8T0J
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![BU of 8t0j by Molmil](/molmil-images/mine/8t0j) | Salmonella Typhimurium ArnD | Descriptor: | Probable 4-deoxy-4-formamido-L-arabinose-phosphoundecaprenol deformylase ArnD | Authors: | Sousa, M.C, Munoz-Escudero, D, Lee, M. | Deposit date: | 2023-06-01 | Release date: | 2023-10-18 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.59 Å) | Cite: | Structure and Function of ArnD. A Deformylase Essential for Lipid A Modification with 4-Amino-4-deoxy-l-arabinose and Polymyxin Resistance. Biochemistry, 62, 2023
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1KYI
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![BU of 1kyi by Molmil](/molmil-images/mine/1kyi) | HslUV (H. influenzae)-NLVS Vinyl Sulfone Inhibitor Complex | Descriptor: | 4-IODO-3-NITROPHENYL ACETYL-LEUCINYL-LEUCINYL-LEUCINYL-VINYLSULFONE, ADENOSINE-5'-TRIPHOSPHATE, ATP-dependent hsl protease ATP-binding subunit hslU, ... | Authors: | Sousa, M.C, Kessler, B.M, Overkleeft, H.S, McKay, D.B. | Deposit date: | 2002-02-04 | Release date: | 2002-05-15 | Last modified: | 2023-08-16 | Method: | X-RAY DIFFRACTION (3.1 Å) | Cite: | Crystal Structure of HslUV Complexed with a Vinyl Sulfone Inhibitor:
Corroboration of a Proposed Mechanism of Allosteric Activation of
HslV by HslU J.Mol.Biol., 318, 2002
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1BUP
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![BU of 1bup by Molmil](/molmil-images/mine/1bup) | T13S MUTANT OF BOVINE 70 KILODALTON HEAT SHOCK PROTEIN | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MAGNESIUM ION, ... | Authors: | Sousa, M.C, Mckay, D.B. | Deposit date: | 1998-09-03 | Release date: | 1998-09-09 | Last modified: | 2023-08-09 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | The hydroxyl of threonine 13 of the bovine 70-kDa heat shock cognate protein is essential for transducing the ATP-induced conformational change. Biochemistry, 37, 1998
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2BUP
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![BU of 2bup by Molmil](/molmil-images/mine/2bup) | T13G Mutant of the ATPASE fragment of Bovine HSC70 | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, CHLORIDE ION, ... | Authors: | Sousa, M.C, Mckay, D.B. | Deposit date: | 1998-09-08 | Release date: | 1998-09-16 | Last modified: | 2024-02-14 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | The hydroxyl of threonine 13 of the bovine 70-kDa heat shock cognate protein is essential for transducing the ATP-induced conformational change. Biochemistry, 37, 1998
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1G3I
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![BU of 1g3i by Molmil](/molmil-images/mine/1g3i) | CRYSTAL STRUCTURE OF THE HSLUV PROTEASE-CHAPERONE COMPLEX | Descriptor: | ADENOSINE-5'-TRIPHOSPHATE, ATP-DEPENDENT HSLU PROTEASE ATP-BINDING SUBUNIT HSLU, ATP-DEPENDENT PROTEASE HSLV | Authors: | Sousa, M.C, Trame, C.B, Tsuruta, H, Wilbanks, S.M, Reddy, V.S, McKay, D.B. | Deposit date: | 2000-10-24 | Release date: | 2000-11-22 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (3.41 Å) | Cite: | Crystal and solution structures of an HslUV protease-chaperone complex. Cell(Cambridge,Mass.), 103, 2000
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1G3K
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![BU of 1g3k by Molmil](/molmil-images/mine/1g3k) | |
8FTN
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![BU of 8ftn by Molmil](/molmil-images/mine/8ftn) | E. coli ArnA dehydrogenase domain mutant - N492A | Descriptor: | Bifunctional UDP-4-amino-4-deoxy-L-arabinose formyltransferase/UDP-glucuronic acid oxidase ArnA, SULFATE ION | Authors: | Sousa, M.C, Mitchell, M.E. | Deposit date: | 2023-01-12 | Release date: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Targeting the Conformational Change in ArnA Dehydrogenase for Selective Inhibition of Polymyxin Resistance. Biochemistry, 62, 2023
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8GJH
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![BU of 8gjh by Molmil](/molmil-images/mine/8gjh) | Salmonella ArnA | Descriptor: | Bifunctional polymyxin resistance protein ArnA, URIDINE-5'-DIPHOSPHATE-GLUCURONIC ACID | Authors: | Sousa, M.C, Mitchell, M.E, Gatzeva-Topalova, P.Z. | Deposit date: | 2023-03-15 | Release date: | 2023-08-02 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (3.6 Å) | Cite: | Targeting the Conformational Change in ArnA Dehydrogenase for Selective Inhibition of Polymyxin Resistance. Biochemistry, 62, 2023
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4LDQ
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![BU of 4ldq by Molmil](/molmil-images/mine/4ldq) | |
4LDR
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![BU of 4ldr by Molmil](/molmil-images/mine/4ldr) | Structure of the S283Y mutant of MRDI | Descriptor: | Methylthioribose-1-phosphate isomerase | Authors: | Sousa, M.C, Templeton, P.D, Metzner, S.I. | Deposit date: | 2013-06-25 | Release date: | 2013-07-31 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.292 Å) | Cite: | Structure of Mediator of RhoA-Dependent Invasion (MRDI) Explains Its Dual Function as a Metabolic Enzyme and a Mediator of Cell Invasion. Biochemistry, 52, 2013
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1JMV
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![BU of 1jmv by Molmil](/molmil-images/mine/1jmv) | |
1JJW
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![BU of 1jjw by Molmil](/molmil-images/mine/1jjw) | |
4OCA
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![BU of 4oca by Molmil](/molmil-images/mine/4oca) | Cryatal structure of ArnB K188A complexted with PLP and UDP-Ara4N | Descriptor: | (2R,3R,4S,5S)-3,4-dihydroxy-5-[({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methyl)amino]tetrahydro-2H-pyr an-2-yl [(2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl dihydrogen diphosphate, UDP-4-amino-4-deoxy-L-arabinose--oxoglutarate aminotransferase | Authors: | Sousa, M.C, Lee, M. | Deposit date: | 2014-01-08 | Release date: | 2014-03-12 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Structural Basis for Substrate Specificity in ArnB. A Key Enzyme in the Polymyxin Resistance Pathway of Gram-Negative Bacteria. Biochemistry, 53, 2014
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4Q3J
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![BU of 4q3j by Molmil](/molmil-images/mine/4q3j) | Crystal structure of NFkB-p65-degrading zinc protease family protein | Descriptor: | MAGNESIUM ION, NFkB-p65-degrading zinc protease family protein, ZINC ION | Authors: | Sousa, M.C, Turco, M.M. | Deposit date: | 2014-04-11 | Release date: | 2014-07-30 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (1.862 Å) | Cite: | The Structure and Specificity of the Type III Secretion System Effector NleC Suggest a DNA Mimicry Mechanism of Substrate Recognition. Biochemistry, 53, 2014
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3EFC
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![BU of 3efc by Molmil](/molmil-images/mine/3efc) | |
4HDJ
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![BU of 4hdj by Molmil](/molmil-images/mine/4hdj) | |
1U2M
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![BU of 1u2m by Molmil](/molmil-images/mine/1u2m) | Crystal Structure of Skp | Descriptor: | Histone-like protein HLP-1 | Authors: | Walton, T.A, Sousa, M.C. | Deposit date: | 2004-07-19 | Release date: | 2004-08-24 | Last modified: | 2017-10-11 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Crystal Structure of Skp, a Prefoldin-like Chaperone that Protects Soluble and Membrane Proteins from Aggregation Mol.Cell, 15, 2004
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1U9J
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![BU of 1u9j by Molmil](/molmil-images/mine/1u9j) | |
1YRW
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![BU of 1yrw by Molmil](/molmil-images/mine/1yrw) | |
1Z7E
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![BU of 1z7e by Molmil](/molmil-images/mine/1z7e) | Crystal structure of full length ArnA | Descriptor: | ADENOSINE-5'-TRIPHOSPHATE, URIDINE-5'-DIPHOSPHATE-GLUCURONIC ACID, protein ArnA | Authors: | Gatzeva-Topalova, P.Z, May, A.P, Sousa, M.C. | Deposit date: | 2005-03-24 | Release date: | 2005-06-07 | Last modified: | 2023-08-23 | Method: | X-RAY DIFFRACTION (3 Å) | Cite: | Structure and Mechanism of ArnA: Conformational Change Implies Ordered Dehydrogenase Mechanism in Key Enzyme for Polymyxin Resistance Structure, 13, 2005
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1Z73
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![BU of 1z73 by Molmil](/molmil-images/mine/1z73) | Crystal Structure of E. coli ArnA dehydrogenase (decarboxylase) domain, S433A mutant | Descriptor: | GLYCEROL, SULFATE ION, protein ArnA | Authors: | Gatzeva-Topalova, P.Z, May, A.P, Sousa, M.C. | Deposit date: | 2005-03-24 | Release date: | 2005-06-07 | Last modified: | 2023-08-23 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structure and Mechanism of ArnA: Conformational Change Implies Ordered Dehydrogenase Mechanism in Key Enzyme for Polymyxin Resistance Structure, 13, 2005
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1Z75
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![BU of 1z75 by Molmil](/molmil-images/mine/1z75) | Crystal Structure of ArnA dehydrogenase (decarboxylase) domain, R619M mutant | Descriptor: | GLYCEROL, SULFATE ION, protein ArnA | Authors: | Gatzeva-Topalova, P.Z, May, A.P, Sousa, M.C. | Deposit date: | 2005-03-24 | Release date: | 2005-06-07 | Last modified: | 2024-02-14 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Structure and Mechanism of ArnA: Conformational Change Implies Ordered Dehydrogenase Mechanism in Key Enzyme for Polymyxin Resistance Structure, 13, 2005
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1Z74
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![BU of 1z74 by Molmil](/molmil-images/mine/1z74) | |
1Z7B
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![BU of 1z7b by Molmil](/molmil-images/mine/1z7b) | |
3OG5
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![BU of 3og5 by Molmil](/molmil-images/mine/3og5) | Crystal Structure of BamA POTRA45 tandem | Descriptor: | Outer membrane protein assembly complex, YaeT protein | Authors: | Gatzeva-Topalova, P.Z, Warner, L.R, Pardi, A, Sousa, M.C. | Deposit date: | 2010-08-16 | Release date: | 2010-11-17 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2.69 Å) | Cite: | Structure and Flexibility of the Complete Periplasmic Domain of BamA: The Protein Insertion Machine of the Outer Membrane Structure, 18, 2010
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