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PDB: 5 件

3K4A
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BU of 3k4a by Molmil
Crystal structure of selenomethionine substituted E. coli beta-glucuronidase
分子名称: Beta-glucuronidase
著者Wallace, B.D, Orans, J, Redinbo, M.R.
登録日2009-10-05
公開日2010-11-17
最終更新日2024-11-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Alleviating cancer drug toxicity by inhibiting a bacterial enzyme.
Science, 330, 2010
3K46
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BU of 3k46 by Molmil
Crystal structure of full-length E. coli beta-glucuronidase
分子名称: Beta-glucuronidase
著者Wallace, B.D, Lane, K.T, Redinbo, M.R.
登録日2009-10-05
公開日2010-11-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Alleviating cancer drug toxicity by inhibiting a bacterial enzyme.
Science, 330, 2010
3LPF
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BU of 3lpf by Molmil
Structure of E. coli beta-Glucuronidase bound with a novel, potent inhibitor 1-((6,7-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl)-1-(2-hydroxyethyl)-3-(3-methoxyphenyl)thiourea
分子名称: 1-[(6,7-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-(2-hydroxyethyl)-3-(3-methoxyphenyl)thiourea, Beta-glucuronidase
著者Wallace, B.D, Redinbo, M.R.
登録日2010-02-05
公開日2010-11-17
最終更新日2024-11-27
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Alleviating cancer drug toxicity by inhibiting a bacterial enzyme.
Science, 330, 2010
3LPG
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BU of 3lpg by Molmil
Structure of E. coli beta-Glucuronidase bound with a novel, potent inhibitor 3-(2-fluorophenyl)-1-(2-hydroxyethyl)-1-((6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl)urea
分子名称: 3-(2-fluorophenyl)-1-(2-hydroxyethyl)-1-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]urea, Beta-glucuronidase
著者Wallace, B.D, Redinbo, M.R.
登録日2010-02-05
公開日2010-11-17
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.425 Å)
主引用文献Alleviating cancer drug toxicity by inhibiting a bacterial enzyme.
Science, 330, 2010
3K4D
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BU of 3k4d by Molmil
Crystal structure of E. coli beta-glucuronidase with the glucaro-d-lactam inhibitor bound
分子名称: (2S,3R,4S,5R)-3,4,5-trihydroxy-6-oxopiperidine-2-carboxylic acid, Beta-glucuronidase
著者Wallace, B.D, Redinbo, M.R.
登録日2009-10-05
公開日2010-11-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.393 Å)
主引用文献Alleviating cancer drug toxicity by inhibiting a bacterial enzyme.
Science, 330, 2010

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件を2025-07-09に公開中

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