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PDB: 5 件

6P11
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BU of 6p11 by Molmil
Structure of spastin AAA domain (T692A mutant) in complex with JNJ-7706621 inhibitor
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1H-1,2,4-triazol-3-yl}amino)benzenesulfonamide, Drosophila melanogaster Spastin AAA domain, ...
著者Pisa, R, Cupido, T, Kapoor, T.M.
登録日2019-05-17
公開日2019-07-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26, 2019
6P10
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BU of 6p10 by Molmil
Structure of spastin AAA domain (N527C mutant) in complex with JNJ-7706621 inhibitor
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1H-1,2,4-triazol-3-yl}amino)benzenesulfonamide, Drosophila melanogaster Spastin AAA domain, ...
著者Pisa, R, Cupido, T, Kapoor, T.M.
登録日2019-05-17
公開日2019-07-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.301 Å)
主引用文献Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26, 2019
6P12
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BU of 6p12 by Molmil
Structure of spastin AAA domain (wild-type) in complex with diaminotriazole-based inhibitor
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 3-{[5-amino-1-(2-fluoro-6-methoxybenzene-1-carbonyl)-1H-1,2,4-triazol-3-yl]amino}-N-methylbenzamide, Drosophila melanogaster Spastin AAA domain, ...
著者Pisa, R, Cupido, T, Kapoor, T.M.
登録日2019-05-17
公開日2019-07-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.94131851 Å)
主引用文献Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26, 2019
6P14
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BU of 6p14 by Molmil
Structure of spastin AAA domain (T692A mutant) in complex with a diaminotriazole-based inhibitor (crystal form B)
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 3-{[5-amino-1-(2-fluoro-6-methoxybenzene-1-carbonyl)-1H-1,2,4-triazol-3-yl]amino}-N-methylbenzamide, ACETATE ION, ...
著者Pisa, R, Cupido, T, Kapoor, T.M.
登録日2019-05-17
公開日2019-07-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.93001127 Å)
主引用文献Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26, 2019
6P13
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BU of 6p13 by Molmil
Structure of spastin AAA domain (T692A mutant) in complex with a diaminotriazole-based inhibitor (crystal form A)
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 3-{[5-amino-1-(2-fluoro-6-methoxybenzene-1-carbonyl)-1H-1,2,4-triazol-3-yl]amino}-N-methylbenzamide, SULFATE ION, ...
著者Pisa, R, Cupido, T, Kapoor, T.M.
登録日2019-05-17
公開日2019-08-07
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26, 2019

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件を2024-07-10に公開中

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