8EUA
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![BU of 8eua by Molmil](/molmil-images/mine/8eua) | Structure of SARS-CoV2 PLpro bound to a covalent inhibitor | 分子名称: | Papain-like protease nsp3, SULFATE ION, ZINC ION, ... | 著者 | Mathews, I.I, Pokhrel, S, Wakatsuki, S. | 登録日 | 2022-10-18 | 公開日 | 2023-04-05 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Potent and selective covalent inhibition of the papain-like protease from SARS-CoV-2. Nat Commun, 14, 2023
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8EU8
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![BU of 8eu8 by Molmil](/molmil-images/mine/8eu8) | Cryo-EM structure of CH848 10.17DT DS-SOSIP-2P Env | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CH848 10.17DT SOSIP Envelope glycoprotein gp160 | 著者 | Wrapp, D, Acharya, P, Haynes, B.F. | 登録日 | 2022-10-18 | 公開日 | 2023-01-04 | 最終更新日 | 2023-02-08 | 実験手法 | ELECTRON MICROSCOPY (3.73 Å) | 主引用文献 | Structure-Based Stabilization of SOSIP Env Enhances Recombinant Ectodomain Durability and Yield. J.Virol., 97, 2023
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8EU3
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![BU of 8eu3 by Molmil](/molmil-images/mine/8eu3) | Cryo-EM structure of cGMP bound human CNGA3/CNGB3 channel in GDN, transition state 1 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CYCLIC GUANOSINE MONOPHOSPHATE, Cyclic nucleotide-gated cation channel alpha-3, ... | 著者 | Hu, Z, Zheng, X, Yang, J. | 登録日 | 2022-10-18 | 公開日 | 2023-08-02 | 実験手法 | ELECTRON MICROSCOPY (3.62 Å) | 主引用文献 | Conformational trajectory of allosteric gating of the human cone photoreceptor cyclic nucleotide-gated channel. Nat Commun, 14, 2023
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8EU2
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![BU of 8eu2 by Molmil](/molmil-images/mine/8eu2) | Class3 of the INO80-Hexasome complex | 分子名称: | DNA (110-MER), Histone H2A type 1, Histone H2B 1.1, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-18 | 公開日 | 2023-07-12 | 最終更新日 | 2024-04-03 | 実験手法 | ELECTRON MICROSCOPY (2.93 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8EU1
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![BU of 8eu1 by Molmil](/molmil-images/mine/8eu1) | |
8ETZ
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![BU of 8etz by Molmil](/molmil-images/mine/8etz) | |
8ETY
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8ETX
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![BU of 8etx by Molmil](/molmil-images/mine/8etx) | |
8ETV
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![BU of 8etv by Molmil](/molmil-images/mine/8etv) | Class2 of the INO80-Hexasome complex | 分子名称: | DNA (110-MER), Histone H2A type 1, Histone H2B 1.1, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-17 | 公開日 | 2023-07-12 | 最終更新日 | 2024-04-03 | 実験手法 | ELECTRON MICROSCOPY (3.16 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8ETT
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![BU of 8ett by Molmil](/molmil-images/mine/8ett) | Class1 of the INO80-Hexasome complex | 分子名称: | DNA (110-MER), Histone H2A type 1, Histone H2B 1.1, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-17 | 公開日 | 2023-07-12 | 最終更新日 | 2024-04-03 | 実験手法 | ELECTRON MICROSCOPY (6.68 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8ETP
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![BU of 8etp by Molmil](/molmil-images/mine/8etp) | Cryo-EM structure of cGMP bound closed state of human CNGA3/CNGB3 channel in GDN | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CYCLIC GUANOSINE MONOPHOSPHATE, Cyclic nucleotide-gated cation channel alpha-3, ... | 著者 | Hu, Z, Zheng, X, Yang, J. | 登録日 | 2022-10-17 | 公開日 | 2023-08-02 | 実験手法 | ELECTRON MICROSCOPY (3.52 Å) | 主引用文献 | Conformational trajectory of allosteric gating of the human cone photoreceptor cyclic nucleotide-gated channel. Nat Commun, 14, 2023
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8ETO
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![BU of 8eto by Molmil](/molmil-images/mine/8eto) | Co-crystal structure of Chaetomium glucosidase with compound 25 | 分子名称: | (1S,2S,3R,4S,5S)-1-(hydroxymethyl)-5-{[(5Z)-6-{[2-nitro-4-(2H-1,2,3-triazol-2-yl)phenyl]amino}hex-5-en-1-yl]amino}cyclohexane-1,2,3,4-tetrol, 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Karade, S.S, Mariuzza, R.A. | 登録日 | 2022-10-17 | 公開日 | 2023-02-22 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure-Based Design of Potent Iminosugar Inhibitors of Endoplasmic Reticulum alpha-Glucosidase I with Anti-SARS-CoV-2 Activity. J.Med.Chem., 66, 2023
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8ETN
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8ETL
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![BU of 8etl by Molmil](/molmil-images/mine/8etl) | Co-crystal structure of Chaetomium glucosidase with compound 24 | 分子名称: | (1S,2S,3R,4S,5S)-5-(butylamino)-1-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol, 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Chaetomium alpha glucosidase, ... | 著者 | Karade, S.S, Mariuzza, R.A. | 登録日 | 2022-10-17 | 公開日 | 2023-02-22 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure-Based Design of Potent Iminosugar Inhibitors of Endoplasmic Reticulum alpha-Glucosidase I with Anti-SARS-CoV-2 Activity. J.Med.Chem., 66, 2023
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8ET8
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![BU of 8et8 by Molmil](/molmil-images/mine/8et8) | Cryo-EM structure of the organic cation transporter 1 in complex with verapamil | 分子名称: | (2S)-2-(3,4-dimethoxyphenyl)-5-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-2-(propan-2-yl)pentanenitrile, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, OCT1 | 著者 | Suo, Y, Wright, N.J, Lee, S.-Y. | 登録日 | 2022-10-16 | 公開日 | 2023-05-31 | 最終更新日 | 2023-08-02 | 実験手法 | ELECTRON MICROSCOPY (3.45 Å) | 主引用文献 | Molecular basis of polyspecific drug and xenobiotic recognition by OCT1 and OCT2. Nat.Struct.Mol.Biol., 30, 2023
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8ESZ
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![BU of 8esz by Molmil](/molmil-images/mine/8esz) | Structure of mitochondrial complex I from Drosophila melanogaster, Helix-locked state | 分子名称: | (2R)-3-{[(S)-hydroxy(3-methylbutoxy)phosphoryl]oxy}-2-(octanoyloxy)propyl decanoate, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, ... | 著者 | Padavannil, A, Letts, J.A. | 登録日 | 2022-10-15 | 公開日 | 2023-03-29 | 最終更新日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Resting mitochondrial complex I from Drosophila melanogaster adopts a helix-locked state. Elife, 12, 2023
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8ESY
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![BU of 8esy by Molmil](/molmil-images/mine/8esy) | D30N mutant HIV protease in complex with benzoxaborolone analog of darunavir | 分子名称: | CHLORIDE ION, GLYCEROL, Protease, ... | 著者 | Windsor, I.W, Graham, B.J, Raines, R.T. | 登録日 | 2022-10-15 | 公開日 | 2023-02-08 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Inhibition of HIV-1 Protease by a Boronic Acid with High Oxidative Stability. Acs Med.Chem.Lett., 14, 2023
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8ESX
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![BU of 8esx by Molmil](/molmil-images/mine/8esx) | HIV protease in complex with benzoxaborolone analog of darunavir | 分子名称: | ACETATE ION, CHLORIDE ION, GLYCEROL, ... | 著者 | Windsor, I.W, Graham, B.J, Raines, R.T. | 登録日 | 2022-10-15 | 公開日 | 2023-02-08 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Inhibition of HIV-1 Protease by a Boronic Acid with High Oxidative Stability. Acs Med.Chem.Lett., 14, 2023
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8ESW
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![BU of 8esw by Molmil](/molmil-images/mine/8esw) | Structure of mitochondrial complex I from Drosophila melanogaster, Flexible-class 1 | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Padavannil, A, Letts, J.A. | 登録日 | 2022-10-15 | 公開日 | 2023-03-29 | 最終更新日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Resting mitochondrial complex I from Drosophila melanogaster adopts a helix-locked state. Elife, 12, 2023
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8ESV
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8ESU
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![BU of 8esu by Molmil](/molmil-images/mine/8esu) | Myoglobin variant Mb-imi complex | 分子名称: | IMIDAZOLE, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Bacik, J.P, Fasan, R, Ando, N. | 登録日 | 2022-10-14 | 公開日 | 2023-12-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.04 Å) | 主引用文献 | Mechanistic manifold in a hemoprotein-catalyzed cyclopropanation reaction with diazoketone. Nat Commun, 14, 2023
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8EST
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![BU of 8est by Molmil](/molmil-images/mine/8est) | REACTION OF PORCINE PANCREATIC ELASTASE WITH 7-SUBSTITUTED 3-ALKOXY-4-CHLOROISOCOUMARINS: DESIGN OF POTENT INHIBITORS USING THE CRYSTAL STRUCTURE OF THE COMPLEX FORMED WITH 4-CHLORO-3-ETHOXY-7-GUANIDINO-ISOCOUMARIN | 分子名称: | CALCIUM ION, ETHYL-(2-CARBOXY-4-GUANIDINIUM-PHENYL)-CHLOROACETATE, PORCINE PANCREATIC ELASTASE, ... | 著者 | Radhakrishnan, R, Powers, J.C, Meyerjunior, E.F. | 登録日 | 1990-02-21 | 公開日 | 1992-10-15 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Reaction of porcine pancreatic elastase with 7-substituted 3-alkoxy-4-chloroisocoumarins: design of potent inhibitors using the crystal structure of the complex formed with 4-chloro-3-ethoxy-7-guanidinoisocoumarin. Biochemistry, 29, 1990
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8ESS
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![BU of 8ess by Molmil](/molmil-images/mine/8ess) | Myoglobin variant Mb-cIII complex | 分子名称: | Myoglobin, SULFATE ION, [2,18-bis(2-carboxyethyl)-7,12-diethenyl-3,8,13,17-tetramethyl-21-(2-oxo-3-phenylpropyl)porphyrin-21-iumato(2-)-kappa~3~N~22~,N~23~,N~24~]iron(2+) | 著者 | Bacik, J.P, Fasan, R, Ando, N. | 登録日 | 2022-10-14 | 公開日 | 2023-12-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Mechanistic manifold in a hemoprotein-catalyzed cyclopropanation reaction with diazoketone. Nat Commun, 14, 2023
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8ESH
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![BU of 8esh by Molmil](/molmil-images/mine/8esh) | Structure of chimeric HLA-A*02:01 bound to CMV peptide | 分子名称: | Beta-2-microglobulin, CMV peptide, HLA-A*02:01 | 著者 | Florio, T.J, Ani, O, Young, M.C, Mallik, L, Sgourakis, N.G. | 登録日 | 2022-10-14 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.72 Å) | 主引用文献 | Decoupling peptide binding from T cell receptor recognition with engineered chimeric MHC-I molecules. Front Immunol, 14, 2023
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8ES5
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