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PDB: 1 results

7M2K
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CDC34A-Ubiquitin-2ab inhibitor complex
Descriptor: 4-[(3',5'-dichloro[1,1'-biphenyl]-4-yl)methyl]-N-ethyl-1-(methoxyacetyl)piperidine-4-carboxamide, Ubiquitin, Ubiquitin-conjugating enzyme E2 R1
Authors:Ceccarelli, D.F, St-Cyr, D, Tyers, M, Sicheri, F.
Deposit date:2021-03-16
Release date:2021-11-03
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.47 Å)
Cite:Identification and optimization of molecular glue compounds that inhibit a noncovalent E2 enzyme-ubiquitin complex.
Sci Adv, 7, 2021

218853

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