3UBD
| Structure of N-terminal domain of RSK2 kinase in complex with flavonoid glycoside SL0101 | 分子名称: | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-chromen-3-yl 3,4-di-O-acetyl-6-deoxy-alpha-L-mannopyranoside, Ribosomal protein S6 kinase alpha-3 | 著者 | Utepbergenov, D, Derewenda, U, Derewenda, Z.S. | 登録日 | 2011-10-24 | 公開日 | 2012-09-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Insights into the Inhibition of the p90 Ribosomal S6 Kinase (RSK) by the Flavonol Glycoside SL0101 from the 1.5 A Crystal Structure of the N-Terminal Domain of RSK2 with Bound Inhibitor. Biochemistry, 51, 2012
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4EL9
| Structure of N-terminal kinase domain of RSK2 with afzelin | 分子名称: | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-chromen-3-yl 6-deoxy-alpha-L-mannopyranoside, Ribosomal protein S6 kinase alpha-3 | 著者 | Utepbergenov, D, Derewenda, U, Derewenda, Z.S. | 登録日 | 2012-04-10 | 公開日 | 2012-09-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Insights into the Inhibition of the p90 Ribosomal S6 Kinase (RSK) by the Flavonol Glycoside SL0101 from the 1.5 A Crystal Structure of the N-Terminal Domain of RSK2 with Bound Inhibitor. Biochemistry, 51, 2012
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4GUE
| Structure of N-terminal kinase domain of RSK2 with flavonoid glycoside quercitrin | 分子名称: | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-3-yl 6-deoxy-alpha-L-mannopyranoside, MAGNESIUM ION, Ribosomal protein S6 kinase alpha-3, ... | 著者 | Derewenda, U, Utepbergenov, D, Szukalska, G, Derewenda, Z.S. | 登録日 | 2012-08-29 | 公開日 | 2013-01-30 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Identification of quercitrin as an inhibitor of the p90 S6 ribosomal kinase (RSK): structure of its complex with the N-terminal domain of RSK2 at 1.8 A resolution. Acta Crystallogr.,Sect.D, 69, 2013
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3G51
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5O1S
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2QR7
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2QR8
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4MAO
| RSK2 T493M C-Terminal Kinase Domain in Complex with RMM58 | 分子名称: | (2Z)-2-(1H-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1H-indazol-5-yl]prop-2-enenitrile, Ribosomal protein S6 kinase alpha-3, SODIUM ION | 著者 | Miller, R.M, Taunton, J. | 登録日 | 2013-08-16 | 公開日 | 2014-10-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Design of reversible, cysteine-targeted Michael acceptors guided by kinetic and computational analysis. J.Am.Chem.Soc., 136, 2014
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4M8T
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