5CHB
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![BU of 5chb by Molmil](/molmil-images/mine/5chb) | Crystal structure of nvPizza2-S16H58 coordinating a CdCl2 nanocrystal | Descriptor: | CADMIUM ION, CHLORIDE ION, SULFATE ION, ... | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2015-07-10 | Release date: | 2015-07-22 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.55 Å) | Cite: | Biomineralization of a Cadmium Chloride Nanocrystal by a Designed Symmetrical Protein Angew.Chem.Int.Ed.Engl., 54, 2015
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5F53
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4ZCN
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![BU of 4zcn by Molmil](/molmil-images/mine/4zcn) | Crystal structure of nvPizza2-S16S58 | Descriptor: | IODIDE ION, SULFATE ION, nvPizza2-S16S58 | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2015-04-16 | Release date: | 2015-07-01 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Crystal structure of nvPizza2-S16S58 To Be Published
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3WW9
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![BU of 3ww9 by Molmil](/molmil-images/mine/3ww9) | Crystal structure of the computationally designed Pizza6 protein | Descriptor: | GLYCEROL, SULFATE ION, pizza6 protein | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.33 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3WW8
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![BU of 3ww8 by Molmil](/molmil-images/mine/3ww8) | Crystal structure of the computationally designed Pizza3 protein | Descriptor: | GLYCEROL, Pizza3 protein, SULFATE ION | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.402 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3WWF
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![BU of 3wwf by Molmil](/molmil-images/mine/3wwf) | Crystal structure of the computationally designed Pizza2-SR protein | Descriptor: | pizza2sr-pb protein | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.601 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3WWB
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![BU of 3wwb by Molmil](/molmil-images/mine/3wwb) | Crystal structure of the computationally designed Pizza2-SR protein | Descriptor: | Pizza2-SR protein | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3WWA
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![BU of 3wwa by Molmil](/molmil-images/mine/3wwa) | Crystal structure of the computationally designed Pizza7 protein after heat treatment | Descriptor: | ISOPROPYL ALCOHOL, Pizza7H protein | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.988 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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3WW7
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![BU of 3ww7 by Molmil](/molmil-images/mine/3ww7) | Crystal structure of the computationally designed Pizza2 protein | Descriptor: | GLYCEROL, Pizza2 protein | Authors: | Voet, A.R.D, Noguchi, H, Addy, C, Simoncini, D, Terada, D, Unzai, S, Park, S.Y, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2014-06-17 | Release date: | 2014-10-08 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.697 Å) | Cite: | Computational design of a self-assembling symmetrical beta-propeller protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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6G6O
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![BU of 6g6o by Molmil](/molmil-images/mine/6g6o) | Crystal structure of the computationally designed Ika8 protein: crystal packing No.1 in P63 | Descriptor: | GLYCEROL, Ika8 | Authors: | Noguchi, H, Addy, C, Simoncini, D, Van Meervelt, L, Schiex, T, Zhang, K.Y.J, Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2018-04-01 | Release date: | 2018-11-28 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Computational design of symmetrical eight-bladed beta-propeller proteins. IUCrJ, 6, 2019
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3LPU
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![BU of 3lpu by Molmil](/molmil-images/mine/3lpu) | HIV integrase | Descriptor: | (2S)-2-(6-chloro-2-methyl-4-phenylquinolin-3-yl)pentanoic acid, 2-[3-[3-(2-hydroxyethoxy)propoxy]propoxy]ethanol, CALCIUM ION, ... | Authors: | Nicolet, S, Christ, F, Voet, A, Marchand, A, Strelkov, S.V, de Maeyer, M, Chaltin, P, Debyzer, Z. | Deposit date: | 2010-02-06 | Release date: | 2010-05-12 | Last modified: | 2021-11-10 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication. Nat.Chem.Biol., 6, 2010
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3LPT
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![BU of 3lpt by Molmil](/molmil-images/mine/3lpt) | HIV integrase | Descriptor: | (6-chloro-2-oxo-4-phenyl-1,2-dihydroquinolin-3-yl)acetic acid, 2-[3-[3-(2-hydroxyethoxy)propoxy]propoxy]ethanol, CALCIUM ION, ... | Authors: | Nicolet, S, Christ, F, Voet, A, Marchand, A, Strelkov, S.V, de Maeyer, M, Chaltin, P, Debyzer, Z. | Deposit date: | 2010-02-05 | Release date: | 2010-05-12 | Last modified: | 2021-11-10 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication. Nat.Chem.Biol., 6, 2010
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6TJG
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![BU of 6tjg by Molmil](/molmil-images/mine/6tjg) | Crystal structure of the computationally designed Cake8 protein | Descriptor: | (4S)-2-METHYL-2,4-PENTANEDIOL, Cake8 | Authors: | Laier, I, Mylemans, B, Noguchi, H, Voet, A.R.D. | Deposit date: | 2019-11-26 | Release date: | 2020-05-06 | Last modified: | 2024-05-01 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Structural plasticity of a designer protein sheds light on beta-propeller protein evolution. Febs J., 288, 2021
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6TJC
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![BU of 6tjc by Molmil](/molmil-images/mine/6tjc) | Crystal structure of the computationally designed Cake3 protein | Descriptor: | Cake3, GLYCEROL, PHOSPHATE ION | Authors: | Laier, I, Mylemans, B, Voet, A.R.D, Noguchi, H. | Deposit date: | 2019-11-26 | Release date: | 2020-05-06 | Last modified: | 2024-05-01 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structural plasticity of a designer protein sheds light on beta-propeller protein evolution. Febs J., 288, 2021
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5NSD
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![BU of 5nsd by Molmil](/molmil-images/mine/5nsd) | Co-crystal structure of NAMPT dimer with KPT-9274 | Descriptor: | (~{E})-3-(6-azanylpyridin-3-yl)-~{N}-[[5-[4-[4,4-bis(fluoranyl)piperidin-1-yl]carbonylphenyl]-7-(4-fluorophenyl)-1-benzofuran-2-yl]methyl]prop-2-enamide, GLYCEROL, Nicotinamide phosphoribosyltransferase, ... | Authors: | Neggers, J.E, Kwanten, B, Dierckx, T, Noguchi, H, Voet, A, Vercruysse, T, Baloglu, E, Senapedis, W, Jacquemyn, M, Daelemans, D. | Deposit date: | 2017-04-26 | Release date: | 2018-02-14 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.046 Å) | Cite: | Target identification of small molecules using large-scale CRISPR-Cas mutagenesis scanning of essential genes. Nat Commun, 9, 2018
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8RM6
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![BU of 8rm6 by Molmil](/molmil-images/mine/8rm6) | Crystal Structure of Human Androgen Receptor DNA Binding Domain Bound to its Response Element: C3(1)ARE | Descriptor: | C3(1)ARE_Chain C, C3(1)ARE_Chain D, Isoform 2 of Androgen receptor, ... | Authors: | Lee, X.Y, Helsen, C, Van Eynde, W, Voet, A, Claessens, F. | Deposit date: | 2024-01-05 | Release date: | 2024-04-24 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Structural mechanism underlying variations in DNA binding by the androgen receptor. J.Steroid Biochem.Mol.Biol., 241, 2024
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8RM7
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![BU of 8rm7 by Molmil](/molmil-images/mine/8rm7) | Crystal Structure of Human Androgen Receptor DNA Binding Domain Bound to its Response Element: MMTV-177 GRE/ARE | Descriptor: | Isoform 2 of Androgen receptor, MMTV-177 GRE/ARE Chain C, MMTV-177 GRE/ARE, ... | Authors: | Lee, X.Y, Helsen, C, Van Eynde, W, Voet, A, Claessens, F. | Deposit date: | 2024-01-05 | Release date: | 2024-04-24 | Method: | X-RAY DIFFRACTION (2.25 Å) | Cite: | Structural mechanism underlying variations in DNA binding by the androgen receptor. J.Steroid Biochem.Mol.Biol., 241, 2024
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5XG5
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![BU of 5xg5 by Molmil](/molmil-images/mine/5xg5) | Crystal structure of Mitsuba-1 with bound NAcGal | Descriptor: | 2-acetamido-2-deoxy-alpha-D-galactopyranose, MITSUBA-1 | Authors: | Terada, D, Voet, A.R.D, Kamata, K, Zhang, K.Y.J, Tame, J.R.H. | Deposit date: | 2017-04-12 | Release date: | 2017-07-12 | Last modified: | 2024-03-27 | Method: | X-RAY DIFFRACTION (1.54 Å) | Cite: | Computational design of a symmetrical beta-trefoil lectin with cancer cell binding activity. Sci Rep, 7, 2017
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5I1Z
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![BU of 5i1z by Molmil](/molmil-images/mine/5i1z) | Structure of nvPizza2-H16S58 | Descriptor: | SULFATE ION, nvPizza2-H16S58 | Authors: | Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2016-02-07 | Release date: | 2017-02-08 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Broken Symmetry: Partial domain swapping in an artificial trimeric protein To Be Published
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6Y7O
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![BU of 6y7o by Molmil](/molmil-images/mine/6y7o) | The complex between the eight-bladed symmetrical designer protein Tako8 and the silicotungstic acid Keggin (STA) | Descriptor: | Keggin (STA), Tako8 | Authors: | Vandebroek, L, Noguchi, H, Parac-Vogt, T.N, Van Meervelt, L, Voet, A.R.D. | Deposit date: | 2020-03-02 | Release date: | 2020-12-16 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Shape and Size Complementarity-Induced Formation of Supramolecular Protein Assemblies with Metal-Oxo Clusters Cryst.Growth Des., 2021
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6Y7P
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![BU of 6y7p by Molmil](/molmil-images/mine/6y7p) | The complex between the eight-bladed symmetrical designer protein Tako8 and 1:2 zirconium(IV) Wells-Dawson (ZrWD) | Descriptor: | Tako8, W-Zr-cluster | Authors: | Vandebroek, L, Noguchi, H, Parac-Vogt, T.N, Van Meervelt, L, Voet, A.R.D. | Deposit date: | 2020-03-02 | Release date: | 2020-12-16 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Shape and Size Complementarity-Induced Formation of Supramolecular Protein Assemblies with Metal-Oxo Clusters Cryst.Growth Des., 2021
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7ZCJ
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![BU of 7zcj by Molmil](/molmil-images/mine/7zcj) | Crystal structure of Pizza6-TNH-TSH with Silicotungstic Acid (STA) polyoxometalate | Descriptor: | Keggin (STA), Pizza6-TNH-TSH | Authors: | Wouters, S.M.L, Kamata, K, Takahashi, K, Vandebroek, L, Parac-Vogt, T.N, Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2022-03-28 | Release date: | 2023-04-19 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.56 Å) | Cite: | Mutational study of a symmetry matched protein-polyoxometalate interface To be published
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7ZPZ
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![BU of 7zpz by Molmil](/molmil-images/mine/7zpz) | Crystal structure of Pizza6-TSR-TSH with Silicotungstic Acid (STA) polyoxometalate | Descriptor: | Keggin (STA), Pizza6-TSR-TSH | Authors: | Wouters, S.M.L, Kamata, K, Takahashi, K, Vandebroek, L, Parac-Vogt, T.N, Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2022-04-29 | Release date: | 2023-05-10 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.57 Å) | Cite: | Mutational study of a symmetry matched protein-polyoxometalate interface To be published
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7ZQ2
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![BU of 7zq2 by Molmil](/molmil-images/mine/7zq2) | Crystal structure of Pizza6-RSH-TSH with Silicotungstic Acid (STA) polyoxometalate | Descriptor: | Keggin (STA), Pizza6-RSH-TSH | Authors: | Wouters, S.M.L, Kamata, K, Takahashi, K, Vandebroek, L, Parac-Vogt, T.N, Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2022-04-29 | Release date: | 2023-05-10 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Mutational study of a symmetry matched protein-polyoxometalate interface To be published
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7ZQG
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![BU of 7zqg by Molmil](/molmil-images/mine/7zqg) | Crystal structure of Pizza6-KSH-TSH with Silicotungstic Acid (STA) polyoxometalate | Descriptor: | Keggin (STA), Pizza6-KSH-TSH | Authors: | Wouters, S.M.L, Kamata, K, Takahashi, K, Vandebroek, L, Parac-Vogt, T.N, Tame, J.R.H, Voet, A.R.D. | Deposit date: | 2022-04-29 | Release date: | 2023-05-10 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Mutational study of a symmetry matched protein-polyoxometalate interface To be published
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