1EAF
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1EAG
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1EAH
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![BU of 1eah by Molmil](/molmil-images/mine/1eah) | PV2L COMPLEXED WITH ANTIVIRAL AGENT SCH48973 | 分子名称: | 1[2-CHLORO-4-METHOXY-PHENYL-OXYMETHYL]-4-[2,6-DICHLORO-PHENYL-OXYMETHYL]-BENZENE, MYRISTIC ACID, POLIOVIRUS TYPE 2 COAT PROTEINS VP1 TO VP4 | 著者 | Lentz, K, Arnold, E. | 登録日 | 1997-07-22 | 公開日 | 1998-09-16 | 最終更新日 | 2023-04-19 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structure of poliovirus type 2 Lansing complexed with antiviral agent SCH48973: comparison of the structural and biological properties of three poliovirus serotypes. Structure, 5, 1997
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1EAI
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![BU of 1eai by Molmil](/molmil-images/mine/1eai) | COMPLEX OF ASCARIS CHYMOTRPSIN/ELASTASE INHIBITOR WITH PORCINE ELASTASE | 分子名称: | PROTEIN (CHYMOTRYPSIN/ELASTASE ISOINHIBITOR 1), PROTEIN (ELASTASE) | 著者 | Huang, K, Strynadka, N.C.J, Bernard, V.D, Peanasky, R.J, James, M.N.G. | 登録日 | 1999-03-25 | 公開日 | 1999-04-05 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The molecular structure of the complex of Ascaris chymotrypsin/elastase inhibitor with porcine elastase. Structure, 2, 1994
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1EAJ
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1EAK
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![BU of 1eak by Molmil](/molmil-images/mine/1eak) | Catalytic domain of proMMP-2 E404Q mutant | 分子名称: | 72 KDA TYPE IV COLLAGENASE, CALCIUM ION, INHIBITOR PEPTIDE, ... | 著者 | Bergmann, U, Tuuttila, A, Tryggvason, K, Morgunova, E. | 登録日 | 2001-07-12 | 公開日 | 2002-08-22 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Crystal Structure of Human Mmp-2 Reveals a New P To be Published
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1EAL
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![BU of 1eal by Molmil](/molmil-images/mine/1eal) | NMR STUDY OF ILEAL LIPID BINDING PROTEIN | 分子名称: | ILEAL LIPID BINDING PROTEIN | 著者 | Luecke, C, Zhang, F, Rueterjans, H, Hamilton, J.A, Sacchettini, J.C. | 登録日 | 1996-08-28 | 公開日 | 1997-01-22 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Flexibility is a likely determinant of binding specificity in the case of ileal lipid binding protein. Structure, 4, 1996
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1EAM
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![BU of 1eam by Molmil](/molmil-images/mine/1eam) | VACCINIA METHYLTRANSFERASE VP39 MUTANT (EC: 2.7.7.19) | 分子名称: | PROTEIN (VP39), S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Hu, G, Hodel, A.E, Gershon, P.D, Quiocho, F.A. | 登録日 | 1999-01-26 | 公開日 | 1999-06-14 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | mRNA cap recognition: dominant role of enhanced stacking interactions between methylated bases and protein aromatic side chains. Proc.Natl.Acad.Sci.USA, 96, 1999
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1EAN
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![BU of 1ean by Molmil](/molmil-images/mine/1ean) | THE RUNX1 Runt domain at 1.70A resolution: A structural switch and specifically bound chloride ions modulate DNA binding | 分子名称: | CHLORIDE ION, RUNT-RELATED TRANSCRIPTION FACTOR 1 | 著者 | Backstrom, S, Wolf-Watz, M, Grundstrom, C, Hard, T, Grundstrom, T, Sauer, U.H. | 登録日 | 2001-07-13 | 公開日 | 2002-09-12 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Runx1 Runt Domain at 1.25 A Resolution: A Structural Switch and Specifically Bound Chloride Ions Modulate DNA Binding J.Mol.Biol., 322, 2002
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1EAO
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![BU of 1eao by Molmil](/molmil-images/mine/1eao) | THE RUNX1 Runt domain at 1.4A resolution: a structural switch and specifically bound chloride ions modulate DNA binding | 分子名称: | BROMIDE ION, RUNT-RELATED TRANSCRIPTION FACTOR 1 | 著者 | Backstrom, S, Wolf-Watz, M, Grundstrom, C, Hard, T.H, Grundstrom, T, Sauer, U.H. | 登録日 | 2001-07-14 | 公開日 | 2002-09-12 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | The Runx1 Runt Domain at 1.25A Resolution: A Structural Switch and Specifically Bound Chloride Ions Modulate DNA Binding J.Mol.Biol., 322, 2002
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1EAP
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![BU of 1eap by Molmil](/molmil-images/mine/1eap) | CRYSTAL STRUCTURE OF A CATALYTIC ANTIBODY WITH A SERINE PROTEASE ACTIVE SITE | 分子名称: | IGG2B-KAPPA 17E8 FAB (HEAVY CHAIN), IGG2B-KAPPA 17E8 FAB (LIGHT CHAIN), PHENYL[1-(N-SUCCINYLAMINO)PENTYL]PHOSPHONATE | 著者 | Zhou, G.W, Guo, J, Huang, W, Scanlan, T.S, Fletterick, R.J. | 登録日 | 1994-08-10 | 公開日 | 1994-12-20 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structure of a catalytic antibody with a serine protease active site. Science, 265, 1994
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1EAQ
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![BU of 1eaq by Molmil](/molmil-images/mine/1eaq) | The RUNX1 Runt domain at 1.25A resolution: A structural switch and specifically bound chloride ions modulate DNA binding | 分子名称: | CHLORIDE ION, RUNT-RELATED TRANSCRIPTION FACTOR 1 | 著者 | Backstrom, S, Wolf-Watz, M, Grundstrom, C, Hard, T, Grundstrom, T, Sauer, U.H. | 登録日 | 2001-07-14 | 公開日 | 2002-09-12 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | The Runx1 Runt Domain at 1.25 A Resolution: A Structural Switch and Specifically Bound Chloride Ions Modulate DNA Binding J.Mol.Biol., 322, 2002
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1EAR
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![BU of 1ear by Molmil](/molmil-images/mine/1ear) | Crystal structure of Bacillus pasteurii UreE at 1.7 A. Type II crystal form. | 分子名称: | UREASE ACCESSORY PROTEIN UREE, ZINC ION | 著者 | Remaut, H, Safarov, N, Ciurli, S, Van Beeumen, J. | 登録日 | 2001-07-16 | 公開日 | 2002-01-04 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural Basis for Ni2+ Transport and Assembly of the Urease Active Site by the Metallochaperone Uree from Bacillus Pasteurii J.Biol.Chem., 276, 2001
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1EAS
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![BU of 1eas by Molmil](/molmil-images/mine/1eas) | NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OF ORALLY ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES | 分子名称: | 3-[[(METHYLAMINO)SULFONYL]AMINO]-2-OXO-6-PHENYL-N-[3,3,3-TRIFLUORO-1-(1-METHYLETHYL)-2-OXOPHENYL]-1(2H)-PYRIDINE ACETAMIDE, PORCINE PANCREATIC ELASTASE, SODIUM ION, ... | 著者 | Ceccarelli, C. | 登録日 | 1994-11-22 | 公開日 | 1995-02-07 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Nonpeptidic inhibitors of human leukocyte elastase. 3. Design, synthesis, X-ray crystallographic analysis, and structure-activity relationships for a series of orally active 3-amino-6-phenylpyridin-2-one trifluoromethyl ketones. J.Med.Chem., 37, 1994
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1EAT
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![BU of 1eat by Molmil](/molmil-images/mine/1eat) | NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY ACTIVE 5-AMINO-PYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYLKETONES | 分子名称: | 2-[5-METHANESULFONYLAMINO-2-(4-AMINOPHENYL)-6-OXO-1,6-DIHYDRO-1-PYRIMIDINYL]-N-(3,3,3-TRIFLUORO-1-ISOPROPYL-2-OXOPROPYL)ACETAMIDE, PORCINE PANCREATIC ELASTASE, SODIUM ION, ... | 著者 | Ceccarelli, C. | 登録日 | 1994-11-22 | 公開日 | 1995-02-07 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Nonpeptidic inhibitors of human leukocyte elastase. 5. Design, synthesis, and X-ray crystallography of a series of orally active 5-aminopyrimidin-6-one-containing trifluoromethyl ketones. J.Med.Chem., 38, 1995
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1EAU
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![BU of 1eau by Molmil](/molmil-images/mine/1eau) | NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 6. DESIGN OF A POTENT, INTRATRACHEALLY ACTIVE, PYRIDONE-BASED TRIFLUOROMETHYL KETONE | 分子名称: | 2-[5-AMINO-6-OXO-2-(2-THIENYL)-1,6-DIHYDROPYRIMIDIN-1-YL)-N-[3,3-DIFLUORO -1-ISOPROPYL-2-OXO-3-(N-(2-MORPHOLINO ETHYL)CARBAMOYL]PROPYL]ACETAMIDE, PORCINE PANCREATIC ELASTASE, SODIUM ION, ... | 著者 | Ceccarelli, C. | 登録日 | 1994-11-22 | 公開日 | 1995-02-07 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Nonpeptidic inhibitors of human leukocyte elastase. 6. Design of a potent, intratracheally active, pyridone-based trifluoromethyl ketone. J.Med.Chem., 38, 1995
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1EAV
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1EAW
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1EAX
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![BU of 1eax by Molmil](/molmil-images/mine/1eax) | Crystal structure of MTSP1 (matriptase) | 分子名称: | BENZAMIDINE, SULFATE ION, SUPPRESSOR OF TUMORIGENICITY 14 | 著者 | Friedrich, R, Bode, W. | 登録日 | 2001-07-17 | 公開日 | 2002-01-28 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Catalytic Domain Structures of Mt-Sp1/Matriptase, a Matrix-Degrading Transmembrane Serine Proteinase. J.Biol.Chem., 277, 2002
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1EAY
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![BU of 1eay by Molmil](/molmil-images/mine/1eay) | CHEY-BINDING (P2) DOMAIN OF CHEA IN COMPLEX WITH CHEY FROM ESCHERICHIA COLI | 分子名称: | CHEA, CHEY | 著者 | Mcevoy, M.M, Hausrath, A.C, Randolph, G.B, Remington, S.J, Dahlquist, F.W. | 登録日 | 1998-04-23 | 公開日 | 1998-07-15 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Two binding modes reveal flexibility in kinase/response regulator interactions in the bacterial chemotaxis pathway. Proc.Natl.Acad.Sci.USA, 95, 1998
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1EAZ
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![BU of 1eaz by Molmil](/molmil-images/mine/1eaz) | Crystal structure of the phosphoinositol (3,4)-bisphosphate binding PH domain of TAPP1 from human. | 分子名称: | CITRIC ACID, TANDEM PH DOMAIN CONTAINING PROTEIN-1 | 著者 | Thomas, C.C, Dowler, S, Deak, M, Alessi, D.R, Van Aalten, D.M.F. | 登録日 | 2001-07-17 | 公開日 | 2002-07-11 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Crystal Structure of the Phosphatidylinositol 3,4-Bisphosphate-Binding Pleckstrin Homology (Ph) Domain of Tandem Ph-Domain-Containing Protein 1 (Tapp1): Molecular Basis of Lipid Specificity Biochem.J., 358, 2001
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1EB0
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![BU of 1eb0 by Molmil](/molmil-images/mine/1eb0) | Crystal structure of Bacillus pasteurii UreE at 1.85 A, phased by SIRAS. Type I crystal form. | 分子名称: | UREASE ACCESSORY PROTEIN UREE, ZINC ION | 著者 | Remaut, H, Safarov, N, Ciurli, S, Van Beeumen, J. | 登録日 | 2001-07-17 | 公開日 | 2002-01-04 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural Basis for Ni2+ Transport and Assembly of the Urease Active Site by the Metallochaperone Uree from Bacillus Pasteurii J.Biol.Chem., 276, 2001
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1EB1
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![BU of 1eb1 by Molmil](/molmil-images/mine/1eb1) | Complex structure of human thrombin with N-methyl-arginine inhibitor | 分子名称: | 3-CYCLOHEXYL-D-ALANYL-L-PROLYL-N~2~-METHYL-L-ARGININE, PEPTIDE INHIBITOR, THROMBIN HEAVY CHAIN, ... | 著者 | Friedrich, R, Steinmetzer, T, Bode, W. | 登録日 | 2001-07-18 | 公開日 | 2002-01-28 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The Methyl Group of N(Alpha)(Me)Arg-Containing Peptides Disturbs the Active-Site Geometry of Thrombin, Impairing Efficient Cleavage J.Mol.Biol., 316, 2002
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1EB2
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![BU of 1eb2 by Molmil](/molmil-images/mine/1eb2) | Trypsin inhibitor complex (BPO) | 分子名称: | 3-[(Z)-AMINO(IMINO)METHYL]-N-[2-(4-BENZOYL-1-PIPERIDINYL)-2-OXO-1-PHENYLETHYL]BENZAMIDE, CALCIUM ION, SULFATE ION, ... | 著者 | Wilkinson, K.W, Young, S.C, Liebeschuetz, J.W, Brady, R.L. | 登録日 | 2001-07-18 | 公開日 | 2002-02-11 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Pro_Select: Combining Structure-Based Drug Design and Array-Based Chemistry for Rapid Lead Discovery. 2. The Development of a Series of Highly Potent and Selective Factor Xa Inhibitors J.Med.Chem., 45, 2002
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1EB3
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![BU of 1eb3 by Molmil](/molmil-images/mine/1eb3) | YEAST 5-AMINOLAEVULINIC ACID DEHYDRATASE 4,7-DIOXOSEBACIC ACID COMPLEX | 分子名称: | 4,7-DIOXOSEBACIC ACID, 5-AMINOLAEVULINIC ACID DEHYDRATASE, ZINC ION | 著者 | Erskine, P.T, Coates, L, Newbold, R, Brindley, A.A, Stauffer, F, Wood, S.P, Warren, M.J, Cooper, J.B, Shoolingin-Jordan, P.M, Neier, R. | 登録日 | 2001-07-18 | 公開日 | 2001-08-02 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | The X-Ray Structure of Yeast 5-Aminolaevulinic Acid Dehydratase Complexed with Two Diacid Inhibitors FEBS Lett., 503, 2001
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