8X2P
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![BU of 8x2p by Molmil](/molmil-images/mine/8x2p) | The Crystal Structure of LCK from Biortus. | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, TETRAETHYLENE GLYCOL, ... | 著者 | Wang, F, Cheng, W, Lv, Z, Meng, Q, Lu, Y. | 登録日 | 2023-11-10 | 公開日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | The Crystal Structure of LCK from Biortus. To Be Published
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8WBS
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![BU of 8wbs by Molmil](/molmil-images/mine/8wbs) | Crystal structure of cis-Epoxysuccinate Hydrolases KlCESH[L]-D48N complexed with sulfate ions | 分子名称: | (S)-2-haloacid dehalogenase, CALCIUM ION, SULFATE ION | 著者 | Dong, S, Xuan, J.S, Feng, Y.G, Cui, Q. | 登録日 | 2023-09-10 | 公開日 | 2024-01-31 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Deciphering the stereo-specific catalytic mechanisms of cis-epoxysuccinate hydrolases producing L(+)-tartaric acid. J.Biol.Chem., 300, 2024
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8X2Q
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![BU of 8x2q by Molmil](/molmil-images/mine/8x2q) | The Crystal Structure of APC from Biortus. | 分子名称: | 1,2-ETHANEDIOL, Adenomatous polyposis coli protein | 著者 | Wang, F, Cheng, W, Lv, Z, Ju, C, Bao, C. | 登録日 | 2023-11-10 | 公開日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The Crystal Structure of APC from Biortus. To Be Published
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8XI8
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![BU of 8xi8 by Molmil](/molmil-images/mine/8xi8) | |
8UTG
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![BU of 8utg by Molmil](/molmil-images/mine/8utg) | An RNA G-Quadruplex from the NS5 gene in the West Nile Virus Genome | 分子名称: | AMMONIUM ION, POTASSIUM ION, RNA (5'-R(*UP*AP*UP*GP*GP*AP*AP*GP*AP*GP*GP*CP*GP*GP*UP*UP*GP*GP*UP*AP*U)-3') | 著者 | Terrell, J.R, Le, T.T, Wilson, W.D, Siemer, J.L. | 登録日 | 2023-10-31 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Structure of an RNA G-quadruplex from the West Nile virus genome. Nat Commun, 15, 2024
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8TXA
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![BU of 8txa by Molmil](/molmil-images/mine/8txa) | Apo Structure of (N1G37) tRNA Methyltransferase from Mycobacterium marinum | 分子名称: | tRNA (guanine-N(1)-)-methyltransferase | 著者 | Balsamo, A, Bruno, C, Edele, C, Fabian, T, Jannotta, R, Lee, R, Schryver, D, Warsaw, J, Warsaw, L, Stojanoff, V, Battaile, K, Perez, A, Bolen, R. | 登録日 | 2023-08-23 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (1.591 Å) | 主引用文献 | Apo Structure of (N1G37) tRNA Methyltransferase from Mycobacterium marinum To Be Published
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8V97
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![BU of 8v97 by Molmil](/molmil-images/mine/8v97) | GII.17 CS-E1 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein VP1, DI(HYDROXYETHYL)ETHER | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 2024
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8YX1
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![BU of 8yx1 by Molmil](/molmil-images/mine/8yx1) | CD40 in complex with Bleselumab Fab | 分子名称: | Bleselumab, heavy chain, light chain, ... | 著者 | Caaveiro, J.M.M, Fernandez-Perez, J, Tsumoto, K. | 登録日 | 2024-04-01 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal structures of human CD40 in complex with monoclonal antibodies dacetuzumab and bleselumab. Biochem.Biophys.Res.Commun., 714, 2024
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8VET
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![BU of 8vet by Molmil](/molmil-images/mine/8vet) | |
8X34
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![BU of 8x34 by Molmil](/molmil-images/mine/8x34) | |
8VEU
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![BU of 8veu by Molmil](/molmil-images/mine/8veu) | |
8VR0
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![BU of 8vr0 by Molmil](/molmil-images/mine/8vr0) | |
8WD2
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![BU of 8wd2 by Molmil](/molmil-images/mine/8wd2) | The Crystal Structure of p53 from Biortus. | 分子名称: | 1,2-ETHANEDIOL, Cellular tumor antigen p53, PHOSPHATE ION, ... | 著者 | Wang, F, Cheng, W, Yuan, Z, Qi, J, Lu, Y. | 登録日 | 2023-09-14 | 公開日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | The Crystal Structure of p53 from Biortus. To Be Published
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8VRV
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![BU of 8vrv by Molmil](/molmil-images/mine/8vrv) | GII.4c H2-tri HBGA norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein, FORMIC ACID, ... | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2024-01-22 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.61 Å) | 主引用文献 | Advancement of norovirus therapies To Be Published
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8XGA
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8TNV
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![BU of 8tnv by Molmil](/molmil-images/mine/8tnv) | Hemocyanin Functional Unit CCHB-g of Concholepas concholepas | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Munoz, S, Vallejos-Baccelliere, G, Manubens, A, Salazar, M, Nascimento, A.F.Z, Ambrosio, A.L.B, Becker, M.I, Guixe, V, Castro-Fernandez, V. | 登録日 | 2023-08-02 | 公開日 | 2024-04-10 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural insights into a functional unit from an immunogenic mollusk hemocyanin. Structure, 32, 2024
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8WBT
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![BU of 8wbt by Molmil](/molmil-images/mine/8wbt) | Crystal structure of cis-Epoxysuccinate Hydrolases KlCESH[L] mutant D48N complexed with L-TA | 分子名称: | (S)-2-haloacid dehalogenase, CALCIUM ION, GLYCEROL, ... | 著者 | Dong, S, Xuan, J.S, Feng, Y.G, Cui, Q. | 登録日 | 2023-09-10 | 公開日 | 2024-01-31 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Deciphering the stereo-specific catalytic mechanisms of cis-epoxysuccinate hydrolases producing L(+)-tartaric acid. J.Biol.Chem., 300, 2024
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8WF7
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![BU of 8wf7 by Molmil](/molmil-images/mine/8wf7) | The Crystal Structure of integrase from Biortus | 分子名称: | ACETATE ION, Integrase, SULFATE ION | 著者 | Wang, F, Cheng, W, Yuan, Z, Qi, J, Li, J. | 登録日 | 2023-09-19 | 公開日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | The Crystal Structure of integrase from Biortus To Be Published
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8X5Z
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8V1O
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![BU of 8v1o by Molmil](/molmil-images/mine/8v1o) | Crystal structure of IRAK4 kinase domain with compound 4 | 分子名称: | CHLORIDE ION, GLYCEROL, Interleukin-1 receptor-associated kinase 4, ... | 著者 | Weiss, M.M, Zheng, X, Browne, C.M, Campbell, V, Chen, D, Enerson, B, Fei, X, Huang, X, Klaus, C.R, Li, H, Mayo, M, McDonald, A.A, Paul, A, Sharma, K, Shi, Y, Slavin, A, Walter, D.M, Yuan, K, Zhang, Y, Zhu, X, Kelleher, J, Ji, N, Walker, D, Mainolfi, N. | 登録日 | 2023-11-21 | 公開日 | 2024-07-03 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.92 Å) | 主引用文献 | Discovery of KT-413, a Targeted Protein Degrader of IRAK4 and IMiD Substrates Targeting MYD88 Mutant Diffuse Large B-Cell Lymphoma. J.Med.Chem., 2024
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8UDC
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![BU of 8udc by Molmil](/molmil-images/mine/8udc) | Crystal structure of TcPINK1 in complex with CYC116 | 分子名称: | (4P)-4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin-4-yl)phenyl]pyrimidin-2-amine, DI(HYDROXYETHYL)ETHER, SULFATE ION, ... | 著者 | Veyron, S, Rasool, S, Trempe, J.F. | 登録日 | 2023-09-28 | 公開日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural Characterization of a small-molecule inhibitor of PINK1, a precursor tool compound for the study of Parkinson's disease To Be Published
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8YJ8
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![BU of 8yj8 by Molmil](/molmil-images/mine/8yj8) | Characerization of a novel format scFvXVHH single-chain Biparatopic antibody against a metal binding protein, MtsA | 分子名称: | Iron ABC transporter substrate-binding lipoprotein MtsA, VHH43, ZINC ION | 著者 | Ito, S, Nagatoishi, S, Nakakido, M, Tsumoto, K. | 登録日 | 2024-03-01 | 公開日 | 2024-06-19 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Characterization of a novel format scFv×VHH single-chain biparatopic antibody against metal binding protein MtsA. Protein Sci., 33, 2024
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8YTR
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![BU of 8ytr by Molmil](/molmil-images/mine/8ytr) | The structure of Cu(II)-CopC from Thioalkalivibrio paradoxus | 分子名称: | COPPER (II) ION, CopC domain-containing protein, DI(HYDROXYETHYL)ETHER | 著者 | Kulikova, O.G, Solovieva, A.Y, Varfolomeeva, L.A, Dergousova, N.I, Nikolaeva, A.Y, Boyko, K.M, Tikhonova, T.V, Popov, V.O. | 登録日 | 2024-03-26 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The structure of Cu(II)-CopC from Thioalkalivibrio paradoxus To Be Published
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8YU9
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![BU of 8yu9 by Molmil](/molmil-images/mine/8yu9) | Tubulin-RB3-TTL in complex with compound SI10 | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(2-chloranylthieno[3,2-d]pyrimidin-4-yl)-7-methoxy-1,3-dihydroquinoxalin-2-one, CALCIUM ION, ... | 著者 | Wu, C.Y, Wang, Y.X. | 登録日 | 2024-03-27 | 公開日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | The crystal structure of tubulin-RB3-TTL in complex with compound AB10 To Be Published
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8V2L
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![BU of 8v2l by Molmil](/molmil-images/mine/8v2l) | Crystal structure of IRAK4 kinase domain with compound 8 | 分子名称: | 1,2-ETHANEDIOL, Interleukin-1 receptor-associated kinase 4, N-{2-[4-(hydroxymethyl)phenyl]-6-(2-hydroxypropan-2-yl)-2H-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide | 著者 | Weiss, M.M, Zheng, X, Browne, C.M, Campbell, V, Chen, D, Enerson, B, Fei, X, Huang, X, Klaus, C.R, Li, H, Mayo, M, McDonald, A.A, Paul, A, Sharma, K, Shi, Y, Slavin, A, Walter, D.M, Yuan, K, Zhang, Y, Zhu, X, Kelleher, J, Ji, N, Walker, D, Mainolfi, N. | 登録日 | 2023-11-22 | 公開日 | 2024-07-03 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | Discovery of KT-413, a Targeted Protein Degrader of IRAK4 and IMiD Substrates Targeting MYD88 Mutant Diffuse Large B-Cell Lymphoma. J.Med.Chem., 2024
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