1F0N
| MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85B | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ANTIGEN 85B | 著者 | Anderson, D.H, Harth, G, Horwitz, M.A, Eisenberg, D, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2000-05-16 | 公開日 | 2001-01-24 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | An interfacial mechanism and a class of inhibitors inferred from two crystal structures of the Mycobacterium tuberculosis 30 kDa major secretory protein (Antigen 85B), a mycolyl transferase. J.Mol.Biol., 307, 2001
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1F0O
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1F0P
| MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85B WITH TREHALOSE | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ANTIGEN 85-B, ... | 著者 | Anderson, D.H, Harth, G, Horwitz, M.A, Eisenberg, D, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2000-05-16 | 公開日 | 2001-01-24 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | An interfacial mechanism and a class of inhibitors inferred from two crystal structures of the Mycobacterium tuberculosis 30 kDa major secretory protein (Antigen 85B), a mycolyl transferase. J.Mol.Biol., 307, 2001
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1F0Q
| CRYSTAL STRUCTURE OF THE ALPHA SUBUNIT OF PROTEIN KINASE CK2 IN COMPLEX WITH THE NUCLEOTIDE COMPETITIVE INHIBITOR EMODIN | 分子名称: | 3-METHYL-1,6,8-TRIHYDROXYANTHRAQUINONE, PROTEIN KINASE CK2, ALPHA SUBUNIT | 著者 | Battistutta, R, Sarno, S, De Moliner, E, Papinutto, E, Zanotti, G, Pinna, L.A. | 登録日 | 2000-05-17 | 公開日 | 2001-05-23 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | The replacement of ATP by the competitive inhibitor emodin induces conformational modifications in the catalytic site of protein kinase CK2. J.Biol.Chem., 275, 2000
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1F0R
| CRYSTAL STRUCTURE OF HUMAN COAGULATION FACTOR XA COMPLEXED WITH RPR208815 | 分子名称: | CALCIUM ION, COAGULATION FACTOR XA, THIENO[3,2-B]PYRIDINE-2-SULFONIC ACID [1-(1-AMINO-ISOQUINOLIN-7-YLMETHYL)-2-OXO-PYRROLDIN-3-YL]-AMIDE | 著者 | Maignan, S, Guilloteau, J.P, Pouzieux, S, Choi-Sledeski, Y.M, Becker, M.R, Klein, S.I, Ewing, W.R, Pauls, H.W, Spada, A.P, Mikol, V. | 登録日 | 2000-05-17 | 公開日 | 2000-09-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structures of human factor Xa complexed with potent inhibitors. J.Med.Chem., 43, 2000
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1F0S
| Crystal Structure of Human Coagulation Factor XA Complexed with RPR208707 | 分子名称: | CALCIUM ION, COAGULATION FACTOR XA, THIENO[3,2-B]PYRIDINE-2-SULFONIC ACID [2-OXO-1-(1H-PYRROLO[2,3-C]PYRIDIN-2-YLMETHYL)-PYRROLIDIN-3-YL]-AMIDE | 著者 | Maignan, S, Guilloteau, J.P, Pouzieux, S, Choi-Sledeski, Y.M, Becker, M.R, Klein, S.I, Ewing, W.R, Pauls, H.W, Spada, A.P, Mikol, V. | 登録日 | 2000-05-17 | 公開日 | 2000-09-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structures of human factor Xa complexed with potent inhibitors. J.Med.Chem., 43, 2000
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1F0T
| BOVINE TRYPSIN COMPLEXED WITH RPR131247 | 分子名称: | 4-HYDROXY-3-[2-OXO-3-(THIENO[3,2-B]PYRIDINE-2-SULFONYLAMINO)-PYRROLIDIN-1-YLMETHYL]-BENZAMIDINE, CALCIUM ION, SULFATE ION, ... | 著者 | Maignan, S, Guilloteau, J.P, Pouzieux, S, Choi-Sledeski, Y.M, Becker, M.R, Klein, S.I, Ewing, W.R, Pauls, H.W, Spada, A.P, Mikol, V. | 登録日 | 2000-05-17 | 公開日 | 2000-09-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structures of human factor Xa complexed with potent inhibitors. J.Med.Chem., 43, 2000
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1F0U
| BOVINE TRYPSIN COMPLEXED WITH RPR128515 | 分子名称: | 3-[(3'-AMINOMETHYL-BIPHENYL-4-CARBONYL)-AMINO]-2-(3-CARBAMIMIDOYL-BENZYL)-BUTYRIC ACID METHYL ESTER, CALCIUM ION, SULFATE ION, ... | 著者 | Maignan, S, Guilloteau, J.P, Pouzieux, S, Choi-Sledeski, Y.M, Becker, M.R, Klein, S.I, Ewing, W.R, Pauls, H.W, Spada, A.P, Mikol, V. | 登録日 | 2000-05-17 | 公開日 | 2000-09-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of human factor Xa complexed with potent inhibitors. J.Med.Chem., 43, 2000
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1F0V
| Crystal structure of an Rnase A dimer displaying a new type of 3D domain swapping | 分子名称: | 5'-D(*CP*G)-3', GLYCEROL, PHOSPHATE ION, ... | 著者 | Liu, Y.S, Gotte, G, Libonati, M, Eisenberg, D.S. | 登録日 | 2000-05-17 | 公開日 | 2001-02-21 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A domain-swapped RNase A dimer with implications for amyloid formation Nat.Struct.Biol., 8, 2001
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1F0W
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1F0X
| CRYSTAL STRUCTURE OF D-LACTATE DEHYDROGENASE, A PERIPHERAL MEMBRANE RESPIRATORY ENZYME. | 分子名称: | D-LACTATE DEHYDROGENASE, FLAVIN-ADENINE DINUCLEOTIDE | 著者 | Dym, O, Pratt, E.A, Ho, C, Eisenberg, D. | 登録日 | 2000-05-17 | 公開日 | 2000-08-23 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The crystal structure of D-lactate dehydrogenase, a peripheral membrane respiratory enzyme. Proc.Natl.Acad.Sci.USA, 97, 2000
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1F0Y
| L-3-HYDROXYACYL-COA DEHYDROGENASE COMPLEXED WITH ACETOACETYL-COA AND NAD+ | 分子名称: | ACETOACETYL-COENZYME A, L-3-HYDROXYACYL-COA DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Barycki, J.J, O'Brien, L.K, Strauss, A.W, Banaszak, L.J. | 登録日 | 2000-05-17 | 公開日 | 2000-09-01 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Sequestration of the active site by interdomain shifting. Crystallographic and spectroscopic evidence for distinct conformations of L-3-hydroxyacyl-CoA dehydrogenase. J.Biol.Chem., 275, 2000
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1F0Z
| SOLUTION STRUCTURE OF THIS, THE SULFUR CARRIER PROTEIN IN E.COLI THIAMIN BIOSYNTHESIS | 分子名称: | THIS PROTEIN | 著者 | Wang, C, Xi, J, Begley, T.P, Nicholson, L.K. | 登録日 | 2000-05-17 | 公開日 | 2001-01-10 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of ThiS and implications for the evolutionary roots of ubiquitin. Nat.Struct.Biol., 8, 2001
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1F10
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1F11
| F124 FAB FRAGMENT FROM A MONOCLONAL ANTI-PRES2 ANTIBODY | 分子名称: | F124 IMMUNOGLOBULIN (IGG1 HEAVY CHAIN), F124 IMMUNOGLOBULIN (KAPPA LIGHT CHAIN) | 著者 | Saul, F.A, Vulliez-Le Normand, B, Passafiume, M, Riottot, M.M, Bentley, G.A. | 登録日 | 2000-05-18 | 公開日 | 2000-08-30 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structure of the Fab fragment from F124, a monoclonal antibody specific for hepatitis B surface antigen. Acta Crystallogr.,Sect.D, 56, 2000
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1F12
| L-3-HYDROXYACYL-COA DEHYDROGENASE COMPLEXED WITH 3-HYDROXYBUTYRYL-COA | 分子名称: | 3-HYDROXYBUTANOYL-COENZYME A, L-3-HYDROXYACYL-COA DEHYDROGENASE | 著者 | Barycki, J.J, O'Brien, L.K, Strauss, A.W, Banaszak, L.J. | 登録日 | 2000-05-18 | 公開日 | 2000-09-27 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Sequestration of the active site by interdomain shifting. Crystallographic and spectroscopic evidence for distinct conformations of L-3-hydroxyacyl-CoA dehydrogenase. J.Biol.Chem., 275, 2000
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1F13
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1F14
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1F15
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1F16
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1F17
| L-3-HYDROXYACYL-COA DEHYDROGENASE COMPLEXED WITH NADH | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, L-3-HYDROXYACYL-COA DEHYDROGENASE | 著者 | Barycki, J.J, O'Brien, L.K, Strauss, A.W, Banaszak, L.J. | 登録日 | 2000-05-18 | 公開日 | 2000-09-27 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Sequestration of the active site by interdomain shifting. Crystallographic and spectroscopic evidence for distinct conformations of L-3-hydroxyacyl-CoA dehydrogenase. J.Biol.Chem., 275, 2000
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1F18
| Crystal structure of yeast copper-zinc superoxide dismutase mutant GLY85ARG | 分子名称: | COPPER (II) ION, COPPER-ZINC SUPEROXIDE DISMUTASE, ZINC ION | 著者 | Hart, P.J, Ogihara, N.L, Liu, H, Nersissian, A.M, Valentine, J.S, Eisenberg, D. | 登録日 | 2000-05-18 | 公開日 | 2002-12-18 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A structure-based mechanism for copper-zinc superoxide dismutase. Biochemistry, 38, 1999
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1F1A
| Crystal structure of yeast H48Q cuznsod fals mutant analog | 分子名称: | COPPER (II) ION, COPPER-ZINC SUPEROXIDE DISMUTASE, ZINC ION | 著者 | Hart, P.J, Ogihara, N.L, Liu, H, Nersissian, A.M, Valentine, J.S, Eisenberg, D. | 登録日 | 2000-05-18 | 公開日 | 2002-12-18 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | A structure-based mechanism for copper-zinc superoxide dismutase. Biochemistry, 38, 1999
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1F1B
| CRYSTAL STRUCTURE OF E. COLI ASPARTATE TRANSCARBAMOYLASE P268A MUTANT IN THE R-STATE IN THE PRESENCE OF N-PHOSPHONACETYL-L-ASPARTATE | 分子名称: | ASPARTATE CARBAMOYLTRANSFERASE CATALYTIC CHAIN, ASPARTATE CARBAMOYLTRANSFERASE REGULATORY CHAIN, N-(PHOSPHONACETYL)-L-ASPARTIC ACID, ... | 著者 | Jin, L, Stec, B, Kantrowitz, E.R. | 登録日 | 2000-05-18 | 公開日 | 2000-11-22 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | A cis-proline to alanine mutant of E. coli aspartate transcarbamoylase: kinetic studies and three-dimensional crystal structures. Biochemistry, 39, 2000
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1F1C
| CRYSTAL STRUCTURE OF CYTOCHROME C549 | 分子名称: | CYTOCHROME C549, HEME C | 著者 | Kerfeld, C.A, Sawaya, M.R, Yeates, T.O, Krogmann, D.W. | 登録日 | 2000-05-18 | 公開日 | 2001-08-08 | 最終更新日 | 2021-03-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structures of cytochrome c-549 and cytochrome c6 from the cyanobacterium Arthrospira maxima. Biochemistry, 40, 2001
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