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2Q9O
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Near-atomic resolution structure of a Melanocarpus albomyces laccase
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ...
著者Hakulinen, N, Rouvinen, J.
登録日2007-06-13
公開日2008-03-25
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献A near atomic resolution structure of a Melanocarpus albomyces laccase.
J.Struct.Biol., 162, 2008
6K4E
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SiaA-PP2C domain of Pseudomonas aeruginosa
分子名称: MAGNESIUM ION, Putative serine phosphatase
著者Lin, J.Q, Lescar, J.
登録日2019-05-23
公開日2019-06-26
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.094 Å)
主引用文献The SiaABC threonine phosphorylation pathway controls biofilm formation in response to carbon availability in Pseudomonas aeruginosa.
Plos One, 15, 2020
1DDJ
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BU of 1ddj by Molmil
CRYSTAL STRUCTURE OF HUMAN PLASMINOGEN CATALYTIC DOMAIN
分子名称: PLASMINOGEN
著者Wang, X, Terzyan, S, Tang, J, Loy, J, Lin, X, Zhang, X.
登録日1999-11-10
公開日2000-02-18
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Human plasminogen catalytic domain undergoes an unusual conformational change upon activation.
J.Mol.Biol., 295, 2000
1DO2
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BU of 1do2 by Molmil
TRIGONAL CRYSTAL FORM OF HEAT SHOCK LOCUS U (HSLU) FROM ESCHERICHIA COLI
分子名称: PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, PROTEIN (HEAT SHOCK LOCUS U)
著者Bochtler, M, Hartmann, C, Song, H.K, Bourenkov, G.P, Bartunik, H.D.
登録日1999-12-18
公開日2000-02-18
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献The structures of HsIU and the ATP-dependent protease HsIU-HsIV.
Nature, 403, 2000
1DD7
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MURINE INDUCIBLE NITRIC OXIDE SYNTHASE OXYGENASE DOMAIN (DELTA 114) (N-[(1,3-BENZODIOXOL-5-YL)METHYL]-1-[2-(1H-IMIDAZOL-1-YL)PYRIMIDIN-4-YL]-4-(METHOXYCARBONYL)-PIPERAZINE-2-ACETAMIDE COMPLEX
分子名称: INDUCIBLE NITRIC OXIDE SYNTHASE, PROTOPORPHYRIN IX CONTAINING FE, SULFITE ION, ...
著者Adler, M, Whitlow, M.
登録日1999-11-08
公開日2000-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Allosteric inhibitors of inducible nitric oxide synthase dimerization discovered via combinatorial chemistry.
Proc.Natl.Acad.Sci.USA, 97, 2000
2OKK
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The X-ray crystal structure of the 65kDa isoform of Glutamic Acid Decarboxylase (GAD65)
分子名称: GAMMA-AMINO-BUTANOIC ACID, GLYCEROL, Glutamate decarboxylase 2
著者Buckle, A.M, Fenalti, G, Law, R.H.P, Whisstock, J.C.
登録日2007-01-17
公開日2007-03-27
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献GABA production by glutamic acid decarboxylase is regulated by a dynamic catalytic loop.
Nat.Struct.Mol.Biol., 14, 2007
2O2E
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BU of 2o2e by Molmil
Mycobacterium tuberculosis tryptophan synthase beta subunit dimer (apoform)
分子名称: Tryptophan synthase beta chain
著者Burenkov, G.P, Kachalova, G.S, Bartunik, H.D, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB)
登録日2006-11-29
公開日2008-04-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure Tryptophan SYNTHASE beta subunit dimer from MYCOBACTERIUM TUBERCULOSIS
To be Published
1DM9
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HEAT SHOCK PROTEIN 15 KD
分子名称: HYPOTHETICAL 15.5 KD PROTEIN IN MRCA-PCKA INTERGENIC REGION, SULFATE ION
著者Staker, B.L, Korber, P, Bardwell, J.C.A, Saper, M.A.
登録日1999-12-14
公開日2000-02-18
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of Hsp15 reveals a novel RNA-binding motif.
EMBO J., 19, 2000
2QNB
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Glycogen Phosphorylase b in complex with N-benzoyl-N'-beta-D-glucopyranosyl urea
分子名称: Glycogen phosphorylase, muscle form, N-[(phenylcarbonyl)carbamoyl]-beta-D-glucopyranosylamine
著者Chrysina, E.D, Tiraidis, C, Alexacou, K.-M, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-18
公開日2008-07-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献N-(4-substituted-benzoyl)-N'-(beta-D-glucopyranosyl)ureas, inhibitors of glycogen phosphorylase: synthesis, kinetic and crystallographic evaluation
To be Published
2P9H
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BU of 2p9h by Molmil
High resolution structure of the Lactose Repressor bound to IPTG
分子名称: 1-methylethyl 1-thio-beta-D-galactopyranoside, Lactose operon repressor
著者Daber, R.
登録日2007-03-26
公開日2007-06-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural analysis of lac repressor bound to allosteric effectors.
J.Mol.Biol., 370, 2007
2OOB
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crystal structure of the UBA domain from Cbl-b ubiquitin ligase in complex with ubiquitin
分子名称: E3 ubiquitin-protein ligase CBL-B, Ubiquitin
著者Kozlov, G, Gehring, K.
登録日2007-01-25
公開日2007-02-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural basis for ubiquitin-mediated dimerization and activation of the ubiquitin protein ligase Cbl-b.
Mol.Cell, 27, 2007
2OQR
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The structure of the response regulator RegX3 from Mycobacterium tuberculosis
分子名称: ACETATE ION, BETA-MERCAPTOETHANOL, LANTHANUM (III) ION, ...
著者King-Scott, J.
登録日2007-02-01
公開日2007-10-16
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献The Structure of a Full-length Response Regulator from Mycobacterium tuberculosis in a Stabilized Three-dimensional Domain-swapped, Activated State.
J.Biol.Chem., 282, 2007
2P8C
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BU of 2p8c by Molmil
Crystal structure of N-succinyl Arg/Lys racemase from Bacillus cereus ATCC 14579 complexed with N-succinyl Arg.
分子名称: MAGNESIUM ION, Mandelate racemase/muconate lactonizing enzyme family protein, N~2~-(3-CARBOXYPROPANOYL)-L-ARGININE
著者Fedorov, A.A, Song, L, Fedorov, E.V, Gerlt, J.A, Almo, S.C.
登録日2007-03-22
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Prediction and assignment of function for a divergent N-succinyl amino acid racemase.
Nat.Chem.Biol., 3, 2007
2P88
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Crystal structure of N-succinyl Arg/Lys racemase from Bacillus cereus ATCC 14579
分子名称: MAGNESIUM ION, Mandelate racemase/muconate lactonizing enzyme family protein
著者Fedorov, A.A, Song, L, Fedorov, E.V, Gerlt, J.A, Almo, S.C.
登録日2007-03-22
公開日2007-07-03
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Prediction and assignment of function for a divergent N-succinyl amino acid racemase.
Nat.Chem.Biol., 3, 2007
2QMP
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BU of 2qmp by Molmil
Crystal Structure of HIV-1 protease complexed with PL-100
分子名称: N-[(5S)-5-{[(4-aminophenyl)sulfonyl](isobutyl)amino}-6-hydroxyhexyl]-Nalpha-(methoxycarbonyl)-beta-phenyl-L-phenylalaninamide, Pol polyprotein
著者Allison, T.J.
登録日2007-07-16
公開日2008-07-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of HIV-1 protease complexed with PL-100
To be Published
2QX3
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Structure of pectate lyase II from Xanthomonas campestris pv. campestris str. ATCC 33913
分子名称: PHOSPHATE ION, Pectate lyase II
著者Garron, M.L, Shaya, D.
登録日2007-08-10
公開日2008-03-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A seductive method to improve the thermostability and activity of an enzyme
To be Published
2QZ6
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BU of 2qz6 by Molmil
First crystal structure of a psychrophile class C beta-lactamase
分子名称: Beta-lactamase
著者Michaux, C, Massant, J, Kerff, F, Charlier, P, Wouters, J.
登録日2007-08-16
公開日2008-03-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Crystal structure of a cold-adapted class C beta-lactamase
Febs J., 275, 2008
2R26
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BU of 2r26 by Molmil
The Structure of the Ternary Complex of Carboxymethyl Coenzyme A and Oxalateacetate with Citrate Synthase from the Thermophilic Archaeonthermoplasma Acidophilum
分子名称: CARBOXYMETHYL COENZYME *A, Citrate Synthase, OXALOACETATE ION
著者Lehmann, C.
登録日2007-08-24
公開日2008-08-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Structure of the Ternary Complex of Carboxymethyl Coenzyme A and Oxalateacetate with Citrate Synthase from the Thermophilic Archaeonthermoplasma Acidophilum
To be Published, 2007
2QLM
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Glycogen phosphorylase in complex with FN67
分子名称: Glycogen phosphorylase, muscle form, N-{[(4-methylphenyl)carbonyl]carbamoyl}-beta-D-glucopyranosylamine
著者Oikonomakos, N.G, Chryina, E.D, Tiraidis, C, Kosmopoulou, M.N, Zographos, S.E, Leonidas, D.D.
登録日2007-07-13
公開日2008-07-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献N-(4-substituted-benzoyl)-N'-(beta-D-glucopyranosyl)ureas, inhibitors of glycogen phosphorylase: synthesis, kinetic and crystallographic evaluation
To be Published
2QY1
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pectate lyase A31G/R236F from Xanthomonas campestris
分子名称: PHOSPHATE ION, Pectate lyase II
著者Garron, M.L, Shaya, D.
登録日2007-08-13
公開日2008-02-26
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Improvement of the thermostability and activity of a pectate lyase by single amino acid substitutions, using a strategy based on melting-temperature-guided sequence alignment.
Appl.Environ.Microbiol., 74, 2008
1VSO
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BU of 1vso by Molmil
Crystal Structure of the Ligand-Binding Core of iGluR5 in Complex With the Antagonist (S)-ATPO at 1.85 A resolution
分子名称: (S)-2-AMINO-3-(5-TERT-BUTYL-3-(PHOSPHONOMETHOXY)-4-ISOXAZOLYL)PROPIONIC ACID, GLYCEROL, Glutamate receptor, ...
著者Hald, H, Naur, P, Gajhede, M, Kastrup, J.S.
登録日2007-03-29
公開日2007-07-03
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: structures of the ligand-binding core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid.
J.Biol.Chem., 282, 2007
2QZL
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Crystal Structure of human Beta Secretase complexed with IXS
分子名称: Beta-secretase 1, N-[(1S)-1-benzyl-2-{[(1S)-2-(isobutylamino)-1-methyl-2-oxoethyl]amino}ethyl]-N'-[(1R)-1-(4-fluorophenyl)ethyl]-5-[methyl(methylsulfonyl)amino]isophthalamide
著者Munshi, S.
登録日2007-08-16
公開日2008-04-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献BACE-1 inhibition by a series of psi[CH2NH] reduced amide isosteres
Bioorg.Med.Chem.Lett., 16, 2006
1CE8
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CARBAMOYL PHOSPHATE SYNTHETASE FROM ESCHERICHIS COLI WITH COMPLEXED WITH THE ALLOSTERIC LIGAND IMP
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, INOSINIC ACID, ...
著者Thoden, J.B, Raushel, F.M, Holden, H.M.
登録日1999-03-18
公開日1999-07-26
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The binding of inosine monophosphate to Escherichia coli carbamoyl phosphate synthetase.
J.Biol.Chem., 274, 1999
2QN3
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Glycogen Phosphorylase in complex with N-4-chlorobenzoyl-N-beta-D-glucopyranosyl urea
分子名称: Glycogen phosphorylase, muscle form, N-{[(4-chlorophenyl)carbonyl]carbamoyl}-beta-D-glucopyranosylamine
著者Chrysina, E.D, Tiraidis, C, Alexacou, K.-M, Zographos, S.E, Leonidas, D.D, Oikonomakos, N.G.
登録日2007-07-17
公開日2008-07-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献N-(4-substituted-benzoyl)-N'-(beta-D-glucopyranosyl)ureas, inhibitors of glycogen phosphorylase: synthesis, kinetic and crystallographic evaluation
To be Published
2OXE
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Structure of the Human Pancreatic Lipase-related Protein 2
分子名称: CALCIUM ION, CHLORIDE ION, Pancreatic lipase-related protein 2, ...
著者Walker, J.R, Davis, T, Seitova, A, Finerty Jr, P.J, Butler-Cole, C, Kozieradzki, I, Weigelt, J, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2007-02-20
公開日2007-03-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of human pancreatic lipase-related protein 2 with the lid in an open conformation.
Biochemistry, 47, 2008

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