7G1W
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![BU of 7g1w by Molmil](/molmil-images/mine/7g1w) | Crystal Structure of human FABP4 binding site mutated to that of FABP5 in complex with 5-(3,5-dichloroanilino)-3,3-dimethyl-5-oxopentanoic acid | 分子名称: | 5-(3,5-dichloroanilino)-3,3-dimethyl-5-oxopentanoic acid, Fatty acid-binding protein, adipocyte | 著者 | Ehler, A, Benz, J, Obst, U, Brunner, M, Rudolph, M.G. | 登録日 | 2023-04-27 | 公開日 | 2023-06-14 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Crystal Structure of a human FABP4 binding site mutated to that of FABP5 complex To be published
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8IVL
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![BU of 8ivl by Molmil](/molmil-images/mine/8ivl) | FABP7 complexed with Cholesterol | 分子名称: | CHOLESTEROL, Fatty acid-binding protein, brain | 著者 | Wei, P.C, Zhao, K, Yin, L. | 登録日 | 2023-03-28 | 公開日 | 2024-02-28 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Fatty acid-binding proteins 3, 7, and 8 bind cholesterol and facilitate its egress from lysosomes. J.Cell Biol., 223, 2024
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8IVF
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![BU of 8ivf by Molmil](/molmil-images/mine/8ivf) | FABP7 complexed with 25-HC | 分子名称: | 25-HYDROXYCHOLESTEROL, Fatty acid-binding protein, brain | 著者 | Wei, P.C, Zhao, K, Yin, L. | 登録日 | 2023-03-27 | 公開日 | 2024-02-28 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Fatty acid-binding proteins 3, 7, and 8 bind cholesterol and facilitate its egress from lysosomes. J.Cell Biol., 223, 2024
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8GEW
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![BU of 8gew by Molmil](/molmil-images/mine/8gew) | H-FABP crystal soaked in a bromo palmitic acid solution | 分子名称: | 2-Bromopalmitic acid, Fatty acid-binding protein, heart, ... | 著者 | Howard, E, Cousido-Siah, A, Alvarez, A, Espinosa, Y, Podjarny, A, Mitschler, A, Carlevaro, M. | 登録日 | 2023-03-07 | 公開日 | 2023-08-30 | 最終更新日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (0.97 Å) | 主引用文献 | Lipid exchange in crystal-confined fatty acid binding proteins: X-ray evidence and molecular dynamics explanation. Proteins, 91, 2023
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8GEU
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![BU of 8geu by Molmil](/molmil-images/mine/8geu) | Crystal structure of human cellular retinol binding protein 1 in complex with methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[(1-methylpyrazol-4-yl)methyl]amine | 分子名称: | 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, N-methyl-1-{3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]methanamine, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-07 | 公開日 | 2023-10-11 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8GEV
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![BU of 8gev by Molmil](/molmil-images/mine/8gev) | Crystal structure of human cellular retinol binding protein 1 in complex with 1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(methoxymethyl)piperidine | 分子名称: | 1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(methoxymethyl)piperidine, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-07 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8GEM
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![BU of 8gem by Molmil](/molmil-images/mine/8gem) | Crystal structure of human cellular retinol binding protein 1 in complex with N-ethyl-N-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(1H-pyrazol-1-yl)ethanamine | 分子名称: | N-ethyl-N-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(1H-pyrazol-1-yl)ethan-1-amine, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-07 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8GEY
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![BU of 8gey by Molmil](/molmil-images/mine/8gey) | Crystal structure of human cellular retinol binding protein 1 in complex with 4-(hydroxymethyl)-1-[(4-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)sulfonyl]piperidin-4-ol | 分子名称: | 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-(hydroxymethyl)-1-(4-methoxy-5,6,7,8-tetrahydronaphthalene-1-sulfonyl)piperidin-4-ol, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-07 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8GDM
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![BU of 8gdm by Molmil](/molmil-images/mine/8gdm) | Crystal structure of human cellular retinol binding protein 1 in complex with {[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine | 分子名称: | (1S)-N-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-1-(thiophen-2-yl)ethan-1-amine, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-06 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8GD2
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![BU of 8gd2 by Molmil](/molmil-images/mine/8gd2) | Crystal structure of human cellular retinol binding protein 1 in complex with N-methyl-1-{3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}-N-(2-thienylmethyl)methanamine | 分子名称: | 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, N-methyl-1-{3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}-N-[(thiophen-2-yl)methyl]methanamine, Retinol-binding protein 1 | 著者 | Plau, J, Golczak, M. | 登録日 | 2023-03-03 | 公開日 | 2023-10-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | Discovery of Nonretinoid Inhibitors of CRBP1: Structural and Dynamic Insights for Ligand-Binding Mechanisms. Acs Chem.Biol., 18, 2023
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8HTA
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![BU of 8hta by Molmil](/molmil-images/mine/8hta) | |
8EPV
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![BU of 8epv by Molmil](/molmil-images/mine/8epv) | 2.2 A crystal structure of the lipocalin cat allergen Fel d 7 | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, Fel d 7 allergen, ... | 著者 | Min, J, Pedersen, L.C, Geoffrey, M.A. | 登録日 | 2022-10-06 | 公開日 | 2023-04-05 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Structural and ligand binding analysis of the pet allergens Can f 1 and Fel d 7. Front Allergy, 4, 2023
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8EPU
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![BU of 8epu by Molmil](/molmil-images/mine/8epu) | |
8B0H
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![BU of 8b0h by Molmil](/molmil-images/mine/8b0h) | 2C9, C5b9-CD59 cryoEM structure | 分子名称: | CD59 glycoprotein, Complement C5, Complement component C6, ... | 著者 | Couves, E.C, Gardner, S, Bubeck, D. | 登録日 | 2022-09-07 | 公開日 | 2023-02-22 | 最終更新日 | 2023-03-01 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Structural basis for membrane attack complex inhibition by CD59. Nat Commun, 14, 2023
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8B0G
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![BU of 8b0g by Molmil](/molmil-images/mine/8b0g) | 2C9, C5b9-CD59 structure | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CD59 glycoprotein, Complement C5, ... | 著者 | Couves, E.C, Gardner, S, Bubeck, D. | 登録日 | 2022-09-07 | 公開日 | 2023-02-22 | 最終更新日 | 2023-03-01 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Structural basis for membrane attack complex inhibition by CD59. Nat Commun, 14, 2023
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8B0F
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![BU of 8b0f by Molmil](/molmil-images/mine/8b0f) | CryoEM structure of C5b8-CD59 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Bubeck, D, Couves, E.C, Gardner, S. | 登録日 | 2022-09-07 | 公開日 | 2023-02-22 | 最終更新日 | 2023-03-01 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structural basis for membrane attack complex inhibition by CD59. Nat Commun, 14, 2023
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8AMC
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![BU of 8amc by Molmil](/molmil-images/mine/8amc) | Crystal Structure of cat allergen Fel d 4 | 分子名称: | Allergen Fel d 4, SULFATE ION | 著者 | Schooltink, L, Sagmeister, T, Gottstein, N, Pavkov-Keller, T, Keller, W. | 登録日 | 2022-08-03 | 公開日 | 2023-08-16 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Crystal Structure of cat allergen Fel d 4 To Be Published
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8AEH
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![BU of 8aeh by Molmil](/molmil-images/mine/8aeh) | |
8AEJ
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![BU of 8aej by Molmil](/molmil-images/mine/8aej) | |
8AEI
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![BU of 8aei by Molmil](/molmil-images/mine/8aei) | |
8DN1
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![BU of 8dn1 by Molmil](/molmil-images/mine/8dn1) | Q108K:K40L:T51C:T53A:R58L:Q38F:Q4F mutant of hCRBPII bound to synthetic fluorophore CM1V at pH 7.2 | 分子名称: | (2E)-3-[7-(diethylamino)-2-oxo-2H-1-benzopyran-3-yl]prop-2-enal, bound form, GLYCEROL, ... | 著者 | Bingham, C.R, Borhan, B, Geiger, J.H. | 登録日 | 2022-07-10 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.32 Å) | 主引用文献 | Light controlled reversible Michael addition of cysteine: a new tool for dynamic site-specific labeling of proteins. Analyst, 148, 2023
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7YF1
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![BU of 7yf1 by Molmil](/molmil-images/mine/7yf1) | |
8DB2
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![BU of 8db2 by Molmil](/molmil-images/mine/8db2) | Q108K:K40L:T51C:T53A:R58L:Q38F mutant of hCRBPII bound to synthetic fluorophore CM1V | 分子名称: | (2E)-3-[7-(diethylamino)-2-oxo-2H-1-benzopyran-3-yl]prop-2-enal, bound form, Retinol-binding protein 2 | 著者 | Bingham, C.R, Geiger, J.H, Borhan, B, Staples, R. | 登録日 | 2022-06-14 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Light controlled reversible Michael addition of cysteine: a new tool for dynamic site-specific labeling of proteins. Analyst, 148, 2023
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8D6H
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![BU of 8d6h by Molmil](/molmil-images/mine/8d6h) | Q108K:K40L:T51C:T53A:R58L:Q38F:Q4F mutant of hCRBPII bound to synthetic fluorophore CM1V after UV irradiation | 分子名称: | (2E)-3-[7-(diethylamino)-2-oxo-2H-1-benzopyran-3-yl]prop-2-enal, bound form, ACETATE ION, ... | 著者 | Bingham, C.R, Geiger, J.H, Borhan, B. | 登録日 | 2022-06-06 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Light controlled reversible Michael addition of cysteine: a new tool for dynamic site-specific labeling of proteins. Analyst, 148, 2023
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8D6N
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![BU of 8d6n by Molmil](/molmil-images/mine/8d6n) | Q108K:K40L:T53A:R58L:Q38F:Q4F mutant of hCRBPII bound to synthetic fluorophore CM1V | 分子名称: | (2E)-3-[7-(diethylamino)-2-oxo-2H-1-benzopyran-3-yl]prop-2-enal, bound form, ACETATE ION, ... | 著者 | Bingham, C.R, Geiger, J.H, Borhan, B. | 登録日 | 2022-06-06 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Light controlled reversible Michael addition of cysteine: a new tool for dynamic site-specific labeling of proteins. Analyst, 148, 2023
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