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PDB: 70 件

6B6A
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BU of 6b6a by Molmil
Beta-Lactamase, 2secs timepoint, mixed, shards crystal form
分子名称: (2R)-2-[(1S)-1-{[(2Z)-2-(2-amino-1,3-thiazol-4-yl)-2-(methoxyimino)acetyl]amino}-2-hydroxyethyl]-5-methylidene-5,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, Beta-lactamase, Ceftriaxone, ...
著者Pandey, S, Schmidt, M.
登録日2017-10-01
公開日2018-06-27
最終更新日2020-01-15
実験手法X-RAY DIFFRACTION (2.298 Å)
主引用文献Enzyme intermediates captured "on the fly" by mix-and-inject serial crystallography.
BMC Biol., 16, 2018
8EC4
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BU of 8ec4 by Molmil
XFEL structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 240ms
分子名称: Beta-lactamase, PHOSPHATE ION, TRANS-ENAMINE INTERMEDIATE OF SULBACTAM
著者Malla, T.N, Schmidt, M.
登録日2022-09-01
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
7K8E
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BU of 7k8e by Molmil
Beta-lactamase mixed with Ceftriaxone, 5ms
分子名称: Beta-lactamase, Ceftriaxone, PHOSPHATE ION
著者Pandey, S, Schmidt, M.
登録日2020-09-26
公開日2021-09-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.40005636 Å)
主引用文献Observation of substrate diffusion and ligand binding in enzyme crystals using high-repetition-rate mix-and-inject serial crystallography
Iucrj, 8, 2021
6B5X
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BU of 6b5x by Molmil
Beta-Lactamase, unmixed shards crystal form
分子名称: Beta-lactamase, PHOSPHATE ION
著者Pandey, S.
登録日2017-09-29
公開日2018-06-27
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Enzyme intermediates captured "on the fly" by mix-and-inject serial crystallography.
BMC Biol., 16, 2018
3VFH
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BU of 3vfh by Molmil
BlaC E166A CDC-1 Acyl-Intermediate
分子名称: (2R)-5-methylidene-2-{(1R)-2-oxo-1-[(phenylacetyl)amino]ethyl}-5,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, Beta-lactamase, PHOSPHATE ION
著者Mire, J.A, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2012-01-09
公開日2012-09-19
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献BlaC-Specific Fluorogenic Probes for Rapid Tuberculosis Detection
To be Published
7K8F
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BU of 7k8f by Molmil
Beta-lactamase mixed with Ceftriaxone, 10ms
分子名称: Beta-lactamase, Ceftriaxone, PHOSPHATE ION
著者Pandey, S, Schmidt, M.
登録日2020-09-26
公開日2021-09-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.60003138 Å)
主引用文献Observation of substrate diffusion and ligand binding in enzyme crystals using high-repetition-rate mix-and-inject serial crystallography
Iucrj, 8, 2021
7K8H
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BU of 7k8h by Molmil
Beta-lactamase mixed with Ceftriaxone, 50ms
分子名称: Beta-lactamase, Ceftriaxone, PHOSPHATE ION
著者Pandey, S, Schmidt, M.
登録日2020-09-27
公開日2021-09-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.60006261 Å)
主引用文献Observation of substrate diffusion and ligand binding in enzyme crystals using high-repetition-rate mix-and-inject serial crystallography
Iucrj, 8, 2021
8GCS
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BU of 8gcs by Molmil
XFEL structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 3 ms
分子名称: Beta-lactamase, PHOSPHATE ION
著者Malla, T.N, Schmidt, M.
登録日2023-03-03
公開日2023-09-20
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
8EBI
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BU of 8ebi by Molmil
XFEL structure of beta lactamase microcrystals mixed with sulbactam solution for 15ms
分子名称: Beta-lactamase, PHOSPHATE ION, TRANS-ENAMINE INTERMEDIATE OF SULBACTAM
著者Malla, T.N, Schmidt, M.
登録日2022-08-31
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
7K8K
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BU of 7k8k by Molmil
Beta-lactamase mixed with Sulbactam, 60ms
分子名称: Beta-lactamase, PHOSPHATE ION, SULBACTAM, ...
著者Pandey, S, Schmidt, M.
登録日2020-09-27
公開日2021-09-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Observation of substrate diffusion and ligand binding in enzyme crystals using high-repetition-rate mix-and-inject serial crystallography
Iucrj, 8, 2021
8ECF
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BU of 8ecf by Molmil
Cryo structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 3 hours
分子名称: Beta-lactamase, PHOSPHATE ION, TRANS-ENAMINE INTERMEDIATE OF SULBACTAM
著者Malla, T.N, Schmidt, M.
登録日2022-09-01
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.736 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
8GCT
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BU of 8gct by Molmil
XFEL structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 6 ms
分子名称: Beta-lactamase, PHOSPHATE ION
著者Malla, T.N, Schmidt, M.
登録日2023-03-03
公開日2023-09-20
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
6B5Y
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BU of 6b5y by Molmil
Beta-lactamase, mixed with Ceftriaxone, 30ms time point, Shards crystal form
分子名称: Beta-lactamase, Ceftriaxone, PHOSPHATE ION
著者Pandey, S, Schmidt, M.
登録日2017-09-29
公開日2018-06-27
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Enzyme intermediates captured "on the fly" by mix-and-inject serial crystallography.
BMC Biol., 16, 2018
3VFF
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BU of 3vff by Molmil
BlaC E166A CDC-OMe Acyl-Intermediate Complex
分子名称: (2R)-2-[(1S)-1-(benzoylamino)-1-methoxy-2-oxoethyl]-5-methylidene-5,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, Beta-lactamase, PHOSPHATE ION
著者Mire, J.A, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2012-01-09
公開日2012-09-19
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.777 Å)
主引用文献BlaC-Specific Fluorogenic Probes for Rapid Tuberculosis Detection
To be Published
8EBR
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BU of 8ebr by Molmil
XFEL structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 30ms
分子名称: Beta-lactamase, PHOSPHATE ION, SULBACTAM, ...
著者Malla, T.N, Schmidt, M.
登録日2022-08-31
公開日2023-03-08
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
3NCK
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BU of 3nck by Molmil
Crystal Structure of BlaC-E166A covalently bound with Nafcillin
分子名称: (2R,4S)-2-[(1R)-1-{[(2-ethoxynaphthalen-1-yl)carbonyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, Beta-lactamase
著者Tremblay, L.W, Blanchard, J.S.
登録日2010-06-04
公開日2011-12-14
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献BlaC-E166A covalently bound with cephalosporins and penicillins
To be Published
7K8L
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BU of 7k8l by Molmil
Beta-lactamase, Unmixed
分子名称: Beta-lactamase, PHOSPHATE ION
著者Pandey, S, Schmidt, M.
登録日2020-09-27
公開日2021-09-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.8000102 Å)
主引用文献Observation of substrate diffusion and ligand binding in enzyme crystals using high-repetition-rate mix-and-inject serial crystallography
Iucrj, 8, 2021
3ZHH
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BU of 3zhh by Molmil
X-ray structure of the full-length beta-lactamase from M.tuberculosis
分子名称: BETA-LACTAMASE, SULFATE ION
著者Feiler, C, Fisher, A.C, Marrichi, M.J, Wright, L, Schmidpeter, P.A.M, Blankenfeldt, W, Pavelka, M, DeLisa, M.P.
登録日2012-12-21
公開日2013-09-25
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Directed Evolution of Mycobacterium Tuberculosis Beta-Lactamase Reveals Gatekeeper Residue that Regulates Antibiotic Resistance and Catalytic Efficiency.
Plos One, 8, 2013
4EBN
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BU of 4ebn by Molmil
BlaC Amoxicillin Acyl-Intermediate Complex
分子名称: 2-{1-[2-AMINO-2-(4-HYDROXY-PHENYL)-ACETYLAMINO]-2-OXO-ETHYL}-5,5-DIMETHYL-THIAZOLIDINE-4-CARBOXYLIC ACID, Beta-lactamase, PHOSPHATE ION
著者Mire, J.A, TB Structural Genomics Consortium (TBSGC)
登録日2012-03-23
公開日2013-04-03
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Faropenem is Effective Against Mycobacterium tuberculosis in vitro and in vivo
To be Published
8GCX
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BU of 8gcx by Molmil
XFEL structure of Mycobacterium tuberculosis beta lactamase microcrystals mixed with sulbactam for 700 ms
分子名称: Beta-lactamase, PHOSPHATE ION, TRANS-ENAMINE INTERMEDIATE OF SULBACTAM
著者Malla, T.N, Schmidt, M.
登録日2023-03-03
公開日2023-09-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Heterogeneity in M. tuberculosis beta-lactamase inhibition by Sulbactam.
Nat Commun, 14, 2023
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件を2024-07-10に公開中

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