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4MGS
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BU of 4mgs by Molmil
BiXyn10A CBM1 APO
分子名称: Putative glycosyl hydrolase family 10
著者Chekan, J.R, Nair, S.K.
登録日2013-08-28
公開日2014-08-20
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Xylan utilization in human gut commensal bacteria is orchestrated by unique modular organization of polysaccharide-degrading enzymes.
Proc.Natl.Acad.Sci.USA, 111, 2014
4EVH
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BU of 4evh by Molmil
Crystal structure of calcium-bound alpha-1 giardin
分子名称: CALCIUM ION, Giardin subunit alpha-1
著者Weeratunga, S, Hofmann, A.
登録日2012-04-26
公開日2012-07-25
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Alpha-1 giardin is an annexin with highly unusual calcium-regulated mechanisms
J.Mol.Biol., 423, 2012
4EVF
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BU of 4evf by Molmil
Crystal structure of apo alpha-1 giardin
分子名称: Giardin subunit alpha-1
著者Weeratunga, S, Hofmann, A.
登録日2012-04-26
公開日2012-07-25
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Alpha-1 giardin is an annexin with highly unusual calcium-regulated mechanisms
J.Mol.Biol., 423, 2012
5KYJ
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BU of 5kyj by Molmil
Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core
分子名称: (6~{R})-5-(5-fluoranyl-2-methoxy-pyrimidin-4-yl)-2-(3-methylsulfonylphenyl)-6-propan-2-yl-4,6-dihydropyrrolo[3,4-c]pyrazole, Oxysterols receptor LXR-beta, Retinoic acid receptor RXR-beta
著者Chen, G, McKeever, B.M.
登録日2016-07-21
公開日2016-09-21
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core.
Bioorg.Med.Chem.Lett., 26, 2016
5KYA
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BU of 5kya by Molmil
Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core
分子名称: Oxysterols receptor LXR-beta, Retinoic acid receptor RXR-beta, [2-[(6~{R})-2-(3-methylsulfonylphenyl)-6-propan-2-yl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]-4-(trifluoromethyl)pyrimidin-5-yl]methanol
著者Chen, G, McKeever, B.M.
登録日2016-07-21
公開日2016-09-21
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.598 Å)
主引用文献Brain penetrant liver X receptor (LXR) modulators based on a 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole core.
Bioorg.Med.Chem.Lett., 26, 2016
5LDY
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BU of 5ldy by Molmil
Structure of Yersinia pseudotuberculosis InvD
分子名称: Ig domain protein group 1 domain protein, PHOSPHATE ION
著者Sadana, P, Scrima, A.
登録日2016-06-28
公開日2017-06-14
最終更新日2020-06-17
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The invasin D protein from Yersinia pseudotuberculosis selectively binds the Fab region of host antibodies and affects colonization of the intestine
J.Biol.Chem., 2018
3PF3
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BU of 3pf3 by Molmil
Crystal structure of a mutant (C202A) of Triosephosphate isomerase from Giardia lamblia derivatized with MMTS
分子名称: CALCIUM ION, GLYCEROL, SULFATE ION, ...
著者Enriquez-Flores, S, Rodriguez-Romero, A, Hernandez-Santoyo, A, Reyes-Vivas, H.
登録日2010-10-27
公開日2011-06-22
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.098 Å)
主引用文献Determining the molecular mechanism of inactivation by chemical modification of triosephosphate isomerase from the human parasite Giardia lamblia: A study for antiparasitic drug design.
Proteins, 79, 2011
5LS9
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BU of 5ls9 by Molmil
Humanized Archaeal ferritin
分子名称: Ferritin, putative, MAGNESIUM ION
著者Baiocco, P, Trabuco, M.C, Boffi, A.
登録日2016-08-23
公開日2016-11-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.93 Å)
主引用文献Humanized archaeal ferritin as a tool for cell targeted delivery.
Nanoscale, 9, 2017
5DEF
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BU of 5def by Molmil
Crystal structure of B*27:04 complex bound to the pVIPR peptide
分子名称: Beta-2-microglobulin, CHLORIDE ION, GLYCEROL, ...
著者Loll, B, Fabian, H, Huser, H, Hee, C.S, Uchanska-Ziegler, B, Ziegler, A.
登録日2015-08-25
公開日2015-11-18
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Increased Conformational Flexibility of HLA-B*27 Subtypes Associated With Ankylosing Spondylitis.
Arthritis Rheumatol, 68, 2016
5OBB
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BU of 5obb by Molmil
Structure of a modified mouse H chain ferritin with a lanthanide binding motif in complex with Terbium
分子名称: Ferritin heavy chain, TERBIUM(III) ION
著者Baiocco, P, Trabuco, M.C.
登録日2017-06-26
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Engineered ferritin for lanthanide binding.
PLoS ONE, 13, 2018
5OBA
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BU of 5oba by Molmil
Structure of a modified mouse H-chain ferritin with a lanthanide binding motif
分子名称: FE (III) ION, Ferritin heavy chain
著者Baiocco, P, Trabuco, M.C.
登録日2017-06-26
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Engineered ferritin for lanthanide binding.
PLoS ONE, 13, 2018
5DEG
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BU of 5deg by Molmil
Crystal structure of B*27:06 bound to the pVIPR peptide
分子名称: Beta-2-microglobulin, GLYCEROL, MHC class I antigen, ...
著者Loll, B, Fabian, H, Hee, C.S, Huser, H, Uchanska-Ziegler, B, Ziegler, A.
登録日2015-08-25
公開日2015-11-18
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Increased Conformational Flexibility of HLA-B*27 Subtypes Associated With Ankylosing Spondylitis.
Arthritis Rheumatol, 68, 2016
5O3I
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BU of 5o3i by Molmil
Human Brd2(BD2) mutant in complex with AL-tBu
分子名称: (2~{S})-1-[(2~{S})-2-oxidanylpropoxy]propan-2-ol, Bromodomain-containing protein 2, CHLORIDE ION, ...
著者Chan, K.-H, Runcie, A.C, Ciulli, A.
登録日2017-05-23
公開日2018-02-14
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition.
Chem Sci, 9, 2018
2WQ1
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BU of 2wq1 by Molmil
GCN4 leucine zipper mutant with three IxxNTxx motifs coordinating bromide
分子名称: BROMIDE ION, GENERAL CONTROL PROTEIN GCN4
著者Hartmann, M.D, Hernandez Alvarez, B, Lupas, A.N.
登録日2009-08-12
公開日2009-11-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.08 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WPR
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BU of 2wpr by Molmil
Salmonella enterica SadA 483-523 fused to GCN4 adaptors (SadAK3b-V1, out-of-register fusion)
分子名称: CHLORIDE ION, TRIMERIC AUTOTRANSPORTER ADHESIN FRAGMENT
著者Hartmann, M.D, Ridderbusch, O, Lupas, A.N, Hernandez Alvarez, B.
登録日2009-08-09
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
4APN
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BU of 4apn by Molmil
Structure of TR from Leishmania infantum in complex with a diarylpirrole-based inhibitor
分子名称: 4-[[1-(4-ethylphenyl)-2-methyl-5-(4-methylsulfanylphenyl)pyrrol-3-yl]methyl]thiomorpholine, FLAVIN-ADENINE DINUCLEOTIDE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Baiocco, P, Ilari, A, Colotti, G, Biava, M.
登録日2012-04-04
公開日2013-04-17
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Inhibition of Leishmania Infantum Trypanothione Reductase by Azole-Based Compounds: A Comparative Analysis with its Physiological Substrate by X-Ray Crystallography.
Chemmedchem, 8, 2013
2WQ2
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BU of 2wq2 by Molmil
GCN4 leucine zipper mutant with three IxxNTxx motifs coordinating iodide
分子名称: GENERAL CONTROL PROTEIN GCN4, IODIDE ION
著者Hartmann, M.D, Hernandez Alvarez, B, Lupas, A.N.
登録日2009-08-12
公開日2009-11-03
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WPZ
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BU of 2wpz by Molmil
GCN4 leucine zipper mutant with two VxxNxxx motifs coordinating chloride
分子名称: CHLORIDE ION, GENERAL CONTROL PROTEIN GCN4
著者Zeth, K, Hartmann, M.D, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B.
登録日2009-08-12
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WPY
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BU of 2wpy by Molmil
GCN4 leucine zipper mutant with one VxxNxxx motif coordinating chloride
分子名称: CHLORIDE ION, GENERAL CONTROL PROTEIN GCN4
著者Zeth, K, Hartmann, M.D, Albrecht, R, Lupas, A.N, Hernandez Alvarez, B.
登録日2009-08-12
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WPQ
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BU of 2wpq by Molmil
Salmonella enterica SadA 479-519 fused to GCN4 adaptors (SadAK3, in- register fusion)
分子名称: CHLORIDE ION, NITRATE ION, TRIMERIC AUTOTRANSPORTER ADHESIN FRAGMENT
著者Hartmann, M.D, Hernandez Alvarez, B, Albrecht, R, Zeth, K, Lupas, A.N.
登録日2009-08-09
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WQ0
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BU of 2wq0 by Molmil
GCN4 leucine zipper mutant with three IxxNTxx motifs coordinating chloride
分子名称: CHLORIDE ION, GENERAL CONTROL PROTEIN GCN4
著者Hartmann, M.D, Hernandez Alvarez, B, Lupas, A.N.
登録日2009-08-12
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WPS
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BU of 2wps by Molmil
Salmonella enterica SadA 483-523 fused to GCN4 adaptors (SadAK3b-V2, out-of-register fusion)
分子名称: CHLORIDE ION, TRIMERIC AUTOTRANSPORTER ADHESIN FRAGMENT
著者Hartmann, M.D, Ridderbusch, O, Lupas, A.N, Hernandez Alvarez, B.
登録日2009-08-09
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
2WQ3
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BU of 2wq3 by Molmil
GCN4 leucine zipper mutant with three IxxNTxx motifs coordinating chloride and nitrate
分子名称: CHLORIDE ION, GENERAL CONTROL PROTEIN GCN4, NITRATE ION
著者Hartmann, M.D, Hernandez Alvarez, B, Lupas, A.N.
登録日2009-08-12
公開日2009-11-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.22 Å)
主引用文献A Coiled-Coil Motif that Sequesters Ions to the Hydrophobic Core.
Proc.Natl.Acad.Sci.USA, 106, 2009
3OMZ
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BU of 3omz by Molmil
Crystal structure of MICA-specific human gamma delta T cell receptor
分子名称: human Vdelta1 gamma delta T cell receptor delta1A/B-3
著者Xu, B, Holmes, M.A, Strong, R.K.
登録日2010-08-27
公開日2011-01-26
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3.04 Å)
主引用文献Crystal structure of a {gamma}{delta} T-cell receptor specific for the human MHC class I homolog MICA.
Proc.Natl.Acad.Sci.USA, 108, 2011
2QVW
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BU of 2qvw by Molmil
Structure of Giardia Dicer refined against twinned data
分子名称: GLP_546_48378_50642, MANGANESE (II) ION
著者Doudna, J.A, MacRae, I.J.
登録日2007-08-09
公開日2007-09-25
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献An unusual case of pseudo-merohedral twinning in orthorhombic crystals of Dicer
Acta Crystallogr.,Sect.D, 63, 2007

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