4PRO
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4PVM
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![BU of 4pvm by Molmil](/molmil-images/mine/4pvm) | Neutron structure of human transthyretin (TTR) at room temperature to 2.0A resolution (Laue) | 分子名称: | Transthyretin | 著者 | Fisher, S.J, Blakeley, M.P, Haupt, M, Mason, S.A, Cooper, J.B, Mitchell, E.P, Forsyth, V.T. | 登録日 | 2014-03-18 | 公開日 | 2014-11-12 | 最終更新日 | 2024-03-20 | 実験手法 | NEUTRON DIFFRACTION (2 Å), X-RAY DIFFRACTION | 主引用文献 | Binding site asymmetry in human transthyretin: insights from a joint neutron and X-ray crystallographic analysis using perdeuterated protein IUCrJ, 1, 2014
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5E6P
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3PCX
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![BU of 3pcx by Molmil](/molmil-images/mine/3pcx) | Caspase-3 E246A, K242A Double Mutant | 分子名称: | Caspase-3, Inhibitor Ac-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-23 | 最終更新日 | 2012-12-12 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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6GPB
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4QTY
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![BU of 4qty by Molmil](/molmil-images/mine/4qty) | Caspase-3 E190A | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, AZIDE ION, Caspase-3, ... | 著者 | Cade, C, Swartz, P.D, MacKenzie, S.H, Clark, A.C. | 登録日 | 2014-07-09 | 公開日 | 2014-11-05 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (1.602 Å) | 主引用文献 | Modifying caspase-3 activity by altering allosteric networks. Biochemistry, 53, 2014
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3M9Z
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![BU of 3m9z by Molmil](/molmil-images/mine/3m9z) | Crystal Structure of extracellular domain of mouse NKR-P1A | 分子名称: | Killer cell lectin-like receptor subfamily B member 1A, PHOSPHATE ION | 著者 | Kolenko, P, Rozbesky, D, Bezouska, K, Hasek, J, Dohnalek, J. | 登録日 | 2010-03-23 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Molecular architecture of mouse activating NKR-P1 receptors. J.Struct.Biol., 175, 2011
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4QU5
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![BU of 4qu5 by Molmil](/molmil-images/mine/4qu5) | Caspase-3 T140V | 分子名称: | ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, Caspase-3 | 著者 | Cade, C, Swartz, P.D, MacKenzie, S.H, Clark, A.C. | 登録日 | 2014-07-10 | 公開日 | 2014-11-05 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (1.908 Å) | 主引用文献 | Modifying caspase-3 activity by altering allosteric networks. Biochemistry, 53, 2014
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4QUI
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![BU of 4qui by Molmil](/molmil-images/mine/4qui) | Caspase-3 F128AV266H | 分子名称: | 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, CHLORIDE ION, ... | 著者 | Cade, C, Swartz, P.D, MacKenzie, S.H, Clark, A.C. | 登録日 | 2014-07-10 | 公開日 | 2014-11-05 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (1.758 Å) | 主引用文献 | Modifying caspase-3 activity by altering allosteric networks. Biochemistry, 53, 2014
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6E6L
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4P2X
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![BU of 4p2x by Molmil](/molmil-images/mine/4p2x) | Swapped Dimer of Mycobacterial Adenylyl cyclase Rv1625c: Form 2 | 分子名称: | Adenylate cyclase, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Barathy, D.V, Mattoo, R, Visweswariah, S.S, Suguna, K. | 登録日 | 2014-03-05 | 公開日 | 2014-09-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | New structural forms of a mycobacterial adenylyl cyclase Rv1625c. Iucrj, 1, 2014
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1Y5X
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![BU of 1y5x by Molmil](/molmil-images/mine/1y5x) | tRNA-guanine Transglycosylase (TGT) in complex with 6-Amino-4-[2-(4-methoxyphenyl)ethyl]-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one | 分子名称: | 6-AMINO-4-[2-(4-METHOXYPHENYL)ETHYL]-1,7-DIHYDRO-8H-IMIDAZO[4,5-G]QUINAZOLIN-8-ONE, Queuine tRNA-ribosyltransferase, ZINC ION | 著者 | Stengl, B, Meyer, E.A, Heine, A, Brenk, R, Diederich, F, Klebe, G. | 登録日 | 2004-12-03 | 公開日 | 2005-12-13 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structures of tRNA-guanine transglycosylase (TGT) in complex with novel and potent inhibitors unravel pronounced induced-fit adaptations and suggest dimer formation upon substrate binding J.Mol.Biol., 370, 2007
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4P2F
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![BU of 4p2f by Molmil](/molmil-images/mine/4p2f) | Monomeric form of a single mutant (F363R) of Mycobacterial Adenylyl cyclase Rv1625c | 分子名称: | 1,2-ETHANEDIOL, Adenylate cyclase, DI(HYDROXYETHYL)ETHER, ... | 著者 | Barathy, D.V, Mattoo, R, Visweswariah, S.S, Suguna, K. | 登録日 | 2014-03-04 | 公開日 | 2014-09-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | New structural forms of a mycobacterial adenylyl cyclase Rv1625c. Iucrj, 1, 2014
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4P2M
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![BU of 4p2m by Molmil](/molmil-images/mine/4p2m) | Swapped Dimer of Mycobacterial Adenylyl cyclase Rv1625c: Form 1 | 分子名称: | Adenylate cyclase, DI(HYDROXYETHYL)ETHER, SULFATE ION | 著者 | Barathy, D.V, Mattoo, R, Visweswariah, S.S, Suguna, K. | 登録日 | 2014-03-04 | 公開日 | 2014-09-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | New structural forms of a mycobacterial adenylyl cyclase Rv1625c. Iucrj, 1, 2014
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6EAT
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![BU of 6eat by Molmil](/molmil-images/mine/6eat) | Crystallographic structure of the cyclic nonapeptide derived from the BTCI inhibitor bound to beta-trypsin in space group P 21 21 21. | 分子名称: | 9MER-PEPTIDE, CALCIUM ION, Cationic trypsin, ... | 著者 | Fernandes, J.C, Valadares, N.F, Freitas, S.M, Barbosa, J.A.R.G. | 登録日 | 2018-08-03 | 公開日 | 2019-03-13 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.149 Å) | 主引用文献 | Crystallographic structure of a complex between trypsin and a nonapeptide derived from a Bowman-Birk inhibitor found in Vigna unguiculata seeds. Arch. Biochem. Biophys., 665, 2019
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6H0F
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![BU of 6h0f by Molmil](/molmil-images/mine/6h0f) | Structure of DDB1-CRBN-pomalidomide complex bound to IKZF1(ZF2) | 分子名称: | DNA damage-binding protein 1,DNA damage-binding protein 1,DNA damage-binding protein 1,DNA damage-binding protein 1, DNA-binding protein Ikaros, Protein cereblon, ... | 著者 | Petzold, G, Bunker, R.D, Thoma, N.H. | 登録日 | 2018-07-09 | 公開日 | 2018-11-07 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Defining the human C2H2 zinc finger degrome targeted by thalidomide analogs through CRBN. Science, 362, 2018
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6E5R
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6E63
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![BU of 6e63 by Molmil](/molmil-images/mine/6e63) | Crystal structure of malaria transmission-blocking antigen Pfs48/45 6C in complex with antibody TB31F | 分子名称: | GLYCEROL, Pf48/45, TB31F Fab heavy chain, ... | 著者 | Kundu, P, Semesi, A, Julien, J.P. | 登録日 | 2018-07-23 | 公開日 | 2018-11-28 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural delineation of potent transmission-blocking epitope I on malaria antigen Pfs48/45. Nat Commun, 9, 2018
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2ZTA
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![BU of 2zta by Molmil](/molmil-images/mine/2zta) | X-RAY STRUCTURE OF THE GCN4 LEUCINE ZIPPER, A TWO-STRANDED, PARALLEL COILED COIL | 分子名称: | GCN4 LEUCINE ZIPPER | 著者 | O'Shea, E.K, Klemm, J.D, Kim, P.S, Alber, T. | 登録日 | 1991-07-05 | 公開日 | 1992-10-15 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | X-ray structure of the GCN4 leucine zipper, a two-stranded, parallel coiled coil. Science, 254, 1991
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3PD1
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![BU of 3pd1 by Molmil](/molmil-images/mine/3pd1) | Caspase-3 K242A | 分子名称: | Caspase-3, Inhibitor Ac-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-23 | 最終更新日 | 2013-02-27 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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6EI8
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3PD0
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![BU of 3pd0 by Molmil](/molmil-images/mine/3pd0) | Caspase-3 E246A | 分子名称: | CHLORIDE ION, Caspase-3, INHIBITOR AC-DEVD-CMK | 著者 | Walters, J, Swartz, P, Mattos, C, Clark, A.C. | 登録日 | 2010-10-22 | 公開日 | 2011-02-16 | 最終更新日 | 2012-12-12 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Thermodynamic, enzymatic and structural effects of removing a salt bridge at the base of loop 4 in (pro)caspase-3. Arch.Biochem.Biophys., 508, 2011
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6H0G
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![BU of 6h0g by Molmil](/molmil-images/mine/6h0g) | Structure of the DDB1-CRBN-pomalidomide complex bound to ZNF692(ZF4) | 分子名称: | DNA damage-binding protein 1,DNA damage-binding protein 1,DNA damage-binding protein 1,DDB1 (DNA damage binding protein 1),DNA damage-binding protein 1,DNA damage-binding protein 1,DNA damage-binding protein 1, Protein cereblon, S-Pomalidomide, ... | 著者 | Bunker, R.D, Petzold, G, Thoma, N.H. | 登録日 | 2018-07-09 | 公開日 | 2018-11-07 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (4.25 Å) | 主引用文献 | Defining the human C2H2 zinc finger degrome targeted by thalidomide analogs through CRBN. Science, 362, 2018
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4TPS
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![BU of 4tps by Molmil](/molmil-images/mine/4tps) | Sporulation Inhibitor of DNA Replication, SirA, in complex with Domain I of DnaA | 分子名称: | ACETATE ION, BETA-MERCAPTOETHANOL, Chromosomal replication initiator protein DnaA, ... | 著者 | Jameson, K.H, Turkenburg, J.P, Fogg, M.J, Grahl, A, Wilkinson, A.J. | 登録日 | 2014-06-09 | 公開日 | 2014-07-30 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Structure and interactions of the Bacillus subtilis sporulation inhibitor of DNA replication, SirA, with domain I of DnaA. Mol.Microbiol., 93, 2014
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5VB0
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![BU of 5vb0 by Molmil](/molmil-images/mine/5vb0) | Crystal structure of fosfomycin resistance protein FosA3 | 分子名称: | Fosfomycin resistance protein FosA3, MANGANESE (II) ION, NICKEL (II) ION | 著者 | Klontz, E, Guenther, S, Silverstein, Z, Sundberg, E. | 登録日 | 2017-03-28 | 公開日 | 2017-08-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.689 Å) | 主引用文献 | Structure and Dynamics of FosA-Mediated Fosfomycin Resistance in Klebsiella pneumoniae and Escherichia coli. Antimicrob. Agents Chemother., 61, 2017
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