6G5H
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![BU of 6g5h by Molmil](/molmil-images/mine/6g5h) | Cryo-EM structure of a late human pre-40S ribosomal subunit - Mature | 分子名称: | 18S ribosomal RNA, 40S ribosomal protein S10, 40S ribosomal protein S11, ... | 著者 | Ameismeier, M, Cheng, J, Berninghausen, O, Beckmann, R. | 登録日 | 2018-03-29 | 公開日 | 2018-06-06 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Visualizing late states of human 40S ribosomal subunit maturation. Nature, 558, 2018
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4BJ5
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![BU of 4bj5 by Molmil](/molmil-images/mine/4bj5) | Crystal structure of Rif2 in complex with the C-terminal domain of Rap1 (Rap1-RCT) | 分子名称: | DNA-BINDING PROTEIN RAP1, PROTEIN RIF2, SULFATE ION | 著者 | Shi, T, Bunker, R.D, Gut, H, Scrima, A, Thoma, N.H. | 登録日 | 2013-04-16 | 公開日 | 2013-06-19 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.29 Å) | 主引用文献 | Rif1 and Rif2 Shape Telomere Funcation and Architecture Through Multivalent RAP1 Interactions Cell(Cambridge,Mass.), 153, 2013
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6HGJ
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7KTR
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![BU of 7ktr by Molmil](/molmil-images/mine/7ktr) | Cryo-EM structure of the human SAGA coactivator complex (TRRAP, core) | 分子名称: | Ataxin-7, INOSITOL HEXAKISPHOSPHATE, Isoform 3 of Transcription factor SPT20 homolog, ... | 著者 | Herbst, D.A, Esbin, M.N, Nogales, E. | 登録日 | 2020-11-24 | 公開日 | 2021-11-10 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (2.93 Å) | 主引用文献 | Structure of the human SAGA coactivator complex. Nat.Struct.Mol.Biol., 28, 2021
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6HHY
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![BU of 6hhy by Molmil](/molmil-images/mine/6hhy) | Klebsiella pneumoniae Seryl-tRNA Synthetase in Complex with 5'-O-(N-(L-seryl)-sulfamoyl)N3-methyluridine | 分子名称: | 1,2-ETHANEDIOL, 5'-O-(N-(L-seryl)-sulfamoyl)N3-methyluridine, CALCIUM ION, ... | 著者 | Pang, L, De Graef, S, Weeks, S.D, Strelkov, S.V. | 登録日 | 2018-08-29 | 公開日 | 2019-12-18 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Structural Insights into the Binding of Natural Pyrimidine-Based Inhibitors of Class II Aminoacyl-tRNA Synthetases. Acs Chem.Biol., 15, 2020
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2CJS
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![BU of 2cjs by Molmil](/molmil-images/mine/2cjs) | Structural Basis for a Munc13-1 Homodimer - Munc13-1 - RIM Heterodimer Switch: C2-domains as Versatile Protein-Protein Interaction Modules | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, REGULATING SYNAPTIC MEMBRANE EXOCYTOSIS PROTEIN 2, ... | 著者 | Lu, J, Machius, M, Dulubova, I, Dai, H, Sudhof, T.C, Tomchick, D.R, Rizo, J. | 登録日 | 2006-04-06 | 公開日 | 2006-06-07 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Structural Basis for a Munc13-1 Homodimer to Munc13-1/Rim Heterodimer Switch. Plos Biol., 4, 2006
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7K04
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![BU of 7k04 by Molmil](/molmil-images/mine/7k04) | Structure of TFIIH/Rad4-Rad23-Rad33/DNA in DNA opening | 分子名称: | CALCIUM ION, DNA repair helicase RAD25, DNA repair helicase RAD3, ... | 著者 | van Eeuwen, T, Min, J.H, Murakami, K. | 登録日 | 2020-09-03 | 公開日 | 2021-07-28 | 実験手法 | ELECTRON MICROSCOPY (9.25 Å) | 主引用文献 | Cryo-EM structure of TFIIH/Rad4-Rad23-Rad33 in damaged DNA opening in nucleotide excision repair. Nat Commun, 12, 2021
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4EEU
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![BU of 4eeu by Molmil](/molmil-images/mine/4eeu) | Crystal structure of phiLOV2.1 | 分子名称: | FLAVIN MONONUCLEOTIDE, Phototropin-2 | 著者 | Hitomi, K, Christie, J.M, Arvai, A.S, Hartfield, K.A, Pratt, A.J, Tainer, J.A, Getzoff, E.D. | 登録日 | 2012-03-28 | 公開日 | 2012-05-16 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.4068 Å) | 主引用文献 | Structural Tuning of the Fluorescent Protein iLOV for Improved Photostability. J.Biol.Chem., 287, 2012
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2OKR
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4E5B
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![BU of 4e5b by Molmil](/molmil-images/mine/4e5b) | |
8IVQ
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![BU of 8ivq by Molmil](/molmil-images/mine/8ivq) | Cryo-EM structure of mouse BIRC6, Global map | 分子名称: | Isoform 2 of Baculoviral IAP repeat-containing protein 6 | 著者 | Liu, S, Jiang, T, Bu, F, Zhao, J, Wang, G, Li, N, Gao, N, Qiu, X. | 登録日 | 2023-03-28 | 公開日 | 2024-01-24 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Molecular mechanisms underlying the BIRC6-mediated regulation of apoptosis and autophagy. Nat Commun, 15, 2024
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2AGA
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![BU of 2aga by Molmil](/molmil-images/mine/2aga) | De-ubiquitinating function of ataxin-3: insights from the solution structure of the Josephin domain | 分子名称: | Machado-Joseph disease protein 1 | 著者 | Mao, Y, Senic-Matuglia, F, Di Fiore, P, Polo, S, Hodsdon, M.E, De Camilli, P. | 登録日 | 2005-07-26 | 公開日 | 2005-08-30 | 最終更新日 | 2024-05-08 | 実験手法 | SOLUTION NMR | 主引用文献 | Deubiquitinating function of ataxin-3: insights from the solution structure of the Josephin domain. Proc.Natl.Acad.Sci.Usa, 102, 2005
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2OCI
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![BU of 2oci by Molmil](/molmil-images/mine/2oci) | Crystal structure of valacyclovir hydrolase complexed with a product analogue | 分子名称: | L-TYROSINAMIDE, MAGNESIUM ION, MANGANESE (II) ION, ... | 著者 | Lai, L, Xu, Z, Amidon, G.L. | 登録日 | 2006-12-20 | 公開日 | 2008-02-05 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Molecular basis of prodrug activation by human valacyclovirase, an alpha-amino acid ester hydrolase. J.Biol.Chem., 283, 2008
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2OCK
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![BU of 2ock by Molmil](/molmil-images/mine/2ock) | Crystal structure of valacyclovir hydrolase D123N mutant | 分子名称: | MAGNESIUM ION, MANGANESE (II) ION, Valacyclovir hydrolase | 著者 | Lai, L, Xu, Z, Amidon, G.L. | 登録日 | 2006-12-20 | 公開日 | 2008-02-05 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Molecular basis of prodrug activation by human valacyclovirase, an alpha-amino acid ester hydrolase. J.Biol.Chem., 283, 2008
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2OCL
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![BU of 2ocl by Molmil](/molmil-images/mine/2ocl) | Crystal structure of valacyclovir hydrolase S122A mutant | 分子名称: | MAGNESIUM ION, MANGANESE (II) ION, Valacyclovir hydrolase | 著者 | Lai, L, Xu, Z, Amidon, G.L. | 登録日 | 2006-12-20 | 公開日 | 2008-02-05 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Molecular basis of prodrug activation by human valacyclovirase, an alpha-amino acid ester hydrolase. J.Biol.Chem., 283, 2008
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4EH3
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![BU of 4eh3 by Molmil](/molmil-images/mine/4eh3) | Human p38 MAP kinase in complex with NP-F2 and RL87 | 分子名称: | Mitogen-activated protein kinase 14, NARINGENIN, N~4~-cyclopropyl-2-phenylquinazoline-4,7-diamine | 著者 | Over, B, Gruetter, C, Waldmann, H, Rauh, D. | 登録日 | 2012-04-02 | 公開日 | 2012-12-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Natural-product-derived fragments for fragment-based ligand discovery. Nat Chem, 5, 2012
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2NS5
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7BC2
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![BU of 7bc2 by Molmil](/molmil-images/mine/7bc2) | BAZ2A bromodomain in complex with triazole compound MS04-TN04 | 分子名称: | 2-(1-methyl-1H-1,2,3-triazol-5-yl)-5-((2-(pyridin-4-yl)pyrrolidin-1-yl)methyl)-1H-benzo[d]imidazole, Bromodomain adjacent to zinc finger domain protein 2A | 著者 | Dalle Vedove, A, Cazzanelli, G, Sedykh, M, Caflisch, A, Lolli, G. | 登録日 | 2020-12-18 | 公開日 | 2021-10-20 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing. Acs Med.Chem.Lett., 13, 2022
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4YWD
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![BU of 4ywd by Molmil](/molmil-images/mine/4ywd) | Structure of rat cytosolic pepck in complex with 2,3-Pyridine dicarboxylic acid | 分子名称: | MANGANESE (II) ION, Phosphoenolpyruvate carboxykinase, cytosolic [GTP], ... | 著者 | Balan, M.D, Johnson, T.A, Mcleod, M.J, Lotosky, W.R, Holyoak, T. | 登録日 | 2015-03-20 | 公開日 | 2015-09-23 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Inhibition and Allosteric Regulation of Monomeric Phosphoenolpyruvate Carboxykinase by 3-Mercaptopicolinic Acid. Biochemistry, 54, 2015
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2E5K
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![BU of 2e5k by Molmil](/molmil-images/mine/2e5k) | Solution structure of SH3 domain in Suppressor of T-cell receptor signaling 1 | 分子名称: | Suppressor of T-cell receptor signaling 1 | 著者 | Sukegawa, S, Tsuda, K, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-12-21 | 公開日 | 2007-06-26 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of SH3 domain in Suppressor of T-cell receptor signaling 1 To be Published
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8J19
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![BU of 8j19 by Molmil](/molmil-images/mine/8j19) | Cryo-EM structure of the LY237-bound GPR84 receptor-Gi complex | 分子名称: | 6-nonylpyridine-2,4-diol, Antibody fragment ScFv16, G-protein coupled receptor 84, ... | 著者 | Liu, H, Yin, W, Xu, H.E. | 登録日 | 2023-04-12 | 公開日 | 2023-06-21 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.23 Å) | 主引用文献 | Structural insights into ligand recognition and activation of the medium-chain fatty acid-sensing receptor GPR84. Nat Commun, 14, 2023
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4H12
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![BU of 4h12 by Molmil](/molmil-images/mine/4h12) | The crystal structure of methyltransferase domain of human SET domain-containing protein 2 in complex with S-adenosyl-L-homocysteine | 分子名称: | CHLORIDE ION, Histone-lysine N-methyltransferase SETD2, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Amaya, M.F, Dong, A, Zeng, H, Mackenzie, F, Bunnage, M, Weigelt, J, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Wu, H, Structural Genomics Consortium (SGC) | 登録日 | 2012-09-10 | 公開日 | 2012-10-03 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Sinefungin Derivatives as Inhibitors and Structure Probes of Protein Lysine Methyltransferase SETD2. J.Am.Chem.Soc., 134, 2012
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6J73
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![BU of 6j73 by Molmil](/molmil-images/mine/6j73) | Crystal structure of IniA from Mycobacterium smegmatis | 分子名称: | Isoniazid inducible gene protein IniA | 著者 | Wang, M.F, Guo, X.Y, Hu, J.J, Li, J, Rao, Z.H. | 登録日 | 2019-01-16 | 公開日 | 2019-09-11 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (3.211 Å) | 主引用文献 | Mycobacterial dynamin-like protein IniA mediates membrane fission. Nat Commun, 10, 2019
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8J18
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![BU of 8j18 by Molmil](/molmil-images/mine/8j18) | Cryo-EM structure of the 3-OH-C12-bound GPR84 receptor-Gi complex | 分子名称: | (3R)-3-HYDROXYDODECANOIC ACID, Antibody fragment ScFv16, G-protein coupled receptor 84, ... | 著者 | Liu, H, Yin, W, Xu, H.E. | 登録日 | 2023-04-12 | 公開日 | 2023-06-21 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (2.89 Å) | 主引用文献 | Structural insights into ligand recognition and activation of the medium-chain fatty acid-sensing receptor GPR84. Nat Commun, 14, 2023
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8J1A
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![BU of 8j1a by Molmil](/molmil-images/mine/8j1a) | Cryo-EM structure of the GPR84 receptor-Gi complex with no ligand modeled | 分子名称: | Antibody fragment ScFv16, G-protein coupled receptor 84, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Liu, H, Yin, W, Xu, H.E. | 登録日 | 2023-04-12 | 公開日 | 2023-06-21 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.24 Å) | 主引用文献 | Structural insights into ligand recognition and activation of the medium-chain fatty acid-sensing receptor GPR84. Nat Commun, 14, 2023
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