4XTJ
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![BU of 4xtj by Molmil](/molmil-images/mine/4xtj) | N-terminal 43 kDa fragment of the E. coli DNA gyrase B subunit grown from 100 mM KCl plus 100 mM NaCl condition | 分子名称: | CHLORIDE ION, DNA gyrase subunit B, MAGNESIUM ION, ... | 著者 | Hearnshaw, S.J, Chung, T.T, Stevenson, C.E.M, Maxwell, A, Lawson, D.M. | 登録日 | 2015-01-23 | 公開日 | 2015-04-08 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | The role of monovalent cations in the ATPase reaction of DNA gyrase Acta Crystallogr.,Sect.D, 71, 2015
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8G3L
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![BU of 8g3l by Molmil](/molmil-images/mine/8g3l) | BceAB-S nucleotide free BceS state 2 | 分子名称: | Bacitracin export ATP-binding protein BceA, Bacitracin export permease protein BceB, OLEIC ACID, ... | 著者 | George, N.L, Orlando, B.J. | 登録日 | 2023-02-08 | 公開日 | 2023-06-21 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Architecture of a complete Bce-type antimicrobial peptide resistance module. Nat Commun, 14, 2023
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8G3A
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![BU of 8g3a by Molmil](/molmil-images/mine/8g3a) | BceAB-S nucleotide free TM state 1 | 分子名称: | Bacitracin export ATP-binding protein BceA, Bacitracin export permease protein BceB, OLEIC ACID, ... | 著者 | George, N.L, Orlando, B.J. | 登録日 | 2023-02-07 | 公開日 | 2023-06-21 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Architecture of a complete Bce-type antimicrobial peptide resistance module. Nat Commun, 14, 2023
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8G4C
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![BU of 8g4c by Molmil](/molmil-images/mine/8g4c) | BceABS ATPgS high res TM | 分子名称: | Bacitracin export ATP-binding protein BceA, Bacitracin export permease protein BceB, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | George, N.L, Orlando, B.J. | 登録日 | 2023-02-09 | 公開日 | 2023-06-21 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Architecture of a complete Bce-type antimicrobial peptide resistance module. Nat Commun, 14, 2023
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8G4D
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![BU of 8g4d by Molmil](/molmil-images/mine/8g4d) | BceABS ATPgS tilted BceS | 分子名称: | Bacitracin export ATP-binding protein BceA, Bacitracin export permease protein BceB, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, ... | 著者 | George, N.L, Orlando, B.J. | 登録日 | 2023-02-09 | 公開日 | 2023-06-21 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Architecture of a complete Bce-type antimicrobial peptide resistance module. Nat Commun, 14, 2023
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1Y4S
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![BU of 1y4s by Molmil](/molmil-images/mine/1y4s) | Conformation rearrangement of heat shock protein 90 upon ADP binding | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Chaperone protein htpG, MAGNESIUM ION | 著者 | Huai, Q, Wang, H, Liu, Y, Kim, H, Toft, D, Ke, H. | 登録日 | 2004-12-01 | 公開日 | 2005-04-19 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structures of the N-terminal and middle domains of E. coli Hsp90 and conformation changes upon ADP binding. Structure, 13, 2005
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4KQV
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![BU of 4kqv by Molmil](/molmil-images/mine/4kqv) | Topoisomerase iv atp binding domain of francisella tularensis in complex with a small molecule inhibitor | 分子名称: | 6-fluoro-4-[(3aR,6aR)-hexahydropyrrolo[3,4-b]pyrrol-5(1H)-yl]-N-methyl-2-[(2-methylpyrimidin-5-yl)oxy]-9H-pyrimido[4,5-b]indol-8-amine, IODIDE ION, Topoisomerase IV, ... | 著者 | Bensen, D.C, Akers-Rodriguez, S, Lam, T, Tari, L.W. | 登録日 | 2013-05-15 | 公開日 | 2014-01-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | A new class of type iia topoisomerase inhibitors with
broad-spectrum antibacterial activity To be Published
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1Y8P
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![BU of 1y8p by Molmil](/molmil-images/mine/1y8p) | Crystal structure of the PDK3-L2 complex | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, ... | 著者 | Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T. | 登録日 | 2004-12-13 | 公開日 | 2005-05-24 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex. Embo J., 24, 2005
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1Y4U
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![BU of 1y4u by Molmil](/molmil-images/mine/1y4u) | Conformation rearrangement of heat shock protein 90 upon ADP binding | 分子名称: | Chaperone protein htpG | 著者 | Huai, Q, Wang, H, Liu, Y, Kim, H, Toft, D, Ke, H. | 登録日 | 2004-12-01 | 公開日 | 2005-04-19 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structures of the N-terminal and middle domains of E. coli Hsp90 and conformation changes upon ADP binding. Structure, 13, 2005
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1ZXM
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![BU of 1zxm by Molmil](/molmil-images/mine/1zxm) | Human Topo IIa ATPase/AMP-PNP | 分子名称: | DNA topoisomerase II, alpha isozyme, MAGNESIUM ION, ... | 著者 | Wei, H, Ruthenburg, A.J, Bechis, S.K, Verdine, G.L. | 登録日 | 2005-06-08 | 公開日 | 2005-08-23 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Nucleotide-dependent Domain Movement in the ATPase Domain of a Human Type IIA DNA Topoisomerase. J.Biol.Chem., 280, 2005
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1Y8N
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![BU of 1y8n by Molmil](/molmil-images/mine/1y8n) | Crystal structure of the PDK3-L2 complex | 分子名称: | DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, POTASSIUM ION, ... | 著者 | Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T. | 登録日 | 2004-12-13 | 公開日 | 2005-05-24 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex. Embo J., 24, 2005
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1Y8O
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![BU of 1y8o by Molmil](/molmil-images/mine/1y8o) | Crystal structure of the PDK3-L2 complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, ... | 著者 | Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T. | 登録日 | 2004-12-13 | 公開日 | 2005-05-24 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.48 Å) | 主引用文献 | Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex. Embo J., 24, 2005
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1ZXN
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![BU of 1zxn by Molmil](/molmil-images/mine/1zxn) | Human DNA topoisomerase IIa ATPase/ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, DNA topoisomerase II, alpha isozyme, ... | 著者 | Wei, H, Ruthenburg, A.J, Bechis, S.K, Verdine, G.L. | 登録日 | 2005-06-08 | 公開日 | 2005-08-23 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Nucleotide-dependent Domain Movement in the ATPase Domain of a Human Type IIA DNA Topoisomerase. J.Biol.Chem., 280, 2005
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7ZBG
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![BU of 7zbg by Molmil](/molmil-images/mine/7zbg) | Human Topoisomerase II Beta ATPase ADP | 分子名称: | 4-[(2S,3R)-3-[3,5-bis(oxidanylidene)piperazin-1-ium-1-yl]butan-2-yl]piperazin-4-ium-2,6-dione, ADENOSINE-5'-DIPHOSPHATE, DNA topoisomerase 2-beta, ... | 著者 | Ling, E.M, Basle, A, Cowell, I.G, Blower, T.R, Austin, C.A. | 登録日 | 2022-03-23 | 公開日 | 2022-05-25 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | A comprehensive structural analysis of the ATPase domain of human DNA topoisomerase II beta bound to AMPPNP, ADP, and the bisdioxopiperazine, ICRF193. Structure, 30, 2022
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7Z9G
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![BU of 7z9g by Molmil](/molmil-images/mine/7z9g) | E.coli gyrase holocomplex with 217 bp DNA and Albi-2 | 分子名称: | 4-[[3-(2-azanylethoxy)-2-oxidanyl-4-[[5-[[(2~{S})-2-[[4-[(6-oxidanylnaphthalen-2-yl)carbonylamino]phenyl]carbonylamino]-3-(1~{H}-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]phenyl]carbonylamino]-3-methoxy-2-oxidanyl-benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ... | 著者 | Ghilarov, D, Heddle, J.G.H. | 登録日 | 2022-03-21 | 公開日 | 2023-02-15 | 最終更新日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.25 Å) | 主引用文献 | Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin. Nat Catal, 6, 2023
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7Z9M
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![BU of 7z9m by Molmil](/molmil-images/mine/7z9m) | E.coli gyrase holocomplex with 217 bp DNA and Albi-1 (site AA) | 分子名称: | 4-[[4-[[5-[[(2S)-2-[[5-[(4-cyanophenyl)carbonylamino]pyridin-2-yl]carbonylamino]-3-(1H-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]-2-oxidanyl-3-propan-2-yloxy-phenyl]carbonylamino]benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ... | 著者 | Ghilarov, D, Heddle, J.G.H. | 登録日 | 2022-03-21 | 公開日 | 2023-02-15 | 最終更新日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin. Nat Catal, 6, 2023
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7Z9C
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![BU of 7z9c by Molmil](/molmil-images/mine/7z9c) | E.coli gyrase holocomplex with 217 bp DNA and albicidin | 分子名称: | DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), DNA (5'-D(P*AP*AP*AP*TP*CP*TP*GP*TP*GP*CP*GP*GP*GP*T)-3'), ... | 著者 | Ghilarov, D, Heddle, J.G.H, Suessmuth, R. | 登録日 | 2022-03-21 | 公開日 | 2023-02-15 | 最終更新日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.06 Å) | 主引用文献 | Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin. Nat Catal, 6, 2023
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7Z9K
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![BU of 7z9k by Molmil](/molmil-images/mine/7z9k) | E.coli gyrase holocomplex with 217 bp DNA and Albi-1 (site TG) | 分子名称: | 4-[[4-[[5-[[(2S)-2-[[5-[(4-cyanophenyl)carbonylamino]pyridin-2-yl]carbonylamino]-3-(1H-1,2,3-triazol-4-yl)propanoyl]amino]pyridin-2-yl]carbonylamino]-2-oxidanyl-3-propan-2-yloxy-phenyl]carbonylamino]benzoic acid, DNA (5'-D(*AP*AP*TP*CP*AP*CP*CP*CP*GP*CP*AP*CP*AP*GP*AP*TP*TP*T)-3'), DNA (5'-D(*GP*AP*TP*TP*TP*TP*AP*TP*GP*CP*CP*TP*GP*AP*TP*TP*CP*T)-3'), ... | 著者 | Ghilarov, D, Heddle, J.G.H. | 登録日 | 2022-03-21 | 公開日 | 2023-03-08 | 最終更新日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.25 Å) | 主引用文献 | Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin. Nat Catal, 6, 2023
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7YQ8
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![BU of 7yq8 by Molmil](/molmil-images/mine/7yq8) | Cryo-EM structure of human topoisomerase II beta in complex with DNA and etoposide | 分子名称: | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol -5-yl 4,6-O-[(1R)-ethylidene]-beta-D-glucopyranoside, 50-mer DNA, DNA topoisomerase 2-beta, ... | 著者 | Naganuma, M, Ehara, H, Kim, D, Nakagawa, R, Cong, A, Bu, H, Jeong, J, Jang, J, Schellenberg, M.J, Bunch, H, Sekine, S. | 登録日 | 2022-08-05 | 公開日 | 2024-01-03 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | ERK2-topoisomerase II regulatory axis is important for gene activation in immediate early genes. Nat Commun, 14, 2023
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7ZP0
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![BU of 7zp0 by Molmil](/molmil-images/mine/7zp0) | |
8A3U
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![BU of 8a3u by Molmil](/molmil-images/mine/8a3u) | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (symmetrical variant, trigonal form with short c-axis) | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, FLAVIN MONONUCLEOTIDE, Putative Sensory box protein,Sensor protein FixL | 著者 | Arinkin, V, Batra-Safferling, R, Granzin, J. | 登録日 | 2022-06-09 | 公開日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (symmetrical variant, trigonal form
with short c-axis) To Be Published
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8A52
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![BU of 8a52 by Molmil](/molmil-images/mine/8a52) | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (asymmetrical variant, trigonal form with long c-axis) | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, FLAVIN MONONUCLEOTIDE, Putative Sensory box protein,Putative Sensory box protein,Sensor protein FixL | 著者 | Batra-Safferling, R, Arinkin, V, Granzin, J. | 登録日 | 2022-06-14 | 公開日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.461 Å) | 主引用文献 | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (asymmetrical variant, trigonal form with long c axis) To Be Published
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8A6X
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![BU of 8a6x by Molmil](/molmil-images/mine/8a6x) | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (asymmetrical variant, trigonal form with long c axis) | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, FLAVIN MONONUCLEOTIDE, Putative Sensory box protein,Sensor protein FixL | 著者 | Arinkin, V, Granzin, J, Batra-Safferling, R. | 登録日 | 2022-06-20 | 公開日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of a chimeric LOV-Histidine kinase SB2F1 (asymmetrical variant, trigonal form with long c axis) To Be Published
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8A7F
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![BU of 8a7f by Molmil](/molmil-images/mine/8a7f) | Crystal structure of a chimeric LOV-Histidine kinase SB2F1-I66R mutant (asymmetrical variant, trigonal form with long c axis) | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, FLAVIN MONONUCLEOTIDE, Putative Sensory box protein,Sensor protein FixL | 著者 | Batra-Safferling, R, Arinkin, V, Granzin, J. | 登録日 | 2022-06-21 | 公開日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.71 Å) | 主引用文献 | Crystal structure of a chimeric LOV-Histidine kinase SB2F1-I66R mutant (asymmetrical variant, trigonal form with long c axis) To Be Published
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8A7H
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![BU of 8a7h by Molmil](/molmil-images/mine/8a7h) | Crystal structure of a chimeric LOV-Histidine kinase SB2F1-I66R mutant (light state; asymmetrical variant, trigonal form with long c axis) | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Flavin mononucleotide (semi-quinone intermediate), Putative Sensory box protein,Sensor protein FixL | 著者 | Arinkin, V, Granzin, J, Batra-Safferling, R. | 登録日 | 2022-06-21 | 公開日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.145 Å) | 主引用文献 | Crystal structure of a chimeric LOV-Histidine kinase SB2F1-I66R mutant (light state; asymmetrical variant, trigonal form with long c axis) To Be Published
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