2C5X
| Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design | 分子名称: | CELL DIVISION PROTEIN KINASE 2, CYCLIN A2, HYDROXY(OXO)(3-{[(2Z)-4-[3-(1H-1,2,4-TRIAZOL-1-YLMETHYL)PHENYL]PYRIMIDIN-2(5H)-YLIDENE]AMINO}PHENYL)AMMONIUM | 著者 | Kontopidis, G, Mcinnes, C, Pandalaneni, S.R, Mcnae, I, Gibson, D, Mezna, M, Thomas, M, Wood, G, Wang, S, Walkinshaw, M.D, Fischer, P.M. | 登録日 | 2005-11-03 | 公開日 | 2006-03-01 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Differential Binding of Inhibitors to Active and Inactive Cdk2 Provides Insights for Drug Design. Chem.Biol., 13, 2006
|
|
2KH5
| Solution Structure of cis-5R,6S-thymine glycol opposite complementary adenine in duplex DNA | 分子名称: | 5'-D(*AP*CP*AP*AP*AP*CP*AP*CP*GP*CP*AP*C)-3', 5'-D(*GP*TP*GP*CP*GP*(CTG)P*GP*TP*TP*TP*GP*T)-3' | 著者 | Brown, K.L. | 登録日 | 2009-03-24 | 公開日 | 2010-03-02 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Binding of the human nucleotide excision repair proteins XPA and XPC/HR23B to the 5R-thymine glycol lesion and structure of the cis-(5R,6S) thymine glycol epimer in the 5'-GTgG-3' sequence: destabilization of two base pairs at the lesion site Nucleic Acids Res., 38, 2010
|
|
2KH7
| |
1WW3
| Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-D-glucopyranosylamine and N-trifluoroacetyl-beta-D-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylase | 分子名称: | Glycogen phosphorylase, muscle form, N-(trifluoroacetyl)-beta-D-glucopyranosylamine, ... | 著者 | Anagnostou, E, Kosmopoulou, M.N, Chrysina, E.D, Leonidas, D.D, Hadjiloi, T, Tiraidis, C, Zographos, S.E, Gyorgydeak, Z, Somsak, L, Docsa, T, Gergely, P, Kolisis, F.N, Oikonomakos, N.G. | 登録日 | 2004-12-31 | 公開日 | 2005-12-13 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-d-glucopyranosylamine and N-trifluoroacetyl-beta-d-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylase Bioorg.Med.Chem., 14, 2006
|
|
1OVV
| |
1IKJ
| 1.27 A CRYSTAL STRUCTURE OF NITROPHORIN 4 FROM RHODNIUS PROLIXUS COMPLEXED WITH IMIDAZOLE | 分子名称: | IMIDAZOLE, NITROPHORIN 4, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Roberts, S.A, Weichsel, A, Qui, Y, Shelnutt, J.A, Walker, F.A, Montfort, W.R. | 登録日 | 2001-05-03 | 公開日 | 2001-10-03 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.27 Å) | 主引用文献 | Ligand-induced heme ruffling and bent no geometry in ultra-high-resolution structures of nitrophorin 4. Biochemistry, 40, 2001
|
|
1P84
| HDBT inhibited Yeast Cytochrome bc1 Complex | 分子名称: | 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, ... | 著者 | Palsdottir, H, Lojero, C.G, Trumpower, B.L, Hunte, C. | 登録日 | 2003-05-06 | 公開日 | 2003-07-29 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of the yeast cytochrome bc1 complex with a hydroxyquinone anion Qo site inhibitor bound J.Biol.Chem., 278, 2003
|
|
1JJT
| IMP-1 METALLO BETA-LACTAMASE FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH A BIARYL SUCCINIC ACID INHIBITOR (1) | 分子名称: | 2,3-BIS-BENZO[1,3]DIOXOL-5-YLMETHYL-SUCCINIC ACID, ACETATE ION, IMP-1 METALLO BETA-LACTAMASE, ... | 著者 | Fitzgerald, P.M.D, Sharma, N. | 登録日 | 2001-07-09 | 公開日 | 2001-07-25 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Succinic acids as potent inhibitors of plasmid-borne IMP-1 metallo-beta-lactamase. J.Biol.Chem., 276, 2001
|
|
1ERD
| THE NMR SOLUTION STRUCTURE OF THE PHEROMONE ER-2 FROM THE CILIATED PROTOZOAN EUPLOTES RAIKOVI | 分子名称: | PHEROMONE ER-2 | 著者 | Ottiger, M, Szyperski, T, Luginbuhl, P, Ortenzi, C, Luporini, P, Bradshaw, R.A, Wuthrich, K. | 登録日 | 1994-02-14 | 公開日 | 1994-10-15 | 最終更新日 | 2022-02-16 | 実験手法 | SOLUTION NMR | 主引用文献 | The NMR solution structure of the pheromone Er-2 from the ciliated protozoan Euplotes raikovi. Protein Sci., 3, 1994
|
|
1ERP
| NUCLEAR MAGNETIC RESONANCE SOLUTION STRUCTURE OF THE PHEROMONE ER-10 FROM THE CILIATED PROTOZOAN EUPLOTES RAIKOVI | 分子名称: | PHEROMONE ER-10 | 著者 | Brown, L.R, Mronga, S, Bradshaw, R, Ortenzi, C, Luporini, P, Wuthrich, K. | 登録日 | 1992-12-02 | 公開日 | 1993-10-31 | 最終更新日 | 2022-02-16 | 実験手法 | SOLUTION NMR | 主引用文献 | Nuclear magnetic resonance solution structure of the pheromone Er-10 from the ciliated protozoan Euplotes raikovi. J.Mol.Biol., 231, 1993
|
|
1WVV
| |
1PJJ
| Complex between the Lactococcus lactis Fpg and an abasic site containing DNA. | 分子名称: | DNA (5'-D(*CP*TP*CP*TP*TP*TP*(3DR)P*TP*TP*TP*CP*TP*CP*G)-3'), DNA (5'-D(*GP*CP*GP*AP*GP*AP*AP*AP*CP*AP*AP*AP*GP*A)-3'), Formamidopyrimidine-DNA glycosylase, ... | 著者 | Serre, L, Pereira de Jesus, K, Boiteux, S, Zelwer, C, Castaing, B. | 登録日 | 2003-06-03 | 公開日 | 2004-06-08 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural insights into abasic site for Fpg specific binding and catalysis: comparative high-resolution crystallographic studies of Fpg bound to various models of abasic site analogues-containing DNA. Nucleic Acids Res., 33, 2005
|
|
1PC3
| |
1X8O
| 1.01 A Crystal Structure Of Nitrophorin 4 From Rhodnius Prolixus Complexed With Nitric Oxide at pH 5.6 | 分子名称: | NITRIC OXIDE, Nitrophorin 4, PHOSPHATE ION, ... | 著者 | Kondrashov, D.A, Roberts, S.A, Weichsel, A, Montfort, W.R. | 登録日 | 2004-08-18 | 公開日 | 2004-10-05 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.01 Å) | 主引用文献 | Protein functional cycle viewed at atomic resolution: conformational change and mobility in nitrophorin 4 as a function of pH and NO binding Biochemistry, 43, 2004
|
|
1PK0
| Crystal Structure of the EF3-CaM complexed with PMEApp | 分子名称: | (ADENIN-9-YL-ETHOXYMETHYL)-HYDROXYPHOSPHINYL-DIPHOSPHATE, CALCIUM ION, Calmodulin, ... | 著者 | Shen, Y, Tang, W.J. | 登録日 | 2003-06-04 | 公開日 | 2004-02-10 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Selective inhibition of anthrax edema factor by adefovir, a drug for chronic hepatitis B virus infection. Proc.Natl.Acad.Sci.USA, 101, 2004
|
|
1ZJ6
| Crystal structure of human ARL5 | 分子名称: | ADP-ribosylation factor-like protein 5, GUANOSINE-3'-MONOPHOSPHATE-5'-DIPHOSPHATE, SULFATE ION | 著者 | Wang, Z.X, Shi, L, Liu, J.F, An, X.M, Chang, W.R, Liang, D.C. | 登録日 | 2005-04-28 | 公開日 | 2005-06-07 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | 2.0A crystal structure of human ARL5-GDP3'P, a novel member of the small GTP-binding proteins Biochem.Biophys.Res.Commun., 332, 2005
|
|
1YYP
| Crystal structure of cytomegalovirus UL44 bound to C-terminal peptide from CMV UL54 | 分子名称: | 1,2-ETHANEDIOL, DNA polymerase, DNA polymerase processivity factor, ... | 著者 | Appleton, B.A, Brooks, J, Loregian, A, Filman, D.J, Coen, D.M, Hogle, J.M. | 登録日 | 2005-02-25 | 公開日 | 2005-12-27 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of the cytomegalovirus DNA polymerase subunit UL44 in complex with the C terminus from the catalytic subunit. Differences in structure and function relative to unliganded UL44. J.Biol.Chem., 281, 2006
|
|
1PYS
| PHENYLALANYL-TRNA SYNTHETASE FROM THERMUS THERMOPHILUS | 分子名称: | MAGNESIUM ION, PHENYLALANYL-TRNA SYNTHETASE | 著者 | Safro, M, Mosyak, L, Goldgur, Y, Reshetnikova, L, Delarue, M. | 登録日 | 1996-11-14 | 公開日 | 1997-11-19 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structure of phenylalanyl-tRNA synthetase from Thermus thermophilus. Nat.Struct.Biol., 2, 1995
|
|
1LCJ
| |
1ZNJ
| INSULIN, MONOCLINIC CRYSTAL FORM | 分子名称: | CHLORIDE ION, INSULIN, PHENOL, ... | 著者 | Turkenburg, M.G.W, Whittingham, J.L, Turkenburg, J.P, Dodson, G.G, Derewenda, U, Smith, G.D, Dodson, E.J, Derewenda, Z.S, Xiao, B. | 登録日 | 1997-09-23 | 公開日 | 1998-01-28 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure Determination and Refinement of Two Crystal Forms of Native Insulins To be Published
|
|
1L9O
| |
1L3I
| MT0146, THE PRECORRIN-6Y METHYLTRANSFERASE (CBIT) HOMOLOG FROM M. THERMOAUTOTROPHICUM, ADOHCY BINARY COMPLEX | 分子名称: | Precorrin-6y methyltransferase/putative decarboxylase, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Keller, J.P, Smith, P.M, Benach, J, Christendat, D, deTitta, G, Hunt, J.F. | 登録日 | 2002-02-27 | 公開日 | 2002-11-27 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | The Crystal Structure of Mt0146/CbiT Suggests that the Putative Precorrin-8W Decarboxylase is a Methyltransferase Structure, 10, 2002
|
|
1YWB
| 0.9 A Structure of NP4 from Rhodnius Prolixus complexed with NO at pH 5.6 | 分子名称: | NITRIC OXIDE, PHOSPHATE ION, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Maes, E.M, Weichsel, A, Roberts, S.A, Montfort, W.R. | 登録日 | 2005-02-17 | 公開日 | 2005-10-04 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (0.97 Å) | 主引用文献 | Ultrahigh Resolution Structures of Nitrophorin 4: Heme Distortion in Ferrous CO and NO Complexes Biochemistry, 44, 2005
|
|
1ZN5
| |
1P9B
| Structure of fully ligated Adenylosuccinate synthetase from Plasmodium falciparum | 分子名称: | 6-O-PHOSPHORYL INOSINE MONOPHOSPHATE, Adenylosuccinate Synthetase, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Eaazhisai, K, Jayalakshmi, R, Gayathri, P, Anand, R.P, Sumathy, K, Balaram, H, Murthy, M.R. | 登録日 | 2003-05-10 | 公開日 | 2004-02-03 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structure of Fully Ligated Adenylosuccinate Synthetase from Plasmodium falciparum. J.Mol.Biol., 335, 2004
|
|