5G4A
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![BU of 5g4a by Molmil](/molmil-images/mine/5g4a) | AadA in complex with ATP and magnesium | 分子名称: | 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, Aminoglycoside (3'') (9) adenylyltransferase, ... | 著者 | Stern, A.L, van der Verren, S, Selmer, M. | 登録日 | 2016-05-07 | 公開日 | 2017-11-29 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural mechanism of AadA, a dual-specificity aminoglycoside adenylyltransferase fromSalmonella enterica. J.Biol.Chem., 293, 2018
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5LUH
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![BU of 5luh by Molmil](/molmil-images/mine/5luh) | AadA E87Q in complex with ATP, calcium and streptomycin | 分子名称: | 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ... | 著者 | Stern, A.L, Van der Verren, S.E, Selmer, M. | 登録日 | 2016-09-08 | 公開日 | 2018-01-17 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Structural mechanism of AadA, a dual-specificity aminoglycoside adenylyltransferase fromSalmonella enterica. J.Biol.Chem., 293, 2018
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5LPA
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![BU of 5lpa by Molmil](/molmil-images/mine/5lpa) | AadA E87Q in complex with ATP, calcium and dihydrostreptomycin | 分子名称: | 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ... | 著者 | Stern, A.L, Van der Verren, S.E, Selmer, M. | 登録日 | 2016-08-12 | 公開日 | 2018-01-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural mechanism of AadA, a dual-specificity aminoglycoside adenylyltransferase fromSalmonella enterica. J.Biol.Chem., 293, 2018
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1FY8
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![BU of 1fy8 by Molmil](/molmil-images/mine/1fy8) | CRYSTAL STRUCTURE OF THE DELTAILE16VAL17 RAT ANIONIC TRYPSINOGEN-BPTI COMPLEX | 分子名称: | CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ... | 著者 | Pasternak, A, White, A, Jeffery, C.J, Ringe, D, Hedstrom, L. | 登録日 | 2000-09-28 | 公開日 | 2000-11-08 | 最終更新日 | 2017-10-04 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity. Protein Sci., 10, 2001
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3TGK
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![BU of 3tgk by Molmil](/molmil-images/mine/3tgk) | TRYPSINOGEN MUTANT D194N AND DELETION OF ILE 16-VAL 17 COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI) | 分子名称: | CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ... | 著者 | Pasternak, A, White, A, Jeffery, C.J, Medina, N, Cahoon, M, Ringe, D, Hedstrom, L. | 登録日 | 1998-07-19 | 公開日 | 2001-07-04 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity. Protein Sci., 10, 2001
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3TGI
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![BU of 3tgi by Molmil](/molmil-images/mine/3tgi) | WILD-TYPE RAT ANIONIC TRYPSIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI) | 分子名称: | BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ... | 著者 | Pasternak, A, Ringe, D, Hedstrom, L. | 登録日 | 1998-07-15 | 公開日 | 1998-12-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Comparison of Anionic and Cationic Trypsinogens: The Anionic Activation Domain is More Flexible in Solution and Differs in its Mode of Bpti Binding in the Crystal Structure Protein Sci., 8, 1999
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3TGJ
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![BU of 3tgj by Molmil](/molmil-images/mine/3tgj) | S195A TRYPSINOGEN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI) | 分子名称: | BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ... | 著者 | Pasternak, A, Ringe, D, Hedstrom, L. | 登録日 | 1998-07-16 | 公開日 | 1998-12-23 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Comparison of Anionic and Cationic Trypsinogens: The Anionic Activation Domain is More Flexible in Solution and Differs in its Mode of Bpti Binding in the Crystal Structure Protein Sci., 8, 1999
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1F5R
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![BU of 1f5r by Molmil](/molmil-images/mine/1f5r) | RAT TRYPSINOGEN MUTANT COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR | 分子名称: | CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, TRYPSIN II, ... | 著者 | Pasternak, A, White, A, Cahoon, M, Ringe, D, Hedstrom, L. | 登録日 | 2000-06-15 | 公開日 | 2001-07-04 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity. Protein Sci., 10, 2001
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1F7Z
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![BU of 1f7z by Molmil](/molmil-images/mine/1f7z) | RAT TRYPSINOGEN K15A COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR | 分子名称: | CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ... | 著者 | Pasternak, A, White, A, Jeffery, C.J, Medina, N, Cahoon, M, Ringe, D, Hedstrom, L. | 登録日 | 2000-06-28 | 公開日 | 2001-07-04 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity. Protein Sci., 10, 2001
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3T2N
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![BU of 3t2n by Molmil](/molmil-images/mine/3t2n) | Human hepsin protease in complex with the Fab fragment of an inhibitory antibody | 分子名称: | Antibody, Fab fragment, Heavy Chain, ... | 著者 | Koschubs, T, Dengl, S, Duerr, H, Kaluza, K, Georges, G, Hartl, C, Jennewein, S, Lanzendoerfer, M, Auer, J, Stern, A, Huang, K.-S, Kostrewa, D, Ries, S, Hansen, S, Kohnert, U, Cramer, P, Mundigl, O. | 登録日 | 2011-07-22 | 公開日 | 2011-12-28 | 最終更新日 | 2012-07-25 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Allosteric antibody inhibition of human hepsin protease. Biochem.J., 442, 2012
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1LSI
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![BU of 1lsi by Molmil](/molmil-images/mine/1lsi) | |
3K8C
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![BU of 3k8c by Molmil](/molmil-images/mine/3k8c) | |
3K7O
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![BU of 3k7o by Molmil](/molmil-images/mine/3k7o) | |
3K7S
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![BU of 3k7s by Molmil](/molmil-images/mine/3k7s) | |
3K7P
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![BU of 3k7p by Molmil](/molmil-images/mine/3k7p) | |
3M1P
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![BU of 3m1p by Molmil](/molmil-images/mine/3m1p) | |
1NPA
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![BU of 1npa by Molmil](/molmil-images/mine/1npa) | crystal structure of HIV-1 protease-hup | 分子名称: | (3S)-TETRAHYDROFURAN-3-YL (1R,2S)-3-[4-((1R)-2-{[(S)-AMINO(HYDROXY)METHYL]OXY}-2,3-DIHYDRO-1H-INDEN-1-YL)-2-BENZYL-3-OXOPYRROLIDIN-2-YL]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, POL polyprotein | 著者 | Smith III, A.B, Hirschmann, R, Pasternak, A, Yao, W, Sprengeler, P.A, Holloway, M.K, Kuo, L.C, Chen, Z, Darke, P.L, Schleif, W.A. | 登録日 | 2003-01-17 | 公開日 | 2004-01-27 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | An orally bioavailable pyrrolinone inhibitor of HIV-1 protease: computational analysis and X-ray crystal structure of the enzyme complex. J.MED.CHEM., 40, 1997
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