1TZE
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1TYM
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1TNL
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1TYN
| ATOMIC STRUCTURE OF THE TRYPSIN-CYCLOTHEONAMIDE A COMPLEX: LESSONS FOR THE DESIGN OF SERINE PROTEASE INHIBITORS | 分子名称: | BETA-TRYPSIN, CYCLOTHEONAMIDE A | 著者 | Lee, A.Y, Hagihara, M, Karmacharya, R, Albers, M.W, Schreiber, S.L, Clardy, J. | 登録日 | 1994-09-19 | 公開日 | 1995-01-26 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Atomic Structure of the Trypsin-Cyclotheonamide a Complex: Lessons for the Design of Serine Protease Inhibitors J.Am.Chem.Soc., 115, 1993
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1TPP
| THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | (2S)-3-(4-carbamimidoylphenyl)-2-hydroxypropanoic acid, BETA-TRYPSIN, CALCIUM ION, ... | 著者 | Walter, J, Bode, W, Huber, R. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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1UCO
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1TNH
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1TPO
| THE GEOMETRY OF THE REACTIVE SITE AND OF THE PEPTIDE GROUPS IN TRYPSIN, TRYPSINOGEN AND ITS COMPLEXES WITH INHIBITORS | 分子名称: | BETA-TRYPSIN, CALCIUM ION | 著者 | Bode, W, Walter, J, Huber, R. | 登録日 | 1982-09-27 | 公開日 | 1983-01-18 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Geometry of the Reactive Site and of the Peptide Groups in Trypsin, Trypsinogen and its Complexes with Inhibitors Acta Crystallogr.,Sect.B, 39, 1983
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5BVF
| Tetrahydropyrrolo-diazepenones as inhibitors of ERK2 kinase | 分子名称: | 2-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1S,3R)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1H-pyrrolo[1,2-a][1,4]diazepin-1-one, Mitogen-activated protein kinase 1, SULFATE ION | 著者 | Ma, X, Steven, S. | 登録日 | 2015-06-05 | 公開日 | 2015-09-09 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Tetrahydropyrrolo-diazepenones as inhibitors of ERK2 kinase. Bioorg.Med.Chem.Lett., 25, 2015
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1UH7
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1UHG
| Crystal Structure of S-Ovalbumin At 1.9 Angstrom Resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Ovalbumin, ... | 著者 | Yamasaki, M, Takahashi, N, Hirose, M. | 登録日 | 2003-07-03 | 公開日 | 2003-07-22 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure of S-ovalbumin as a Non-loop-inserted Thermostabilized Serpin Form J.Biol.Chem., 278, 2003
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5C1Q
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1UH9
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1UHS
| Solution structure of mouse homeodomain-only protein HOP | 分子名称: | homeodomain only protein | 著者 | Saito, K, Koshiba, S, Inoue, M, Shirouzu, M, Terada, T, Yabuki, T, Aoki, M, Matsuda, T, Seki, E, Hirota, H, Yoshida, M, Tanaka, A, Osanai, T, Arakawa, T, Carninci, P, Kawai, J, Hayashizaki, Y, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2003-07-10 | 公開日 | 2004-07-10 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of mouse homeodomain-only protein HOP To be Published
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1UIH
| ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LYSOZYME | 著者 | Motoshima, H, Ohmura, T, Ueda, T, Imoto, T. | 登録日 | 1996-11-26 | 公開日 | 1997-11-26 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Fluctuations in free or substrate-complexed lysozyme and a mutant of it detected on x-ray crystallography and comparison with those detected on NMR. J.Biochem.(Tokyo), 131, 2002
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3S4Q
| P38 alpha kinase complexed with a pyrazolo-triazine based inhibitor | 分子名称: | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-N-cyclopropyl-4-methylbenzamide, Mitogen-activated protein kinase 14 | 著者 | Sack, J.S. | 登録日 | 2011-05-20 | 公開日 | 2012-02-01 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitors. Bioorg.Med.Chem.Lett., 21, 2011
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1UIB
| ANALYSIS OF THE STABILIZATION OF HEN LYSOZYME WITH THE HELIX DIPOLE AND CHARGED SIDE CHAINS | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LYSOZYME | 著者 | Motoshima, H, Ohmura, T, Ueda, T, Imoto, T. | 登録日 | 1996-11-26 | 公開日 | 1997-11-26 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Fluctuations in free or substrate-complexed lysozyme and a mutant of it detected on x-ray crystallography and comparison with those detected on NMR. J.Biochem.(Tokyo), 131, 2002
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3SA0
| Complex of ERK2 with norathyriol | 分子名称: | Mitogen-activated protein kinase 1, SULFATE ION, norathyriol | 著者 | Kurinov, I, Malakhova, M. | 登録日 | 2011-06-02 | 公開日 | 2011-12-14 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.5947 Å) | 主引用文献 | Norathyriol Suppresses Skin Cancers Induced by Solar Ultraviolet Radiation by Targeting ERK Kinases. Cancer Res., 72, 2012
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1UIF
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1UID
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1UH8
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1UHF
| Solution Structure of the third SH3 domain of human intersectin 2(KIAA1256) | 分子名称: | INTERSECTIN 2 | 著者 | Suzuki, S, Hatanaka, H, Koshiba, S, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2003-07-03 | 公開日 | 2004-08-10 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution Structure of the third SH3 domain of human intersectin 2(KIAA1256) To be Published
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1UHB
| Crystal structure of porcine alpha trypsin bound with auto catalyticaly produced native peptide at 2.15 A resolution | 分子名称: | 9-mer peptide from Trypsin, ACETATE ION, CALCIUM ION, ... | 著者 | Pattabhi, V, Syed Ibrahim, B, Shamaladevi, N. | 登録日 | 2003-06-27 | 公開日 | 2004-07-27 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Trypsin activity reduced by an autocatalytically produced nonapeptide. J.Biomol.Struct.Dyn., 21, 2004
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1UHZ
| Solution structure of dsRNA binding domain in Staufen homolog 2 | 分子名称: | staufen (RNA binding protein) homolog 2 | 著者 | He, F, Muto, Y, Obayashi, N, Shirouzu, M, Terada, T, Kigawa, T, Inoue, M, Yabuki, T, Aoki, M, Seki, E, Matsuda, T, Hirota, H, Yoshida, M, Koboyashi, N, Tanaka, A, Osanai, T, Matsuo, Y, Hayashizaki, Y, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2003-07-14 | 公開日 | 2004-08-03 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of dsRNA binding domain in Staufen homolog 2 To be Published
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1UN5
| ARH-II, AN ANGIOGENIN/RNASE A CHIMERA | 分子名称: | ANGIOGENIN, CITRIC ACID | 著者 | Holloway, D.E, Baker, M.D, Acharya, K.R. | 登録日 | 2003-09-04 | 公開日 | 2004-02-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystallographic Studies on Structural Features that Determine the Enzymatic Specificity and Potency of Human Angiogenin: Thr44, Thr80 and Residues 38-41 Biochemistry, 43, 2004
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