6XOG
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![BU of 6xog by Molmil](/molmil-images/mine/6xog) | Structure of SUMO1-ML786519 adduct bound to SAE | 分子名称: | SULFATE ION, SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ... | 著者 | Sintchak, M, Lane, W, Bump, N. | 登録日 | 2020-07-07 | 公開日 | 2021-03-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer. J.Med.Chem., 64, 2021
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6XOI
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![BU of 6xoi by Molmil](/molmil-images/mine/6xoi) | Structure of SUMO1-ML00752641 adduct bound to SAE | 分子名称: | SULFATE ION, SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ... | 著者 | Sintchak, M, Lane, W, Bump, N. | 登録日 | 2020-07-07 | 公開日 | 2021-03-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer. J.Med.Chem., 64, 2021
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5FQ2
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![BU of 5fq2 by Molmil](/molmil-images/mine/5fq2) | |
6XOH
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![BU of 6xoh by Molmil](/molmil-images/mine/6xoh) | Structure of SUMO1-ML00789344 adduct bound to SAE | 分子名称: | SULFATE ION, SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ... | 著者 | Sintchak, M, Lane, W, Bump, N. | 登録日 | 2020-07-07 | 公開日 | 2021-03-24 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.226 Å) | 主引用文献 | Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer. J.Med.Chem., 64, 2021
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1Y8Q
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![BU of 1y8q by Molmil](/molmil-images/mine/1y8q) | SUMO E1 ACTIVATING ENZYME SAE1-SAE2-MG-ATP COMPLEX | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Ubiquitin-like 1 activating enzyme E1A, ... | 著者 | Lois, L.M, Lima, C.D. | 登録日 | 2004-12-13 | 公開日 | 2005-01-25 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structures of the SUMO E1 provide mechanistic insights into SUMO activation and E2 recruitment to E1 Embo J., 24, 2005
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3KYC
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![BU of 3kyc by Molmil](/molmil-images/mine/3kyc) | Human SUMO E1 complex with a SUMO1-AMP mimic | 分子名称: | 5'-deoxy-5'-(sulfamoylamino)adenosine, SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ... | 著者 | Lima, C.D. | 登録日 | 2009-12-05 | 公開日 | 2010-02-16 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Active site remodelling accompanies thioester bond formation in the SUMO E1. Nature, 463, 2010
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6CWY
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![BU of 6cwy by Molmil](/molmil-images/mine/6cwy) | Crystal structure of SUMO E1 in complex with an allosteric inhibitor | 分子名称: | GLYCEROL, MAGNESIUM ION, SULFATE ION, ... | 著者 | Lv, Z, Yuan, L, Atkison, J.H, Williams, K.M, Olsen, S.K. | 登録日 | 2018-04-01 | 公開日 | 2019-01-16 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.462 Å) | 主引用文献 | Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme. Nat Commun, 9, 2018
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4W5V
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![BU of 4w5v by Molmil](/molmil-images/mine/4w5v) | Crystal structure of Human SUMO E2-conjugating enzyme (Ubc9) in complex with E1-activating enzyme (Uba2) ubiquitin fold domain (Ufd) | 分子名称: | FORMIC ACID, GLYCEROL, POTASSIUM ION, ... | 著者 | Boucher, L.E, Reiter, K.H, Matunis, M.J, Bosch, J. | 登録日 | 2014-08-19 | 公開日 | 2015-09-09 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of human SUMO complex To Be Published
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3KYD
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![BU of 3kyd by Molmil](/molmil-images/mine/3kyd) | Human SUMO E1~SUMO1-AMP tetrahedral intermediate mimic | 分子名称: | 1,2-ETHANEDIOL, 5'-{[(3-aminopropyl)sulfonyl]amino}-5'-deoxyadenosine, SUMO-activating enzyme subunit 1, ... | 著者 | Lima, C.D. | 登録日 | 2009-12-05 | 公開日 | 2010-02-16 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Active site remodelling accompanies thioester bond formation in the SUMO E1. Nature, 463, 2010
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1Y8R
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![BU of 1y8r by Molmil](/molmil-images/mine/1y8r) | |
6CWZ
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![BU of 6cwz by Molmil](/molmil-images/mine/6cwz) | Crystal structure of apo SUMO E1 | 分子名称: | SUMO-activating enzyme subunit 1, SUMO-activating enzyme subunit 2, ZINC ION | 著者 | Lv, Z, Yuan, L, Atkison, J.H, Williams, K.M, Olsen, S.K. | 登録日 | 2018-04-01 | 公開日 | 2019-01-16 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme. Nat Commun, 9, 2018
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2PX9
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![BU of 2px9 by Molmil](/molmil-images/mine/2px9) | The intrinsic affinity between E2 and the Cys domain of E1 in Ubiquitin-like modifications | 分子名称: | SUMO-activating enzyme subunit 2, SUMO-conjugating enzyme UBC9 | 著者 | Wang, J.H, Hu, W.D, Cai, S, Lee, B, Song, J, Chen, Y. | 登録日 | 2007-05-14 | 公開日 | 2007-07-24 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | The intrinsic affinity between E2 and the Cys domain of E1 in ubiquitin-like modifications. Mol.Cell, 27, 2007
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