8K1L
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![BU of 8k1l by Molmil](/molmil-images/mine/8k1l) | Cryo-EM structure of Na+,K+-ATPase alpha2 from Artemia salina in cation-free E2P form | 分子名称: | Na+,K+-ATPase alpha2KK, Na+,K+-ATPase beta2, TETRAFLUOROALUMINATE ION | 著者 | Abe, K, Artigas, P. | 登録日 | 2023-07-11 | 公開日 | 2023-11-29 | 最終更新日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.44 Å) | 主引用文献 | A Na pump with reduced stoichiometry is up-regulated by brine shrimp in extreme salinities. Proc.Natl.Acad.Sci.USA, 120, 2023
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8IJM
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![BU of 8ijm by Molmil](/molmil-images/mine/8ijm) | Cyo-EM structure of K794A non-gastric proton pump in Na+ bound E1AMPPCP state | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, ... | 著者 | Abe, K. | 登録日 | 2023-02-27 | 公開日 | 2023-08-02 | 最終更新日 | 2023-08-09 | 実験手法 | ELECTRON MICROSCOPY (3.13 Å) | 主引用文献 | An unusual conformation from Na + -sensitive non-gastric proton pump mutants reveals molecular mechanisms of cooperative Na + -binding. Biochim Biophys Acta Mol Cell Res, 1870, 2023
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8OX5
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![BU of 8ox5 by Molmil](/molmil-images/mine/8ox5) | Cryo-EM structure of ATP8B1-CDC50A in E1P-ADP conformation | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-DIPHOSPHATE, Cell cycle control protein 50A, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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8OX9
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![BU of 8ox9 by Molmil](/molmil-images/mine/8ox9) | Cryo-EM structure of ATP8B1-CDC50A in E2P active conformation with bound PC | 分子名称: | (2R)-3-{[(R)-{[(1S,2S,3R,4S,5S,6S)-2,6-dihydroxy-3,4,5-tris(phosphonooxy)cyclohexyl]oxy}(hydroxy)phosphoryl]oxy}propane -1,2-diyl dioctanoate, (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.72 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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8OX8
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![BU of 8ox8 by Molmil](/molmil-images/mine/8ox8) | Cryo-EM structure of ATP8B1-CDC50A in E2P autoinhibited "open" conformation | 分子名称: | (2R)-3-{[(R)-{[(1S,2S,3R,4S,5S,6S)-2,6-dihydroxy-3,4,5-tris(phosphonooxy)cyclohexyl]oxy}(hydroxy)phosphoryl]oxy}propane -1,2-diyl dioctanoate, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cell cycle control protein 50A, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.98 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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8OXC
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![BU of 8oxc by Molmil](/molmil-images/mine/8oxc) | Cryo-EM structure of ATP8B1-CDC50A in E2-Pi conformation with occluded PI | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOINOSITOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cell cycle control protein 50A, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.58 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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8OX7
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![BU of 8ox7 by Molmil](/molmil-images/mine/8ox7) | Cryo-EM structure of ATP8B1-CDC50A in E2P autoinhibited "closed" conformation | 分子名称: | (2R)-3-{[(R)-{[(1S,2S,3R,4S,5S,6S)-2,6-dihydroxy-3,4,5-tris(phosphonooxy)cyclohexyl]oxy}(hydroxy)phosphoryl]oxy}propane -1,2-diyl dioctanoate, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cell cycle control protein 50A, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.56 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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8OXA
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![BU of 8oxa by Molmil](/molmil-images/mine/8oxa) | Cryo-EM structure of ATP8B1-CDC50A in E2-Pi conformation with occluded PS | 分子名称: | (2~{S})-2-azanyl-3-[[(2~{R})-3-hexadecanoyloxy-2-[(~{Z})-octadec-9-enoyl]oxy-propoxy]-oxidanyl-phosphoryl]oxy-propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cell cycle control protein 50A, ... | 著者 | Dieudonne, T, Kummerer, F, Juknaviciute Laursen, M, Stock, C, Kock Flygaard, R, Khalid, S, Lenoir, G, Lyons, J.A, Lindorff-Larsen, K, Nissen, P. | 登録日 | 2023-05-01 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.76 Å) | 主引用文献 | Activation and substrate specificity of the human P4-ATPase ATP8B1. Nat Commun, 14, 2023
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7VH6
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![BU of 7vh6 by Molmil](/molmil-images/mine/7vh6) | Cryo-EM structure of the hexameric plasma membrane H+-ATPase in the active state (pH 6.0, BeF3-, conformation 1, C1 symmetry) | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, BERYLLIUM TRIFLUORIDE ION, Plasma membrane ATPase 1 | 著者 | Zhao, P, Zhao, C, Chen, D, Yun, C, Li, H, Bai, L. | 登録日 | 2021-09-21 | 公開日 | 2021-11-24 | 最終更新日 | 2022-02-16 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Structure and activation mechanism of the hexameric plasma membrane H + -ATPase. Nat Commun, 12, 2021
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7VH5
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![BU of 7vh5 by Molmil](/molmil-images/mine/7vh5) | Cryo-EM structure of the hexameric plasma membrane H+-ATPase in the autoinhibited state (pH 7.4, C1 symmetry) | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, Plasma membrane ATPase 1, SPHINGOSINE | 著者 | Zhao, P, Zhao, C, Chen, D, Yun, C, Li, H, Bai, L. | 登録日 | 2021-09-21 | 公開日 | 2021-11-24 | 最終更新日 | 2022-02-16 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structure and activation mechanism of the hexameric plasma membrane H + -ATPase. Nat Commun, 12, 2021
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7VPI
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![BU of 7vpi by Molmil](/molmil-images/mine/7vpi) | Cryo-EM structure of the human ATP13A2 (E1-ATP state) | 分子名称: | MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, Polyamine-transporting ATPase 13A2 | 著者 | Tomita, A, Yamashita, K, Nishizawa, T, Nureki, O. | 登録日 | 2021-10-17 | 公開日 | 2021-12-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Cryo-EM reveals mechanistic insights into lipid-facilitated polyamine export by human ATP13A2. Mol.Cell, 81, 2021
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7VSH
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![BU of 7vsh by Molmil](/molmil-images/mine/7vsh) | |
7VPJ
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![BU of 7vpj by Molmil](/molmil-images/mine/7vpj) | Cryo-EM structure of the human ATP13A2 (E1P-ADP state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Tomita, A, Yamashita, K, Nishizawa, T, Nureki, O. | 登録日 | 2021-10-17 | 公開日 | 2021-12-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Cryo-EM reveals mechanistic insights into lipid-facilitated polyamine export by human ATP13A2. Mol.Cell, 81, 2021
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7VPL
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![BU of 7vpl by Molmil](/molmil-images/mine/7vpl) | Cryo-EM structure of the human ATP13A2 (SPM-bound E2Pi state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, MAGNESIUM ION, Polyamine-transporting ATPase 13A2, ... | 著者 | Tomita, A, Yamashita, K, Nishizawa, T, Nureki, O. | 登録日 | 2021-10-17 | 公開日 | 2021-12-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Cryo-EM reveals mechanistic insights into lipid-facilitated polyamine export by human ATP13A2. Mol.Cell, 81, 2021
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7VSG
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![BU of 7vsg by Molmil](/molmil-images/mine/7vsg) | |
7VPK
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![BU of 7vpk by Molmil](/molmil-images/mine/7vpk) | Cryo-EM structure of the human ATP13A2 (SPM-bound E2P state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, BERYLLIUM TRIFLUORIDE ION, MAGNESIUM ION, ... | 著者 | Tomita, A, Yamashita, K, Nishizawa, T, Nureki, O. | 登録日 | 2021-10-17 | 公開日 | 2021-12-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Cryo-EM reveals mechanistic insights into lipid-facilitated polyamine export by human ATP13A2. Mol.Cell, 81, 2021
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7W48
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![BU of 7w48 by Molmil](/molmil-images/mine/7w48) | |
7W49
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![BU of 7w49 by Molmil](/molmil-images/mine/7w49) | |
7W47
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![BU of 7w47 by Molmil](/molmil-images/mine/7w47) | Crystal structure of the gastric proton pump complexed with tegoprazan | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, MAGNESIUM ION, Potassium-transporting ATPase alpha chain 1, ... | 著者 | Abe, K, Tanaka, S, Morita, M, Yamagishi, T. | 登録日 | 2021-11-26 | 公開日 | 2022-01-05 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural Basis for Binding of Potassium-Competitive Acid Blockers to the Gastric Proton Pump. J.Med.Chem., 65, 2022
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7WYX
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![BU of 7wyx by Molmil](/molmil-images/mine/7wyx) | Cryo-EM structure of Na+,K+-ATPase in the E2P state formed by ATP with istaroxime | 分子名称: | (3E,5S,8R,9S,10R,13S,14S)-3-(2-azanylethoxyimino)-10,13-dimethyl-1,2,4,5,7,8,9,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthrene-6,17-dione, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kanai, R, Cornelius, F, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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7WZ0
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![BU of 7wz0 by Molmil](/molmil-images/mine/7wz0) | Cryo-EM structure of Na+,K+-ATPase in the E2P state formed by inorganic phosphate with ouabain | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kanai, R, Cornelius, F, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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7WYW
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![BU of 7wyw by Molmil](/molmil-images/mine/7wyw) | Cryo-EM structure of Na+,K+-ATPase in the E2P state formed by inorganic phosphate | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kanai, R, Cornelius, F, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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7WYZ
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![BU of 7wyz by Molmil](/molmil-images/mine/7wyz) | Cryo-EM structure of Na+,K+-ATPase in the E2P state formed by ATP with ouabain | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kanai, R, Cornelius, F, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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7WYS
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![BU of 7wys by Molmil](/molmil-images/mine/7wys) | Crystal structures of Na+,K+-ATPase in complex with istaroxime | 分子名称: | (3E,5S,8R,9S,10R,13S,14S)-3-(2-azanylethoxyimino)-10,13-dimethyl-1,2,4,5,7,8,9,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthrene-6,17-dione, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Ogawa, H, Cornelius, F, Kanai, R, Motoyama, K, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-05-04 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.71 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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7WYT
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![BU of 7wyt by Molmil](/molmil-images/mine/7wyt) | Crystal structures of Na+,K+-ATPase in complex with ouabain | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Ogawa, H, Cornelius, F, Kanai, R, Motoyama, K, Vilsen, B, Toyoshima, C. | 登録日 | 2022-02-16 | 公開日 | 2022-05-04 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Cryoelectron microscopy of Na + ,K + -ATPase in the two E2P states with and without cardiotonic steroids. Proc.Natl.Acad.Sci.USA, 119, 2022
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