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PDB: 8 件

7MF4
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BU of 7mf4 by Molmil
Crystal structure of Trypanosoma cruzi cytosolic Malic Enzyme
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CITRIC ACID, Malic enzyme
著者Ranzani, A.T, Cordeiro, A.T.
登録日2021-04-08
公開日2021-07-28
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W29
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BU of 6w29 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC013)
分子名称: 3,5-bis(fluoranyl)-~{N}-[3-[(4-methoxyphenyl)sulfamoyl]phenyl]benzamide, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CITRIC ACID, ...
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-05
公開日2021-03-10
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W2N
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BU of 6w2n by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC009)
分子名称: 3,5-bis(fluoranyl)-~{N}-[3-[(2-fluoranyl-4-methoxy-phenyl)sulfamoyl]phenyl]benzamide, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CITRIC ACID, ...
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-06
公開日2021-03-10
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W59
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BU of 6w59 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC063)
分子名称: 3,5-bis(fluoranyl)-~{N}-[3-[[4-(trifluoromethyloxy)phenyl]sulfamoyl]phenyl]benzamide, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Malic enzyme
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-12
公開日2021-03-17
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W49
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BU of 6w49 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC010)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CITRIC ACID, Malic enzyme, ...
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-10
公開日2021-04-07
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W57
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BU of 6w57 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC069)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Malic enzyme, ~{N}-[5-[[4-[bis(fluoranyl)methoxy]phenyl]sulfamoyl]-2-chloranyl-phenyl]-3,5-bis(fluoranyl)benzamide
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-12
公開日2021-04-07
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W53
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BU of 6w53 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC070)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Malic enzyme, N-(2-chloro-5-{[4-(trifluoromethoxy)phenyl]sulfamoyl}phenyl)-3,5-difluorobenzamide
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-12
公開日2021-04-07
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021
6W56
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BU of 6w56 by Molmil
Trypanosoma cruzi Malic Enzyme in complex with inhibitor (MEC062)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Malic enzyme, ~{N}-[3-[[4-[bis(fluoranyl)methoxy]phenyl]sulfamoyl]phenyl]-3,5-bis(fluoranyl)benzamide
著者Mercaldi, G.F, Fagundes, M, Faria, J.N, Cordeiro, A.T.
登録日2020-03-12
公開日2021-04-07
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Trypanosoma cruzi Malic Enzyme Is the Target for Sulfonamide Hits from the GSK Chagas Box.
Acs Infect Dis., 7, 2021

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件を2024-06-26に公開中

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