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PDB: 9 件

3UBD
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Structure of N-terminal domain of RSK2 kinase in complex with flavonoid glycoside SL0101
分子名称: 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-chromen-3-yl 3,4-di-O-acetyl-6-deoxy-alpha-L-mannopyranoside, Ribosomal protein S6 kinase alpha-3
著者Utepbergenov, D, Derewenda, U, Derewenda, Z.S.
登録日2011-10-24
公開日2012-09-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Insights into the Inhibition of the p90 Ribosomal S6 Kinase (RSK) by the Flavonol Glycoside SL0101 from the 1.5 A Crystal Structure of the N-Terminal Domain of RSK2 with Bound Inhibitor.
Biochemistry, 51, 2012
4EL9
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Structure of N-terminal kinase domain of RSK2 with afzelin
分子名称: 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-chromen-3-yl 6-deoxy-alpha-L-mannopyranoside, Ribosomal protein S6 kinase alpha-3
著者Utepbergenov, D, Derewenda, U, Derewenda, Z.S.
登録日2012-04-10
公開日2012-09-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Insights into the Inhibition of the p90 Ribosomal S6 Kinase (RSK) by the Flavonol Glycoside SL0101 from the 1.5 A Crystal Structure of the N-Terminal Domain of RSK2 with Bound Inhibitor.
Biochemistry, 51, 2012
4GUE
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Structure of N-terminal kinase domain of RSK2 with flavonoid glycoside quercitrin
分子名称: 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-3-yl 6-deoxy-alpha-L-mannopyranoside, MAGNESIUM ION, Ribosomal protein S6 kinase alpha-3, ...
著者Derewenda, U, Utepbergenov, D, Szukalska, G, Derewenda, Z.S.
登録日2012-08-29
公開日2013-01-30
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Identification of quercitrin as an inhibitor of the p90 S6 ribosomal kinase (RSK): structure of its complex with the N-terminal domain of RSK2 at 1.8 A resolution.
Acta Crystallogr.,Sect.D, 69, 2013
3G51
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Structural diversity of the active conformation of the N-terminal kinase domain of p90 ribosomal S6 kinase 2
分子名称: PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Ribosomal protein S6 kinase alpha-3
著者Kurinov, I.
登録日2009-02-04
公開日2009-12-15
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural diversity of the active N-terminal kinase domain of p90 ribosomal S6 kinase 2
Plos One, 4, 2009
5O1S
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Dimethyl fumarate is an allosteric covalent inhibitor of the p90 ribosomal S6 kinases
分子名称: Dimethyl fumarate, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Andersen, J.L, Nissen, P.
登録日2017-05-19
公開日2018-05-30
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Dimethyl fumarate is an allosteric covalent inhibitor of the p90 ribosomal S6 kinases.
Nat Commun, 9, 2018
2QR7
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2.0A X-ray structure of C-terminal kinase domain of p90 ribosomal S6 kinase 2: Se-Met derivative
分子名称: Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Malakhova, M, Tereshko, V, Dong, Z.
登録日2007-07-27
公開日2007-12-11
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for activation of the autoinhibitory C-terminal kinase domain of p90 RSK2.
Nat.Struct.Mol.Biol., 15, 2008
2QR8
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2.0A X-ray structure of C-terminal kinase domain of p90 ribosomal S6 kinase 2 (RSK2)
分子名称: Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Tereshko, V, Malakhova, M, Dong, Z.
登録日2007-07-27
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural basis for activation of the autoinhibitory C-terminal kinase domain of p90 RSK2.
Nat.Struct.Mol.Biol., 15, 2008
4MAO
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RSK2 T493M C-Terminal Kinase Domain in Complex with RMM58
分子名称: (2Z)-2-(1H-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1H-indazol-5-yl]prop-2-enenitrile, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Miller, R.M, Taunton, J.
登録日2013-08-16
公開日2014-10-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Design of reversible, cysteine-targeted Michael acceptors guided by kinetic and computational analysis.
J.Am.Chem.Soc., 136, 2014
4M8T
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RSK2 T493M C-Terminal Kinase Domain in complex with 3-(3-(1H-pyrazol-4-yl)phenyl)-2-cyanoacrylamide
分子名称: (2E)-2-cyano-3-[3-(1H-pyrazol-4-yl)phenyl]prop-2-enamide, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Miller, R.M, Taunton, J.
登録日2013-08-13
公開日2014-10-22
最終更新日2014-11-26
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Covalent docking of large libraries for the discovery of chemical probes.
Nat.Chem.Biol., 10, 2014

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件を2024-07-10に公開中

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