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1C8L
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SYNERGISTIC INHIBITION OF GLYCOGEN PHOSPHORYLASE A BY A POTENTIAL ANTIDIABETIC DRUG AND CAFFEINE
分子名称: 2,3-DICARBOXY-4-(2-CHLORO-PHENYL)-1-ETHYL-5-ISOPROPOXYCARBONYL-6-METHYL-PYRIDINIUM, CAFFEINE, GLYCEROL, ...
著者Tsitsanou, K.E, Skamnaki, V.T, Oikonomakos, N.G.
登録日2000-05-16
公開日2000-05-31
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis of the synergistic inhibition of glycogen phosphorylase a by caffeine and a potential antidiabetic drug.
Arch.Biochem.Biophys., 384, 2000
5FMC
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Structure of D80A-fructofuranosidase from Xanthophyllomyces dendrorhous complexed with fructose and BIS-TRIS propane buffer
分子名称: 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Ramirez-Escudero, M, Sanz-Aparicio, J.
登録日2015-11-02
公開日2016-02-10
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Structural Analysis of Beta-Fructofuranosidase from Xanthophyllomyces Dendrorhous Reveals Unique Features and the Crucial Role of N-Glycosylation in Oligomerization and Activity
J.Biol.Chem., 291, 2016
1C93
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Endo-Beta-N-Acetylglucosaminidase H, D130N/E132Q Double Mutant
分子名称: ENDO-BETA-N-ACETYLGLUCOSAMINIDASE H
著者Rao, V, Cui, T, Guan, C, Van Roey, P.
登録日1999-07-30
公開日1999-11-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Mutations of endo-beta-N-acetylglucosaminidase H active site residues Asp130 and Glu132: activities and conformations.
Protein Sci., 8, 1999
1CDI
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BU of 1cdi by Molmil
STRUCTURES OF AN HIV AND MHC BINDING FRAGMENT FROM HUMAN CD4 AS REFINED IN TWO CRYSTAL LATTICES
分子名称: T CELL SURFACE GLYCOPROTEIN CD4
著者Ryu, S.E, Truneh, A, Sweet, R.W, Hendrickson, W.A.
登録日1994-01-26
公開日1994-04-30
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structures of an HIV and MHC binding fragment from human CD4 as refined in two crystal lattices.
Structure, 2, 1994
1BS3
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P.SHERMANII SOD(FE+3) FLUORIDE
分子名称: FE (III) ION, FLUORIDE ION, SUPEROXIDE DISMUTASE
著者Schmidt, M.
登録日1998-08-31
公開日1999-06-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Manipulating the coordination mumber of the ferric iron within the cambialistic superoxide dismutase of Propionibacterium shermanii by changing the pH-value A crystallographic analysis
Eur.J.Biochem., 262, 1999
7CJI
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Photosystem II structure in the S1 state
分子名称: 1,2-DI-O-ACYL-3-O-[6-DEOXY-6-SULFO-ALPHA-D-GLUCOPYRANOSYL]-SN-GLYCEROL, 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-DISTEAROYL-MONOGALACTOSYL-DIGLYCERIDE, ...
著者Li, H, Shen, J.-R, Suga, M.
登録日2020-07-11
公開日2021-04-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Capturing structural changes of the S 1 to S 2 transition of photosystem II using time-resolved serial femtosecond crystallography.
Iucrj, 8, 2021
5OJT
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Structure-Activity Relationships and Biological Characterization of a Novel, Potent and Serum Stable C-X-C chemokine receptor type 4 (CXCR4) Antagonist
分子名称: ACE-ARG-ALA-(D)CYS-ARG-BNA-HIS-PEN
著者Brancaccio, D, Carotenuto, A.
登録日2017-07-24
公開日2017-11-22
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Structure-Activity Relationships and Biological Characterization of a Novel, Potent, and Serum Stable C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonist.
J. Med. Chem., 60, 2017
7CBM
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Cryo-EM structure of the flagellar distal rod with partial hook from Salmonella
分子名称: Flagellar basal-body rod protein FlgF, Flagellar basal-body rod protein FlgG, Flagellar hook protein FlgE
著者Tan, J.X, Chang, S.H, Wang, X.F, Xu, C.H, Zhou, Y, Zhang, X, Zhu, Y.Q.
登録日2020-06-12
公開日2021-04-28
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structural basis of assembly and torque transmission of the bacterial flagellar motor.
Cell, 184, 2021
7CAV
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Versatile cis-prenyltransferase MM_0014 from Methanosarcina mazei (crystal type: co-FG+DMAPP)
分子名称: 2-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propane-1,3-diol, DIMETHYLALLYL DIPHOSPHATE, DIPHOSPHATE, ...
著者Unno, H, Hemmi, H.
登録日2020-06-10
公開日2021-04-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献A versatile cis-prenyltransferase from Methanosarcina mazei catalyzes both C- and O-prenylations.
J.Biol.Chem., 296, 2021
1BN4
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CARBONIC ANHYDRASE II INHIBITOR
分子名称: CARBONIC ANHYDRASE, MERCURY (II) ION, N-[(4-METHOXYPHENYL)METHYL]2,5-THIOPHENEDESULFONAMIDE, ...
著者Boriack-Sjodin, P.A, Zeitlin, S, Christianson, D.W.
登録日1998-07-31
公開日1999-05-18
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural analysis of inhibitor binding to human carbonic anhydrase II.
Protein Sci., 7, 1998
5GAG
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RNC in complex with SRP-SR in the closed state
分子名称: 1A9L SS, 23S rRNA, 50S ribosomal protein L10, ...
著者Jomaa, A, Boehringer, D, Leibundgut, M, Ban, N.
登録日2015-11-26
公開日2016-01-27
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Structures of the E. coli translating ribosome with SRP and its receptor and with the translocon.
Nat Commun, 7, 2016
1BQM
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BU of 1bqm by Molmil
HIV-1 RT/HBY 097
分子名称: (S)-4-ISOPROPOXYCARBONYL-6-METHOXY-3-METHYLTHIOMETHYL-3,4-DIHYDROQUINOXALIN-2(1H)-THIONE, REVERSE TRANSCRIPTASE
著者Hsiou, Y, Das, K, Ding, J, Arnold, E.
登録日1998-08-17
公開日1999-01-06
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structures of Tyr188Leu mutant and wild-type HIV-1 reverse transcriptase complexed with the non-nucleoside inhibitor HBY 097: inhibitor flexibility is a useful design feature for reducing drug resistance.
J.Mol.Biol., 284, 1998
1BQN
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TYR 188 LEU HIV-1 RT/HBY 097
分子名称: (S)-4-ISOPROPOXYCARBONYL-6-METHOXY-3-METHYLTHIOMETHYL-3,4-DIHYDROQUINOXALIN-2(1H)-THIONE, REVERSE TRANSCRIPTASE
著者Hsiou, Y, Das, K, Ding, J, Arnold, E.
登録日1998-08-17
公開日1999-01-06
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structures of Tyr188Leu mutant and wild-type HIV-1 reverse transcriptase complexed with the non-nucleoside inhibitor HBY 097: inhibitor flexibility is a useful design feature for reducing drug resistance.
J.Mol.Biol., 284, 1998
7CC3
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Versatile cis-prenyltransferase MM_0014 from Methanosarcina mazei (crystal type: co-FG)
分子名称: (2R)-3-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propane-1,2-diol, (2S)-3-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propane-1,2-diol, 2-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propane-1,3-diol, ...
著者Unno, H, Hemmi, H.
登録日2020-06-16
公開日2021-04-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献A versatile cis-prenyltransferase from Methanosarcina mazei catalyzes both C- and O-prenylations.
J.Biol.Chem., 296, 2021
5G1S
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Open conformation of Francisella tularensis ClpP at 1.7 A
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, ACETATE ION, ...
著者Diaz-Saez, L, Pankov, G, Hunter, W.N.
登録日2016-03-30
公開日2016-10-19
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Open and compressed conformations of Francisella tularensis ClpP.
Proteins, 85, 2017
1BRY
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BRYODIN TYPE I RIP
分子名称: BRYODIN I
著者Klei, H.E, Chang, C.Y.
登録日1997-02-14
公開日1998-03-04
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Molecular, biological, and preliminary structural analysis of recombinant bryodin 1, a ribosome-inactivating protein from the plant Bryonia dioica.
Biochemistry, 36, 1997
1BQ2
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E. COLI THYMIDYLATE SYNTHASE MUTANT N177A
分子名称: PHOSPHATE ION, THYMIDYLATE SYNTHASE
著者Reyes, C.L, Sage, C.R, Rutenber, E.E, Finer-Moore, J.S, Stroud, R.M.
登録日1998-08-20
公開日1999-04-27
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Inactivity of N229A thymidylate synthase due to water-mediated effects: isolating a late stage in methyl transfer.
J.Mol.Biol., 284, 1998
1BSM
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P.SHERMANII SOD(FE+3) 140K PH8
分子名称: FE (III) ION, SUPEROXIDE DISMUTASE
著者Schmidt, M.
登録日1998-08-28
公開日1999-06-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Manipulating the coordination mumber of the ferric iron within the cambialistic superoxide dismutase of Propionibacterium shermanii by changing the pH-value A crystallographic analysis
Eur.J.Biochem., 262, 1999
7CJJ
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Photosystem II structure in the S2 state
分子名称: 1,2-DI-O-ACYL-3-O-[6-DEOXY-6-SULFO-ALPHA-D-GLUCOPYRANOSYL]-SN-GLYCEROL, 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-DISTEAROYL-MONOGALACTOSYL-DIGLYCERIDE, ...
著者Li, H, Shen, J.-R, Suga, M.
登録日2020-07-11
公開日2021-04-28
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Capturing structural changes of the S 1 to S 2 transition of photosystem II using time-resolved serial femtosecond crystallography.
Iucrj, 8, 2021
5OBA
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Structure of a modified mouse H-chain ferritin with a lanthanide binding motif
分子名称: FE (III) ION, Ferritin heavy chain
著者Baiocco, P, Trabuco, M.C.
登録日2017-06-26
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Engineered ferritin for lanthanide binding.
PLoS ONE, 13, 2018
1BIU
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HIV-1 INTEGRASE CORE DOMAIN COMPLEXED WITH MG++
分子名称: HIV-1 INTEGRASE, MAGNESIUM ION
著者Goldgur, Y, Dyda, F, Hickman, A.B, Jenkins, T.M, Craigie, R, Davies, D.R.
登録日1998-06-19
公開日1998-08-19
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Three new structures of the core domain of HIV-1 integrase: an active site that binds magnesium.
Proc.Natl.Acad.Sci.USA, 95, 1998
5G2T
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BT1596 in complex with its substrate 4,5 unsaturated uronic acid alpha 1,4 D-Glucosamine-2-N, 6-O-disulfate
分子名称: 1,2-ETHANEDIOL, 2-O GLYCOSAMINOGLYCAN SULFATASE, 4-deoxy-2-O-sulfo-alpha-L-threo-hex-4-enopyranuronic acid, ...
著者Cartmell, A, Lowe, E.C, Basle, A, Crouch, L.I, Czjzek, M, Turnbull, J, Henrissat, B, Terrapon, N, Thomas, S, Murray, H, Firbank, S.J, Bolam, D.N.
登録日2016-04-13
公開日2017-05-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献How members of the human gut microbiota overcome the sulfation problem posed by glycosaminoglycans.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
1CDY
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STRUCTURE OF T-CELL SURFACE GLYCOPROTEIN CD4 MUTANT WITH GLY 47 REPLACED BY SER
分子名称: T-CELL SURFACE GLYCOPROTEIN CD4
著者Wu, H, Myszka, D, Tendian, S.W, Brouillette, C.G, Sweet, R.W, Chaiken, I.M, Hendrickson, W.A.
登録日1996-11-11
公開日1997-04-01
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinetic and structural analysis of mutant CD4 receptors that are defective in HIV gp120 binding.
Proc.Natl.Acad.Sci.USA, 93, 1996
7COU
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Structure of cyanobacterial photosystem II in the dark S1 state
分子名称: 1,2-DI-O-ACYL-3-O-[6-DEOXY-6-SULFO-ALPHA-D-GLUCOPYRANOSYL]-SN-GLYCEROL, 1,2-DIPALMITOYL-PHOSPHATIDYL-GLYCEROLE, 1,2-DISTEAROYL-MONOGALACTOSYL-DIGLYCERIDE, ...
著者Li, H, Shen, J.-R, Suga, M.
登録日2020-08-05
公開日2021-04-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Capturing structural changes of the S 1 to S 2 transition of photosystem II using time-resolved serial femtosecond crystallography.
Iucrj, 8, 2021
1BMS
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CRYSTAL STRUCTURE OF MS2 CAPSIDS WITH MUTATIONS IN THE SUBUNIT FG LOOP
分子名称: BACTERIOPHAGE MS2 CAPSID
著者Liljas, L, Stonehouse, N.J.
登録日1995-08-29
公開日1996-03-08
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structures of MS2 capsids with mutations in the subunit FG loop.
J.Mol.Biol., 256, 1996

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