7A2N
 
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7A2M
 
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7A2R
 
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2HDA
 
 | Yes SH3 domain | Descriptor: | Proto-oncogene tyrosine-protein kinase Yes, SULFATE ION | Authors: | Camara-Artigas, A, Luque, I, Ruiz-Sanz, J, Mateo, P.L, Martin-Garcia, J.M. | Deposit date: | 2006-06-20 | Release date: | 2007-04-17 | Last modified: | 2023-08-30 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Crystallographic structure of the SH3 domain of the human c-Yes tyrosine kinase: Loop flexibility and amyloid aggregation. Febs Lett., 581, 2007
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8P8K
 
 | Acyl-ACP thioesterase from Lemna paucicostata in complex with a thiazolopyridine | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-[2,6-bis(fluoranyl)phenyl]-6-chloranyl-[1,3]thiazolo[4,5-b]pyridine, Acyl-ACP thioesterase | Authors: | Freigang, J. | Deposit date: | 2023-06-01 | Release date: | 2023-09-20 | Last modified: | 2023-12-06 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | A Study in Scaffold Hopping: Discovery and Optimization of Thiazolopyridines as Potent Herbicides That Inhibit Acyl-ACP Thioesterase. J.Agric.Food Chem., 71, 2023
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7ZLX
 
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8QRT
 
 | Acyl-ACP thioesterase from Lemna paucicostata in complex with a spirolactam | Descriptor: | (5~{S})-7-[[2,6-bis(fluoranyl)phenyl]methyl]-3-(3-methylthiophen-2-yl)-1-oxa-2,7-diazaspiro[4.4]non-2-en-6-one, Acyl-acp thioesterase | Authors: | Freigang, J. | Deposit date: | 2023-10-09 | Release date: | 2024-02-21 | Last modified: | 2025-04-16 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Discovery and optimization of spirocyclic lactams that inhibit acyl-ACP thioesterase. Pest Manag Sci, 81, 2025
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8QS0
 
 | Acyl-ACP thioesterase from Lemna paucicostata in complex with a spirolactam | Descriptor: | (5~{S})-9-[[2,6-bis(fluoranyl)phenyl]methyl]-3-(3-methylthiophen-2-yl)-1-oxa-2,9-diazaspiro[4.5]dec-2-en-10-one, Acyl-acp thioesterase | Authors: | Freigang, J. | Deposit date: | 2023-10-10 | Release date: | 2024-02-21 | Last modified: | 2025-04-16 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Discovery and optimization of spirocyclic lactams that inhibit acyl-ACP thioesterase. Pest Manag Sci, 81, 2025
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2FQX
 
 | PnrA from Treponema pallidum complexed with guanosine | Descriptor: | GUANOSINE, Membrane lipoprotein tmpC | Authors: | Brautigam, C.A, Deka, R.K, Tomchick, D.R, Machius, M, Norgard, M.V. | Deposit date: | 2006-01-18 | Release date: | 2006-02-14 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | The PnrA (Tp0319; TmpC) lipoprotein represents a new family of bacterial purine nucleoside receptor encoded within an ATP-binding cassette (ABC)-like operon in Treponema pallidum J.Biol.Chem., 281, 2006
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2FQW
 
 | PnrA from Treponema pallidum as purified from E. coli (bound to inosine) | Descriptor: | INOSINE, Membrane lipoprotein tmpC | Authors: | Brautigam, C.A, Deka, R.K, Tomchick, D.R, Machius, M, Norgard, M.V. | Deposit date: | 2006-01-18 | Release date: | 2006-02-14 | Last modified: | 2024-02-14 | Method: | X-RAY DIFFRACTION (1.71 Å) | Cite: | The PnrA (Tp0319; TmpC) lipoprotein represents a new family of bacterial purine nucleoside receptor encoded within an ATP-binding cassette (ABC)-like operon in Treponema pallidum J.Biol.Chem., 281, 2006
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5OAZ
 
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5OAV
 
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8OJW
 
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8OJX
 
 | Streptavidin S112YK121E artificial metalloenzyme for carboamination | Descriptor: | IRIDIUM ION, Streptavidin, trichloro{(1,2,3,4,5-eta)-1,2,3,4-tetramethyl-5-[2-({5-[(3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentanoyl}amino)ethyl]cyclopentadienyl}rhodium(1+) | Authors: | Igareta, N.V, Ward, T.R. | Deposit date: | 2023-03-25 | Release date: | 2024-04-03 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Streptavidin WT artificial metalloenzyme for carboamination To Be Published
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5OB0
 
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5OB2
 
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2G93
 
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5OB1
 
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7PVR
 
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7PVQ
 
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7PVX
 
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7PW2
 
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7PVS
 
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7PVV
 
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7PW0
 
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