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PDB: 32 件

2KSM
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BU of 2ksm by Molmil
Central B domain of Rv0899 from Mycobacterium tuberculosis
分子名称: MYCOBACTERIUM TUBERCULOSIS RV0899/MT0922/OmpATb
著者Teriete, P, Yao, Y, Kolodzik, A, Yu, J, Song, H, Niederweis, M, Marassi, F.M.
登録日2010-01-07
公開日2010-02-02
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Mycobacterium tuberculosis Rv0899 adopts a mixed alpha/beta-structure and does not form a transmembrane beta-barrel.
Biochemistry, 49, 2010
4I3K
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BU of 4i3k by Molmil
Crystal structure of a metabolic reductase with 1-hydroxy-6-(4-hydroxybenzyl)-4-methylpyridin-2(1H)-one
分子名称: 1-hydroxy-6-(4-hydroxybenzyl)-4-methylpyridin-2(1H)-one, Isocitrate dehydrogenase [NADP] cytoplasmic, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Zheng, B, Yao, Y, Liu, Z, Deng, L, Anglin, J.L, Jiang, H, Prasad, B.V.V, Song, Y.
登録日2012-11-26
公開日2013-05-22
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.3056 Å)
主引用文献Crystallographic Investigation and Selective Inhibition of Mutant Isocitrate Dehydrogenase.
ACS Med Chem Lett, 4, 2013
2QC1
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BU of 2qc1 by Molmil
Crystal structure of the extracellular domain of the nicotinic acetylcholine receptor 1 subunit bound to alpha-bungarotoxin at 1.9 A resolution
分子名称: Acetylcholine receptor subunit alpha, Alpha-bungarotoxin, alpha-D-mannopyranose-(1-2)-alpha-D-mannopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]alpha-D-mannopyranose-(1-6)]alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
著者Dellisanti, C.D, Yao, Y, Stroud, J.C, Wang, Z, Chen, L.
登録日2007-06-18
公開日2007-08-07
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Crystal structure of the extracellular domain of nAChR alpha1 bound to alpha-bungarotoxin at 1.94 A resolution.
Nat.Neurosci., 10, 2007
2LCA
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Solution structure of the C domain of RV0899 from mycobacterium tuberculosis
分子名称: Uncharacterized protein Rv0899/MT0922
著者Marassi, F, Yao, Y.
登録日2011-04-26
公開日2012-01-04
最終更新日2023-12-06
実験手法SOLUTION NMR
主引用文献Molecular Structure and Peptidoglycan Recognition of Mycobacterium tuberculosis ArfA (Rv0899).
J.Mol.Biol., 416, 2012
4ID7
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BU of 4id7 by Molmil
ACK1 kinase in complex with the inhibitor cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol
分子名称: Activated CDC42 kinase 1, SULFATE ION, cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol
著者Jin, M, Wang, J, Kleinberg, A, Kadalbajoo, M, Siu, K, Cooke, A, Bittner, M, Yao, Y, Thelemann, A, Ji, Q, Bhagwat, S, Crew, A.P, Pachter, J, Epstein, D, Mulvihill, M.J.
登録日2012-12-11
公開日2013-01-30
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Discovery of potent, selective and orally bioavailable imidazo[1,5-a]pyrazine derived ACK1 inhibitors.
Bioorg.Med.Chem.Lett., 23, 2013
8Z3B
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BU of 8z3b by Molmil
Crystal structure of GSTd2
分子名称: Glutathione S-transferase delta
著者Mo, X, Yao, Y.
登録日2024-04-15
公開日2024-07-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Characterization of a Plutella xylostella GZTd2, evolved in isothiocyanate detoxification
To be published
5Z4U
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BU of 5z4u by Molmil
Crystal Structure of T2R-TTL complex with 7a3
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 4-(4-ethoxyphenyl)-1-methyl-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole, CALCIUM ION, ...
著者Lai, Q, Wang, Y, Yang, J, Yao, Y.
登録日2018-01-14
公開日2019-01-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.18 Å)
主引用文献Crystal Structure of T2R-TTL complex with 7a3
To Be Published
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件を2024-09-04に公開中

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