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9ESM
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Archaellum filament from the Halobacterium salinarum deltaAgl26 strain
分子名称: Archaellin, beta-D-glucopyranuronic acid-(1-4)-beta-D-glucopyranose
著者Grosmann-Haham, I, Shahar, A.
登録日2024-03-26
公開日2024-07-17
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.06 Å)
主引用文献Perturbed N-glycosylation of Halobacterium salinarum archaellum filaments leads to filament bundling and compromised cell motility.
Nat Commun, 15, 2024
8ZHJ
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BU of 8zhj by Molmil
SARS-CoV-2 spike trimer (6P) in complex with three H18 Fabs, head-to-head aggregate (C1 symmetry)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Heavy chain of H18 Fab, ...
著者Yan, Q, Gao, X, Liu, B, Hou, R, He, P, Li, Z, Chen, Q, Wang, J, He, J, Chen, L, Zhao, J, Xiong, X.
登録日2024-05-11
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (8.45 Å)
主引用文献Antibodies utilizing VL6-57 light chains target a convergent cryptic epitope on SARS-CoV-2 spike protein helping to drive the genesis of Omicron variants
To Be Published
9FWG
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BU of 9fwg by Molmil
LSD1/CoREST bound to bomedemstat
分子名称: Bomedemstat FAD adduct, Lysine-specific histone demethylase 1A, REST corepressor 1
著者Speranzini, V, Mattevi, A.
登録日2024-06-30
公開日2024-07-10
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Characterization of structural, biochemical, pharmacokinetic, and pharmacodynamic properties of the LSD1 inhibitor bomedemstat in preclinical models.
Prostate, 84, 2024
9FX5
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BU of 9fx5 by Molmil
Crystal structure of Cryo2RT Thaumatin at 296K
分子名称: L(+)-TARTARIC ACID, Thaumatin I
著者Huang, C.Y, Aumonier, S, Olieric, V, Wang, M.
登録日2024-07-01
公開日2024-07-31
最終更新日2024-08-14
実験手法X-RAY DIFFRACTION (1.592 Å)
主引用文献Cryo2RT: a high-throughput method for room-temperature macromolecular crystallography from cryo-cooled crystals.
Acta Crystallogr D Struct Biol, 80, 2024
9ETU
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BU of 9etu by Molmil
Archaellum filament from the Halobacterium salinarum deltaAgl27 strain
分子名称: 3-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-beta-D-glucopyranuronic acid-(1-4)-beta-D-glucopyranose, Archaellin
著者Grossman-Haham, I, Shahar, A.
登録日2024-03-27
公開日2024-07-17
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.33 Å)
主引用文献Perturbed N-glycosylation of Halobacterium salinarum archaellum filaments leads to filament bundling and compromised cell motility.
Nat Commun, 15, 2024
8ZHF
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BU of 8zhf by Molmil
SARS-CoV-2 spike trimer (6P) in complex with R1-26 Fab, head-to-head aggregate
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Heavy chain of R1-26 Fab, ...
著者Yan, Q, Gao, X, Liu, B, Hou, R, He, P, Li, Z, Chen, Q, Wang, J, He, J, Chen, L, Zhao, J, Xiong, X.
登録日2024-05-10
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (5.26 Å)
主引用文献Antibodies utilizing VL6-57 light chains target a convergent cryptic epitope on SARS-CoV-2 spike protein helping to drive the genesis of Omicron variants
To Be Published
9BEW
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BU of 9bew by Molmil
Cryo-EM structure of the HIV-1 BG505 IDL Env trimer in complex with 3BNC117 and 10-1074 Fabs
分子名称: 10-1074 heavy chain, 10-1074 light chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Gorman, J, Kwong, P.D.
登録日2024-04-16
公開日2024-07-31
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Design of soluble HIV-1 envelope trimers free of covalent gp120-gp41 bonds with prevalent native-like conformation.
Cell Rep, 43, 2024
9F3W
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BU of 9f3w by Molmil
CutC choline lyase in complex with fluoromethylcholine
分子名称: Choline trimethylamine-lyase, fluoromethylcholine
著者Kalnins, G.
登録日2024-04-26
公開日2024-05-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献CutC choline lyase in complex with fluoromethylcholine
To Be Published
7QZJ
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BU of 7qzj by Molmil
1.55 A X-ray crystallographic structure of SapH from Streptomyces sp. (HPH0547) involved in Pseudouridimycin biosynthesis
分子名称: 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, Aspartate aminotransferase family protein, GLYCEROL, ...
著者Schnell, R, Schneider, G.
登録日2022-01-31
公開日2023-02-15
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Pseudouridine-Modifying Enzymes SapB and SapH Control Entry into the Pseudouridimycin Biosynthetic Pathway.
Acs Chem.Biol., 18, 2023
9G48
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BU of 9g48 by Molmil
Staphylococcus aureus MazF in complex with Nanobody 6
分子名称: 2-(2-METHOXYETHOXY)ETHANOL, CADMIUM ION, Endoribonuclease MazF, ...
著者Zorzini, V, Haesaerts, S, Loris, R.
登録日2024-07-15
公開日2024-07-24
実験手法X-RAY DIFFRACTION (2.143536 Å)
主引用文献Nanobody-mediated activation and inhibition of Staphylococcus aureus MazF
To Be Published
9CKV
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BU of 9ckv by Molmil
Cryo-EM structure of alpha5beta1 integrin in complex with NeoNectin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Werther, R, Nguyen, A, Estrada Alamo, K.A, Wang, X, Campbell, M.G.
登録日2024-07-09
公開日2024-07-17
実験手法ELECTRON MICROSCOPY (3.19 Å)
主引用文献De Novo Design of Integrin alpha5beta1 Modulating Proteins for Regenerative Medicine
To Be Published
9FX4
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BU of 9fx4 by Molmil
Crystal structure of Cryo2RT Thaumatin at 100K
分子名称: L(+)-TARTARIC ACID, Thaumatin I
著者Huang, C.Y, Aumonier, S, Olieric, V, Wang, M.
登録日2024-07-01
公開日2024-07-31
最終更新日2024-08-14
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Cryo2RT: a high-throughput method for room-temperature macromolecular crystallography from cryo-cooled crystals.
Acta Crystallogr D Struct Biol, 80, 2024
8ZHK
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BU of 8zhk by Molmil
SARS-CoV-2 spike trimer (6P) in complex with three H18 Fabs, head-to-head aggregate (C3 symmetry)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Heavy chain of H18 Fab, ...
著者Yan, Q, Gao, X, Liu, B, Hou, R, He, P, Li, Z, Chen, Q, Wang, J, He, J, Chen, L, Zhao, J, Xiong, X.
登録日2024-05-11
公開日2024-08-21
実験手法ELECTRON MICROSCOPY (6.3 Å)
主引用文献Antibodies utilizing VL6-57 light chains target a convergent cryptic epitope on SARS-CoV-2 spike protein helping to drive the genesis of Omicron variants
To Be Published
8CHH
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BU of 8chh by Molmil
SH3 domain solved by the exact solid-state method from the Bruker Dynamics Center using the correction method for spin-diffusion with PDB 2NUZ as reference
分子名称: Spectrin alpha chain, non-erythrocytic 1
著者Soeldner, B.
登録日2023-02-08
公開日2023-03-08
最終更新日2024-06-19
実験手法SOLID-STATE NMR
主引用文献Integrated Assessment of the Structure and Dynamics of Solid Proteins.
J Phys Chem Lett, 14, 2023
9F3Y
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BU of 9f3y by Molmil
CutC choline lyase in complex with difluorocholine
分子名称: Choline trimethylamine-lyase, difluorocholine
著者Kalnins, G.
登録日2024-04-26
公開日2024-05-08
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献CutC choline lyase in complex with difluorocholine
To Be Published
8ZM1
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BU of 8zm1 by Molmil
Structure of human pyruvate dehydrogenase kinase 2 complexed with compound 6
分子名称: (5~{R})-5-propan-2-ylindeno[1,2-b]pyridin-5-ol, [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial
著者Akai, S, Orita, T, Nomura, A, Adachi, T.
登録日2024-05-22
公開日2024-06-19
最終更新日2024-07-03
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase.
Bioorg.Med.Chem.Lett., 109, 2024
9EQ7
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BU of 9eq7 by Molmil
Halobacterium salinarum archaellum filament
分子名称: 2-O-sulfo-beta-D-glucopyranuronic acid-(1-4)-3-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-beta-D-glucopyranuronic acid-(1-4)-beta-D-glucopyranose, Archaellin
著者Grossman-Haham, I, Shahar, A.
登録日2024-03-21
公開日2024-07-17
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.23 Å)
主引用文献Perturbed N-glycosylation of Halobacterium salinarum archaellum filaments leads to filament bundling and compromised cell motility.
Nat Commun, 15, 2024
8C3N
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BU of 8c3n by Molmil
Stapled peptide SP30 in complex with humanised RadA mutant HumRadA22
分子名称: 4,6-diethylpyrimidin-2-amine, ADENOSINE-5'-DIPHOSPHATE, Breast cancer type 2 susceptibility protein, ...
著者Pantelejevs, T, Hyvonen, M.
登録日2022-12-27
公開日2023-03-08
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献A recombinant approach for stapled peptide discovery yields inhibitors of the RAD51 recombinase.
Chem Sci, 14, 2023
9BVS
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BU of 9bvs by Molmil
NMR structure of TLP-1 in solution
分子名称: Temporin-1Tl
著者Jia, R, McShan, A.C.
登録日2024-05-20
公開日2024-06-05
実験手法SOLUTION NMR
主引用文献Design and Development of Temporin L Analogues to Inhibit the Main Protease of SARS-CoV-2
To Be Published
8CF4
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BU of 8cf4 by Molmil
SH3 domain solved by the exact solid-state method from the Bruker Dynamics Center using the combined correction method with PDB 2NUZ
分子名称: Spectrin alpha chain, non-erythrocytic 1
著者Soeldner, B.
登録日2023-02-02
公開日2023-03-08
最終更新日2024-06-19
実験手法SOLID-STATE NMR
主引用文献Integrated Assessment of the Structure and Dynamics of Solid Proteins.
J Phys Chem Lett, 14, 2023
8CHG
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BU of 8chg by Molmil
SH3 domain solved by the exact solid-state method from the Bruker Dynamics Center using the correction for dipolar truncation with PDB 2NUZ
分子名称: Spectrin alpha chain, non-erythrocytic 1
著者Soeldner, B.
登録日2023-02-08
公開日2023-03-08
最終更新日2024-06-19
実験手法SOLID-STATE NMR
主引用文献Integrated Assessment of the Structure and Dynamics of Solid Proteins.
J Phys Chem Lett, 14, 2023
9FTW
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BU of 9ftw by Molmil
Crystal structure of calcium-activated EndoU
分子名称: 1,2-ETHANEDIOL, ACETATE ION, CALCIUM ION, ...
著者Fribourg, S, Campagne, S.
登録日2024-06-25
公開日2024-08-14
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Molecular Basis for the Calcium-Dependent Activation of the Ribonuclease EndoU.
Res Sq, 2024
9BRD
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BU of 9brd by Molmil
Synaptic Vesicle V-ATPase with synaptophysin and SidK, State 3
分子名称: (7R)-4,7-DIHYDROXY-N,N,N-TRIMETHYL-10-OXO-3,5,9-TRIOXA-4-PHOSPHAHEPTACOSAN-1-AMINIUM 4-OXIDE, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Coupland, C.E, Rubinstein, J.L.
登録日2024-05-11
公開日2024-06-26
最終更新日2024-07-24
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献High-resolution electron cryomicroscopy of V-ATPase in native synaptic vesicles.
Science, 385, 2024
9F3X
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BU of 9f3x by Molmil
CutC choline lyase in complex with cyclopropylcholine
分子名称: Choline trimethylamine-lyase, cyclopropylcholine
著者Kalnins, G.
登録日2024-04-26
公開日2024-05-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献CutC choline lyase in complex with fluoromethylcholine
To Be Published
9G4G
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BU of 9g4g by Molmil
Staphylococcus aureus MazF in complex with Nanobody 9
分子名称: Endoribonuclease MazF, Nanobody 9, SULFATE ION
著者Zorzini, V, Haesaerts, S, Loris, R.
登録日2024-07-15
公開日2024-07-24
実験手法X-RAY DIFFRACTION (2.8957293 Å)
主引用文献Nanobody-mediated activation and inhibition of Staphylococcus aureus MazF
To Be Published

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件を2024-08-28に公開中

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