1BFI
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![BU of 1bfi by Molmil](/molmil-images/mine/1bfi) | SOLUTION STRUCTURE OF THE C-TERMINAL SH2 DOMAIN OF THE P85ALPHA REGULATORY SUBUNIT OF PHOSPHOINOSITIDE 3-KINASE, NMR, 30 STRUCTURES | 分子名称: | P85 ALPHA | 著者 | Siegal, G, Davis, B, Kristensen, S.M, Sankar, A, Linacre, J, Stein, R.C, Panayotou, G, Waterfield, M.D, Driscoll, P.C. | 登録日 | 1997-11-18 | 公開日 | 1998-02-25 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the C-terminal SH2 domain of the p85 alpha regulatory subunit of phosphoinositide 3-kinase. J.Mol.Biol., 276, 1998
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4XSX
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4XKA
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4XCZ
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![BU of 4xcz by Molmil](/molmil-images/mine/4xcz) | X-ray structure of the N-formyltransferase QdtF from Providencia alcalifaciens in complex with TDP-Qui3n and N5-THF | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, N-{[4-({[(6R)-2-amino-5-formyl-4-oxo-1,4,5,6,7,8-hexahydropteridin-6-yl]methyl}amino)phenyl]carbonyl}-L-glutamic acid, ... | 著者 | Thoden, J.B, Woodford, C.R, Holden, H.M. | 登録日 | 2014-12-18 | 公開日 | 2015-01-21 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | New Role for the Ankyrin Repeat Revealed by a Study of the N-Formyltransferase from Providencia alcalifaciens. Biochemistry, 54, 2015
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4XD8
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4XKO
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4XUR
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4XUO
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4XUQ
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4XUT
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![BU of 4xut by Molmil](/molmil-images/mine/4xut) | Structure of the CBM22-2 xylan-binding domain in complex with 1,3:1,4 Beta-glucotetraose B from Paenibacillus barcinonensis Xyn10C | 分子名称: | CALCIUM ION, Endo-1,4-beta-xylanase C, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Sainz-Polo, M.A, Sanz-Aparicio, J. | 登録日 | 2015-01-26 | 公開日 | 2015-06-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Exploring Multimodularity in Plant Cell Wall Deconstruction: STRUCTURAL AND FUNCTIONAL ANALYSIS OF Xyn10C CONTAINING THE CBM22-1-CBM22-2 TANDEM. J.Biol.Chem., 290, 2015
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4XSQ
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![BU of 4xsq by Molmil](/molmil-images/mine/4xsq) | Structure of a variable lymphocyte receptor-like protein Bf66946 from Branchiostoma floridae | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, variable lymphocyte receptor-like protein Bf66946 | 著者 | Cao, D.D, Cheng, W, Jiang, Y.L, Wang, W.J, Li, Q, Chen, Y, Zhou, C.Z. | 登録日 | 2015-01-22 | 公開日 | 2016-03-23 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Structure of a variable lymphocyte receptor-like protein from the amphioxus Branchiostoma floridae. Sci Rep, 6, 2016
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4XSY
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![BU of 4xsy by Molmil](/molmil-images/mine/4xsy) | Crystal structure of CBR 9379 bound to Escherichia coli RNA polymerase holoenzyme | 分子名称: | 3-{[(2,6-dichlorophenyl)carbamoyl]amino}-N-hydroxy-N'-phenyl-5-(trifluoromethyl)benzenecarboximidamide, DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ... | 著者 | Bae, B, Darst, S.A. | 登録日 | 2015-01-22 | 公開日 | 2015-07-22 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (4.007 Å) | 主引用文献 | CBR antimicrobials inhibit RNA polymerase via at least two bridge-helix cap-mediated effects on nucleotide addition. Proc.Natl.Acad.Sci.USA, 112, 2015
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4XUP
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8OWC
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4XUN
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4XXD
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![BU of 4xxd by Molmil](/molmil-images/mine/4xxd) | Crystal Structure of mid-region amyloid beta capture by solanezumab | 分子名称: | Amyloid-beta fragment, Fab Heavy Chain, Fab Light Chain | 著者 | Hermans, S.J, Crespi, G.A.N, Parker, M.W, Miles, L.A. | 登録日 | 2015-01-30 | 公開日 | 2015-04-29 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Molecular basis for mid-region amyloid-beta capture by leading Alzheimer's disease immunotherapies. Sci Rep, 5, 2015
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8JP1
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![BU of 8jp1 by Molmil](/molmil-images/mine/8jp1) | Crystal structure of AKR1C3 in complex with DFV | 分子名称: | 7-HYDROXY-2-(4-HYDROXY-PHENYL)-CHROMAN-4-ONE, Aldo-keto reductase family 1 member C3, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Zheng, X.H, Liu, H, Yao, Z.Q, Zhang, L.P. | 登録日 | 2023-06-10 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Inhibition of AKR1Cs by liquiritigenin and the structural basis. Chem.Biol.Interact., 385, 2023
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4YFT
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![BU of 4yft by Molmil](/molmil-images/mine/4yft) | HUab-20bp | 分子名称: | DNA-binding protein HU-alpha, DNA-binding protein HU-beta, synthetic DNA strand | 著者 | Hammel, M, Reyes, F.E, Parpana, R, Tainer, J.A, Adhya, S, Amlanjyoti, D. | 登録日 | 2015-02-25 | 公開日 | 2016-06-29 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.914 Å) | 主引用文献 | HU multimerization shift controls nucleoid compaction. Sci Adv, 2, 2016
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4YLK
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![BU of 4ylk by Molmil](/molmil-images/mine/4ylk) | Crystal structure of DYRK1A in complex with 10-Chloro-substituted 11H-indolo[3,2-c]quinolone-6-carboxylic acid inhibitor 5s | 分子名称: | 1,2-ETHANEDIOL, 10-chloro-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, ... | 著者 | Chaikuad, A, Falke, H, Krojer, T, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2015-03-05 | 公開日 | 2015-03-25 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | 10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A. J.Med.Chem., 58, 2015
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4YO9
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![BU of 4yo9 by Molmil](/molmil-images/mine/4yo9) | HKU4 3CLpro unbound structure | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 3C-like proteinase, ACETATE ION, ... | 著者 | St John, S.E, Mesecar, A. | 登録日 | 2015-03-11 | 公開日 | 2015-08-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Targeting zoonotic viruses: Structure-based inhibition of the 3C-like protease from bat coronavirus HKU4-The likely reservoir host to the human coronavirus that causes Middle East Respiratory Syndrome (MERS). Bioorg.Med.Chem., 23, 2015
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4YOE
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![BU of 4yoe by Molmil](/molmil-images/mine/4yoe) | Structure of UP1 bound to RNA 5'-AGU-3' | 分子名称: | ACETATE ION, Heterogeneous nuclear ribonucleoprotein A1, RNA AGU, ... | 著者 | Meagher, J.L, Stuckey, J.A. | 登録日 | 2015-03-11 | 公開日 | 2015-06-10 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | The First Crystal Structure of the UP1 Domain of hnRNP A1 Bound to RNA Reveals a New Look for an Old RNA Binding Protein. J.Mol.Biol., 427, 2015
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4YEW
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![BU of 4yew by Molmil](/molmil-images/mine/4yew) | HUab-19bp | 分子名称: | DNA-binding protein HU-alpha, DNA-binding protein HU-beta, synthetic DNA strand | 著者 | Hammel, M, Reyes, F.E, Parpana, R, Tainer, J.A, Adhya, S, Amlanjyoti, D. | 登録日 | 2015-02-24 | 公開日 | 2016-06-29 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.683 Å) | 主引用文献 | HU multimerization shift controls nucleoid compaction. Sci Adv, 2, 2016
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4YLJ
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![BU of 4ylj by Molmil](/molmil-images/mine/4ylj) | Crystal structure of DYRK1A in complex with 10-Iodo-substituted 11H-indolo[3,2-c]quinoline-6-carboxylic acid inhibitor 5j | 分子名称: | 10-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acid, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, SULFATE ION, ... | 著者 | Chaikuad, A, Falke, H, Nowak, R, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2015-03-05 | 公開日 | 2015-03-25 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.58 Å) | 主引用文献 | 10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A. J.Med.Chem., 58, 2015
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4YO0
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![BU of 4yo0 by Molmil](/molmil-images/mine/4yo0) | Crystal structure of monoclonal anti-human podoplanin antibody NZ-1 with bound PA peptide | 分子名称: | 1,2-ETHANEDIOL, Heavy chain of antigen binding fragment, Fab, ... | 著者 | Fujii, Y, Kitago, Y, Arimori, T, Takagi, J. | 登録日 | 2015-03-11 | 公開日 | 2016-03-02 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Tailored placement of a turn-forming PA tag into the structured domain of a protein to probe its conformational state J.Cell.Sci., 129, 2016
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4YOJ
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![BU of 4yoj by Molmil](/molmil-images/mine/4yoj) | HKU4 3CLpro bound to non-covalent inhibitor 2A | 分子名称: | 3C-like proteinase, ACETATE ION, FORMIC ACID, ... | 著者 | St John, S.E, Mesecar, A. | 登録日 | 2015-03-11 | 公開日 | 2015-08-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Targeting zoonotic viruses: Structure-based inhibition of the 3C-like protease from bat coronavirus HKU4-The likely reservoir host to the human coronavirus that causes Middle East Respiratory Syndrome (MERS). Bioorg.Med.Chem., 23, 2015
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