8TDE
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8TDD
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8TDC
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![BU of 8tdc by Molmil](/molmil-images/mine/8tdc) | Structure of PYCR1 complexed with NADH and 1,3-dithiane-2-carboxylic acid | 分子名称: | 1,3-dithiane-2-carboxylic acid, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Pyrroline-5-carboxylate reductase 1, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Screening a knowledge-based library of low molecular weight compounds against the proline biosynthetic enzyme 1-pyrroline-5-carboxylate 1 (PYCR1) Protein Sci., 33, 2024
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8TDB
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8TDA
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8TD9
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![BU of 8td9 by Molmil](/molmil-images/mine/8td9) | Structure of PYCR1 complexed with NADH and L-pipecolic acid | 分子名称: | (2S)-piperidine-2-carboxylic acid, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Pyrroline-5-carboxylate reductase 1, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Screening a knowledge-based library of low molecular weight compounds against the proline biosynthetic enzyme 1-pyrroline-5-carboxylate 1 (PYCR1) Protein Sci., 33, 2024
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8TD8
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![BU of 8td8 by Molmil](/molmil-images/mine/8td8) | Structure of PYCR1 complexed with NADH and 2S-Hydroxy-3,3-dimethylbutyric acid | 分子名称: | (2S)-2-hydroxy-3,3-dimethylbutanoic acid, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Pyrroline-5-carboxylate reductase 1, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Screening a knowledge-based library of low molecular weight compounds against the proline biosynthetic enzyme 1-pyrroline-5-carboxylate 1 (PYCR1) Protein Sci., 33, 2024
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8TD7
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8TD6
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![BU of 8td6 by Molmil](/molmil-images/mine/8td6) | |
8TD5
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8TD4
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![BU of 8td4 by Molmil](/molmil-images/mine/8td4) | Structure of PYCR1 complexed with NADH and 1,3-Dithiolane-2-carboxylic acid | 分子名称: | 1,3-dithiolane-2-carboxylic acid, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Pyrroline-5-carboxylate reductase 1, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Screening a knowledge-based library of low molecular weight compounds against the proline biosynthetic enzyme 1-pyrroline-5-carboxylate 1 (PYCR1) Protein Sci., 33, 2024
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8TD3
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8TD2
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![BU of 8td2 by Molmil](/molmil-images/mine/8td2) | Structure of PYCR1 complexed with NADH and cyclobutane-1,1-dicarboxylic acid | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Screening a knowledge-based library of low molecular weight compounds against the proline biosynthetic enzyme 1-pyrroline-5-carboxylate 1 (PYCR1) Protein Sci., 33, 2024
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8TD1
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8TD0
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![BU of 8td0 by Molmil](/molmil-images/mine/8td0) | Structure of PYCR1 complexed with 5-oxo-7a-phenyl-hexahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylic acid | 分子名称: | (3R,4S,7aR)-5-oxo-7a-phenylhexahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-03-06 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCZ
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8TCY
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![BU of 8tcy by Molmil](/molmil-images/mine/8tcy) | Structure of PYCR1 complexed with 7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid | 分子名称: | 7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid, DI(HYDROXYETHYL)ETHER, Pyrroline-5-carboxylate reductase 1, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-03-06 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCX
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![BU of 8tcx by Molmil](/molmil-images/mine/8tcx) | Structure of PYCR1 complexed with 2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carboxylic acid | 分子名称: | 2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-03-06 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCW
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8TCV
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![BU of 8tcv by Molmil](/molmil-images/mine/8tcv) | Structure of PYCR1 complexed with 4-bromobenzene-1,3-dicarboxylic acid | 分子名称: | 4-bromobenzene-1,3-dicarboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | 著者 | Tanner, J.J, Meeks, K.R. | 登録日 | 2023-07-02 | 公開日 | 2024-03-06 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCU
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8TCT
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![BU of 8tct by Molmil](/molmil-images/mine/8tct) | Structure of 3K-GlcH bound Bacteroides thetaiotaomicron 3-Keto-beta-glucopyranoside-1,2-Lyase BT1 | 分子名称: | 1,5-anhydro-D-ribo-hex-3-ulose, COBALT (II) ION, PHOSPHATE ION, ... | 著者 | Lazarski, A.C, Worrall, L.J, Strynadka, N.C.J. | 登録日 | 2023-07-02 | 公開日 | 2024-06-12 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | An alternative broad-specificity pathway for glycan breakdown in bacteria. Nature, 631, 2024
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8TCS
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![BU of 8tcs by Molmil](/molmil-images/mine/8tcs) | Structure of trehalose bound Alistipes sp. 3-Keto-beta-glucopyranoside-1,2-Lyase AL1 | 分子名称: | ACETATE ION, COBALT (II) ION, Xylose isomerase-like TIM barrel domain-containing protein, ... | 著者 | Lazarski, A.C, Worrall, L.J, Strynadka, N.C.J. | 登録日 | 2023-07-02 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | An alternative broad-specificity pathway for glycan breakdown in bacteria. Nature, 631, 2024
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8TCR
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![BU of 8tcr by Molmil](/molmil-images/mine/8tcr) | Structure of glucose bound Alistipes sp. 3-Keto-beta-glucopyranoside-1,2-Lyase AL1 | 分子名称: | COBALT (II) ION, MALONATE ION, Sugar phosphate isomerase, ... | 著者 | Lazarski, A.C, Worrall, L.J, Strynadka, N.C.J. | 登録日 | 2023-07-02 | 公開日 | 2024-06-12 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | An alternative broad-specificity pathway for glycan breakdown in bacteria. Nature, 631, 2024
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8TCO
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