4UD7
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![BU of 4ud7 by Molmil](/molmil-images/mine/4ud7) | Structure of the stapled peptide YS-02 bound to MDM2 | 分子名称: | MDM2, YS-02 | 著者 | Tan, Y.S, Reeks, J, Brown, C.J, Jennings, C.E, Eapen, R.S, Tng, Q.S, Thean, D, Ying, Y.T, Gago, F.J.F, Lane, D.P, Noble, M.E.M, Verma, C. | 登録日 | 2014-12-08 | 公開日 | 2016-01-13 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Benzene Probes in Molecular Dynamics Simulations Reveal Novel Binding Sites for Ligand Design. J Phys Chem Lett, 7, 2016
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4UE1
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![BU of 4ue1 by Molmil](/molmil-images/mine/4ue1) | Structure of the stapled peptide YS-01 bound to MDM2 | 分子名称: | E3 UBIQUITIN-PROTEIN LIGASE MDM2, YS-01 | 著者 | Tan, Y.S, Reeks, J, Brown, C.J, Jennings, C.E, Eapen, R.S, Tng, Q.S, Thean, D, Ying, Y.T, Gago, F.J.F, Lane, D.P, Noble, M.E.M, Verma, C. | 登録日 | 2014-12-14 | 公開日 | 2016-01-13 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Benzene Probes in Molecular Dynamics Simulations Reveal Novel Binding Sites for Ligand Design. J Phys Chem Lett, 7, 2016
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5WED
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8HP3
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![BU of 8hp3 by Molmil](/molmil-images/mine/8hp3) | Crystal structure of meso-diaminopimelate dehydrogenase from Prevotella timonensis | 分子名称: | 1,2-ETHANEDIOL, Meso-diaminopimelate D-dehydrogenase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Tan, Y, Song, W. | 登録日 | 2022-12-11 | 公開日 | 2023-12-13 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (3.07 Å) | 主引用文献 | Rational Design of Meso -Diaminopimelate Dehydrogenase with Enhanced Reductive Amination Activity for Efficient Production of d- p -Hydroxyphenylglycine. Appl.Environ.Microbiol., 89, 2023
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8HP0
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5I1Q
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![BU of 5i1q by Molmil](/molmil-images/mine/5i1q) | Second bromodomain of TAF1 bound to a pyrrolopyridone compound | 分子名称: | 3-[6-(but-3-en-1-yl)-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl]-N,N-dimethylbenzamide, Transcription initiation factor TFIID subunit 1 | 著者 | Tang, Y, Poy, F, Bellon, S.F. | 登録日 | 2016-01-09 | 公開日 | 2016-06-08 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains. J.Med.Chem., 59, 2016
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5I29
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![BU of 5i29 by Molmil](/molmil-images/mine/5i29) | TAF1(2) bound to a pyrrolopyridone compound | 分子名称: | CALCIUM ION, N,N-dimethyl-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)benzamide, Transcription initiation factor TFIID subunit 1 | 著者 | Tang, Y, Poy, F, Bellon, S.F. | 登録日 | 2016-02-08 | 公開日 | 2016-06-08 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.21 Å) | 主引用文献 | Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains. J.Med.Chem., 59, 2016
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7YPD
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7VU8
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![BU of 7vu8 by Molmil](/molmil-images/mine/7vu8) | L7-Tir domain with bound ligand | 分子名称: | 2',3'- cyclic AMP, Flax rust resistance protein | 著者 | Tan, Y, Xu, C, Yu, D, Song, W, Wu, B, Schulze-Lefert, P, Chai, J. | 登録日 | 2021-11-01 | 公開日 | 2022-06-01 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | TIR domains of plant immune receptors are 2',3'-cAMP/cGMP synthetases mediating cell death. Cell, 185, 2022
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7X5L
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![BU of 7x5l by Molmil](/molmil-images/mine/7x5l) | Tir-dsDNA complex, the initial binding state | 分子名称: | DNA (5'-D(*AP*TP*AP*AP*AP*TP*TP*A)-3'), DNA (5'-D(*TP*TP*AP*AP*TP*TP*AP*A)-3'), Flax rust resistance protein | 著者 | Tan, Y, Xu, C, Yu, D, Song, W, Wu, B, Schulze-Lefert, P, Chai, J. | 登録日 | 2022-03-04 | 公開日 | 2022-06-01 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | TIR domains of plant immune receptors are 2',3'-cAMP/cGMP synthetases mediating cell death. Cell, 185, 2022
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7X5M
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![BU of 7x5m by Molmil](/molmil-images/mine/7x5m) | Tir-dsDNA complex, the initial binding state | 分子名称: | 2',3'- cyclic AMP, DNA (5'-D(P*AP*TP*TP*AP*A)-3'), DNA (5'-D(P*AP*TP*TP*TP*A)-3'), ... | 著者 | Tan, Y, Xu, C, Yu, D, Song, W, Wu, B, Schulze-Lefert, P, Chai, J. | 登録日 | 2022-03-05 | 公開日 | 2022-06-01 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.42 Å) | 主引用文献 | TIR domains of plant immune receptors are 2',3'-cAMP/cGMP synthetases mediating cell death. Cell, 185, 2022
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7X5K
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![BU of 7x5k by Molmil](/molmil-images/mine/7x5k) | Tir-dsDNA complex, the initial binding state | 分子名称: | DNA (43-MER), Flax rust resistance protein | 著者 | Tan, Y, Xu, C, Yu, D, Song, W, Wu, B, Schulze-Lefert, P, Chai, J. | 登録日 | 2022-03-04 | 公開日 | 2022-06-08 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | TIR domains of plant immune receptors are 2',3'-cAMP/cGMP synthetases mediating cell death. Cell, 185, 2022
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7X5H
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![BU of 7x5h by Molmil](/molmil-images/mine/7x5h) | Serotonin 5A (5-HT5A) receptor-Gi protein complex | 分子名称: | 3-(2-azanylethyl)-1H-indole-5-carboxamide, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ... | 著者 | Tan, Y, Xu, P, Huang, S, Xu, H.E, Jiang, Y. | 登録日 | 2022-03-04 | 公開日 | 2022-09-14 | 最終更新日 | 2022-09-21 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural insights into the ligand binding and G i coupling of serotonin receptor 5-HT 5A . Cell Discov, 8, 2022
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3VVP
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3VVR
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![BU of 3vvr by Molmil](/molmil-images/mine/3vvr) | Crystal structure of MATE in complex with MaD5 | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein, macrocyclic peptide | 著者 | Tanaka, Y, Ishitani, R, Nureki, O. | 登録日 | 2012-07-27 | 公開日 | 2013-04-03 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural basis for the drug extrusion mechanism by a MATE multidrug transporter. Nature, 496, 2013
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4GA4
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![BU of 4ga4 by Molmil](/molmil-images/mine/4ga4) | Crystal structure of AMP phosphorylase N-terminal deletion mutant | 分子名称: | PHOSPHATE ION, Putative thymidine phosphorylase | 著者 | Nishitani, Y, Aono, R, Nakamura, A, Sato, T, Atomi, H, Imanaka, T, Miki, K. | 登録日 | 2012-07-25 | 公開日 | 2013-05-15 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.51 Å) | 主引用文献 | Structure analysis of archaeal AMP phosphorylase reveals two unique modes of dimerization J.Mol.Biol., 425, 2013
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4GA5
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![BU of 4ga5 by Molmil](/molmil-images/mine/4ga5) | Crystal structure of AMP phosphorylase C-terminal deletion mutant in the apo-form | 分子名称: | Putative thymidine phosphorylase | 著者 | Nishitani, Y, Aono, R, Nakamura, A, Sato, T, Atomi, H, Imanaka, T, Miki, K. | 登録日 | 2012-07-25 | 公開日 | 2013-05-15 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Structure analysis of archaeal AMP phosphorylase reveals two unique modes of dimerization J.Mol.Biol., 425, 2013
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6LEP
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![BU of 6lep by Molmil](/molmil-images/mine/6lep) | Crystal structure of thiosulfate transporter YeeE inactive mutant - C91A | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Sulf_transp domain-containing protein, THIOSULFATE | 著者 | Tanaka, Y, Tsukazaki, T, Yoshikaie, K, Sugano, Y, Takeuchi, A, Uchino, S. | 登録日 | 2019-11-26 | 公開日 | 2020-09-02 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of a YeeE/YedE family protein engaged in thiosulfate uptake. Sci Adv, 6, 2020
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6LEO
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![BU of 6leo by Molmil](/molmil-images/mine/6leo) | Crystal structure of thiosulfate transporter YeeE from Spirochaeta thermophila | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Sulf_transp domain-containing protein, THIOSULFATE | 著者 | Tanaka, Y, Tsukazaki, T, Yoshikaie, K, Takeuchi, A, Uchino, S, Sugano, Y. | 登録日 | 2019-11-26 | 公開日 | 2020-09-02 | 最終更新日 | 2020-09-30 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | Crystal structure of a YeeE/YedE family protein engaged in thiosulfate uptake. Sci Adv, 6, 2020
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3VU4
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![BU of 3vu4 by Molmil](/molmil-images/mine/3vu4) | |
3VLU
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![BU of 3vlu by Molmil](/molmil-images/mine/3vlu) | Crystal structure of Sphingomonas sp. A1 alginate-binding protein AlgQ1 in complex with saturated trimannuronate | 分子名称: | AlgQ1, CALCIUM ION, beta-D-mannopyranuronic acid-(1-4)-beta-D-mannopyranuronic acid-(1-4)-beta-D-mannopyranuronic acid | 著者 | Nishitani, Y, Maruyama, Y, Itoh, T, Mikami, B, Hashimoto, W, Murata, K. | 登録日 | 2011-12-05 | 公開日 | 2012-01-25 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Recognition of heteropolysaccharide alginate by periplasmic solute-binding proteins of a bacterial ABC transporter Biochemistry, 51, 2012
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5ZOI
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![BU of 5zoi by Molmil](/molmil-images/mine/5zoi) | Crystal Structure of alpha1,3-Fucosyltransferase | 分子名称: | Alpha-(1,3)-fucosyltransferase FucT, [[(2S,3R,4S,5R)-5-(2-azanyl-6-oxidanylidene-1H-purin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2S,3S,4S,5R,6R)-6-methyl-3,4,5-tris(oxidanyl)oxan-2-yl] hydrogen phosphate | 著者 | Tan, Y, Yang, G. | 登録日 | 2018-04-13 | 公開日 | 2019-06-26 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (3.19 Å) | 主引用文献 | Directed evolution of an alpha 1,3-fucosyltransferase using a single-cell ultrahigh-throughput screening method. Sci Adv, 5, 2019
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7D79
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![BU of 7d79 by Molmil](/molmil-images/mine/7d79) | The structure of DcsB complex with its substrate analogue | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DltD domain-containing protein, ... | 著者 | Tang, Y, Zhou, J.H, Wang, G.Q. | 登録日 | 2020-10-03 | 公開日 | 2021-01-27 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.10411429 Å) | 主引用文献 | A Polyketide Cyclase That Forms Medium-Ring Lactones. J.Am.Chem.Soc., 143, 2021
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7DKG
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![BU of 7dkg by Molmil](/molmil-images/mine/7dkg) | Influenza H5N1 nucleoprotein (truncated) in complex with nucleotides | 分子名称: | Nucleoprotein, RNA (5'-R(P*(OMU)P*(OMU)P*(OMU))-3') | 著者 | Tang, Y.S, Xu, S, Chen, Y.W, Wang, J.H, Shaw, P.C. | 登録日 | 2020-11-24 | 公開日 | 2021-04-14 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal structures of influenza nucleoprotein complexed with nucleic acid provide insights into the mechanism of RNA interaction. Nucleic Acids Res., 49, 2021
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7DQK
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![BU of 7dqk by Molmil](/molmil-images/mine/7dqk) | A nicotine MATE transporter, Nicotiana tabacum MATE2 (NtMATE2) | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Tanaka, Y, Tsukazaki, T, Sasaki, A, Iwaki, S. | 登録日 | 2020-12-24 | 公開日 | 2021-06-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Crystal structures of a nicotine MATE transporter provide insight into its mechanism of substrate transport. Febs Lett., 595, 2021
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