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6V3I
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BU of 6v3i by Molmil
K2P2.1(TREK-1)I110D:RuR bound channel structure
分子名称: CADMIUM ION, DODECANE, HEXANE, ...
著者Pope, L, Lolicato, M, Minor, D.L.
登録日2019-11-25
公開日2020-02-26
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Polynuclear Ruthenium Amines Inhibit K2PChannels via a "Finger in the Dam" Mechanism.
Cell Chem Biol, 2020
6V3C
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BU of 6v3c by Molmil
K2P2.1(TREK-1)I110D:Ru360 bound channel structure
分子名称: CADMIUM ION, HEXANE, N-OCTANE, ...
著者Pope, L, Lolicato, M, Minor, D.L.
登録日2019-11-25
公開日2020-02-26
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.51 Å)
主引用文献Polynuclear Ruthenium Amines Inhibit K2PChannels via a "Finger in the Dam" Mechanism.
Cell Chem Biol, 2020
6V37
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BU of 6v37 by Molmil
K2P2.1(TREK-1)I110D:RuR:ML335 bound channel structure
分子名称: CADMIUM ION, DODECANE, HEXANE, ...
著者Pope, L, Lolicato, M, Minor, D.L.
登録日2019-11-25
公開日2020-02-26
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Polynuclear Ruthenium Amines Inhibit K2PChannels via a "Finger in the Dam" Mechanism.
Cell Chem Biol, 2020
6V36
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BU of 6v36 by Molmil
K2P2.1(TREK-1)I110D apo channel structure
分子名称: CADMIUM ION, N-OCTANE, POTASSIUM ION, ...
著者Pope, L, Lolicato, M, Minor, D.L.
登録日2019-11-25
公開日2020-02-26
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Polynuclear Ruthenium Amines Inhibit K2PChannels via a "Finger in the Dam" Mechanism.
Cell Chem Biol, 2020
6UXB
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BU of 6uxb by Molmil
MthK N-terminal truncation state 3 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-07
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.9 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UXA
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BU of 6uxa by Molmil
MthK N-terminal truncation state 2 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-07
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UX7
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BU of 6ux7 by Molmil
MthK N-terminal truncation state 1 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-06
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (6.7 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UX4
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BU of 6ux4 by Molmil
MthK N-terminal truncation RCK domain state 2 bound with calcium
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-06
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UWN
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BU of 6uwn by Molmil
MthK N-terminal truncation RCK domain state 1 bound with calcium
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-05
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UFE
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BU of 6ufe by Molmil
The structure of a potassium selective ion channel at atomic resolution
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, POTASSIUM ION, Transporter
著者Langan, P.S, Vandavasi, V.G, Sullivan, B, Afonine, P.V, Weiss, K.L.
登録日2019-09-24
公開日2020-08-05
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献The structure of a potassium-selective ion channel reveals a hydrophobic gate regulating ion permeation.
Iucrj, 7, 2020
6U9Z
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BU of 6u9z by Molmil
Wild-type MthK pore in 6 mM K+
分子名称: Calcium-gated potassium channel MthK, HEXANE-1,6-DIOL, POTASSIUM ION
著者Posson, D.J, Nimigean, C.M.
登録日2019-09-09
公開日2020-11-04
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.954 Å)
主引用文献Selectivity filter ion binding affinity determines inactivation in a potassium channel.
Proc.Natl.Acad.Sci.USA, 117, 2020
6U9Y
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BU of 6u9y by Molmil
Wild-type MthK pore in 11 mM K+
分子名称: Calcium-gated potassium channel MthK, HEXANE-1,6-DIOL, POTASSIUM ION
著者Posson, D.J, Nimigean, C.M.
登録日2019-09-09
公開日2020-11-04
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Selectivity filter ion binding affinity determines inactivation in a potassium channel.
Proc.Natl.Acad.Sci.USA, 117, 2020
6U9T
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BU of 6u9t by Molmil
Wild-type MthK pore in 50 mM K+
分子名称: Calcium-gated potassium channel MthK, HEXANE-1,6-DIOL, POTASSIUM ION
著者Posson, D.J, Nimigean, C.M.
登録日2019-09-09
公開日2020-11-04
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Selectivity filter ion binding affinity determines inactivation in a potassium channel.
Proc.Natl.Acad.Sci.USA, 117, 2020
6U9P
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BU of 6u9p by Molmil
Wild-type MthK pore in ~150 mM K+
分子名称: Calcium-gated potassium channel MthK, HEXANE-1,6-DIOL, POTASSIUM ION
著者Posson, D.J, Nimigean, C.M.
登録日2019-09-09
公開日2020-11-04
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Selectivity filter ion binding affinity determines inactivation in a potassium channel.
Proc.Natl.Acad.Sci.USA, 117, 2020
6U6H
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BU of 6u6h by Molmil
Calcium-bound MthK open-inactivated state 3
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-08-29
公開日2020-04-22
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U6E
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BU of 6u6e by Molmil
Calcium-bound MthK open-inactivated state 2
分子名称: Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-29
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (6.3 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U6D
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BU of 6u6d by Molmil
MthK closed state with EDTA
分子名称: Calcium-gated potassium channel MthK, POTASSIUM ION
著者Fan, C, Rheinberger, J, Nimigean, C.M.
登録日2019-08-29
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U68
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BU of 6u68 by Molmil
Calcium-bound MthK open-inactivated state 1
分子名称: Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-29
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U5R
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BU of 6u5r by Molmil
Calcium-bound MthK closed state
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U5P
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BU of 6u5p by Molmil
Calcium-bound MthK gating ring state 1
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U5N
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BU of 6u5n by Molmil
Calcium-bound MthK gating ring state 2
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6RV4
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BU of 6rv4 by Molmil
Crystal structure of the human two pore domain potassium ion channel TASK-1 (K2P3.1) in a closed conformation with a bound inhibitor BAY 2341237
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CHOLESTEROL HEMISUCCINATE, POTASSIUM ION, ...
著者Rodstrom, K.E.J, Pike, A.C.W, Zhang, W, Quigley, A, Speedman, D, Mukhopadhyay, S.M.M, Shrestha, L, Chalk, R, Venkaya, S, Bushell, S.R, Tessitore, A, Burgess-Brown, N, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2019-05-30
公開日2019-08-07
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献A lower X-gate in TASK channels traps inhibitors within the vestibule.
Nature, 582, 2020
6RV3
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BU of 6rv3 by Molmil
Crystal structure of the human two pore domain potassium ion channel TASK-1 (K2P3.1) in a closed conformation with a bound inhibitor BAY 1000493
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CHOLESTEROL HEMISUCCINATE, DECYL-BETA-D-MALTOPYRANOSIDE, ...
著者Rodstrom, K.E.J, Pike, A.C.W, Zhang, W, Quigley, A, Speedman, D, Mukhopadhyay, S.M.M, Shrestha, L, Chalk, R, Venkaya, S, Bushell, S.R, Tessitore, A, Burgess-Brown, N, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2019-05-30
公開日2019-08-07
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A lower X-gate in TASK channels traps inhibitors within the vestibule.
Nature, 582, 2020
6RV2
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BU of 6rv2 by Molmil
Crystal structure of the human two pore domain potassium ion channel TASK-1 (K2P3.1) in a closed conformation
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CHOLESTEROL HEMISUCCINATE, DECYL-BETA-D-MALTOPYRANOSIDE, ...
著者Rodstrom, K.E.J, Pike, A.C.W, Zhang, W, Quigley, A, Speedman, D, Mukhopadhyay, S.M.M, Shrestha, L, Chalk, R, Venkaya, S, Bushell, S.R, Tessitore, A, Burgess-Brown, N, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2019-05-30
公開日2019-08-07
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A lower X-gate in TASK channels traps inhibitors within the vestibule.
Nature, 582, 2020
6PIS
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BU of 6pis by Molmil
Mouse two pore domain K+ channel TRAAK (K2P4.1) - Fab complex structure
分子名称: ANTIBODY FAB FRAGMENT HEAVY CHAIN, ANTIBODY FAB FRAGMENT LIGHT CHAIN, POTASSIUM ION, ...
著者Brohawn, S.G.
登録日2019-06-27
公開日2019-12-25
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.77 Å)
主引用文献The mechanosensitive ion channel TRAAK is localized to the mammalian node of Ranvier.
Elife, 8, 2019

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