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1ANN
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ANNEXIN IV
分子名称: ANNEXIN IV, CALCIUM ION
著者Sutton, R.B, Sprang, S.R.
登録日1995-09-21
公開日1996-01-29
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Three Dimensional Structure of Annexin IV
Annexins: Molecular Structure to Cellular Function, 1996
1A5I
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CATALYTIC DOMAIN OF VAMPIRE BAT (DESMODUS ROTUNDUS) SALIVA PLASMINOGEN ACTIVATOR IN COMPLEX WITH EGR-CMK (GLU-GLY-ARG CHLOROMETHYL KETONE)
分子名称: L-alpha-glutamyl-N-{(1S)-4-{[amino(iminio)methyl]amino}-1-[(1S)-2-chloro-1-hydroxyethyl]butyl}glycinamide, PLASMINOGEN ACTIVATOR
著者Renatus, M, Stubbs, M.T, Bode, W.
登録日1998-02-17
公開日1999-03-23
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Catalytic domain structure of vampire bat plasminogen activator: a molecular paradigm for proteolysis without activation cleavage.
Biochemistry, 36, 1997
1BP1
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CRYSTAL STRUCTURE OF BPI, THE HUMAN BACTERICIDAL PERMEABILITY-INCREASING PROTEIN
分子名称: 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, BACTERICIDAL/PERMEABILITY-INCREASING PROTEIN
著者Beamer, L.J, Carroll, S.F, Eisenberg, D.
登録日1997-04-08
公開日1997-09-04
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of human BPI and two bound phospholipids at 2.4 angstrom resolution.
Science, 276, 1997
1BNB
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SOLUTION STRUCTURE OF BOVINE NEUTROPHIL BETA-DEFENSIN 12: THE PEPTIDE FOLD OF THE BETA-DEFENSINS IS IDENTICAL TO THAT OF THE CLASSICAL DEFENSINS
分子名称: BOVINE NEUTROPHIL BETA-DEFENSIN 12
著者Zimmermann, G.R, Legault, P, Selsted, M.E, Pardi, A.
登録日1995-03-08
公開日1995-10-15
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献Solution structure of bovine neutrophil beta-defensin-12: the peptide fold of the beta-defensins is identical to that of the classical defensins.
Biochemistry, 34, 1995
1C2O
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ELECTROPHORUS ELECTRICUS ACETYLCHOLINESTERASE
分子名称: ACETYLCHOLINESTERASE
著者Bourne, Y, Marchot, P.
登録日1999-07-26
公開日2000-01-19
最終更新日2021-06-02
実験手法X-RAY DIFFRACTION (4.2 Å)
主引用文献Conformational flexibility of the acetylcholinesterase tetramer suggested by x-ray crystallography.
J.Biol.Chem., 274, 1999
1BX2
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CRYSTAL STRUCTURE OF HLA-DR2 (DRA*0101,DRB1*1501) COMPLEXED WITH A PEPTIDE FROM HUMAN MYELIN BASIC PROTEIN
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, PROTEIN (HLA-DR2)
著者Smith, K.J, Pyrdol, J, Gauthier, L, Wiley, D.C, Wucherpfennig, K.
登録日1998-10-12
公開日1998-10-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structure of HLA-DR2 (DRA*0101, DRB1*1501) complexed with a peptide from human myelin basic protein.
J.Exp.Med., 188, 1998
1A60
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NMR STRUCTURE OF A CLASSICAL PSEUDOKNOT: INTERPLAY OF SINGLE-AND DOUBLE-STRANDED RNA, 24 STRUCTURES
分子名称: TYMV PSEUDOKNOT
著者Kolk, M.H, Van Der Graaf, M, Wijmenga, S.S, Pleij, C.W.A, Heus, H.A, Hilbers, C.W.
登録日1998-03-04
公開日1998-05-27
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR structure of a classical pseudoknot: interplay of single- and double-stranded RNA.
Science, 280, 1998
1DGN
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SOLUTION STRUCTURE OF ICEBERG, AN INHIBITOR OF INTERLEUKIN-1BETA GENERATION
分子名称: ICEBERG (PROTEASE INHIBITOR)
著者Humke, E.W, Shriver, S.K, Starovasnik, M.A, Fairbrother, W.J, Dixit, V.M.
登録日1999-11-24
公開日2000-10-09
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献ICEBERG: a novel inhibitor of interleukin-1beta generation.
Cell(Cambridge,Mass.), 103, 2000
1DQZ
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CRYSTAL STRUCTURE OF ANTIGEN 85C FROM MYCOBACTERIUM TUBERCULOSIS
分子名称: PROTEIN (ANTIGEN 85-C)
著者Ronning, D.R, Klabunde, T, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2000-01-05
公開日2000-07-12
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structure of the secreted form of antigen 85C reveals potential targets for mycobacterial drugs and vaccines.
Nat.Struct.Biol., 7, 2000
1ATN
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Atomic structure of the actin:DNASE I complex
分子名称: ACTIN, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ...
著者Kabsch, W, Mannherz, H.G, Suck, D, Pai, E, Holmes, K.C.
登録日1991-03-08
公開日1992-07-15
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Atomic structure of the actin:DNase I complex.
Nature, 347, 1990
1BIM
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CRYSTALLOGRAPHIC STUDIES ON THE BINDING MODES OF P2-P3 BUTANEDIAMIDE RENIN INHIBITORS
分子名称: (2S)-2-[(2-amino-1,3-thiazol-4-yl)methyl]-N~1~-{(1S,2S)-1-(cyclohexylmethyl)-2-hydroxy-2-[(3R)-1,5,5-trimethyl-2-oxopyrrolidin-3-yl]ethyl}-N~4~-[2-(dimethylamino)-2-oxoethyl]-N~4~-[(1S)-1-phenylethyl]butanediamide, Renin
著者Tong, L.
登録日1995-09-27
公開日1996-01-29
最終更新日2022-03-09
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystallographic studies on the binding modes of P2-P3 butanediamide renin inhibitors.
J.Biol.Chem., 270, 1995
1CUA
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CUTINASE, N172K MUTANT
分子名称: CUTINASE
著者Longhi, S, Cambillau, C.
登録日1995-11-16
公開日1996-07-11
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Dynamics of Fusarium solani cutinase investigated through structural comparison among different crystal forms of its variants.
Proteins, 26, 1996
1CP7
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AMINOPEPTIDASE FROM STREPTOMYCES GRISEUS
分子名称: AMINOPEPTIDASE, CALCIUM ION, ZINC ION
著者Gilboa, R, Greenblatt, H.M, Perach, M, Spungin-Bialik, A, Lessel, U, Schomburg, D, Blumberg, S, Shoham, G.
登録日1999-06-10
公開日2000-05-03
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Interactions of Streptomyces griseus aminopeptidase with a methionine product analogue: a structural study at 1.53 A resolution.
Acta Crystallogr.,Sect.D, 56, 2000
1D3Q
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CRYSTAL STRUCTURE OF HUMAN ALPHA THROMBIN IN COMPLEX WITH BENZO[B]THIOPHENE INHIBITOR 2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[4-(2-PYRROLIDIN-1-YL-ETHOXY)-BENZYL]-2-4-(2-PYRROLIDIN-1-YL-ETHOXY)-PHENYL] -BENZO[B]THIOPHENE, ALPHA-THROMBIN, ...
著者Chirgadze, N.Y.
登録日1999-09-30
公開日2000-10-04
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献The crystal structures of human alpha-thrombin complexed with active site-directed diamino benzo[b]thiophene derivatives: a binding mode for a structurally novel class of inhibitors.
Protein Sci., 9, 2000
1CUI
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CUTINASE, S120A MUTANT
分子名称: CUTINASE
著者Martinez, C, Cambillau, C.
登録日1995-11-16
公開日1996-07-11
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Dynamics of Fusarium solani cutinase investigated through structural comparison among different crystal forms of its variants.
Proteins, 26, 1996
1CJ1
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GROWTH FACTOR RECEPTOR BINDING PROTEIN SH2 DOMAIN (HUMAN) COMPLEXED WITH A PHOSPHOTYROSYL DERIVATIVE
分子名称: PROTEIN (GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2), [1-[1-(6-CARBAMOYL-CYCLOHEX-2-ENYLCARBAMOYL)-CYCLOHEXYLCARBAMOYL]-2-(4-PHOSPHONOOXY-PHENYL)- ETHYL]-CARBAMIC ACID 3-AMINOBENZYLESTER
著者Rahuel, J.
登録日1999-04-21
公開日1999-12-22
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure-based design, synthesis, and X-ray crystallography of a high-affinity antagonist of the Grb2-SH2 domain containing an asparagine mimetic.
J.Med.Chem., 42, 1999
1DNK
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THE X-RAY STRUCTURE OF THE DNASE I-D(GGTATACC)2 COMPLEX AT 2.3 ANGSTROMS RESOLUTION
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DNA (5'-D(*GP*GP*TP*AP*TP*AP*C)-3'), DNA (5'-D(*GP*GP*TP*AP*TP*AP*CP*C)-3'), ...
著者Weston, S.A, Lahm, A, Suck, D.
登録日1992-08-10
公開日1994-01-31
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献X-ray structure of the DNase I-d(GGTATACC)2 complex at 2.3 A resolution.
J.Mol.Biol., 226, 1992
1DQY
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CRYSTAL STRUCTURE OF ANTIGEN 85C FROM MYCOBACTERIUM TUBERCULOSIS WITH DIETHYL PHOSPHATE INHIBITOR
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, DIETHYL PHOSPHONATE, PROTEIN (ANTIGEN 85-C)
著者Ronning, D.R, Klabunde, T, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2000-01-05
公開日2000-07-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献Crystal structure of the secreted form of antigen 85C reveals potential targets for mycobacterial drugs and vaccines.
Nat.Struct.Biol., 7, 2000
1DTG
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HUMAN TRANSFERRIN N-LOBE MUTANT H249E
分子名称: CARBONATE ION, FE (III) ION, TRANSFERRIN
著者MacGillivray, R.T, Bewley, M.C, Smith, C.A, He, Q.Y, Mason, A.B.
登録日2000-01-12
公開日2000-01-21
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Mutation of the iron ligand His 249 to Glu in the N-lobe of human transferrin abolishes the dilysine "trigger" but does not significantly affect iron release.
Biochemistry, 39, 2000
1DEU
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CRYSTAL STRUCTURE OF HUMAN PROCATHEPSIN X: A CYSTEINE PROTEASE WITH THE PROREGION COVALENTLY LINKED TO THE ACTIVE SITE CYSTEINE
分子名称: PROCATHEPSIN X
著者Sivaraman, J, Nagler, D.K, Zhang, R, Menard, R, Cygler, M.
登録日1999-11-15
公開日2000-02-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of human procathepsin X: a cysteine protease with the proregion covalently linked to the active site cysteine.
J.Mol.Biol., 295, 2000
1DPO
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STRUCTURE OF RAT TRYPSIN
分子名称: BENZAMIDINE, CALCIUM ION, SULFATE ION, ...
著者Stroud, R.M.
登録日1997-03-31
公開日1997-07-07
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献1.59 A structure of trypsin at 120 K: comparison of low temperature and room temperature structures.
Proteins, 10, 1991
1D48
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STRUCTURE OF THE PURE-SPERMINE FORM OF Z-DNA (MAGNESIUM FREE) AT 1 ANGSTROM RESOLUTION
分子名称: DNA (5'-D(*CP*GP*CP*GP*CP*G)-3'), SPERMINE
著者Egli, M, Williams, L.D, Gao, Q, Rich, A.
登録日1991-09-11
公開日1992-04-15
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献Structure of the pure-spermine form of Z-DNA (magnesium free) at 1-A resolution.
Biochemistry, 30, 1991
1ESB
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DIRECT STRUCTURE OBSERVATION OF AN ACYL-ENZYME INTERMEDIATE IN THE HYDROLYSIS OF AN ESTER SUBSTRATE BY ELASTASE
分子名称: CALCIUM ION, N-[(BENZYLOXY)CARBONYL]-L-ALANINE, PORCINE PANCREATIC ELASTASE, ...
著者Ding, X, Rasmussen, B, Petsko, G.A, Ringe, D.
登録日1994-02-04
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Direct structural observation of an acyl-enzyme intermediate in the hydrolysis of an ester substrate by elastase.
Biochemistry, 33, 1994
1EJN
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UROKINASE PLASMINOGEN ACTIVATOR B-CHAIN INHIBITOR COMPLEX
分子名称: N-(1-ADAMANTYL)-N'-(4-GUANIDINOBENZYL)UREA, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
著者Sperl, S, Jacob, U, Arroyo de Prada, N, Stuerzebecher, J, Wilhelm, O.G, Bode, W, Magdolen, V, Huber, R, Moroder, L.
登録日2000-04-22
公開日2000-05-17
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献(4-aminomethyl)phenylguanidine derivatives as nonpeptidic highly selective inhibitors of human urokinase.
Proc.Natl.Acad.Sci.USA, 97, 2000
1EOV
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FREE ASPARTYL-TRNA SYNTHETASE (ASPRS) (E.C. 6.1.1.12) FROM YEAST
分子名称: ASPARTYL-TRNA SYNTHETASE
著者Sauter, C, Lorber, B, Cavarelli, J, Moras, D, Giege, R.
登録日2000-03-24
公開日2000-09-24
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The free yeast aspartyl-tRNA synthetase differs from the tRNA(Asp)-complexed enzyme by structural changes in the catalytic site, hinge region, and anticodon-binding domain.
J.Mol.Biol., 299, 2000

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