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PDB: 2 results

3VW6
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BU of 3vw6 by Molmil
Crystal structure of human apoptosis signal-regulating kinase 1 (ASK1) with imidazopyridine inhibitor
Descriptor: 4-tert-butyl-N-[6-(1H-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide, Mitogen-activated protein kinase kinase kinase 5
Authors:Terao, Y, Suzuki, H, Yoshikawa, M, Yashiro, H, Takekawa, S, Fujitani, Y, Okada, K, Inoue, Y, Yamamoto, Y, Nakagawa, H, Yao, S, Kawamoto, T, Uchikawa, O.
Deposit date:2012-08-06
Release date:2012-10-31
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Design and biological evaluation of imidazo[1,2-a]pyridines as novel and potent ASK1 inhibitors.
Bioorg. Med. Chem. Lett., 22, 2012
3WWG
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BU of 3wwg by Molmil
Crystal structure of the N-glycan-deficient variant N448A of isopullulanase complexed with isopanose
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Isopullulanase, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ...
Authors:Miyazaki, T, Yashiro, H, Nishikawa, A, Tonozuka, T.
Deposit date:2014-06-17
Release date:2014-11-12
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:The side chain of a glycosylated asparagine residue is important for the stability of isopullulanase
J.Biochem., 157, 2015

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