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PDB: 3 件

7NI4
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BU of 7ni4 by Molmil
Human ATM kinase domain with bound M4076 inhibitor
分子名称: 8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-one, Serine-protein kinase ATM, ZINC ION
著者Stakyte, K, Rotheneder, M.
登録日2021-02-11
公開日2021-09-01
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Molecular basis of human ATM kinase inhibition.
Nat.Struct.Mol.Biol., 28, 2021
7NI5
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BU of 7ni5 by Molmil
Human ATM kinase with bound inhibitor KU-55933
分子名称: 2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one, Serine-protein kinase ATM, ZINC ION
著者Bartho, J.D, Stakyte, K, Rotheneder, M, Lammens, K, Hopfner, K.P.
登録日2021-02-11
公開日2021-09-01
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.78 Å)
主引用文献Molecular basis of human ATM kinase inhibition.
Nat.Struct.Mol.Biol., 28, 2021
7NI6
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BU of 7ni6 by Molmil
Human ATM kinase with bound ATPyS
分子名称: MAGNESIUM ION, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, Serine-protein kinase ATM, ...
著者Stakyte, K, Rotheneder, M, Lammens, K, Bartho, J.D.
登録日2021-02-11
公開日2021-09-01
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Molecular basis of human ATM kinase inhibition.
Nat.Struct.Mol.Biol., 28, 2021

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件を2024-07-10に公開中

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