARIUM ION, DNA (5'-D(*GP*GP*GP*GP*CP*CP*GP*GP*GP*GP*CP*C)-3') | 著者 | Geng, Y, Liu, C, Cai, Q, Luo, Z, Zhu, G. | 登録日 | 2021-03-12 | 公開日 | 2021-06-09 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Crystal structure of parallel G-quadruplex formed by the two-repeat ALS- and FTD-related GGGGCC sequence. Nucleic Acids Res., 49, 2021
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