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PDB: 2 results

6FYM
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BU of 6fym by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK1
Descriptor: 7,8-dimethyl-2-(pyrimidin-2-ylsulfanylmethyl)-3~{H}-quinazolin-4-one, NITRATE ION, Poly [ADP-ribose] polymerase 14
Authors:Karlberg, T, Thorsell, A.G, Kirby, I.T, Sreenivasan, R, Cohen, M.S, Schuler, H.
Deposit date:2018-03-12
Release date:2019-02-20
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:A Potent and Selective PARP11 Inhibitor Suggests Coupling between Cellular Localization and Catalytic Activity.
Cell Chem Biol, 25, 2018
6FZM
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BU of 6fzm by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK6
Descriptor: 4-[(8-methyl-4-oxidanylidene-7-prop-1-ynyl-3~{H}-quinazolin-2-yl)methylsulfanyl]benzoic acid, Poly [ADP-ribose] polymerase 14
Authors:Karlberg, T, Thorsell, A.G, Kirby, I.T, Sreenivasan, R, Cohen, M.S, Schuler, H.
Deposit date:2018-03-15
Release date:2019-02-20
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.67 Å)
Cite:A Potent and Selective PARP11 Inhibitor Suggests Coupling between Cellular Localization and Catalytic Activity.
Cell Chem Biol, 25, 2018

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