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6FH6
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Crystal Structure of BAZ2B bromodomain in complex with 1-methylpyridinone compound 1
分子名称: Bromodomain adjacent to zinc finger domain protein 2B, ~{N}-(2-azanylethyl)-1-methyl-6-oxidanylidene-pyridine-3-carboxamide
著者Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A.
登録日2018-01-12
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.082 Å)
主引用文献Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains.
ChemMedChem, 13, 2018
6FGU
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Crystal Structure of BAZ2B bromodomain in complex with 1-methylpyridinone compound 4
分子名称: 1-methyl-6-oxidanylidene-~{N}-(2-pyrrolidin-1-ylethyl)pyridine-3-carboxamide, Bromodomain adjacent to zinc finger domain protein 2B
著者Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A.
登録日2018-01-11
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains.
ChemMedChem, 13, 2018
6FG6
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Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridinone compound 1
分子名称: Bromodomain adjacent to zinc finger domain protein 2A, ~{N}-(2-azanylethyl)-1-methyl-6-oxidanylidene-pyridine-3-carboxamide
著者Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A.
登録日2018-01-10
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains.
ChemMedChem, 13, 2018
6FGW
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BU of 6fgw by Molmil
Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridinone compound 4
分子名称: 1-methyl-6-oxidanylidene-~{N}-(2-pyrrolidin-1-ylethyl)pyridine-3-carboxamide, Bromodomain adjacent to zinc finger domain protein 2A
著者Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A.
登録日2018-01-11
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.725 Å)
主引用文献Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains.
ChemMedChem, 13, 2018
6FGG
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Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridinone compound 5
分子名称: Bromodomain adjacent to zinc finger domain protein 2A, ~{N}-[3-[2-(dimethylamino)ethyl]-2-oxidanylidene-1,3-benzoxazol-5-yl]-1-methyl-6-oxidanylidene-pyridine-3-carboxamide
著者Dalle Vedove, A, Spiliotopoulos, D, Lolli, G, Caflisch, A.
登録日2018-01-10
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains.
ChemMedChem, 13, 2018
7TGG
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BU of 7tgg by Molmil
Cryo-EM structure of PilA-N and PilA-C from Geobacter sulfurreducens
分子名称: Geopilin domain 1 protein, Geopilin domain 2 protein
著者Wang, F, Mustafa, K, Chan, C.H, Joshi, K, Bond, D.R, Hochbaum, A.I, Egelman, E.H.
登録日2022-01-07
公開日2022-02-23
最終更新日2024-06-05
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Cryo-EM structure of an extracellular Geobacter OmcE cytochrome filament reveals tetrahaem packing.
Nat Microbiol, 7, 2022
6TDB
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BU of 6tdb by Molmil
Neuropilin2-b1 domain in a complex with the C-terminal VEGFB167 peptide
分子名称: 1,2-ETHANEDIOL, ACETYL GROUP, C-terminal VEGFB167 peptide, ...
著者Eldrid, C, Yu, L, Yelland, T, Fotinou, C, Djordjevic, S.
登録日2019-11-08
公開日2020-11-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献NRP2-b1 domain in a complex with the C-terminal VEGFB167 peptide
To Be Published
6TJT
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Neuropilin2-b1 domain in a complex with the C-terminal VEGFC peptide
分子名称: 1,2-ETHANEDIOL, Neuropilin-2, SULFATE ION, ...
著者Eldrid, C, Yu, L, Yelland, T, Fotinou, C, Djordjevic, S.
登録日2019-11-26
公開日2020-12-16
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.31 Å)
主引用文献NRP2-b1 domain in a complex with the C-terminal VEGFC peptide
To Be Published
8HWJ
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BU of 8hwj by Molmil
Bacterial STING from Epilithonimonas lactis in complex with 3'3'-c-di-AMP
分子名称: (2R,3R,3aS,5R,7aR,9R,10R,10aS,12R,14aR)-2,9-bis(6-amino-9H-purin-9-yl)octahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8 ]tetraoxadiphosphacyclododecine-3,5,10,12-tetrol 5,12-dioxide, CD-NTase-associated protein 12
著者Wang, Y.-C, Yang, C.-S, Hou, M.-H, Chen, Y.
登録日2022-12-30
公開日2024-01-03
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.553 Å)
主引用文献Structural insights into the regulation, ligand recognition, and oligomerization of bacterial STING.
Nat Commun, 14, 2023
8HY8
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BU of 8hy8 by Molmil
Bacterial STING from Epilithonimonas lactis
分子名称: CD-NTase-associated protein 12
著者Wang, Y.-C, Yang, C.-S, Hou, M.-H, Chen, Y.
登録日2023-01-06
公開日2024-01-10
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.568 Å)
主引用文献Structural insights into the regulation, ligand recognition, and oligomerization of bacterial STING.
Nat Commun, 14, 2023
4J3O
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BU of 4j3o by Molmil
Crystal structure of the FimD usher traversed by the pilus tip complex assembly composed of FimC:FimF:FimG:FimH
分子名称: Chaperone protein FimC, Outer membrane usher protein FimD, Protein FimF, ...
著者Geibel, S, Waksman, G.
登録日2013-02-06
公開日2013-04-10
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Structural and energetic basis of folded-protein transport by the FimD usher.
Nature, 496, 2013
2XTL
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BU of 2xtl by Molmil
Structure of the major pilus backbone protein from Streptococcus Agalactiae
分子名称: CELL WALL SURFACE ANCHOR FAMILY PROTEIN, POTASSIUM ION
著者Rinauda, D, Gourlay, L.J, Soriano, M, Grandi, G, Bolognesi, M.
登録日2010-10-11
公開日2011-07-06
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structure-Based Approach to Rationally Design a Chimeric Protein for an Effective Vaccine Against Group B Streptococcus Infections.
Proc.Natl.Acad.Sci.USA, 108, 2011
8EXH
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BU of 8exh by Molmil
Agrobacterium tumefaciens Tpilus
分子名称: (14S,17R)-20-amino-17-hydroxy-11,17-dioxo-12,16,18-trioxa-17lambda~5~-phosphaicosan-14-yl tetradecanoate, Protein virB2
著者Beltran, L.C, Egelman, E.H.
登録日2022-10-25
公開日2023-03-22
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Archaeal DNA-import apparatus is homologous to bacterial conjugation machinery
Nat Commun, 14, 2023
3F84
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BU of 3f84 by Molmil
Structure of fusion complex of major pilin CfaB and major pilin CfaB of CFA/I pilus from ETEC E. coli
分子名称: CFA/I fimbrial subunit B
著者Xia, D, Li, Y.F.
登録日2008-11-11
公開日2009-08-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structure of CFA/I fimbriae from enterotoxigenic Escherichia coli.
Proc.Natl.Acad.Sci.USA, 106, 2009
2VQI
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BU of 2vqi by Molmil
Structure of the P pilus usher (PapC) translocation pore
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, LAURYL DIMETHYLAMINE-N-OXIDE, OUTER MEMBRANE USHER PROTEIN PAPC
著者Remaut, H, Tang, C, Henderson, N.S, Pinkner, J.S, Wang, T, Hultgren, S.J, Thanassi, D.G, Li, H, Waksman, G.
登録日2008-03-16
公開日2008-05-27
最終更新日2019-01-16
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Fiber formation across the bacterial outer membrane by the chaperone/usher pathway.
Cell, 133, 2008
1P5V
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BU of 1p5v by Molmil
X-ray structure of the Caf1M:Caf1 chaperone:subunit preassembly complex
分子名称: Chaperone protein Caf1M, F1 capsule antigen
著者Zavialov, A.V, Berglund, J, Pudney, A.F, Fooks, L.J, Ibrahim, T.M, MacIntyre, S, Knight, S.D.
登録日2003-04-28
公開日2003-06-24
最終更新日2018-03-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure and Biogenesis of the Capsular F1 Antigen from Yersinia pestis. Preserved Folding Energy Drives Fiber Formation
Cell(Cambridge,Mass.), 113, 2003
1P5U
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BU of 1p5u by Molmil
X-ray structure of the ternary Caf1M:Caf1:Caf1 chaperone:subunit:subunit complex
分子名称: Chaperone protein Caf1M, F1 capsule antigen
著者Zavialov, A.V, Berglund, J, Pudney, A.F, Fooks, L.J, Ibrahim, T.M, MacIntyre, S, Knight, S.D.
登録日2003-04-28
公開日2003-06-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Structure and Biogenesis of the Capsular F1 Antigen from Yersinia pestis. Preserved Folding Energy Drives Fiber Formation
Cell(Cambridge,Mass.), 113, 2003
6AOX
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BU of 6aox by Molmil
F9 pilus adhesin FmlH lectin domain from E. coli UTI89 co-crystallized with TF antigen
分子名称: Fml fimbrial adhesin FmlD, beta-D-galactopyranose-(1-3)-2-acetamido-2-deoxy-alpha-D-galactopyranose
著者Kalas, V, Hultgren, S.J.
登録日2017-08-16
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure-based discovery of glycomimetic FmlH ligands as inhibitors of bacterial adhesion during urinary tract infection.
Proc.Natl.Acad.Sci.USA, 115, 2018
6ARN
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BU of 6arn by Molmil
F9 pilus adhesin FmlH lectin domain from E. coli UTI89 co-crystallized with o-methoxyphenyl beta-galactoside (OMPG)
分子名称: 2-methoxyphenyl beta-D-galactopyranoside, Putative Fml fimbrial adhesin FmlD, SULFATE ION
著者Kalas, V, Hultgren, S.J.
登録日2017-08-22
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Structure-based discovery of glycomimetic FmlH ligands as inhibitors of bacterial adhesion during urinary tract infection.
Proc.Natl.Acad.Sci.USA, 115, 2018
6AS8
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BU of 6as8 by Molmil
F9 pilus adhesin FmlH lectin domain from E. coli UTI89 co-crystallized with ortho-biphenyl-2'-carboxyl N-acetyl-beta-galactosaminoside
分子名称: Fml fimbrial adhesin FmlD, ortho-biphenyl-2'-carboxyl N-acetyl-beta-galactosaminoside
著者Kalas, V, Hultgren, S.J.
登録日2017-08-23
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.101 Å)
主引用文献Structure-based discovery of glycomimetic FmlH ligands as inhibitors of bacterial adhesion during urinary tract infection.
Proc.Natl.Acad.Sci.USA, 115, 2018
6AOY
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BU of 6aoy by Molmil
F9 pilus adhesin FmlH lectin domain from E. coli UTI89 co-crystallized with o-nitrophenyl beta-galactoside (ONPG)
分子名称: 2-nitrophenyl beta-D-galactopyranoside, Fml fimbrial adhesin FmlD, SULFATE ION
著者Kalas, V, Hultgren, S.J.
登録日2017-08-16
公開日2018-02-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based discovery of glycomimetic FmlH ligands as inhibitors of bacterial adhesion during urinary tract infection.
Proc.Natl.Acad.Sci.USA, 115, 2018
4Y2O
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BU of 4y2o by Molmil
Structure of CFA/I pili chaperone-major subunit complex (CfaA-CfaB)
分子名称: CFA/I fimbrial subunit B, CfA/I fimbrial subunit A (Colonization factor antigen subunit A putative chaperone), NICKEL (II) ION, ...
著者Bao, R, Xia, D.
登録日2015-02-10
公開日2016-08-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.419 Å)
主引用文献Off-pathway assembly of fimbria subunits is prevented by chaperone CfaA of CFA/I fimbriae from enterotoxigenic E. coli.
Mol. Microbiol., 102, 2016
4Y2N
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BU of 4y2n by Molmil
Structure of CFA/I pili major subunit CfaB trimer
分子名称: 1,2-ETHANEDIOL, CFA/I fimbrial subunit B, MAGNESIUM ION
著者Bao, R, Xia, D.
登録日2015-02-10
公開日2016-08-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Off-pathway assembly of fimbria subunits is prevented by chaperone CfaA of CFA/I fimbriae from enterotoxigenic E. coli.
Mol. Microbiol., 102, 2016
4Y2L
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Structure of CFA/I pili major subunit CfaB trimer
分子名称: CALCIUM ION, CFA/I fimbrial subunit B, ISOPROPYL ALCOHOL
著者Bao, R, Xia, D.
登録日2015-02-10
公開日2016-08-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.746 Å)
主引用文献Off-pathway assembly of fimbria subunits is prevented by chaperone CfaA of CFA/I fimbriae from enterotoxigenic E. coli.
Mol. Microbiol., 102, 2016
3GEW
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BU of 3gew by Molmil
FaeE-FaeG chaperone-major pilin complex of F4 ad fimbriae
分子名称: Chaperone protein faeE, GLYCEROL, K88 fimbrial protein AD, ...
著者Van Molle, I, Moonens, K, Garcia-Pino, A, Buts, L, Bouckaert, J, De Greve, H.
登録日2009-02-26
公開日2009-10-20
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and thermodynamic characterization of pre- and postpolymerization states in the F4 fimbrial subunit FaeG
J.Mol.Biol., 394, 2009

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件を2024-09-18に公開中

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