6AP9
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![BU of 6ap9 by Molmil](/molmil-images/mine/6ap9) | |
8SC9
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![BU of 8sc9 by Molmil](/molmil-images/mine/8sc9) | Structure of PPARG in complex with MTX-531 | 分子名称: | N-[(5P)-2-chloro-5-(4-{[(1R)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide, Peroxisome proliferator-activated receptor gamma, SULFATE ION, ... | 著者 | Whitehead, C.E, Leopold, J. | 登録日 | 2023-04-05 | 公開日 | 2024-06-12 | 実験手法 | X-RAY DIFFRACTION (1.855 Å) | 主引用文献 | Structure of PPARG in complex with MTX-531 To Be Published
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5FLX
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![BU of 5flx by Molmil](/molmil-images/mine/5flx) | Mammalian 40S HCV-IRES complex | 分子名称: | 18S RRNA, 40S RIBOSOMAL PROTEIN S10, 40S RIBOSOMAL PROTEIN S11, ... | 著者 | Yamamoto, H, Collier, M, Loerke, J, Ismer, J, Schmidt, A, Hilal, T, Sprink, T, Yamamoto, K, Mielke, T, Burger, J, Shaikh, T.R, Dabrowski, M, Hildebrand, P.W, Scheerer, P, Spahn, C.M.T. | 登録日 | 2015-10-28 | 公開日 | 2015-12-23 | 最終更新日 | 2017-08-30 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | Molecular Architecture of the Ribosome-Bound Hepatitis C Virus Internal Ribosomal Entry Site RNA. Embo J., 34, 2015
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6ZMN
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![BU of 6zmn by Molmil](/molmil-images/mine/6zmn) | |
3CGO
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![BU of 3cgo by Molmil](/molmil-images/mine/3cgo) | IRAK-4 Inhibitors (Part II)- A structure based assessment of imidazo[1,2 a]pyridine binding | 分子名称: | 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-N-methylacetamide, Mitogen-activated protein kinase 10 | 著者 | Ceska, T.A, Platt, A, Fortunato, M, Dickson, K.M, Beevers, R. | 登録日 | 2008-03-06 | 公開日 | 2008-06-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | IRAK-4 inhibitors. Part II: A structure-based assessment of imidazo[1,2-a]pyridine binding Bioorg.Med.Chem.Lett., 18, 2008
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7SFT
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![BU of 7sft by Molmil](/molmil-images/mine/7sft) | Filamin complex-2 | 分子名称: | Filamin-A, Integrin alpha-IIb light chain, form 2 | 著者 | Liu, J, Qin, J. | 登録日 | 2021-10-04 | 公開日 | 2023-04-12 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | A mechanism of platelet integrin alpha IIb beta 3 outside-in signaling through a novel integrin alpha IIb subunit-filamin-actin linkage. Blood, 141, 2023
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3ELJ
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![BU of 3elj by Molmil](/molmil-images/mine/3elj) | Jnk1 complexed with a bis-anilino-pyrrolopyrimidine inhibitor. | 分子名称: | 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide, Mitogen-activated protein kinase 8 | 著者 | Chamberlain, S, Atkins, C, Deanda, F, Dumble, M, Gerding, R, Groy, A, Korenchuk, S, Kumar, R, Lei, H, Mook, R, Moorthy, G, Redman, A, Rowland, J, Shewchuk, L, Vicentini, G, Mosley, J. | 登録日 | 2008-09-22 | 公開日 | 2008-12-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Optimization of 4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine IGF-1R tyrosine kinase inhibitors towards JNK selectivity. Bioorg.Med.Chem.Lett., 19, 2009
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3DD3
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![BU of 3dd3 by Molmil](/molmil-images/mine/3dd3) | |
3CSH
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![BU of 3csh by Molmil](/molmil-images/mine/3csh) | |
3CSJ
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![BU of 3csj by Molmil](/molmil-images/mine/3csj) | Human glutathione s-transferase p1-1 in complex with chlorambucil | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORAMBUCIL, CHLORIDE ION, ... | 著者 | Parker, L.J. | 登録日 | 2008-04-09 | 公開日 | 2008-07-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The anti-cancer drug chlorambucil as a substrate for the human polymorphic enzyme glutathione transferase P1-1: kinetic properties and crystallographic characterisation of allelic variants. J.Mol.Biol., 380, 2008
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3CSI
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![BU of 3csi by Molmil](/molmil-images/mine/3csi) | |
3DGQ
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![BU of 3dgq by Molmil](/molmil-images/mine/3dgq) | |
2MAJ
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![BU of 2maj by Molmil](/molmil-images/mine/2maj) | |
2MAK
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![BU of 2mak by Molmil](/molmil-images/mine/2mak) | |
2OAD
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![BU of 2oad by Molmil](/molmil-images/mine/2oad) | |
2OAC
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![BU of 2oac by Molmil](/molmil-images/mine/2oac) | |
2OA7
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![BU of 2oa7 by Molmil](/molmil-images/mine/2oa7) | |
2PGT
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![BU of 2pgt by Molmil](/molmil-images/mine/2pgt) | CRYSTAL STRUCTURE OF HUMAN GLUTATHIONE S-TRANSFERASE P1-1[V104] COMPLEXED WITH (9R,10R)-9-(S-GLUTATHIONYL)-10-HYDROXY-9,10-DIHYDROPHENANTHRENE | 分子名称: | (9R,10R)-9-(S-GLUTATHIONYL)-10-HYDROXY-9,10-DIHYDROPHENANTHRENE, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLUTATHIONE S-TRANSFERASE, ... | 著者 | Ji, X. | 登録日 | 1997-02-17 | 公開日 | 1997-09-04 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure and function of the xenobiotic substrate-binding site and location of a potential non-substrate-binding site in a class pi glutathione S-transferase. Biochemistry, 36, 1997
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2M6Y
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![BU of 2m6y by Molmil](/molmil-images/mine/2m6y) | The solution structure of the J-domain of human DnaJA1 | 分子名称: | DnaJ homolog subfamily A member 1 | 著者 | Stark, J.L, Mehla, K, Chaika, N, Acton, T.B, Xiao, R, Singh, P.K, Montelione, G.T, Powers, R, Northeast Structural Genomics Consortium (NESG) | 登録日 | 2013-04-14 | 公開日 | 2013-06-26 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure and function of human DnaJ homologue subfamily a member 1 (DNAJA1) and its relationship to pancreatic cancer. Biochemistry, 53, 2014
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6Y1E
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![BU of 6y1e by Molmil](/molmil-images/mine/6y1e) | Crystal structure of human glutathione transferase P1-1 (hGSTP1-1) that was co-crystallised in the presence of indanyloxyacetic acid-94 (IAA-94) | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-[[6,7-bis(chloranyl)-2-cyclopentyl-2-methyl-1-oxidanylidene-3~{H}-inden-5-yl]oxy]ethanoic acid, GLUTATHIONE, ... | 著者 | Pandian, R, Worth, R, Thangaraj, V, Sayed, Y, Dirr, H.W. | 登録日 | 2020-02-12 | 公開日 | 2020-03-11 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.402 Å) | 主引用文献 | The interaction of IAA-94 with the soluble conformation of the CLIC1 protein and its structural homolog hGSTP1-1 To Be Published
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6GSS
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![BU of 6gss by Molmil](/molmil-images/mine/6gss) | |
7GSS
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![BU of 7gss by Molmil](/molmil-images/mine/7gss) | |
7KSJ
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![BU of 7ksj by Molmil](/molmil-images/mine/7ksj) | |
7KSI
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![BU of 7ksi by Molmil](/molmil-images/mine/7ksi) | |
7KSK
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![BU of 7ksk by Molmil](/molmil-images/mine/7ksk) | |