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1TZE
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SIGNAL TRANSDUCTION ADAPTOR GROWTH FACTOR, GRB2 SH2 DOMAIN COMPLEXED WITH PHOSPHOTYROSYL HEPTAPEPTIDE LYS-PRO-PHE-PTYR-VAL-ASN-VAL-NH2 (KFPPYVNC-NH2)
分子名称: GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2, PHOSPHOTYROSYL HEPTAPEPTIDE LYS-PRO-PHE-PTYR-VAL-ASN-VAL-NH2
著者Rahuel, J, Grutter, M.G.
登録日1996-06-06
公開日1997-07-07
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural basis for specificity of Grb2-SH2 revealed by a novel ligand binding mode.
Nat.Struct.Biol., 3, 1996
1TYM
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THE STRUCTURE OF A COMPLEX OF HEXAMERIC INSULIN AND 4'-HYDROXYACETANILIDE
分子名称: CHLORIDE ION, INSULIN, N-(4-HYDROXYPHENYL)ACETAMIDE (TYLENOL), ...
著者Smith, G.D, Ciszak, E.
登録日1994-06-21
公開日1994-09-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The structure of a complex of hexameric insulin and 4'-hydroxyacetanilide.
Proc.Natl.Acad.Sci.USA, 91, 1994
1TNL
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PREDICTION OF NOVEL SERINE PROTEASE INHIBITORS
分子名称: CALCIUM ION, TRANS-2-PHENYLCYCLOPROPYLAMINE, TRYPSIN
著者Kurinov, I, Harrison, R.W.
登録日1994-07-21
公開日1994-11-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Prediction of new serine proteinase inhibitors.
Nat.Struct.Biol., 1, 1994
1TYN
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ATOMIC STRUCTURE OF THE TRYPSIN-CYCLOTHEONAMIDE A COMPLEX: LESSONS FOR THE DESIGN OF SERINE PROTEASE INHIBITORS
分子名称: BETA-TRYPSIN, CYCLOTHEONAMIDE A
著者Lee, A.Y, Hagihara, M, Karmacharya, R, Albers, M.W, Schreiber, S.L, Clardy, J.
登録日1994-09-19
公開日1995-01-26
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Atomic Structure of the Trypsin-Cyclotheonamide a Complex: Lessons for the Design of Serine Protease Inhibitors
J.Am.Chem.Soc., 115, 1993
1TPP
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THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS
分子名称: (2S)-3-(4-carbamimidoylphenyl)-2-hydroxypropanoic acid, BETA-TRYPSIN, CALCIUM ION, ...
著者Walter, J, Bode, W, Huber, R.
登録日1982-09-27
公開日1983-01-18
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors
Acta Crystallogr.,Sect.B, 39, 1983
1UCO
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HEN EGG-WHITE LYSOZYME, LOW HUMIDITY FORM
分子名称: LYSOZYME
著者Nagendra, H.G, Sudarsanakumar, C, Vijayan, M.
登録日1995-12-31
公開日1996-07-11
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An X-ray analysis of native monoclinic lysozyme. A case study on the reliability of refined protein structures and a comparison with the low-humidity form in relation to mobility and enzyme action.
Acta Crystallogr.,Sect.D, 52, 1996
1TNH
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PREDICTION OF NOVEL SERINE PROTEASE INHIBITORS
分子名称: 4-FLUOROBENZYLAMINE, CALCIUM ION, TRYPSIN
著者Kurinov, I, Harrison, R.W.
登録日1994-07-21
公開日1994-11-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Prediction of new serine proteinase inhibitors.
Nat.Struct.Biol., 1, 1994
1TPO
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THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS
分子名称: BETA-TRYPSIN, CALCIUM ION
著者Bode, W, Walter, J, Huber, R.
登録日1982-09-27
公開日1983-01-18
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors
Acta Crystallogr.,Sect.B, 39, 1983
5BVF
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Tetrahydropyrrolo-diazepenones as inhibitors of ERK2 kinase
分子名称: 2-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1S,3R)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepin-1-one, Mitogen-activated protein kinase 1, SULFATE ION
著者Ma, X, Steven, S.
登録日2015-06-05
公開日2015-09-09
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Tetrahydropyrrolo-diazepenones as inhibitors of ERK2 kinase.
Bioorg.Med.Chem.Lett., 25, 2015
1UH7
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Crystal structure of rhizopuspepsin at pH 4.6
分子名称: hizopuspepsin I
著者Prasad, B.V.L.S, Suguna, K.
登録日2003-06-26
公開日2004-06-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Effect of pH on the structure of rhizopuspepsin.
Acta Crystallogr.,Sect.D, 59, 2003
1UHG
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Crystal Structure of S-Ovalbumin At 1.9 Angstrom Resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Ovalbumin, ...
著者Yamasaki, M, Takahashi, N, Hirose, M.
登録日2003-07-03
公開日2003-07-22
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal Structure of S-ovalbumin as a Non-loop-inserted Thermostabilized Serpin Form
J.Biol.Chem., 278, 2003
5C1Q
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Serine/threonine-protein kinase pim-1
分子名称: 3-methoxy[1]benzothieno[2,3-c]quinolin-6(5H)-one, Serine/threonine-protein kinase pim-1
著者Li, W, Wan, X, Huang, N.
登録日2015-06-15
公開日2015-12-16
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Serine/threonine-protein kinase pim-1
To Be Published
1UH9
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Crystal structure of rhizopuspepsin at pH 7.0
分子名称: hizopuspepsin I
著者Prasad, B.V.L.S, Suguna, K.
登録日2003-06-26
公開日2004-06-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Effect of pH on the structure of rhizopuspepsin.
Acta Crystallogr.,Sect.D, 59, 2003
1UHS
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Solution structure of mouse homeodomain-only protein HOP
分子名称: homeodomain only protein
著者Saito, K, Koshiba, S, Inoue, M, Shirouzu, M, Terada, T, Yabuki, T, Aoki, M, Matsuda, T, Seki, E, Hirota, H, Yoshida, M, Tanaka, A, Osanai, T, Arakawa, T, Carninci, P, Kawai, J, Hayashizaki, Y, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2003-07-10
公開日2004-07-10
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Solution structure of mouse homeodomain-only protein HOP
To be Published
1UIH
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ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LYSOZYME
著者Motoshima, H, Ohmura, T, Ueda, T, Imoto, T.
登録日1996-11-26
公開日1997-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Fluctuations in free or substrate-complexed lysozyme and a mutant of it detected on x-ray crystallography and comparison with those detected on NMR.
J.Biochem.(Tokyo), 131, 2002
3S4Q
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P38 alpha kinase complexed with a pyrazolo-triazine based inhibitor
分子名称: 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-N-cyclopropyl-4-methylbenzamide, Mitogen-activated protein kinase 14
著者Sack, J.S.
登録日2011-05-20
公開日2012-02-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitors.
Bioorg.Med.Chem.Lett., 21, 2011
1UIB
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ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LYSOZYME
著者Motoshima, H, Ohmura, T, Ueda, T, Imoto, T.
登録日1996-11-26
公開日1997-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献Fluctuations in free or substrate-complexed lysozyme and a mutant of it detected on x-ray crystallography and comparison with those detected on NMR.
J.Biochem.(Tokyo), 131, 2002
3SA0
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Complex of ERK2 with norathyriol
分子名称: Mitogen-activated protein kinase 1, SULFATE ION, norathyriol
著者Kurinov, I, Malakhova, M.
登録日2011-06-02
公開日2011-12-14
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.5947 Å)
主引用文献Norathyriol Suppresses Skin Cancers Induced by Solar Ultraviolet Radiation by Targeting ERK Kinases.
Cancer Res., 72, 2012
1UIF
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ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS
分子名称: LYSOZYME
著者Motoshima, H, Ohmura, T, Ueda, T, Imoto, T.
登録日1996-11-26
公開日1997-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Analysis of the stability of mutant lysozymes at position 15 using X-ray crystallography.
J.Biochem.(Tokyo), 122, 1997
1UID
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ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS
分子名称: LYSOZYME
著者Motoshima, H, Ohmura, T, Ueda, T, Imoto, T.
登録日1996-11-26
公開日1997-11-26
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Analysis of the stability of mutant lysozymes at position 15 using X-ray crystallography.
J.Biochem.(Tokyo), 122, 1997
1UH8
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Crystal structure of rhizopuspepsin at pH 8.0
分子名称: hizopuspepsin I
著者Prasad, B.V.L.S, Suguna, K.
登録日2003-06-26
公開日2004-06-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Effect of pH on the structure of rhizopuspepsin.
Acta Crystallogr.,Sect.D, 59, 2003
1UHF
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Solution Structure of the third SH3 domain of human intersectin 2(KIAA1256)
分子名称: INTERSECTIN 2
著者Suzuki, S, Hatanaka, H, Koshiba, S, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2003-07-03
公開日2004-08-10
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Solution Structure of the third SH3 domain of human intersectin 2(KIAA1256)
To be Published
1UHB
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Crystal structure of porcine alpha trypsin bound with auto catalyticaly produced native peptide at 2.15 A resolution
分子名称: 9-mer peptide from Trypsin, ACETATE ION, CALCIUM ION, ...
著者Pattabhi, V, Syed Ibrahim, B, Shamaladevi, N.
登録日2003-06-27
公開日2004-07-27
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Trypsin activity reduced by an autocatalytically produced nonapeptide.
J.Biomol.Struct.Dyn., 21, 2004
1UHZ
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Solution structure of dsRNA binding domain in Staufen homolog 2
分子名称: staufen (RNA binding protein) homolog 2
著者He, F, Muto, Y, Obayashi, N, Shirouzu, M, Terada, T, Kigawa, T, Inoue, M, Yabuki, T, Aoki, M, Seki, E, Matsuda, T, Hirota, H, Yoshida, M, Koboyashi, N, Tanaka, A, Osanai, T, Matsuo, Y, Hayashizaki, Y, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2003-07-14
公開日2004-08-03
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Solution structure of dsRNA binding domain in Staufen homolog 2
To be Published
1UN5
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ARH-II, AN ANGIOGENIN/RNASE A CHIMERA
分子名称: ANGIOGENIN, CITRIC ACID
著者Holloway, D.E, Baker, M.D, Acharya, K.R.
登録日2003-09-04
公開日2004-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystallographic Studies on Structural Features that Determine the Enzymatic Specificity and Potency of Human Angiogenin: Thr44, Thr80 and Residues 38-41
Biochemistry, 43, 2004

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件を2024-09-11に公開中

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