2EJJ
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7MXV
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7MXT
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7MXQ
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2C37
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8FUI
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![BU of 8fui by Molmil](/molmil-images/mine/8fui) | HIV-1 wild type protease with GRL-02519A, with N-(2,5-dimethylphenyl)-4-(pyridin-3-yl)pyrimidin-2-amine as P2-P3 group | 分子名称: | ACETATE ION, CHLORIDE ION, FORMIC ACID, ... | 著者 | Wang, Y.-F, Wong-Sam, A.E, Ghosh, A.K, Weber, I.T. | 登録日 | 2023-01-17 | 公開日 | 2023-05-24 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Exploration of imatinib and nilotinib-derived templates as the P2-Ligand for HIV-1 protease inhibitors: Design, synthesis, protein X-ray structural studies, and biological evaluation. Eur.J.Med.Chem., 255, 2023
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8FUJ
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![BU of 8fuj by Molmil](/molmil-images/mine/8fuj) | HIV-1 wild type protease with GRL-03419A, with N-(2,5-dimethylphenyl)-4-(pyridin-3-yl)pyrimidin-2-amine as P2-P3 group and 3,5-difluorophenylmethyl as the P1 group | 分子名称: | CHLORIDE ION, FORMIC ACID, GLYCEROL, ... | 著者 | Wang, Y.-F, Agniswamy, J, Ghosh, A.K, Weber, I.T. | 登録日 | 2023-01-17 | 公開日 | 2023-05-24 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.12 Å) | 主引用文献 | Exploration of imatinib and nilotinib-derived templates as the P2-Ligand for HIV-1 protease inhibitors: Design, synthesis, protein X-ray structural studies, and biological evaluation. Eur.J.Med.Chem., 255, 2023
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8POB
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![BU of 8pob by Molmil](/molmil-images/mine/8pob) | Crystal structure of Hen Egg White Lysozyme co-crystallized with 10 mM TbXo4-SO3 | 分子名称: | 6-[[4-[(6-carboxypyridin-2-yl)methyl]-7-(3-sulfopropyl)-1,4,7-triazonan-1-yl]methyl]pyridine-2-carboxylic acid, CHLORIDE ION, Lysozyme C, ... | 著者 | Alsalman, Z, Girard, E. | 登録日 | 2023-07-04 | 公開日 | 2024-07-10 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Influence of Chemical Modifications of the Crystallophore on Protein Nucleating Properties and Supramolecular Interactions Network. Chemistry, 30, 2024
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7NQ6
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8PUJ
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![BU of 8puj by Molmil](/molmil-images/mine/8puj) | The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin. | 分子名称: | COB(II)INAMIDE, HYDROXIDE ION, SODIUM ION, ... | 著者 | Whittaker, J, Martinez-Felices, J.M, Guskov, A, Slotboom, D.J. | 登録日 | 2023-07-17 | 公開日 | 2024-07-24 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The surface-exposed lipo-protein of BtuG3 in complex with cyanocobinamide. To Be Published
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8PTF
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![BU of 8ptf by Molmil](/molmil-images/mine/8ptf) | The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin. | 分子名称: | COB(II)INAMIDE, SODIUM ION, YncE family protein, ... | 著者 | Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J. | 登録日 | 2023-07-14 | 公開日 | 2024-07-24 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | The surface-exposed lipo-protein of BtuG1 in complex with cyanocobinamide. To Be Published
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7NQA
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![BU of 7nqa by Molmil](/molmil-images/mine/7nqa) | Crystal structure of Nucleoporin-98 nanobody MS98-6 complex solved at 2.2A resolution | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Anti-Nup98 Nanobody MS98-6, Nuclear pore complex protein Nup98-Nup96, ... | 著者 | Sola-Colom, M, Trakhanov, S, Goerlich, D. | 登録日 | 2021-03-01 | 公開日 | 2021-07-21 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | A checkpoint function for Nup98 in nuclear pore formation suggested by novel inhibitory nanobodies. Embo J., 2024
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2BJB
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![BU of 2bjb by Molmil](/molmil-images/mine/2bjb) | Mycobacterium Tuberculosis Epsp Synthase In Unliganded State | 分子名称: | 3-PHOSPHOSHIKIMATE 1-CARBOXYVINYLTRANSFERASE, ACETATE ION, SODIUM ION | 著者 | Bourenkov, G.P, Kachalova, G.S, Strizhov, N, Bruning, M, Vagin, A, Bartunik, H.D. | 登録日 | 2005-02-01 | 公開日 | 2006-03-09 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Mycobacterium Tuberculosis Epsp Synthase in Unliganded State To be Published
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8PNX
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![BU of 8pnx by Molmil](/molmil-images/mine/8pnx) | Crystal structure of D-amino acid aminotransferase from Blastococcus saxobsidens in PMP form | 分子名称: | 1,2-ETHANEDIOL, 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, Branched-chain amino acid aminotransferase/4-amino-4-deoxychorismate lyase, ... | 著者 | Matyuta, I.O, Boyko, K.M, Nikolaeva, A.Y, Shilova, S.A, Popov, V.O. | 登録日 | 2023-07-03 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural determinants of dual substrate recognition in the transaminase from Blastococcus saxobsidens specific to D-amino acids and R-amines To Be Published
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8PIW
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![BU of 8piw by Molmil](/molmil-images/mine/8piw) | Crystal structure of Hen Egg White Lysozyme co-crystallized with 10 mM TbXo4-NMet2 | 分子名称: | 6-[[4-[(6-carboxypyridin-2-yl)methyl]-7-[3-(dimethylamino)propyl]-1,4,7-triazonan-1-yl]methyl]pyridine-2-carboxylic acid, CHLORIDE ION, Lysozyme C, ... | 著者 | Alsalman, Z, Girard, E. | 登録日 | 2023-06-22 | 公開日 | 2024-07-10 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Influence of Chemical Modifications of the Crystallophore on Protein Nucleating Properties and Supramolecular Interactions Network. Chemistry, 30, 2024
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8PJD
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![BU of 8pjd by Molmil](/molmil-images/mine/8pjd) | Crystal Structure of Mus musculus Protein Arginine Methyltransferase 2 94-445 | 分子名称: | ACETATE ION, Protein arginine N-methyltransferase 2, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Cura, V, Troffer-Charlier, N, Marechal, N, Bonnefond, L, Cavarelli, J. | 登録日 | 2023-06-23 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Crystal Structure of Mus musculus Protein Arginine Methyltransferase 2 94-445 To Be Published
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7O1U
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8PTD
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![BU of 8ptd by Molmil](/molmil-images/mine/8ptd) | The surface-exposed lipo-protein of BtuG1 in complex with cyanocobalamin. | 分子名称: | COBALAMIN, GLYCEROL, HYDROXIDE ION, ... | 著者 | Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J. | 登録日 | 2023-07-14 | 公開日 | 2024-07-24 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | The surface-exposed lipo-protein of BtuG1 in complex with cyanocobalamin. To Be Published
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7O86
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![BU of 7o86 by Molmil](/molmil-images/mine/7o86) | 1.73A X-ray crystal structure of the conserved C-terminal (CCT) of human SPAK | 分子名称: | CALCIUM ION, MAGNESIUM ION, SODIUM ION, ... | 著者 | Elvers, K.T, Bax, B.D, Lipka-Lloyd, M, Mehellou, Y. | 登録日 | 2021-04-14 | 公開日 | 2021-09-22 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Structures of the Human SPAK and OSR1 Conserved C-Terminal (CCT) Domains. Chembiochem, 23, 2022
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2C21
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![BU of 2c21 by Molmil](/molmil-images/mine/2c21) | Specificity of the Trypanothione-dependednt Leishmania major Glyoxalase I: Structure and biochemical comparison with the human enzyme | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, NICKEL (II) ION, ... | 著者 | Ariza, A, Vickers, T.J, Greig, N, Armour, K.A, Eggleston, I.M, Fairlamb, A.H, Bond, C.S. | 登録日 | 2005-09-23 | 公開日 | 2006-02-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Specificity of the Trypanothione-Dependent Leishmania Major Glyoxalase I: Structure and Biochemical Comparison with the Human Enzyme. Mol.Microbiol., 59, 2006
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8PWK
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![BU of 8pwk by Molmil](/molmil-images/mine/8pwk) | human HINT1 in complex with compound AT8003 | 分子名称: | Histidine triad nucleotide-binding protein 1, SODIUM ION, [(2~{R},3~{R},4~{R},5~{R})-5-[2-azanyl-6-(methylamino)purin-9-yl]-4-fluoranyl-4-methyl-3-oxidanyl-oxolan-2-yl]methyl dihydrogen phosphate | 著者 | Zimberger, C, Canard, B, Ferron, F. | 登録日 | 2023-07-20 | 公開日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (2.095 Å) | 主引用文献 | The activation chain of the broad-spectrum antiviral bemnifosbuvir at atomic resolution Plos Biol., 2024
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7OG3
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![BU of 7og3 by Molmil](/molmil-images/mine/7og3) | IRED-88 | 分子名称: | NAD(P)-dependent oxidoreductase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, SODIUM ION | 著者 | Faller, M, Koch, E. | 登録日 | 2021-05-06 | 公開日 | 2021-10-06 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.904 Å) | 主引用文献 | Machine-Directed Evolution of an Imine Reductase for Activity and Stereoselectivity Acs Catalysis, 2021
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2BPU
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![BU of 2bpu by Molmil](/molmil-images/mine/2bpu) | The Kedge Holmium Derivative of Hen Egg-White Lysozyme at high resolution from Single Wavelength Anomalous Diffraction | 分子名称: | CHLORIDE ION, HOLMIUM ATOM, LYSOZYME C, ... | 著者 | Jakoncic, J, Di Michiel, M, Zhong, Z, Honkimaki, V, Jouanneau, Y, Stojanoff, V. | 登録日 | 2005-04-25 | 公開日 | 2006-08-24 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Anomalous Diffraction at Ultra-High Energy for Protein Crystallography. J.Appl.Crystallogr., 39, 2006
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8Q1F
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![BU of 8q1f by Molmil](/molmil-images/mine/8q1f) | D10N,P146A variant of beta-phosphoglucomutase from Lactococcus lactis in complex with native beta-glucose 1,6-bisphosphate intermediate | 分子名称: | 1,2-ETHANEDIOL, 1,6-di-O-phosphono-beta-D-glucopyranose, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ... | 著者 | Cruz-Navarrete, F.A, Baxter, N.J, Flinders, A.J, Buzoianu, A, Cliff, M.J, Baker, P.J, Waltho, J.P. | 登録日 | 2023-07-31 | 公開日 | 2024-08-07 | 実験手法 | X-RAY DIFFRACTION (1.01 Å) | 主引用文献 | Peri active site catalysis of proline isomerisation is the molecular basis of allomorphy in beta-phosphoglucomutase. Commun Biol, 7, 2024
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1AT5
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![BU of 1at5 by Molmil](/molmil-images/mine/1at5) | HEN EGG WHITE LYSOZYME WITH A SUCCINIMIDE RESIDUE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, LYSOZYME, ... | 著者 | Noguchi, S, Miyawaki, K, Satow, Y. | 登録日 | 1997-08-18 | 公開日 | 1998-02-25 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Succinimide and isoaspartate residues in the crystal structures of hen egg-white lysozyme complexed with tri-N-acetylchitotriose. J.Mol.Biol., 278, 1998
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