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8D20
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BU of 8d20 by Molmil
Crystal structure of Plasmodium falciparum GRP78 in complex with 5'-Methylthioadenosine
分子名称: 5'-DEOXY-5'-METHYLTHIOADENOSINE, Chaperone DnaK, SULFATE ION
著者Mrozek, A, Park, H.W.
登録日2022-05-27
公開日2023-05-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献A non-traditional crystal-based compound screening method targeting the ATP binding site of Plasmodium falciparum GRP78 for identification of novel nucleoside analogues.
Front Mol Biosci, 9, 2022
8D1S
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BU of 8d1s by Molmil
Crystal structure of Plasmodium falciparum GRP78 in complex with Toyocamycin
分子名称: 4-amino-7-(beta-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile, Chaperone DnaK, SULFATE ION
著者Mrozek, A, Chen, Y, Antoshchenko, T, Park, H.W.
登録日2022-05-27
公開日2023-05-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献A non-traditional crystal-based compound screening method targeting the ATP binding site of Plasmodium falciparum GRP78 for identification of novel nucleoside analogues.
Front Mol Biosci, 9, 2022
4AM6
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BU of 4am6 by Molmil
C-TERMINAL DOMAIN OF ACTIN-RELATED PROTEIN ARP8 FROM S. CEREVISIAE
分子名称: ACTIN-LIKE PROTEIN ARP8, SULFATE ION
著者Wuerges, J, Saravanan, M, Bose, D, Cook, N.J, Zhang, X, Wigley, D.B.
登録日2012-03-07
公開日2012-12-12
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Interactions between the Nucleosome Histone Core and Arp8 in the Ino80 Chromatin Remodeling Complex.
Proc.Natl.Acad.Sci.USA, 109, 2012
4AM7
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BU of 4am7 by Molmil
ADP-BOUND C-TERMINAL DOMAIN OF ACTIN-RELATED PROTEIN ARP8 FROM S. CEREVISIAE
分子名称: ACTIN-LIKE PROTEIN ARP8, ADENOSINE-5'-DIPHOSPHATE
著者Wuerges, J, Saravanan, M, Bose, D, Cook, N.J, Zhang, X, Wigley, D.B.
登録日2012-03-07
公開日2012-12-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Interactions between the Nucleosome Histone Core and Arp8 in the Ino80 Chromatin Remodeling Complex.
Proc.Natl.Acad.Sci.USA, 109, 2012
8D22
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BU of 8d22 by Molmil
Crystal structure of Plasmodium falciparum GRP78-NBD in complex with Piclidenoson
分子名称: Chaperone DnaK, Piclidenoson, SULFATE ION
著者Mrozek, A, Park, H.W.
登録日2022-05-27
公開日2023-05-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A non-traditional crystal-based compound screening method targeting the ATP binding site of Plasmodium falciparum GRP78 for identification of novel nucleoside analogues.
Front Mol Biosci, 9, 2022
9CB7
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BU of 9cb7 by Molmil
DeltaNhp10 INO80 bound to S.c 0/40 nucleosome, Ino80-Nucleosome
分子名称: Chromatin-remodeling ATPase INO80, DNA (227-MER), Histone H2A.1, ...
著者Wu, H, Kaur, U, Narlikar, G.J, Cheng, Y.F.
登録日2024-06-18
公開日2025-07-16
実験手法ELECTRON MICROSCOPY (4.04 Å)
主引用文献Autoinhibition imposed by a large conformational switch of INO80 regulates nucleosome positioning
Science, 2025
4A0X
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BU of 4a0x by Molmil
Structure of the global transcription regulator FapR from Staphylococcus aureus
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ACETATE ION, TRANSCRIPTION FACTOR FAPR, ...
著者Albanesi, D, Guerin, M.E, Buschiazzo, A, de Mendoza, D, Alzari, P.M.
登録日2011-09-13
公開日2012-09-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Basis for Feed-Forward Transcriptional Regulation of Membrane Lipid Homeostasis in Staphylococcus Aureus.
Plos Pathog., 9, 2013
8D5D
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BU of 8d5d by Molmil
Structure of Y430F D-ornithine/D-lysine decarboxylase complex with D-arginine
分子名称: (E)-N~2~-({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methylidene)-D-arginine, D-ornithine/D-lysine decarboxylase, DIMETHYL SULFOXIDE, ...
著者Phillips, R.S, Nguyen Hoang, K.N.
登録日2022-06-04
公開日2022-11-16
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献The Y430F mutant of Salmonella d-ornithine/d-lysine decarboxylase has altered stereospecificity and a putrescine allosteric activation site.
Arch.Biochem.Biophys., 731, 2022
8D88
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BU of 8d88 by Molmil
Structure of Y430F D-ornithine/D-lysine decarboxylase complex with D-lysine
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, D-ornithine/D-lysine decarboxylase, ...
著者Phillips, R.S, Nguyen Hoang, K.N.
登録日2022-06-08
公開日2022-11-16
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献The Y430F mutant of Salmonella d-ornithine/d-lysine decarboxylase has altered stereospecificity and a putrescine allosteric activation site.
Arch.Biochem.Biophys., 731, 2022
6TJ6
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BU of 6tj6 by Molmil
T. gondii myosin A trimeric complex with ELC1, calcium-free
分子名称: Calmodulin, putative, IMIDAZOLE, ...
著者Pazicky, S, Loew, C.
登録日2019-11-25
公開日2020-10-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural role of essential light chains in the apicomplexan glideosome.
Commun Biol, 3, 2020
6TJ5
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BU of 6tj5 by Molmil
T. gondii myosin A trimeric complex with ELC1
分子名称: CALCIUM ION, CHLORIDE ION, Calmodulin, ...
著者Pazicky, S, Loew, C.
登録日2019-11-25
公開日2020-10-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.394 Å)
主引用文献Structural role of essential light chains in the apicomplexan glideosome.
Commun Biol, 3, 2020
7E5T
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BU of 7e5t by Molmil
Crystal structure of Fsa2
分子名称: Diels-Alderase fsa2, ETHANOL, PENTAETHYLENE GLYCOL, ...
著者Fujiyama, K, Kato, N, Kinugasa, K, Hino, T, Takahashi, S, Nagano, S.
登録日2021-02-20
公開日2021-06-30
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.16977525 Å)
主引用文献Molecular Basis for Two Stereoselective Diels-Alderases that Produce Decalin Skeletons*.
Angew.Chem.Int.Ed.Engl., 60, 2021
3F4M
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BU of 3f4m by Molmil
Crystal structure of TIPE2
分子名称: CHLORIDE ION, Tumor necrosis factor, alpha-induced protein 8-like protein 2
著者Zhang, X, Wang, J, Shi, Y.
登録日2008-11-01
公開日2009-03-17
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.696 Å)
主引用文献Crystal structure of TIPE2 provides insights into immune homeostasis
Nat.Struct.Mol.Biol., 16, 2009
6Y1M
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BU of 6y1m by Molmil
Crystal structure of the paraoxon-modified A.17 antibody FAB fragment - L47K mutant
分子名称: DIETHYL PHOSPHONATE, FAB A.17 L47K mutant HEAVY CHAIN, FAB A.17 L47K mutant Light CHAIN
著者Chatziefthimiou, S, Mokrushina, Y, Smirnov, I, Gabibov, A, Wilmanns, M.
登録日2020-02-12
公開日2020-09-16
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Multiscale computation delivers organophosphorus reactivity and stereoselectivity to immunoglobulin scavengers.
Proc.Natl.Acad.Sci.USA, 117, 2020
6ZYI
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BU of 6zyi by Molmil
Crystal structure of HSP70 ATPase domain in complex with ADP and calcium
分子名称: ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, Heat shock 70kDa protein 1A variant
著者Yan, Y, Preissler, S, Ron, D.
登録日2020-08-01
公開日2020-12-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.52 Å)
主引用文献Calcium depletion challenges endoplasmic reticulum proteostasis by destabilising BiP-substrate complexes.
Elife, 9, 2020
6ZYJ
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BU of 6zyj by Molmil
Crystal structure of Hsc70 ATPase domain in complex with ADP and calcium
分子名称: ACETATE ION, ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, ...
著者Yan, Y, Preissler, S, Ron, D.
登録日2020-08-01
公開日2020-12-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Calcium depletion challenges endoplasmic reticulum proteostasis by destabilising BiP-substrate complexes.
Elife, 9, 2020
4A0Z
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BU of 4a0z by Molmil
Structure of the global transcription regulator FapR from Staphylococcus aureus in complex with malonyl-CoA
分子名称: MALONYL-COENZYME A, TRANSCRIPTION FACTOR FAPR
著者Albanesi, D, Guerin, M.E, Buschiazzo, A, de Mendoza, D, Alzari, P.M.
登録日2011-09-13
公開日2012-09-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Basis for Feed-Forward Transcriptional Regulation of Membrane Lipid Homeostasis in Staphylococcus Aureus.
Plos Pathog., 9, 2013
7A4V
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BU of 7a4v by Molmil
Crystal structure of lid-truncated ADP-bound BiP in an oligomeric state
分子名称: ADENOSINE-5'-DIPHOSPHATE, Endoplasmic reticulum chaperone BiP, GLYCEROL, ...
著者Perera, L.A, Ron, D.
登録日2020-08-20
公開日2020-12-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Calcium depletion challenges endoplasmic reticulum proteostasis by destabilising BiP-substrate complexes.
Elife, 9, 2020
6ZYH
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BU of 6zyh by Molmil
Crystal structure of GRP78 (70kDa heat shock protein 5 / BiP) ATPase domain in complex with ADP and calcium
分子名称: ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, Endoplasmic reticulum chaperone BiP
著者Yan, Y, Preissler, S, Ron, D.
登録日2020-08-01
公開日2020-12-16
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Calcium depletion challenges endoplasmic reticulum proteostasis by destabilising BiP-substrate complexes.
Elife, 9, 2020
3VOK
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BU of 3vok by Molmil
X-ray Crystal Structure of Wild Type HrtR in the Apo Form with the Target DNA.
分子名称: 5'-D(*AP*TP*GP*AP*CP*AP*CP*TP*GP*TP*GP*TP*CP*AP*T)-3', Transcriptional regulator
著者Sawai, H, Sugimoto, H, Shiro, Y, Aono, S.
登録日2012-01-27
公開日2012-07-25
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Basis for the Transcriptional Regulation of Heme Homeostasis in Lactococcus lactis.
J.Biol.Chem., 287, 2012
3VOX
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BU of 3vox by Molmil
X-ray Crystal Structure of Wild Type HrtR in the Apo Form
分子名称: Transcriptional regulator
著者Sawai, H, Sugimoto, H, Shiro, Y, Aono, S.
登録日2012-02-23
公開日2012-07-25
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for the Transcriptional Regulation of Heme Homeostasis in Lactococcus lactis.
J.Biol.Chem., 287, 2012
7L1G
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BU of 7l1g by Molmil
PRMT5-MEP50 Complexed with SAM
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Methylosome protein 50, ...
著者Palte, R.L.
登録日2020-12-14
公開日2021-04-14
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献Development of a Flexible and Robust Synthesis of Tetrahydrofuro[3,4- b ]furan Nucleoside Analogues.
J.Org.Chem., 86, 2021
8UQE
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BU of 8uqe by Molmil
Crystal structure of RNF168 (RING)-UbcH5c fused to H2A-H2B via a 26-residue linker (RING not modeled in density)
分子名称: E3 ubiquitin-protein ligase RNF168,Ubiquitin-conjugating enzyme E2 D3,Histone H2B type 2-E,Histone H2A type 1-B/E
著者Hu, Q, Botuyan, M.V, Mer, G.
登録日2023-10-23
公開日2024-01-17
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (3.562 Å)
主引用文献Mechanisms of RNF168 nucleosome recognition and ubiquitylation.
Mol.Cell, 84, 2024
8UQA
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Crystal structure of RNF168 (RING)-UbcH5c fused to H2A-H2B via a 12-residue linker
分子名称: CHLORIDE ION, E3 ubiquitin-protein ligase RNF168,Ubiquitin-conjugating enzyme E2 D3,Histone H2B type 2-E,Histone H2A type 1-B/E, SODIUM ION, ...
著者Hu, Q, Botuyan, M.V, Mer, G.
登録日2023-10-23
公開日2024-01-17
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.049 Å)
主引用文献Mechanisms of RNF168 nucleosome recognition and ubiquitylation.
Mol.Cell, 84, 2024
8UQB
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Crystal structure of RNF168 (RING)-UbcH5c fused to H2A-H2B via a 20-residue linker (crystallization condition 1)
分子名称: CHLORIDE ION, E3 ubiquitin-protein ligase RNF168,Ubiquitin-conjugating enzyme E2 D3,Histone H2B type 2-E,Histone H2A type 1-B/E, ZINC ION
著者Hu, Q, Botuyan, M.V, Mer, G.
登録日2023-10-23
公開日2024-01-17
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.484 Å)
主引用文献Mechanisms of RNF168 nucleosome recognition and ubiquitylation.
Mol.Cell, 84, 2024

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