8JG2
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![BU of 8jg2 by Molmil](/molmil-images/mine/8jg2) | |
8JF5
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![BU of 8jf5 by Molmil](/molmil-images/mine/8jf5) | Crystal structure of Lysine Specific Demethylase 1 (LSD1) with TAS1440 | 分子名称: | 4-[5-[(3~{R})-3-azanylpyrrolidin-1-yl]carbonyl-2-[2-fluoranyl-4-(2-methyl-2-oxidanyl-propyl)phenyl]phenyl]-2-fluoranyl-benzenecarbonitrile, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ... | 著者 | Fukushima, H, Machida, T, Yamashita, S, Suzuki, T. | 登録日 | 2023-05-17 | 公開日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | TAS1440, a histone H3 competitive LSD1 inhibitor, activates both TGF-beta and notch signaling pathways via INSM1 dissociation in neuroendocrine small cell lung cancer To Be Published
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8JE4
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![BU of 8je4 by Molmil](/molmil-images/mine/8je4) | Crystal structure of LimF prenyltransferase (H239G/W273T mutant) bound with the thiodiphosphate moiety of farnesyl S-thiolodiphosphate (FSPP) | 分子名称: | MAGNESIUM ION, TRIHYDROGEN THIODIPHOSPHATE, prenyltransferase, ... | 著者 | Hamada, K, Oguni, A, Zhang, Y, Satake, M, Goto, Y, Suga, H, Ogata, K, Sengoku, T. | 登録日 | 2023-05-15 | 公開日 | 2023-11-08 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Switching Prenyl Donor Specificities of Cyanobactin Prenyltransferases. J.Am.Chem.Soc., 145, 2023
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8JCD
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![BU of 8jcd by Molmil](/molmil-images/mine/8jcd) | |
8JCC
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![BU of 8jcc by Molmil](/molmil-images/mine/8jcc) | |
8JC4
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![BU of 8jc4 by Molmil](/molmil-images/mine/8jc4) | Crystal structure of the P450 BM3 heme domain mutant F87A-T268V in complex with Pyd-Pid-Phe and hydroxylamine | 分子名称: | 1-pyridin-4-ylpiperidine-4-carboxylic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, HYDROXYAMINE, ... | 著者 | Jiang, Y, Dong, S, Feng, Y, Cong, Z. | 登録日 | 2023-05-10 | 公開日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.64 Å) | 主引用文献 | C(sp3)-H hydroxylation of Broad-Spectrum Alkanes Catalyzed by an Artificial P450 Peroxygenase Driven by omega-Pyridyl Fatty Acyl Amino Acids. Mol Catal, 550, 2023
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8JC3
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![BU of 8jc3 by Molmil](/molmil-images/mine/8jc3) | Crystal structure of the P450 BM3 heme domain mutant F87A-T268V in complex with Pyd-N-C4-Phe and hydroxylamine | 分子名称: | 4-(pyridin-4-ylamino)butanoic acid, Bifunctional cytochrome P450/NADPH--P450 reductase, HYDROXYAMINE, ... | 著者 | Jiang, Y, Dong, S, Feng, Y, Cong, Z. | 登録日 | 2023-05-10 | 公開日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | C(sp3)-H hydroxylation of Broad-Spectrum Alkanes Catalyzed by an Artificial P450 Peroxygenase Driven by omega-Pyridyl Fatty Acyl Amino Acids. Mol Catal, 550, 2023
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8JBX
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![BU of 8jbx by Molmil](/molmil-images/mine/8jbx) | |
8JA6
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![BU of 8ja6 by Molmil](/molmil-images/mine/8ja6) | |
8J71
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![BU of 8j71 by Molmil](/molmil-images/mine/8j71) | |
8J70
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![BU of 8j70 by Molmil](/molmil-images/mine/8j70) | Native SAND domain of protein SP140 with DNA | 分子名称: | DNA (5'-D(*GP*GP*GP*CP*GP*GP*CP*CP*GP*CP*CP*CP*T)-3'), Nuclear body protein SP140, selenourea | 著者 | Li, H.T, Liu, W.Q. | 登録日 | 2023-04-26 | 公開日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Molecular basis for Speckled protein SP140 bivalent recognition of histone H3 and DNA. To Be Published
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8J6T
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![BU of 8j6t by Molmil](/molmil-images/mine/8j6t) | Cryo-EM structure of the double CAF-1 bound right-handed Di-tetrasome | 分子名称: | Chromatin assembly factor 1 subunit A, Chromatin assembly factor 1 subunit B, Histone H3.1, ... | 著者 | Liu, C.P, Yu, Z.Y, Xu, R.M. | 登録日 | 2023-04-26 | 公開日 | 2023-08-16 | 最終更新日 | 2023-09-06 | 実験手法 | ELECTRON MICROSCOPY (6.6 Å) | 主引用文献 | Structural insights into histone binding and nucleosome assembly by chromatin assembly factor-1. Science, 381, 2023
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8J6S
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![BU of 8j6s by Molmil](/molmil-images/mine/8j6s) | Cryo-EM structure of the single CAF-1 bound right-handed Di-tetrasome | 分子名称: | Chromatin assembly factor 1 subunit A, Chromatin assembly factor 1 subunit B, Histone H3.1, ... | 著者 | Liu, C.P, Yu, Z.Y, Xu, R.M. | 登録日 | 2023-04-26 | 公開日 | 2023-08-16 | 最終更新日 | 2023-09-06 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Structural insights into histone binding and nucleosome assembly by chromatin assembly factor-1. Science, 381, 2023
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8J5M
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![BU of 8j5m by Molmil](/molmil-images/mine/8j5m) | |
8J4L
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![BU of 8j4l by Molmil](/molmil-images/mine/8j4l) | |
8J24
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![BU of 8j24 by Molmil](/molmil-images/mine/8j24) | Cryo-EM structure of FFAR2 complex bound with acetic acid | 分子名称: | ACETATE ION, Free fatty acid receptor 2, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Tai, L, Li, F, Tang, W, Sun, X, Wang, J. | 登録日 | 2023-04-14 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-10 | 実験手法 | ELECTRON MICROSCOPY (2.6 Å) | 主引用文献 | Molecular recognition and activation mechanism of short-chain fatty acid receptors FFAR2/3. Cell Res., 34, 2024
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8J0H
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![BU of 8j0h by Molmil](/molmil-images/mine/8j0h) | |
8J07
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![BU of 8j07 by Molmil](/molmil-images/mine/8j07) | |
8IYJ
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![BU of 8iyj by Molmil](/molmil-images/mine/8iyj) | Cryo-EM structure of the 48-nm repeat doublet microtubule from mouse sperm | 分子名称: | Cilia and flagella-associated protein 77, Cilia- and flagella-associated protein 107, Cilia- and flagella-associated protein 141, ... | 著者 | Zhou, L.N, Gui, M, Wu, J.P. | 登録日 | 2023-04-05 | 公開日 | 2023-07-05 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structures of sperm flagellar doublet microtubules expand the genetic spectrum of male infertility. Cell, 186, 2023
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8IYC
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![BU of 8iyc by Molmil](/molmil-images/mine/8iyc) | Structure insight into substrate recognition and catalysis by feruloyl esterase from Aspergillus sydowii | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETATE ION, ... | 著者 | Phienluphon, A, Kondo, K, Mikami, B, Nagata, T, Katahira, M. | 登録日 | 2023-04-04 | 公開日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural insights into the molecular mechanisms of substrate recognition and hydrolysis by feruloyl esterase from Aspergillus sydowii. Int.J.Biol.Macromol., 253, 2023
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8IYB
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![BU of 8iyb by Molmil](/molmil-images/mine/8iyb) | Structure insight into substrate recognition and catalysis by feruloyl esterase from Aspergillus sydowii | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-(4-HYDROXY-3-METHOXYPHENYL)-2-PROPENOIC ACID, ... | 著者 | Phienluphon, A, Kondo, K, Mikami, B, Nagata, T, Katahira, M. | 登録日 | 2023-04-04 | 公開日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural insights into the molecular mechanisms of substrate recognition and hydrolysis by feruloyl esterase from Aspergillus sydowii. Int.J.Biol.Macromol., 253, 2023
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8IYA
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![BU of 8iya by Molmil](/molmil-images/mine/8iya) | |
8IY8
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![BU of 8iy8 by Molmil](/molmil-images/mine/8iy8) | Structure insight into substrate recognition and catalysis by feruloyl esterase from Aspergillus sydowii | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETATE ION, Feruloyl esterase | 著者 | Phienluphon, A, Kondo, K, Mikami, B, Nagata, T, Katahira, M. | 登録日 | 2023-04-04 | 公開日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural insights into the molecular mechanisms of substrate recognition and hydrolysis by feruloyl esterase from Aspergillus sydowii. Int.J.Biol.Macromol., 253, 2023
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8ITV
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![BU of 8itv by Molmil](/molmil-images/mine/8itv) | KL2.1 in complex with CRM1-Ran-RanBP1 | 分子名称: | (3~{S},5~{R},6~{E},8~{Z},10~{R},12~{E},14~{E},16~{S})-3,16-bis(azanyl)-8,10,12-trimethyl-16-[(2~{S},4~{R},5~{S},6~{S})-5-methyl-4-oxidanyl-6-[(~{E})-prop-1-enyl]oxan-2-yl]-5-oxidanyl-hexadeca-6,8,12,14-tetraenoic acid, ACETATE ION, CHLORIDE ION, ... | 著者 | Sun, Q, Jian, L. | 登録日 | 2023-03-23 | 公開日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | KL2.1 in complex with CRM1-Ran-RanBP1 To Be Published
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8IS4
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![BU of 8is4 by Molmil](/molmil-images/mine/8is4) | Structure of an Isocytosine specific deaminase Vcz in complexed with 5-FU | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 5-FLUOROURACIL, GLYCEROL, ... | 著者 | Guo, W.T, Li, X.J, Wu, B.X. | 登録日 | 2023-03-20 | 公開日 | 2023-08-30 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural characterization of an isocytosine-specific deaminase VCZ reveals its application potential in the anti-cancer therapy. Iscience, 26, 2023
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