6ZJ0
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![BU of 6zj0 by Molmil](/molmil-images/mine/6zj0) | CRYSTAL STRUCTURE OF HRAS-G12D IN COMPLEX WITH GCP AND COMPOUND 18 | 分子名称: | (3~{S})-3-[2-[(dimethylamino)methyl]-1~{H}-indol-3-yl]-5-oxidanyl-2,3-dihydroisoindol-1-one, GTPase HRas, MAGNESIUM ION, ... | 著者 | Kessler, D, Fischer, G, Boettcher, J. | 登録日 | 2020-06-26 | 公開日 | 2020-08-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.763 Å) | 主引用文献 | Drugging all RAS isoforms with one pocket. Future Med Chem, 12, 2020
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6ZJ7
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![BU of 6zj7 by Molmil](/molmil-images/mine/6zj7) | Trehalose transferase (TreT) from Thermoproteus uzoniensis soaked with Mg | 分子名称: | GLYCEROL, TETRAETHYLENE GLYCOL, THIOCYANATE ION, ... | 著者 | Bento, I, Mestrom, L, Marsden, S.R, van der Eijk, H, Laustsen, J.U, Jeffries, C.M, Svergun, D.I, Hagedoorn, P.-H, Hanefeld, U. | 登録日 | 2020-06-28 | 公開日 | 2020-09-30 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Anomeric Selectivity of Trehalose Transferase with Rare l-Sugars. Acs Catalysis, 10, 2020
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6ZJJ
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6ZJY
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![BU of 6zjy by Molmil](/molmil-images/mine/6zjy) | Respiratory complex I from Thermus thermophilus, NAD+ dataset, minor state | 分子名称: | FE2/S2 (INORGANIC) CLUSTER, IRON/SULFUR CLUSTER, NADH-quinone oxidoreductase subunit 1, ... | 著者 | Kaszuba, K, Tambalo, M, Gallagher, G.T, Sazanov, L.A. | 登録日 | 2020-06-29 | 公開日 | 2020-09-02 | 最終更新日 | 2024-05-01 | 実験手法 | ELECTRON MICROSCOPY (5.5 Å) | 主引用文献 | Key role of quinone in the mechanism of respiratory complex I. Nat Commun, 11, 2020
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6ZIA
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![BU of 6zia by Molmil](/molmil-images/mine/6zia) | Ultrafast Structural Response to Charge Redistribution Within a Photosynthetic Reaction Centre - 8 us structure | 分子名称: | 15-cis-1,2-dihydroneurosporene, BACTERIOCHLOROPHYLL B, BACTERIOPHEOPHYTIN B, ... | 著者 | Baath, P, Dods, R, Braenden, G, Neutze, R. | 登録日 | 2020-06-25 | 公開日 | 2020-12-09 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Ultrafast structural changes within a photosynthetic reaction centre. Nature, 589, 2021
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6D78
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![BU of 6d78 by Molmil](/molmil-images/mine/6d78) | The complex between high-affinity TCR DMF5(alpha-D26Y,beta-L98W) and human Class I MHC HLA-A2 with the bound MART-1(27-35)peptide | 分子名称: | Beta-2-microglobulin, DMF5 alpha chain,DMF5 alpha chain, DMF5 beta chain,DMF5 beta chain, ... | 著者 | Hellman, L.M, Singh, N.K. | 登録日 | 2018-04-24 | 公開日 | 2019-04-03 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.347 Å) | 主引用文献 | Improving T Cell Receptor On-Target Specificity via Structure-Guided Design. Mol. Ther., 27, 2019
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6ZK6
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![BU of 6zk6 by Molmil](/molmil-images/mine/6zk6) | Protein Phosphatase 1 (PP1) T320E mutant | 分子名称: | FE (III) ION, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Salvi, F, Barabas, O, Koehn, M. | 登録日 | 2020-06-29 | 公開日 | 2020-11-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Towards Dissecting the Mechanism of Protein Phosphatase-1 Inhibition by Its C-Terminal Phosphorylation. Chembiochem, 22, 2021
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6DA3
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![BU of 6da3 by Molmil](/molmil-images/mine/6da3) | Human CYP3A4 bound to an inhibitor | 分子名称: | Cytochrome P450 3A4, PROTOPORPHYRIN IX CONTAINING FE, tert-butyl [(2R)-1-{[(2R)-1-oxo-3-phenyl-1-{[(pyridin-3-yl)methyl]amino}propan-2-yl]sulfanyl}-3-phenylpropan-2-yl]carbamate | 著者 | Sevrioukova, I.F. | 登録日 | 2018-05-01 | 公開日 | 2019-04-03 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structure-Activity Relationships of Rationally Designed Ritonavir Analogues: Impact of Side-Group Stereochemistry, Headgroup Spacing, and Backbone Composition on the Interaction with CYP3A4. Biochemistry, 58, 2019
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5DF6
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![BU of 5df6 by Molmil](/molmil-images/mine/5df6) | Crystal structure of PTPN11 tandem SH2 domains in complex with a TXNIP peptide | 分子名称: | Tyrosine-protein phosphatase non-receptor type 11, UNKNOWN ATOM OR ION, txnip | 著者 | Dong, A, Li, W, Tempel, W, Liu, Y, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2015-08-26 | 公開日 | 2015-09-23 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Structural basis for the regulatory role of the PPxY motifs in the thioredoxin-interacting protein TXNIP. Biochem.J., 473, 2016
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6ZFD
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![BU of 6zfd by Molmil](/molmil-images/mine/6zfd) | 14-3-3 zeta bound to the phosphorylated 18E6 C-terminus | 分子名称: | 14-3-3 protein zeta/delta,Protein E6, GLYCEROL | 著者 | Gogl, G, Tugaeva, K.V, Sluchanko, N.N, Trave, G. | 登録日 | 2020-06-17 | 公開日 | 2021-02-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Hierarchized phosphotarget binding by the seven human 14-3-3 isoforms. Nat Commun, 12, 2021
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6ZCF
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6ZG6
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![BU of 6zg6 by Molmil](/molmil-images/mine/6zg6) | COPII on membranes, outer coat vertex | 分子名称: | Protein transport protein SEC13, Protein transport protein SEC31 | 著者 | Zanetti, G, Hutchings, J. | 登録日 | 2020-06-18 | 公開日 | 2021-02-17 | 最終更新日 | 2024-05-01 | 実験手法 | ELECTRON MICROSCOPY (12 Å) | 主引用文献 | Structure of the complete, membrane-assembled COPII coat reveals a complex interaction network. Nat Commun, 12, 2021
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8R9A
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![BU of 8r9a by Molmil](/molmil-images/mine/8r9a) | A soakable crystal form of human CDK7 in complex with AMP-PNP | 分子名称: | (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol, Cyclin-dependent kinase 7, DI(HYDROXYETHYL)ETHER | 著者 | Mukherjee, M, Cleasby, A. | 登録日 | 2023-11-30 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 2024
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6ZL0
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6ZG5
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6ZFG
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![BU of 6zfg by Molmil](/molmil-images/mine/6zfg) | 14-3-3 zeta chimera with 18E6 and fusicoccin | 分子名称: | 14-3-3 protein zeta/delta,Protein E6, FUSICOCCIN, GLYCEROL | 著者 | Gogl, G, Tugaeva, K, Sluchanko, N.N, Trave, G. | 登録日 | 2020-06-17 | 公開日 | 2021-02-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Hierarchized phosphotarget binding by the seven human 14-3-3 isoforms. Nat Commun, 12, 2021
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8R9B
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6ZCG
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6ZCH
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8SFG
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![BU of 8sfg by Molmil](/molmil-images/mine/8sfg) | Crystal Structure of the Open Unbound Catalytically Inactive Makes Caterpillars Floppy-like (MCF) Effector from Vibrio vulnificus CMCP6 | 分子名称: | Autotransporter adhesin, CHLORIDE ION, SULFATE ION | 著者 | Minasov, G, Shuvalova, L, Rosas-Lemus, M, Herrera, A, Satchell, K.J.F, Center for Structural Biology of Infectious Diseases (CSBID) | 登録日 | 2023-04-11 | 公開日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal Structure of the Open Unbound Catalytically Inactive Makes Caterpillars Floppy-like (MCF) Effector from Vibrio vulnificus CMCP6. To Be Published
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6D4L
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6YSP
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![BU of 6ysp by Molmil](/molmil-images/mine/6ysp) | Arabidopsis aspartate transcarbamoylase complex with PALA and carbamoyl phosphate | 分子名称: | GLYCEROL, N-(PHOSPHONACETYL)-L-ASPARTIC ACID, PHOSPHORIC ACID MONO(FORMAMIDE)ESTER, ... | 著者 | Ramon Maiques, S, Del Cano Ochoa, F, Bellin, L, Mohlmann, T. | 登録日 | 2020-04-23 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.38 Å) | 主引用文献 | Mechanisms of feedback inhibition and sequential firing of active sites in plant aspartate transcarbamoylase. Nat Commun, 12, 2021
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6YW9
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![BU of 6yw9 by Molmil](/molmil-images/mine/6yw9) | Arabidopsis aspartate transcarbamoylase mutant F161A complex with PALA | 分子名称: | GLYCEROL, N-(PHOSPHONACETYL)-L-ASPARTIC ACID, PYRB | 著者 | Ramon Maiques, S, Del Cano Ochoa, F, Bellin, L, Mohlmann, T. | 登録日 | 2020-04-29 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Mechanisms of feedback inhibition and sequential firing of active sites in plant aspartate transcarbamoylase. Nat Commun, 12, 2021
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4FHV
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6YVB
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![BU of 6yvb by Molmil](/molmil-images/mine/6yvb) | Arabidopsis aspartate transcarbamoylase complex with carbamoyl phosphate | 分子名称: | ACETATE ION, GLYCEROL, PHOSPHORIC ACID MONO(FORMAMIDE)ESTER, ... | 著者 | Ramon Maiques, S, Del Cano Ochoa, F, Bellin, L, Mohlmann, T. | 登録日 | 2020-04-28 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.826 Å) | 主引用文献 | Mechanisms of feedback inhibition and sequential firing of active sites in plant aspartate transcarbamoylase. Nat Commun, 12, 2021
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