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PDB: 287 件

4OCQ
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BU of 4ocq by Molmil
N-acetylhexosamine 1-phosphate kinase in complex with GalNAc
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, N-acetylhexosamine 1-phosphate kinase
著者Li, T.L, Wang, K.C, Lyu, S.Y, Liu, Y.C, Chang, C.Y, Wu, C.J.
登録日2014-01-09
公開日2014-05-14
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.878 Å)
主引用文献Insights into the binding specificity and catalytic mechanism of N-acetylhexosamine 1-phosphate kinases through multiple reaction complexes.
Acta Crystallogr.,Sect.D, 70, 2014
7V3P
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BU of 7v3p by Molmil
Cryo-EM structure of the IGF1R/insulin complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Insulin A chain, Insulin B chain, ...
著者Zhang, J, Liu, C, Zhang, X, Wei, T, Wu, C.
登録日2021-08-11
公開日2022-08-17
最終更新日2024-10-16
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Cryo-EM structure of the IGF1R/insulin complex
To Be Published
7DV3
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BU of 7dv3 by Molmil
Structure of Sulfolobus solfataricus SegA-AMPPNP protein
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, SOJ protein (Soj)
著者Yen, C.Y, Lin, M.G, Wu, C.T, Hsiao, C.D, Sun, Y.J.
登録日2021-01-12
公開日2021-12-22
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Chromosome segregation in Archaea: SegA- and SegB-DNA complex structures provide insights into segrosome assembly.
Nucleic Acids Res., 49, 2021
7CEM
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BU of 7cem by Molmil
Crystal Structure of YbeA CP74 W7F
分子名称: Ribosomal RNA large subunit methyltransferase H,Ribosomal RNA large subunit methyltransferase H
著者Liu, C.Y, Wu, C.Y, Lai, C.H, Hsu, S.T.D, Lyu, P.C.
登録日2020-06-23
公開日2021-06-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.4251 Å)
主引用文献Crystal Structure of YbeA CP74 W7F
To Be Published
5Z0V
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BU of 5z0v by Molmil
Structural insight into the Zika virus capsid encapsulating the viral genome
分子名称: Extracellular solute-binding protein family 1,viral genome protein, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose
著者Li, T, Zhao, Q, Yang, X, Chen, C, Yang, K, Wu, C, Zhang, T, Duan, Y, Xue, X, Mi, K, Ji, X, Wang, Z, Yang, H.
登録日2017-12-21
公開日2018-04-11
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.913 Å)
主引用文献Structural insight into the Zika virus capsid encapsulating the viral genome.
Cell Res., 28, 2018
7XR0
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BU of 7xr0 by Molmil
Crystal structure of T2R-TTL-27a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-5-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of T2R-TTL-27a complex
To Be Published
7XQX
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BU of 7xqx by Molmil
Crystal structure of T2R-TTL-27a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-7-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.36 Å)
主引用文献Crystal structure of T2R-TT complex
To Be Published
7XR1
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BU of 7xr1 by Molmil
Crystal structure of T2R-TTL-3a complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-6-fluoranyl-N-(4-methoxyphenyl)-N-methyl-quinazolin-4-amine, CALCIUM ION, ...
著者Lun, T, Wu, C.Y.
登録日2022-05-09
公開日2023-05-17
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.81 Å)
主引用文献Crystal structure of T2R-TTL-3a complex
To Be Published
4LC7
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BU of 4lc7 by Molmil
Aminooxazoline inhibitor of BACE-1
分子名称: (3aR,7aR)-3a-[3-(5-chloropyridin-3-yl)phenyl]-3a,4,5,6,7,7a-hexahydro-1,3-benzoxazol-2-amine, Beta-Secretase-1, NICKEL (II) ION
著者Huestis, M.P, Liu, W, Volgraf, M, Purkey, H.E, Wu, C, Wang, W, Smith, D, Vigers, G.P.A, Dutcher, D, Hunt, K.W, Siu, M.
登録日2013-06-21
公開日2013-09-18
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Diethylaminosulfur Trifluoride-Mediated Intramolecular Cyclization of 2-hydroxycycloalkylureas to Fused Bicyclic Aminooxazoline Compounds and Evaluation of Their Biochemical Activity Against β-Secretase-1 (BACE-1)
Tetrahedron Lett., 2013
7CNM
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BU of 7cnm by Molmil
YDX in complex with tubulin
分子名称: (2~{S},4~{S})-4-[[2-[(1~{R},3~{R})-1-acetyloxy-4-methyl-3-[[(2~{S},3~{S})-3-methyl-2-[[(2~{R})-1-methylpiperidin-2-yl]carbonylamino]pentanoyl]amino]pentyl]-1,3-thiazol-4-yl]carbonylamino]-5-cyclohexyl-2-methyl-pentanoic acid, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Wang, Y.X, Wu, C.Y.
登録日2020-08-02
公開日2021-08-04
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献The high-resolution X-ray structure of vinca-domain inhibitors of microtubules provides a rational approach for drug design.
Febs Lett., 595, 2021
7CIW
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BU of 7ciw by Molmil
Crystal Structure of Agmatine N-Acetyltransferase mutant S171A in complex with Ac-Agm and CoA
分子名称: Agmatine N-acetyltransferase, COENZYME A, N-(4-carbamimidamidobutyl)ethanamide
著者Chen, J.J, Hu, I.C, Wu, C.Y, Lyu, P.C.
登録日2020-07-08
公開日2021-07-21
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal Structure of Agmatine N-Acetyltransferase mutant S171A in complex with Ac-Agm and CoA
To Be Published
7CNN
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BU of 7cnn by Molmil
vinorelbine in complex with tubulin
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, CHLORIDE ION, ...
著者Wang, Y.X, Wu, C.Y.
登録日2020-08-02
公開日2021-08-04
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The high-resolution X-ray structure of vinca-domain inhibitors of microtubules provides a rational approach for drug design.
Febs Lett., 595, 2021

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件を2024-10-16に公開中

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