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1QZ2
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Crystal Structure of FKBP52 C-terminal Domain complex with the C-terminal peptide MEEVD of Hsp90
分子名称: 5-mer peptide from Heat shock protein HSP 90, FK506-binding protein 4
著者Wu, B, Li, P, Lou, Z, Liu, Y, Ding, Y, Shu, C, Shen, B, Rao, Z.
登録日2003-09-15
公開日2004-06-22
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献3D structure of human FK506-binding protein 52: Implications for the assembly of the glucocorticoid receptor/Hsp90/immunophilin heterocomplex.
Proc.Natl.Acad.Sci.USA, 101, 2004
1Q6H
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Crystal structure of a truncated form of FkpA from Escherichia coli
分子名称: FKBP-type peptidyl-prolyl cis-trans isomerase fkpA
著者Saul, F.A, Arie, J.-P, Vulliez-le Normand, B, Kahn, R, Betton, J.-M, Bentley, G.A.
登録日2003-08-13
公開日2004-01-13
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Structural and functional studies of FkpA from Escherichia coli, a cis/trans peptidyl-prolyl isomerase with chaperone activity.
J.Mol.Biol., 335, 2004
1Q6U
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Crystal structure of FkpA from Escherichia coli
分子名称: CESIUM ION, FKBP-type peptidyl-prolyl cis-trans isomerase fkpA
著者Saul, F.A, Arie, J.-P, Vulliez-le Normand, B, Kahn, R, Betton, J.-M, Bentley, G.A.
登録日2003-08-14
公開日2004-01-13
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structural and functional studies of FkpA from Escherichia coli, a cis/trans peptidyl-prolyl isomerase with chaperone activity.
J.Mol.Biol., 335, 2004
1Q6I
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Crystal structure of a truncated form of FkpA from Escherichia coli, in complex with immunosuppressant FK506
分子名称: 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN, FKBP-type peptidyl-prolyl cis-trans isomerase fkpA
著者Saul, F.A, Arie, J.-P, Vulliez-le Normand, B, Kahn, R, Betton, J.-M, Bentley, G.A.
登録日2003-08-13
公開日2004-01-13
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structural and functional studies of FkpA from Escherichia coli, a cis/trans peptidyl-prolyl isomerase with chaperone activity.
J.Mol.Biol., 335, 2004
1R9H
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Structural Genomics of C.elegans: FKBP-type Peptidylprolyl Isomerase
分子名称: FK506 Binding protein family
著者Li, S, Southeast Collaboratory for Structural Genomics (SECSG)
登録日2003-10-29
公開日2003-12-02
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural Genomics of C.elegans: FKBP-type Peptidylprolyl Isomerase
To be Published
1L1P
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Solution Structure of the PPIase Domain from E. coli Trigger Factor
分子名称: trigger factor
著者Kozlov, G, Trempe, J.-F, Perreault, A, Wong, M, Denisov, A, Ghandi, S, Gehring, K, Ekiel, I, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI)
登録日2002-02-19
公開日2003-06-24
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution Structure of the Closed Form of a Peptidyl-Prolyl Isomerase Reveals the Mechanism of Protein Folding
To be Published
1IX5
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Solution structure of the Methanococcus thermolithotrophicus FKBP
分子名称: FKBP
著者Suzuki, R, Nagata, K, Kawakami, M, Nemoto, N, Furutani, M, Adachi, K, Maruyama, T, Tanokura, M.
登録日2002-06-12
公開日2003-06-10
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Three-dimensional Solution Structure of an Archaeal FKBP with a Dual Function of Peptidyl Prolyl cis-trans Isomerase and Chaperone-like Activities
J.MOL.BIOL., 328, 2003
1J4I
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crystal structure analysis of the FKBP12 complexed with 000308 small molecule
分子名称: 4-METHYL-2-{[4-(TOLUENE-4-SULFONYL)-THIOMORPHOLINE-3-CARBONYL]-AMINO}-PENTANOIC ACID, FKBP12
著者Li, P, Ding, Y, Wang, L, Wu, B, Shu, C, Li, S, Shen, B, Rao, Z.
登録日2001-09-30
公開日2003-06-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Design and structure-based study of new potential FKBP12 inhibitors.
Biophys.J., 85, 2003
1J4H
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crystal structure analysis of the FKBP12 complexed with 000107 small molecule
分子名称: 3-PHENYL-2-{[4-(TOLUENE-4-SULFONYL)-THIOMORPHOLINE-3-CARBONYL]-AMINO}-PROPIONIC ACID ETHYL ESTER, FKBP12
著者Li, P, Ding, Y, Wang, L, Wu, B, Shu, C, Li, S, Shen, B, Rao, Z.
登録日2001-09-30
公開日2003-06-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Design and structure-based study of new potential FKBP12 inhibitors.
Biophys.J., 85, 2003
1KT1
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Structure of the Large FKBP-like Protein, FKBP51, Involved in Steroid Receptor Complexes
分子名称: FK506-binding protein FKBP51, SULFATE ION
著者Sinars, C.R, Cheung-Flynn, J, Rimerman, R.A, Scammell, J.G, Smith, D.F, Clardy, J.C.
登録日2002-01-14
公開日2003-02-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献STRUCTURE OF THE LARGE FK506-BINDING PROTEIN FKBP51, AN HSP90-BINDING PROTEIN AND A COMPONENT OF STEROID RECEPTOR COMPLEXES
Proc.Natl.Acad.Sci.USA, 100, 2003
1KT0
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Structure of the Large FKBP-like Protein, FKBP51, Involved in Steroid Receptor Complexes
分子名称: 51 KDA FK506-BINDING PROTEIN, SULFATE ION
著者Sinars, C.R, Cheung-Flynn, J, Rimerman, R.A, Scammell, J.G, Smith, D.F, Clardy, J.C.
登録日2002-01-14
公開日2003-02-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the large FK506-binding protein FKBP51, an Hsp90-binding protein and a component of steroid receptor complexes
Proc.Natl.Acad.Sci.USA, 100, 2003
1N1A
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Crystal Structure of the N-terminal domain of human FKBP52
分子名称: FKBP52
著者Li, P, Ding, Y, Wu, B, Shu, C, Shen, B, Rao, Z.
登録日2002-10-16
公開日2002-12-30
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of the N-terminal domain of human FKBP52.
Acta Crystallogr.,Sect.D, 59, 2003
1JVW
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TRYPANOSOMA CRUZI MACROPHAGE INFECTIVITY POTENTIATOR (TCMIP)
分子名称: MACROPHAGE INFECTIVITY POTENTIATOR
著者Pereira, P.J.B, Vega, M.C, Gonzalez-Rey, E, Fernandez-Carazo, R, Macedo-Ribeiro, S, Gomis-Rueth, F.X, Gonzalez, A, Coll, M.
登録日2001-08-31
公開日2002-06-05
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Trypanosoma cruzi macrophage infectivity potentiator has a rotamase core and a highly exposed alpha-helix.
EMBO Rep., 3, 2002
1HXV
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PPIASE DOMAIN OF THE MYCOPLASMA GENITALIUM TRIGGER FACTOR
分子名称: TRIGGER FACTOR
著者Vogtherr, M, Parac, T.N, Maurer, M, Pahl, A, Fiebig, K.
登録日2001-01-17
公開日2002-05-29
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR solution structure and dynamics of the peptidyl-prolyl cis-trans isomerase domain of the trigger factor from Mycoplasma genitalium compared to FK506-binding protein.
J.Mol.Biol., 318, 2002
1J4R
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FK506 BINDING PROTEIN COMPLEXED WITH FKB-001
分子名称: 1-[2,2-DIFLUORO-2-(3,4,5-TRIMETHOXY-PHENYL)-ACETYL]-PIPERIDINE-2-CARBOXYLIC ACID 4-PHENYL-1-(3-PYRIDIN-3-YL-PROPYL)-BUTYL ESTER, FK506-BINDING PROTEIN, GLYCEROL, ...
著者Sheriff, S.
登録日2001-10-29
公開日2001-12-19
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献2-Aryl-2,2-difluoroacetamide FKBP12 ligands: synthesis and X-ray structural studies.
Org.Lett., 3, 2001
1FD9
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CRYSTAL STRUCTURE OF THE MACROPHAGE INFECTIVITY POTENTIATOR PROTEIN (MIP) A MAJOR VIRULENCE FACTOR FROM LEGIONELLA PNEUMOPHILA
分子名称: PROTEIN (MACROPHAGE INFECTIVITY POTENTIATOR PROTEIN), ZINC ION
著者Riboldi-Tunnicliffe, A, Jessen, S, Konig, B, Rahfeld, J, Hacker, J, Fischer, G, Hilgenfeld, R.
登録日2000-07-20
公開日2001-07-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Crystal structure of Mip, a prolylisomerase from Legionella pneumophila
Nat.Struct.Biol., 8, 2001
1F40
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SOLUTION STRUCTURE OF FKBP12 COMPLEXED WITH GPI-1046, A NEUROTROPHIC LIGAND
分子名称: (2S)-[3-PYRIDYL-1-PROPYL]-1-[3,3-DIMETHYL-1,2-DIOXOPENTYL]-2-PYRROLIDINECARBOXYLATE, FK506 BINDING PROTEIN (FKBP12)
著者Sich, C, Improta, S, Cowley, D.J, Guenet, C, Merly, J.P, Teufel, M, Saudek, V.
登録日2000-06-07
公開日2000-11-08
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of a neurotrophic ligand bound to FKBP12 and its effects on protein dynamics.
Eur.J.Biochem., 267, 2000
4FAP
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ATOMIC STRUCTURES OF THE RAPAMYCIN ANALOGS IN COMPLEX WITH BOTH HUMAN FKBP12 AND FRB DOMAIN OF FRAP
分子名称: C15-(R)-METHYLTHIENYL RAPAMYCIN, FK506-BINDING PROTEIN, FKBP12-RAPAMYCIN ASSOCIATED PROTEIN
著者Liang, J, Clardy, J.
登録日1999-05-06
公開日2000-09-13
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Refined structure of the FKBP12-rapamycin-FRB ternary complex at 2.2 A resolution.
Acta Crystallogr.,Sect.D, 55, 1999
3FAP
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ATOMIC STRUCTURES OF THE RAPAMYCIN ANALOGS IN COMPLEX WITH BOTH HUMAN FKBP12 AND FRB DOMAIN OF FRAP
分子名称: C15-(R)-METHYLTHIENYL RAPAMYCIN, FK506-BINDING PROTEIN, FKBP12-RAPAMYCIN ASSOCIATED PROTEIN
著者Liang, J, Clardy, J.
登録日1999-05-06
公開日2000-09-13
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Refined structure of the FKBP12-rapamycin-FRB ternary complex at 2.2 A resolution.
Acta Crystallogr.,Sect.D, 55, 1999
1EYM
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FK506 BINDING PROTEIN MUTANT, HOMODIMERIC COMPLEX
分子名称: FK506 BINDING PROTEIN
著者Rollins, C.T, Rivera, V.M, Woolfson, D.N, Keenan, T, Hatada, M, Adams, S.E, Andrade, L.J, Yaeger, D, van Schravendijk, M.R, Holt, D.A, Gilman, M, Clackson, T.
登録日2000-05-07
公開日2000-08-09
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A ligand-reversible dimerization system for controlling protein-protein interactions.
Proc.Natl.Acad.Sci.USA, 97, 2000
1C9H
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CRYSTAL STRUCTURE OF FKBP12.6 IN COMPLEX WITH RAPAMYCIN
分子名称: FKBP12.6, RAPAMYCIN IMMUNOSUPPRESSANT DRUG
著者Deivanayagam, C.C.S, Carson, M, Thotakura, A, Narayana, S.V.L, Chodavarapu, C.S.
登録日1999-08-02
公開日2000-08-03
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of FKBP12.6 in complex with rapamycin.
Acta Crystallogr.,Sect.D, 56, 2000
1D7H
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FKBP COMPLEXED WITH DMSO
分子名称: AMMONIUM ION, DIMETHYL SULFOXIDE, PROTEIN (FK506-BINDING PROTEIN), ...
著者Burkhard, P, Taylor, P, Walkinshaw, M.D.
登録日1999-10-18
公開日1999-10-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献X-ray structures of small ligand-FKBP complexes provide an estimate for hydrophobic interaction energies.
J.Mol.Biol., 295, 2000
1D7J
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FKBP COMPLEXED WITH 4-HYDROXY-2-BUTANONE
分子名称: 4-HYDROXY-2-BUTANONE, AMMONIUM ION, PROTEIN (FK506-BINDING PROTEIN), ...
著者Burkhard, P, Taylor, P, Walkinshaw, M.D.
登録日1999-10-18
公開日1999-10-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献X-ray structures of small ligand-FKBP complexes provide an estimate for hydrophobic interaction energies.
J.Mol.Biol., 295, 2000
1D6O
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NATIVE FKBP
分子名称: AMMONIUM ION, PROTEIN (FK506-BINDING PROTEIN), SULFATE ION
著者Burkhard, P, Taylor, P, Walkinshaw, M.D.
登録日1999-10-15
公開日1999-10-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献X-ray structures of small ligand-FKBP complexes provide an estimate for hydrophobic interaction energies.
J.Mol.Biol., 295, 2000
1D7I
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FKBP COMPLEXED WITH METHYL METHYLSULFINYLMETHYL SULFIDE (DSS)
分子名称: AMMONIUM ION, METHYL METHYLSULFINYLMETHYL SULFIDE, PROTEIN (FK506-BINDING PROTEIN), ...
著者Burkhard, P, Taylor, P, Walkinshaw, M.D.
登録日1999-10-18
公開日1999-10-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献X-ray structures of small ligand-FKBP complexes provide an estimate for hydrophobic interaction energies.
J.Mol.Biol., 295, 2000

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